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中文名称 英文名称 CAS号 化学式 结构式图片
—— [(2R)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)methanone —— C13H18N2O2S
[(2R)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)methanone
—— 2-[4-chloro-2-[1-[(3R)-1-oxaspiro[4.4]nonan-3-yl]triazol-4-yl]phenoxy]acetamide —— C18H21ClN4O3
2-[4-chloro-2-[1-[(3R)-1-oxaspiro[4.4]nonan-3-yl]triazol-4-yl]phenoxy]acetamide
—— (3R)-3-butyl-1-methyl-4-[4-(1H-1,2,4-triazol-5-yl)benzoyl]piperazin-2-one —— C18H23N5O2
(3R)-3-butyl-1-methyl-4-[4-(1H-1,2,4-triazol-5-yl)benzoyl]piperazin-2-one
—— N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-(2-phenylimidazol-1-yl)acetamide —— C20H19N3O3
N-[[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-(2-phenylimidazol-1-yl)acetamide
—— 3-(2-amino-1,3-thiazol-4-yl)-N-[(1S)-1-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]ethyl]propanamide —— C19H23N5OS
3-(2-amino-1,3-thiazol-4-yl)-N-[(1S)-1-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]ethyl]propanamide
—— 5-cyclopropyl-N-[(4S)-6,6-dimethyl-1-phenyl-5,7-dihydro-4H-indazol-4-yl]-1H-pyrazole-3-carboxamide —— C22H25N5O
5-cyclopropyl-N-[(4S)-6,6-dimethyl-1-phenyl-5,7-dihydro-4H-indazol-4-yl]-1H-pyrazole-3-carboxamide
—— (3S)-3-butyl-1-methyl-4-[4-(1H-1,2,4-triazol-5-yl)benzoyl]piperazin-2-one —— C18H23N5O2
(3S)-3-butyl-1-methyl-4-[4-(1H-1,2,4-triazol-5-yl)benzoyl]piperazin-2-one
—— [(3S)-3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone —— C21H21N3O2
[(3S)-3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-[4-(1H-pyrazol-5-yl)phenyl]methanone
—— [3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-[(3R)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone —— C19H22N6O2
[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-[(3R)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone
—— 5-(3-fluorophenyl)-N-[(1S)-1-imidazo[1,2-a]pyrimidin-2-ylpropyl]-1H-pyrazole-4-carboxamide —— C19H17FN6O
5-(3-fluorophenyl)-N-[(1S)-1-imidazo[1,2-a]pyrimidin-2-ylpropyl]-1H-pyrazole-4-carboxamide
—— N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C20H25N5O2
N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— N-methyl-2-(1-methylimidazol-2-yl)-N-[[(3S)-1-phenylpyrrolidin-3-yl]methyl]benzamide —— C23H26N4O
N-methyl-2-(1-methylimidazol-2-yl)-N-[[(3S)-1-phenylpyrrolidin-3-yl]methyl]benzamide
—— [(2S)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)methanone —— C13H18N2O2S
[(2S)-2-(hydroxymethyl)-2,5-dihydropyrrol-1-yl]-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)methanone
—— 3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(1S)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide —— C20H24FN5O
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(1S)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide
—— N,3-dimethyl-N-[(1R)-1-(3-phenyl-1H-pyrazol-5-yl)ethyl]-1-propylpyrazole-4-carboxamide —— C20H25N5O
N,3-dimethyl-N-[(1R)-1-(3-phenyl-1H-pyrazol-5-yl)ethyl]-1-propylpyrazole-4-carboxamide
—— N-methyl-2-(1-methylimidazol-2-yl)-N-[[(3R)-1-phenylpyrrolidin-3-yl]methyl]benzamide —— C23H26N4O
N-methyl-2-(1-methylimidazol-2-yl)-N-[[(3R)-1-phenylpyrrolidin-3-yl]methyl]benzamide
—— [(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-[1-(2-methoxyphenyl)pyrazol-4-yl]methanone —— C20H22N4O3
[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-[1-(2-methoxyphenyl)pyrazol-4-yl]methanone
