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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[3-(5-methyl-1H-pyrazol-4-yl)propyl]-3-[[(2R)-oxolan-2-yl]methyl]urea —— C13H22N4O2
1-[3-(5-methyl-1H-pyrazol-4-yl)propyl]-3-[[(2R)-oxolan-2-yl]methyl]urea
—— 3-methyl-N-[(1S)-1-(2-propan-2-yl-1,3-thiazol-4-yl)ethyl]pyridazine-4-carboxamide —— C14H18N4OS
3-methyl-N-[(1S)-1-(2-propan-2-yl-1,3-thiazol-4-yl)ethyl]pyridazine-4-carboxamide
—— 2-[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]-N-[[(1R,2S)-2-phenylcyclopropyl]methyl]acetamide —— C20H20N2O3
2-[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]-N-[[(1R,2S)-2-phenylcyclopropyl]methyl]acetamide
—— 5-methyl-1-[4-[(2S)-2-phenylazetidine-1-carbonyl]phenyl]pyrazole-4-carboxylic acid —— C21H19N3O3
5-methyl-1-[4-[(2S)-2-phenylazetidine-1-carbonyl]phenyl]pyrazole-4-carboxylic acid
—— (1S,2S)-2-(4-chlorophenyl)-N-[2-(2,5-dimethyl-1,3-oxazol-4-yl)ethyl]cyclopropane-1-carboxamide —— C17H19ClN2O2
(1S,2S)-2-(4-chlorophenyl)-N-[2-(2,5-dimethyl-1,3-oxazol-4-yl)ethyl]cyclopropane-1-carboxamide
—— 3-methyl-N-[(1R)-1-(2-propan-2-yl-1,3-thiazol-4-yl)ethyl]pyridazine-4-carboxamide —— C14H18N4OS
3-methyl-N-[(1R)-1-(2-propan-2-yl-1,3-thiazol-4-yl)ethyl]pyridazine-4-carboxamide
—— [(1S)-3-methyl-1-pyridin-2-ylbutyl] 1,5-dimethylpyrazole-4-carboxylate —— C16H21N3O2
[(1S)-3-methyl-1-pyridin-2-ylbutyl] 1,5-dimethylpyrazole-4-carboxylate
—— 1-(4-bromophenyl)-N-[(1R,2S)-1-hydroxy-2,3-dihydro-1H-inden-2-yl]-5-methylpyrazole-4-carboxamide —— C20H18BrN3O2
1-(4-bromophenyl)-N-[(1R,2S)-1-hydroxy-2,3-dihydro-1H-inden-2-yl]-5-methylpyrazole-4-carboxamide
—— N-[[1-[(2S)-2-hydroxypropyl]piperidin-4-yl]methyl]-N-methyl-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetamide —— C22H31N3O3
N-[[1-[(2S)-2-hydroxypropyl]piperidin-4-yl]methyl]-N-methyl-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetamide
—— 3-[(2R,6R)-2,6-dimethyloxan-4-yl]sulfanyl-5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazole —— C20H23N3O2S
3-[(2R,6R)-2,6-dimethyloxan-4-yl]sulfanyl-5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazole
—— [(2R)-1-[[(1S)-1-(2,4-dichlorophenyl)ethyl]amino]-1-oxopropan-2-yl] 5-methyl-1-pyridin-4-ylpyrazole-4-carboxylate —— C21H20Cl2N4O3
[(2R)-1-[[(1S)-1-(2,4-dichlorophenyl)ethyl]amino]-1-oxopropan-2-yl] 5-methyl-1-pyridin-4-ylpyrazole-4-carboxylate
—— 1-[3-(5-methyl-1H-pyrazol-4-yl)propyl]-3-[(1R)-1-[(2R)-oxolan-2-yl]ethyl]urea —— C14H24N4O2
1-[3-(5-methyl-1H-pyrazol-4-yl)propyl]-3-[(1R)-1-[(2R)-oxolan-2-yl]ethyl]urea
—— 1-[3-(5-methyl-1H-pyrazol-4-yl)propyl]-3-[[(2S)-oxolan-2-yl]methyl]urea —— C13H22N4O2
1-[3-(5-methyl-1H-pyrazol-4-yl)propyl]-3-[[(2S)-oxolan-2-yl]methyl]urea
—— (1-tert-butyl-5-methylpyrazol-4-yl)-[(2R)-2,4-dimethylpiperazin-1-yl]methanone —— C15H26N4O
(1-tert-butyl-5-methylpyrazol-4-yl)-[(2R)-2,4-dimethylpiperazin-1-yl]methanone
—— N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-5-methyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide —— C17H22FN3O2
N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-5-methyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
—— (4S)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-oxoimidazolidine-4-carboxamide —— C16H18FN5O2
(4S)-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-oxoimidazolidine-4-carboxamide
