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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[4-[(2S,4S,5R,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]acetamide —— C36H34N2O5S
N-[4-[(2S,4S,5R,6R)-4-[(4,5-diphenyl-1,3-oxazol-2-yl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]acetamide
—— 2-cyclopentyl-N-[(2S,3R)-3-hydroxy-4-phenylbutan-2-yl]-4-methyl-1,3-thiazole-5-carboxamide —— C20H26N2O2S
2-cyclopentyl-N-[(2S,3R)-3-hydroxy-4-phenylbutan-2-yl]-4-methyl-1,3-thiazole-5-carboxamide
—— N-[(2R,4R)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-4-methyl-2-(1-methylpyrazol-4-yl)-1,3-thiazole-5-carboxamide —— C17H20N4O3S
N-[(2R,4R)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-4-methyl-2-(1-methylpyrazol-4-yl)-1,3-thiazole-5-carboxamide
—— 1-[2-[(R)-tert-butylsulfinyl]ethyl]-3-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]urea —— C14H25N3O2S2
1-[2-[(R)-tert-butylsulfinyl]ethyl]-3-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]urea
—— (2S,3R)-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2,3-dimethylthiomorpholine-4-carboxamide —— C12H19N3OS2
(2S,3R)-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2,3-dimethylthiomorpholine-4-carboxamide
—— N-[(2S,4R)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-4-methyl-2-(1-methylpyrazol-4-yl)-1,3-thiazole-5-carboxamide —— C17H20N4O3S
N-[(2S,4R)-4-(furan-2-yl)-4-hydroxybutan-2-yl]-4-methyl-2-(1-methylpyrazol-4-yl)-1,3-thiazole-5-carboxamide
—— 1-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-3-[(2S)-1-thiophen-2-ylpropan-2-yl]urea —— C15H21N3OS2
1-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-3-[(2S)-1-thiophen-2-ylpropan-2-yl]urea
—— (1R)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)ethanamine —— C17H20N4OS
(1R)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)ethanamine
—— 2-(methoxymethyl)-N-[(2R)-2-(2-methoxyphenyl)-2-piperidin-1-ylethyl]-4-methyl-1,3-thiazole-5-carboxamide —— C21H29N3O3S
2-(methoxymethyl)-N-[(2R)-2-(2-methoxyphenyl)-2-piperidin-1-ylethyl]-4-methyl-1,3-thiazole-5-carboxamide
—— (1R)-N-methyl-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)-N-[2-(1,2,4-triazol-1-yl)ethyl]ethanamine —— C17H21N5S
(1R)-N-methyl-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)-N-[2-(1,2,4-triazol-1-yl)ethyl]ethanamine
—— 2-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-5-methyl-1,3-dioxan-2-yl]phenyl]isoindole-1,3-dione —— C34H29N5O6S
2-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-5-methyl-1,3-dioxan-2-yl]phenyl]isoindole-1,3-dione
—— methyl (2S)-2-[1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-3,5-dimethylpyrazol-4-yl]propanoate —— C15H21N3O2S
methyl (2S)-2-[1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-3,5-dimethylpyrazol-4-yl]propanoate
—— [(1R)-1-[2-(4-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]ethyl] 3-methoxythiophene-2-carboxylate —— C18H16FNO3S2
[(1R)-1-[2-(4-fluorophenyl)-4-methyl-1,3-thiazol-5-yl]ethyl] 3-methoxythiophene-2-carboxylate
—— N-methyl-N-[(1S)-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)ethyl]-2-(1,2-oxazol-3-yl)acetamide —— C18H19N3O2S
N-methyl-N-[(1S)-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)ethyl]-2-(1,2-oxazol-3-yl)acetamide
—— N-[(1R,2S)-2-(4-fluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide —— C16H14FN5OS
N-[(1R,2S)-2-(4-fluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide
—— (1S)-N-methyl-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)-N-[2-(1,2,4-triazol-1-yl)ethyl]ethanamine —— C17H21N5S
(1S)-N-methyl-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)-N-[2-(1,2,4-triazol-1-yl)ethyl]ethanamine