—— 5-(3-fluorophenyl)-N-[(1R)-1-imidazo[1,2-a]pyrimidin-2-ylpropyl]-1H-pyrazole-4-carboxamide —— C19H17FN6O
5-(3-fluorophenyl)-N-[(1R)-1-imidazo[1,2-a]pyrimidin-2-ylpropyl]-1H-pyrazole-4-carboxamide
—— [3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-[(3S)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone —— C19H22N6O2
[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]-[(3S)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]methanone
—— 3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(1R)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide —— C20H24FN5O
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(1R)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]propanamide
—— (2S)-N-[2-[2-(methylsulfanylmethyl)-1,3-thiazol-4-yl]ethyl]-2-pyrazol-1-ylbutanamide —— C14H20N4OS2
(2S)-N-[2-[2-(methylsulfanylmethyl)-1,3-thiazol-4-yl]ethyl]-2-pyrazol-1-ylbutanamide
—— N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-(2-phenylimidazol-1-yl)acetamide —— C20H19N3O3
N-[[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]methyl]-2-(2-phenylimidazol-1-yl)acetamide
—— 5-cyclopropyl-N-[(4R)-6,6-dimethyl-1-phenyl-5,7-dihydro-4H-indazol-4-yl]-1H-pyrazole-3-carboxamide —— C22H25N5O
5-cyclopropyl-N-[(4R)-6,6-dimethyl-1-phenyl-5,7-dihydro-4H-indazol-4-yl]-1H-pyrazole-3-carboxamide
—— 2-[4-chloro-2-[1-[(3S)-1-oxaspiro[4.4]nonan-3-yl]triazol-4-yl]phenoxy]acetamide —— C18H21ClN4O3
2-[4-chloro-2-[1-[(3S)-1-oxaspiro[4.4]nonan-3-yl]triazol-4-yl]phenoxy]acetamide
—— (3R)-3-[2-(2-methoxyphenyl)-1,2,4-triazol-3-yl]-3,4-dihydro-2H-1lambda6,2-benzothiazine 1,1-dioxide —— C17H16N4O3S
(3R)-3-[2-(2-methoxyphenyl)-1,2,4-triazol-3-yl]-3,4-dihydro-2H-1lambda6,2-benzothiazine 1,1-dioxide
—— 3-(3-methoxyphenyl)-N-[(3R)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide —— C21H24N4O2S
3-(3-methoxyphenyl)-N-[(3R)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
—— N-[(1S)-1-[1-(2,4-difluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-methoxypyrimidine-5-carboxamide —— C18H17F2N5O2
N-[(1S)-1-[1-(2,4-difluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-methoxypyrimidine-5-carboxamide
—— (3S)-3-[2-(2-methoxyphenyl)-1,2,4-triazol-3-yl]-3,4-dihydro-2H-1lambda6,2-benzothiazine 1,1-dioxide —— C17H16N4O3S
(3S)-3-[2-(2-methoxyphenyl)-1,2,4-triazol-3-yl]-3,4-dihydro-2H-1lambda6,2-benzothiazine 1,1-dioxide
—— 3-(2-amino-1,3-thiazol-4-yl)-N-[(1R)-1-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]ethyl]propanamide —— C19H23N5OS
3-(2-amino-1,3-thiazol-4-yl)-N-[(1R)-1-[5-methyl-1-(2-methylphenyl)pyrazol-4-yl]ethyl]propanamide
—— (5R)-2-(1-phenyltriazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5R)-2-(1-phenyltriazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— 2-[(2R)-2-[4-(7-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)triazol-1-yl]propyl]-3-methylpyridine —— C21H24N4O3
2-[(2R)-2-[4-(7-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)triazol-1-yl]propyl]-3-methylpyridine
—— ethyl (2S)-2-[3-(4-fluorophenyl)triazolo[4,5-d]pyrimidin-7-yl]sulfanylbutanoate —— C16H16FN5O2S
ethyl (2S)-2-[3-(4-fluorophenyl)triazolo[4,5-d]pyrimidin-7-yl]sulfanylbutanoate
—— N-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]cyclopropanesulfonamide —— C18H23N3O2S
N-[(4S)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]cyclopropanesulfonamide