—— N,2-dimethyl-6-oxo-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1H-pyridine-3-carboxamide —— C18H19N5O2
N,2-dimethyl-6-oxo-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1H-pyridine-3-carboxamide
—— N,2-dimethyl-6-oxo-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1H-pyridine-3-carboxamide —— C18H19N5O2
N,2-dimethyl-6-oxo-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]-1H-pyridine-3-carboxamide
—— (2S)-3-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]propane-1,2-diol —— C14H17NO3S
(2S)-3-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]propane-1,2-diol
—— methyl (2R)-2-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methylsulfanyl]propanoate —— C13H15NO4S
methyl (2R)-2-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methylsulfanyl]propanoate
—— 1-(4-fluorophenyl)-5-methyl-N-[(1R)-1-[4-(triazol-1-yl)phenyl]ethyl]pyrazole-4-carboxamide —— C21H19FN6O
1-(4-fluorophenyl)-5-methyl-N-[(1R)-1-[4-(triazol-1-yl)phenyl]ethyl]pyrazole-4-carboxamide
—— N-[(S)-(3-chlorophenyl)-pyridin-2-ylmethyl]-5-methyl-1H-pyrazole-4-carboxamide —— C17H15ClN4O
N-[(S)-(3-chlorophenyl)-pyridin-2-ylmethyl]-5-methyl-1H-pyrazole-4-carboxamide
—— [(1R)-1-(1-phenylpyrazol-4-yl)ethyl] 1,5-dimethylpyrazole-4-carboxylate —— C17H18N4O2
[(1R)-1-(1-phenylpyrazol-4-yl)ethyl] 1,5-dimethylpyrazole-4-carboxylate
—— N-[(1R)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-1,5-dimethylpyrazole-4-carboxamide —— C13H18N6O
N-[(1R)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-1,5-dimethylpyrazole-4-carboxamide
—— N-[(1S)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-1,5-dimethylpyrazole-4-carboxamide —— C13H18N6O
N-[(1S)-1-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-yl)ethyl]-1,5-dimethylpyrazole-4-carboxamide
—— N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-5-methyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide —— C17H22FN3O2
N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]-5-methyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
—— 3-[(2S,6S)-2,6-dimethyloxan-4-yl]sulfanyl-5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazole —— C20H23N3O2S
3-[(2S,6S)-2,6-dimethyloxan-4-yl]sulfanyl-5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazole
—— N-[(1S)-1-(1-phenyltriazol-4-yl)ethyl]thian-4-amine —— C15H20N4S
N-[(1S)-1-(1-phenyltriazol-4-yl)ethyl]thian-4-amine
—— 5-methyl-N-[(3S,4R)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]-1H-pyrazole-4-carboxamide —— C16H23N5OS
5-methyl-N-[(3S,4R)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]-1H-pyrazole-4-carboxamide
—— 3-(1,3-dimethylpyrazol-4-yl)-1-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]propan-1-one —— C16H22N4O
3-(1,3-dimethylpyrazol-4-yl)-1-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]propan-1-one
—— 2-(3-methoxyphenyl)-5-methyl-N-[(2S)-2-methyl-3-morpholin-4-ylpropyl]-1H-imidazole-4-carboxamide —— C20H28N4O3
2-(3-methoxyphenyl)-5-methyl-N-[(2S)-2-methyl-3-morpholin-4-ylpropyl]-1H-imidazole-4-carboxamide
—— [(1S)-1-(1-phenylpyrazol-4-yl)ethyl] 1,5-dimethylpyrazole-4-carboxylate —— C17H18N4O2
[(1S)-1-(1-phenylpyrazol-4-yl)ethyl] 1,5-dimethylpyrazole-4-carboxylate
—— 1-(4-bromophenyl)-N-[(1R,2R)-1-hydroxy-2,3-dihydro-1H-inden-2-yl]-5-methylpyrazole-4-carboxamide —— C20H18BrN3O2
1-(4-bromophenyl)-N-[(1R,2R)-1-hydroxy-2,3-dihydro-1H-inden-2-yl]-5-methylpyrazole-4-carboxamide
