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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2S,3R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-(2-methoxyethyl)-3,4-dihydro-2H-pyran-6-carboxamide —— C28H41N3O8
(2S,3R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-(2-methoxyethyl)-3,4-dihydro-2H-pyran-6-carboxamide
—— 4-[(2S,3R,4R)-2-ethoxy-3-(3-hydroxypropyl)-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C26H35N3O6
4-[(2S,3R,4R)-2-ethoxy-3-(3-hydroxypropyl)-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— (2S,3R,4R)-N-(cyclopropylmethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxamide —— C26H35N3O5
(2S,3R,4R)-N-(cyclopropylmethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,3R,4S)-N-[5-(2-aminoanilino)-5-oxopentyl]-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxamide —— C33H43N5O6
(2R,3R,4S)-N-[5-(2-aminoanilino)-5-oxopentyl]-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-6-carboxamide
—— (1R,6S)-9-methyl-N-[(1-phenylpyrazol-4-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide —— C19H25N5O
(1R,6S)-9-methyl-N-[(1-phenylpyrazol-4-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
—— (2S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamide —— C36H38N4O6
(2S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2S)-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]propanamide —— C13H15N3OS
(2S)-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]propanamide
—— 1-methyl-1-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-3-[(2-pyrazol-1-ylphenyl)methyl]urea —— C18H25N5O
1-methyl-1-[[(3R)-1-methylpyrrolidin-3-yl]methyl]-3-[(2-pyrazol-1-ylphenyl)methyl]urea
—— 4-[(2S,4S)-2-[2-(2-hydroxyethoxy)ethoxy]-6-(4-piperidin-1-ylpiperidine-1-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C31H44N4O6
4-[(2S,4S)-2-[2-(2-hydroxyethoxy)ethoxy]-6-(4-piperidin-1-ylpiperidine-1-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— (2S,3R,4R)-N-[5-(2-aminoanilino)-5-oxopentyl]-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide —— C36H49N5O8
(2S,3R,4R)-N-[5-(2-aminoanilino)-5-oxopentyl]-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2S,3S,4R)-N-(2-bicyclo[2.2.1]heptanyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide —— C32H45N3O7
(2S,3S,4R)-N-(2-bicyclo[2.2.1]heptanyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide
—— 4-[(2S,3R,4R)-6-[4-(1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C37H48N4O9
4-[(2S,3R,4R)-6-[4-(1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— (2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(4-hydroxybutoxy)-N-[2-[(5-nitropyridin-2-yl)amino]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide —— C28H34N6O7
(2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(4-hydroxybutoxy)-N-[2-[(5-nitropyridin-2-yl)amino]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide
—— 1-methyl-1-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-3-[(2-pyrazol-1-ylphenyl)methyl]urea —— C18H25N5O
1-methyl-1-[[(3S)-1-methylpyrrolidin-3-yl]methyl]-3-[(2-pyrazol-1-ylphenyl)methyl]urea
—— (2S,4S)-N-(2-aminophenyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carboxamide —— C27H32N4O5
(2S,4S)-N-(2-aminophenyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,4R)-N-(1H-benzimidazol-2-ylmethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide —— C29H33N5O6
(2R,4R)-N-(1H-benzimidazol-2-ylmethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2S)-N,N-dimethyl-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]propanamide —— C15H19N3OS
(2S)-N,N-dimethyl-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]propanamide
—— 4-[(2R,4R)-6-(azocane-1-carbonyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C32H39N3O5
4-[(2R,4R)-6-(azocane-1-carbonyl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— (2R)-N,N-dimethyl-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]propanamide —— C15H19N3OS