—— (5S)-2-(1-phenyltriazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one —— C20H25N5O2
(5S)-2-(1-phenyltriazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
—— [(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-(5-propyl-1H-pyrazol-3-yl)methanone —— C20H23N5O2
[(3R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-(5-propyl-1H-pyrazol-3-yl)methanone
—— 2-[(2S)-2-[4-(7-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)triazol-1-yl]propyl]-3-methylpyridine —— C21H24N4O3
2-[(2S)-2-[4-(7-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-8-yl)triazol-1-yl]propyl]-3-methylpyridine
—— N-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]cyclopropanesulfonamide —— C18H23N3O2S
N-[(4R)-1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]cyclopropanesulfonamide
—— N-[(1R)-1-[1-(2,4-difluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-methoxypyrimidine-5-carboxamide —— C18H17F2N5O2
N-[(1R)-1-[1-(2,4-difluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-methoxypyrimidine-5-carboxamide
—— 3-(3-methoxyphenyl)-N-[(3S)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide —— C21H24N4O2S
3-(3-methoxyphenyl)-N-[(3S)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
—— N-[(1S)-1-[1-(2,4-difluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(5-methylpyrazol-1-yl)acetamide —— C18H19F2N5O
N-[(1S)-1-[1-(2,4-difluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(5-methylpyrazol-1-yl)acetamide
—— (3S)-3-butyl-1-methyl-4-(2-methyl-5-phenylpyrazole-3-carbonyl)piperazin-2-one —— C20H26N4O2
(3S)-3-butyl-1-methyl-4-(2-methyl-5-phenylpyrazole-3-carbonyl)piperazin-2-one
—— 3-(2-methylpropyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1,2-oxazole-5-carboxamide —— C18H21N5O2
3-(2-methylpropyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1,2-oxazole-5-carboxamide
—— 2-(1-adamantyl)-N-[(2R)-1-(1,3-thiazol-5-yl)propan-2-yl]acetamide —— C18H26N2OS
2-(1-adamantyl)-N-[(2R)-1-(1,3-thiazol-5-yl)propan-2-yl]acetamide
—— 3-(4-methoxyphenyl)-N-methyl-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide —— C17H18N4O3
3-(4-methoxyphenyl)-N-methyl-N-[(1R)-1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
—— (3R)-3-butyl-1-methyl-4-(2-methyl-5-phenylpyrazole-3-carbonyl)piperazin-2-one —— C20H26N4O2
(3R)-3-butyl-1-methyl-4-(2-methyl-5-phenylpyrazole-3-carbonyl)piperazin-2-one
—— 3-(3-methoxyphenyl)-N-[(1S)-1-(2-methylpyrazol-3-yl)propyl]-1H-pyrazole-5-carboxamide —— C18H21N5O2
3-(3-methoxyphenyl)-N-[(1S)-1-(2-methylpyrazol-3-yl)propyl]-1H-pyrazole-5-carboxamide
—— 5-(3-fluorophenyl)-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide —— C13H12FN7O
5-(3-fluorophenyl)-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
—— 5-(3-fluorophenyl)-N-[(1R)-1-(2H-tetrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide —— C13H12FN7O
5-(3-fluorophenyl)-N-[(1R)-1-(2H-tetrazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
—— 3-(2-methylpropyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1,2-oxazole-5-carboxamide —— C18H21N5O2
3-(2-methylpropyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1,2-oxazole-5-carboxamide
—— (3S,5R,8S)-3-methyl-8-(pentoxymethyl)-3-[2-(prop-2-enylamino)-1,3-thiazol-4-yl]-2,7-dioxaspiro[4.4]nonane-1,6-dione —— C20H28N2O5S
(3S,5R,8S)-3-methyl-8-(pentoxymethyl)-3-[2-(prop-2-enylamino)-1,3-thiazol-4-yl]-2,7-dioxaspiro[4.4]nonane-1,6-dione