—— [(4aR,8aR)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-(2,4-dimethyl-1,3-thiazol-5-yl)methanone —— C13H18N2O2S2
[(4aR,8aR)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-(2,4-dimethyl-1,3-thiazol-5-yl)methanone
—— (2R,3S)-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2,3-dimethylthiomorpholine-4-carboxamide —— C12H19N3OS2
(2R,3S)-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2,3-dimethylthiomorpholine-4-carboxamide
—— 1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-3-[(1S)-1-(furan-2-yl)-2-methoxyethyl]urea —— C14H19N3O3S
1-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-3-[(1S)-1-(furan-2-yl)-2-methoxyethyl]urea
—— N-[(1S,2R)-2-(4-fluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide —— C16H14FN5OS
N-[(1S,2R)-2-(4-fluorophenyl)cyclopropyl]-4-methyl-2-(1H-1,2,4-triazol-5-yl)-1,3-thiazole-5-carboxamide
—— 1-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-3-[(2S)-2-methyl-3-pyrazol-1-ylpropyl]urea —— C15H23N5OS
1-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-3-[(2S)-2-methyl-3-pyrazol-1-ylpropyl]urea
—— N-methyl-N-[(1R)-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)ethyl]thiadiazole-5-carboxamide —— C16H16N4OS2
N-methyl-N-[(1R)-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)ethyl]thiadiazole-5-carboxamide
—— 2,4-dimethyl-5-[[(1S,6R)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl]-1,3-thiazole —— C16H27N3S
2,4-dimethyl-5-[[(1S,6R)-9-propan-2-yl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl]-1,3-thiazole
—— [(2S)-2,4-dimethylpiperazin-1-yl]-(4-methyl-2-pyrimidin-2-yl-1,3-thiazol-5-yl)methanone —— C15H19N5OS
[(2S)-2,4-dimethylpiperazin-1-yl]-(4-methyl-2-pyrimidin-2-yl-1,3-thiazol-5-yl)methanone
—— 1-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-3-[(2R)-2-methyl-3-pyrazol-1-ylpropyl]urea —— C15H23N5OS
1-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-3-[(2R)-2-methyl-3-pyrazol-1-ylpropyl]urea
—— N-methyl-N-[(1R)-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)ethyl]-2-(1,2-oxazol-3-yl)acetamide —— C18H19N3O2S
N-methyl-N-[(1R)-1-(4-methyl-2-phenyl-1,3-thiazol-5-yl)ethyl]-2-(1,2-oxazol-3-yl)acetamide
—— 1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(2S,4R)-4-hydroxy-4-phenylbutan-2-yl]urea —— C18H25N3O2S
1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(2S,4R)-4-hydroxy-4-phenylbutan-2-yl]urea
—— 1-[(2S)-2-cyclohexyl-1-hydroxypropan-2-yl]-3-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]urea —— C16H27N3O2S
1-[(2S)-2-cyclohexyl-1-hydroxypropan-2-yl]-3-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]urea
—— 1-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-3-[(2S)-2-thiophen-3-ylpropyl]urea —— C15H21N3OS2
1-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-3-[(2S)-2-thiophen-3-ylpropyl]urea
—— (2S,3S)-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2,3-dimethylthiomorpholine-4-carboxamide —— C12H19N3OS2
(2S,3S)-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2,3-dimethylthiomorpholine-4-carboxamide
—— [(4aR,8aS)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-(2,4-dimethyl-1,3-thiazol-5-yl)methanone —— C13H18N2O2S2
[(4aR,8aS)-3,4a,5,7,8,8a-hexahydro-2H-pyrano[3,4-b][1,4]thiazin-1-yl]-(2,4-dimethyl-1,3-thiazol-5-yl)methanone
—— 1-methyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(1S)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]urea —— C15H23N5O2S
1-methyl-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(1S)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]urea
—— N-[(2R,3R)-3-hydroxy-4-phenylbutan-2-yl]-2-[(1S)-1-methoxyethyl]-4-methyl-1,3-thiazole-5-carboxamide —— C18H24N2O3S