(2R)-N,N-dimethyl-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]propanamide
—— N-[2-[[(2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-6-[4-(2-oxo-3H-benzimidazol-1-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-pyran-2-yl]oxy]ethyl]-N-(2-hydroxyethyl)-4-methoxybenzenesulfonamide —— C40H46N6O9S
N-[2-[[(2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-6-[4-(2-oxo-3H-benzimidazol-1-yl)piperidine-1-carbonyl]-3,4-dihydro-2H-pyran-2-yl]oxy]ethyl]-N-(2-hydroxyethyl)-4-methoxybenzenesulfonamide
—— 3-[1-[(2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carbonyl]piperidin-4-yl]-1H-benzimidazol-2-one —— C37H39N5O6
3-[1-[(2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carbonyl]piperidin-4-yl]-1H-benzimidazol-2-one
—— tert-butyl N-[(2S)-2-methyl-3-[(1-methyl-3-phenylpyrazole-4-carbonyl)amino]propyl]carbamate —— C20H28N4O3
tert-butyl N-[(2S)-2-methyl-3-[(1-methyl-3-phenylpyrazole-4-carbonyl)amino]propyl]carbamate
—— 4-[(2S,3S,4R)-6-(azocane-1-carbonyl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C29H41N3O5
4-[(2S,3S,4R)-6-(azocane-1-carbonyl)-2-ethoxy-3-(3-hydroxypropyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— (2S,3R,4R)-N-benzyl-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide —— C32H41N3O7
(2S,3R,4R)-N-benzyl-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,3R,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-(2-hydroxyphenyl)-3,4-dihydro-2H-pyran-6-carboxamide —— C31H39N3O8
(2R,3R,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-(2-hydroxyphenyl)-3,4-dihydro-2H-pyran-6-carboxamide
—— (2S,3S,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]-3,4-dihydro-2H-pyran-6-carboxamide —— C29H40N4O6
(2S,3S,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,4R)-N-(2-bicyclo[2.2.1]heptanyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide —— C28H37N3O6
(2R,4R)-N-(2-bicyclo[2.2.1]heptanyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,4R)-N-benzyl-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide —— C28H33N3O6
(2R,4R)-N-benzyl-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,4R)-N-(2,2-dimethoxyethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(4-hydroxybutoxy)-N-methyl-3,4-dihydro-2H-pyran-6-carboxamide —— C26H37N3O7
(2R,4R)-N-(2,2-dimethoxyethyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(4-hydroxybutoxy)-N-methyl-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,3S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamide —— C36H46N4O8
(2R,3S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-3,4-dihydro-2H-pyran-6-carboxamide
—— 4-[(2S,3S,4R)-2-ethoxy-3-(3-hydroxypropyl)-6-(4-piperidin-1-ylpiperidine-1-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C32H46N4O5
4-[(2S,3S,4R)-2-ethoxy-3-(3-hydroxypropyl)-6-(4-piperidin-1-ylpiperidine-1-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— (2R,3R,4S)-N-(2-aminophenyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide —— C31H40N4O7
(2R,3R,4S)-N-(2-aminophenyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carboxamide
—— 8-[(2S,3S,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carbonyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one —— C38H49N5O8
8-[(2S,3S,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-3,4-dihydro-2H-pyran-6-carbonyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
—— N-[2-[[(2R,4R)-6-[4-(1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3,4-dihydro-2H-pyran-2-yl]oxy]ethyl]-N-(2-hydroxyethyl)-4-methoxybenzenesulfonamide —— C40H47N5O10S
N-[2-[[(2R,4R)-6-[4-(1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3,4-dihydro-2H-pyran-2-yl]oxy]ethyl]-N-(2-hydroxyethyl)-4-methoxybenzenesulfonamide
—— N-[2-[[(2S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-pyran-2-yl]oxy]ethyl]-N-(2-hydroxyethyl)-4-methoxybenzenesulfonamide —— C32H40N4O9S