—— 5-methyl-N-[(3S,4S)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]-1H-pyrazole-4-carboxamide —— C16H23N5OS
5-methyl-N-[(3S,4S)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]-1H-pyrazole-4-carboxamide
—— 1-[3-(5-methyl-1H-pyrazol-4-yl)propyl]-3-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]urea —— C14H24N4O2
1-[3-(5-methyl-1H-pyrazol-4-yl)propyl]-3-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]urea
—— 3-[(2S,6R)-2,6-dimethyloxan-4-yl]sulfanyl-5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazole —— C20H23N3O2S
3-[(2S,6R)-2,6-dimethyloxan-4-yl]sulfanyl-5-(2-methylfuran-3-yl)-4-phenyl-1,2,4-triazole
—— N-[(1S)-1-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]ethyl]-2-methyl-1H-pyrrole-3-carboxamide —— C16H15ClN4O2
N-[(1S)-1-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]ethyl]-2-methyl-1H-pyrrole-3-carboxamide
—— 1-(3,5-dimethyl-1,2-oxazol-4-yl)-3-[(1R)-1-(4-imidazol-1-ylphenyl)ethyl]-1-methylurea —— C18H21N5O2
1-(3,5-dimethyl-1,2-oxazol-4-yl)-3-[(1R)-1-(4-imidazol-1-ylphenyl)ethyl]-1-methylurea
—— 1-benzyl-3-[[4-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]urea —— C42H39N3O5S
1-benzyl-3-[[4-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methyl]urea
—— 4-[[4-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-4-oxobutanoic acid —— C38H36N2O7S
4-[[4-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]methylamino]-4-oxobutanoic acid
—— 1-(3,5-dimethyl-1,2-oxazol-4-yl)-3-[(1S)-1-(4-imidazol-1-ylphenyl)ethyl]-1-methylurea —— C18H21N5O2
1-(3,5-dimethyl-1,2-oxazol-4-yl)-3-[(1S)-1-(4-imidazol-1-ylphenyl)ethyl]-1-methylurea
—— 5-[(1S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsulfonyl]ethyl]-3-methyl-1,2,4-oxadiazole —— C11H15N3O4S
5-[(1S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsulfonyl]ethyl]-3-methyl-1,2,4-oxadiazole
—— N-[3-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]acetamide —— C35H32N2O5S
N-[3-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]acetamide
—— N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]pyridine-3-carboxamide —— C32H30N6O5S
N-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]pyridine-3-carboxamide
—— 1-benzyl-3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea —— C33H32N6O5S
1-benzyl-3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea
—— 1-[3-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]-3-ethylurea —— C36H35N3O5S
1-[3-[(2S,4S,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-1,3-dioxan-2-yl]phenyl]-3-ethylurea
—— 1-benzyl-3-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]urea —— C34H34N6O4S
1-benzyl-3-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methyl]urea
—— 4-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methylamino]-4-oxobutanoic acid —— C30H31N5O7S
4-[[4-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]methylamino]-4-oxobutanoic acid
—— 1-ethyl-3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea —— C28H30N6O4S
1-ethyl-3-[3-[(2S,4R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[(1-phenyltetrazol-5-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]urea
—— 5-[(1R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsulfonyl]ethyl]-3-methyl-1,2,4-oxadiazole —— C11H15N3O4S
5-[(1R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsulfonyl]ethyl]-3-methyl-1,2,4-oxadiazole