N-[(2R,3R)-3-hydroxy-4-phenylbutan-2-yl]-2-[(1S)-1-methoxyethyl]-4-methyl-1,3-thiazole-5-carboxamide
—— (1S)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)-N-(thiophen-3-ylmethyl)ethanamine —— C14H20N2S2
(1S)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)-N-(thiophen-3-ylmethyl)ethanamine
—— 1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(2S,4S)-4-hydroxy-4-phenylbutan-2-yl]urea —— C18H25N3O2S
1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(2S,4S)-4-hydroxy-4-phenylbutan-2-yl]urea
—— prop-2-enyl N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]carbamate —— C29H29N5O6S
prop-2-enyl N-[3-[(2R,4S,6R)-4-[4-(hydroxymethyl)phenyl]-6-[[1-(4-hydroxyphenyl)tetrazol-5-yl]sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]carbamate
—— (3S)-N-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-pyridin-3-yloxypyrrolidine-1-carboxamide —— C17H22N4O2S
(3S)-N-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-pyridin-3-yloxypyrrolidine-1-carboxamide
—— 3-imidazol-1-yl-N-[(1R)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]propan-1-amine —— C15H24N4S
3-imidazol-1-yl-N-[(1R)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]propan-1-amine
—— [(3R)-1-benzyl-5-oxopyrrolidin-3-yl]methyl 2,4-dimethyl-1,3-thiazole-5-carboxylate —— C18H20N2O3S
[(3R)-1-benzyl-5-oxopyrrolidin-3-yl]methyl 2,4-dimethyl-1,3-thiazole-5-carboxylate
—— 1-methyl-3-(1-methyl-2-oxopyridin-3-yl)-1-[(1S)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]urea —— C17H24N4O2S
1-methyl-3-(1-methyl-2-oxopyridin-3-yl)-1-[(1S)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]urea
—— 3-imidazol-1-yl-N-[(1S)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]propan-1-amine —— C15H24N4S
3-imidazol-1-yl-N-[(1S)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]propan-1-amine
—— (3S)-N-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-3-pyridin-4-yloxypyrrolidine-1-carboxamide —— C16H20N4O3
(3S)-N-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-3-pyridin-4-yloxypyrrolidine-1-carboxamide
—— N-[(2S)-2-[4-(difluoromethoxy)phenyl]-2-hydroxyethyl]-2,4-dimethyl-1,3-oxazole-5-carboxamide —— C15H16F2N2O4
N-[(2S)-2-[4-(difluoromethoxy)phenyl]-2-hydroxyethyl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
—— (5R)-2-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione —— C13H16N2O3S
(5R)-2-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione
—— 1-[(R)-cyclopropyl-(4-methoxyphenyl)methyl]-3-(4,5-dimethyl-1,3-oxazol-2-yl)urea —— C17H21N3O3
1-[(R)-cyclopropyl-(4-methoxyphenyl)methyl]-3-(4,5-dimethyl-1,3-oxazol-2-yl)urea
—— N-methyl-N-[(1R)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]-1,2-oxazole-3-carboxamide —— C14H19N3O2S
N-methyl-N-[(1R)-1-(4-methyl-2-propan-2-yl-1,3-thiazol-5-yl)ethyl]-1,2-oxazole-3-carboxamide
—— (3S)-N-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-3-(2-methylpropoxy)pyrrolidine-1-carboxamide —— C15H25N3O3
(3S)-N-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-3-(2-methylpropoxy)pyrrolidine-1-carboxamide
—— 4-methyl-5-[(1S)-1-[methyl(sulfamoyl)amino]ethyl]-2-propan-2-yl-1,3-thiazole —— C10H19N3O2S2
4-methyl-5-[(1S)-1-[methyl(sulfamoyl)amino]ethyl]-2-propan-2-yl-1,3-thiazole
—— (3S)-N-[[1-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]piperidin-4-yl]methyl]oxolane-3-carboxamide —— C17H27N3O3
(3S)-N-[[1-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]piperidin-4-yl]methyl]oxolane-3-carboxamide
—— 1-[(1S)-cyclohex-2-en-1-yl]-3-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]urea —— C13H19N3O2
1-[(1S)-cyclohex-2-en-1-yl]-3-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]urea