N-[2-[[(2S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-pyran-2-yl]oxy]ethyl]-N-(2-hydroxyethyl)-4-methoxybenzenesulfonamide
—— 4-[(2R,4R)-2-[2-(2-hydroxyethoxy)ethoxy]-6-(4-piperidin-1-ylpiperidine-1-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C31H44N4O6
4-[(2R,4R)-2-[2-(2-hydroxyethoxy)ethoxy]-6-(4-piperidin-1-ylpiperidine-1-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— 4-[(2S,4S)-2-[2-(2-hydroxyethoxy)ethoxy]-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C25H33N3O7
4-[(2S,4S)-2-[2-(2-hydroxyethoxy)ethoxy]-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— 3-[[(1S)-cyclohex-3-en-1-yl]methyl]-1-(3-imidazol-1-ylpropyl)-1-methylurea —— C15H24N4O
3-[[(1S)-cyclohex-3-en-1-yl]methyl]-1-(3-imidazol-1-ylpropyl)-1-methylurea
—— 4-[(2S,4S)-2-(4-hydroxybutoxy)-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C31H45N3O9
4-[(2S,4S)-2-(4-hydroxybutoxy)-6-(1,4,7,10-tetraoxa-13-azacyclopentadecane-13-carbonyl)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— (2R,3R,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-N-(2-methoxyethyl)-3,4-dihydro-2H-pyran-6-carboxamide —— C25H35N3O6
(2R,3R,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-N-(2-methoxyethyl)-3,4-dihydro-2H-pyran-6-carboxamide
—— 2-[[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl-methylamino]methyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C17H18N4O3
2-[[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl-methylamino]methyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— 4-[(2R,4R)-6-(azocane-1-carbonyl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C28H39N3O6
4-[(2R,4R)-6-(azocane-1-carbonyl)-2-[2-(2-hydroxyethoxy)ethoxy]-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— (2R,3R,4S)-N-cyclohexyl-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-methyl-3,4-dihydro-2H-pyran-6-carboxamide —— C32H47N3O7
(2R,3R,4S)-N-cyclohexyl-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-[2-[2-(2-hydroxyethoxy)ethoxy]ethyl]-N-methyl-3,4-dihydro-2H-pyran-6-carboxamide
—— (2S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-N-(2-methoxyethyl)-3,4-dihydro-2H-pyran-6-carboxamide —— C28H33N3O6
(2S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-N-(2-methoxyethyl)-3,4-dihydro-2H-pyran-6-carboxamide
—— (2R,3S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-3,4-dihydro-2H-pyran-6-carboxamide —— C36H38N4O5S
(2R,3S,4S)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-ethoxy-3-(3-hydroxypropyl)-N-[4-(6-methyl-1,3-benzothiazol-2-yl)phenyl]-3,4-dihydro-2H-pyran-6-carboxamide
—— (2S,4S)-N-(2-bicyclo[2.2.1]heptanyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carboxamide —— C32H37N3O5
(2S,4S)-N-(2-bicyclo[2.2.1]heptanyl)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-[[4-(hydroxymethyl)phenyl]methoxy]-3,4-dihydro-2H-pyran-6-carboxamide
—— 4-[(2R,4R)-6-[4-(1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one —— C33H40N4O7
4-[(2R,4R)-6-[4-(1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-4-yl]-1,5-dimethyl-2-phenylpyrazol-3-one
—— N-[2-[[(2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-6-(4-piperidin-1-ylpiperidine-1-carbonyl)-3,4-dihydro-2H-pyran-2-yl]oxy]ethyl]-N-(2-hydroxyethyl)-4-methoxybenzenesulfonamide —— C38H51N5O8S
N-[2-[[(2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-6-(4-piperidin-1-ylpiperidine-1-carbonyl)-3,4-dihydro-2H-pyran-2-yl]oxy]ethyl]-N-(2-hydroxyethyl)-4-methoxybenzenesulfonamide
—— 3-[1-[(2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carbonyl]piperidin-4-yl]-1H-benzimidazol-2-one —— C33H39N5O6
3-[1-[(2R,4R)-4-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-2-(4-hydroxybutoxy)-3,4-dihydro-2H-pyran-6-carbonyl]piperidin-4-yl]-1H-benzimidazol-2-one
—— tert-butyl N-[(2R)-2-methyl-3-[(1-methyl-3-phenylpyrazole-4-carbonyl)amino]propyl]carbamate —— C20H28N4O3
tert-butyl N-[(2R)-2-methyl-3-[(1-methyl-3-phenylpyrazole-4-carbonyl)amino]propyl]carbamate