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中文名称 英文名称 CAS号 化学式 结构式图片
—— [(3S,4S)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-(5-methoxy-1,3-dimethylpyrazol-4-yl)methanone —— C17H28N4O3
[(3S,4S)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-(5-methoxy-1,3-dimethylpyrazol-4-yl)methanone
—— [(3S,4S)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-[3-methyl-5-(methylamino)-1,2-thiazol-4-yl]methanone —— C16H26N4O2S
[(3S,4S)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-[3-methyl-5-(methylamino)-1,2-thiazol-4-yl]methanone
—— (1-ethyl-3,5-dimethylpyrazol-4-yl)-[(3S,4R)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C18H30N4O2
(1-ethyl-3,5-dimethylpyrazol-4-yl)-[(3S,4R)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— [(3R,4R)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-[3-methyl-5-(methylamino)-1,2-thiazol-4-yl]methanone —— C16H26N4O2S
[(3R,4R)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-[3-methyl-5-(methylamino)-1,2-thiazol-4-yl]methanone
—— [(3S,4R)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-(5-methoxy-1,3-dimethylpyrazol-4-yl)methanone —— C17H28N4O3
[(3S,4R)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-(5-methoxy-1,3-dimethylpyrazol-4-yl)methanone
—— (1-ethyl-3,5-dimethylpyrazol-4-yl)-[(3R,4R)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C18H30N4O2
(1-ethyl-3,5-dimethylpyrazol-4-yl)-[(3R,4R)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— (1-ethyl-3,5-dimethylpyrazol-4-yl)-[(3S,4S)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C18H30N4O2
(1-ethyl-3,5-dimethylpyrazol-4-yl)-[(3S,4S)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— (1-ethyl-3,5-dimethylpyrazol-4-yl)-[(3R,4S)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone —— C18H30N4O2
(1-ethyl-3,5-dimethylpyrazol-4-yl)-[(3R,4S)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]methanone
—— [(3S,4R)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-[3-methyl-5-(methylamino)-1,2-thiazol-4-yl]methanone —— C16H26N4O2S
[(3S,4R)-3-ethyl-4-morpholin-4-ylpyrrolidin-1-yl]-[3-methyl-5-(methylamino)-1,2-thiazol-4-yl]methanone
—— [(3R,4R)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-[1-ethyl-5-(trifluoromethyl)pyrazol-4-yl]methanone —— C15H23F3N4O
[(3R,4R)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-[1-ethyl-5-(trifluoromethyl)pyrazol-4-yl]methanone
—— [(3S,4S)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-[1-ethyl-5-(trifluoromethyl)pyrazol-4-yl]methanone —— C15H23F3N4O
[(3S,4S)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-[1-ethyl-5-(trifluoromethyl)pyrazol-4-yl]methanone
—— 2-[3-[(3R,4S)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C17H25N5O2
2-[3-[(3R,4S)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— (6R)-3-[[1-(difluoromethyl)imidazol-2-yl]methyl]-6-ethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-one —— C14H17F2N3OS
(6R)-3-[[1-(difluoromethyl)imidazol-2-yl]methyl]-6-ethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-one
—— 2-[3-[(3S,4S)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C17H25N5O2
2-[3-[(3S,4S)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— [(3R,4S)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-[1-ethyl-5-(trifluoromethyl)pyrazol-4-yl]methanone —— C15H23F3N4O
[(3R,4S)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-[1-ethyl-5-(trifluoromethyl)pyrazol-4-yl]methanone
—— 2-[3-[(3R,4R)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C17H25N5O2
2-[3-[(3R,4R)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— (6S)-3-[[1-(difluoromethyl)imidazol-2-yl]methyl]-6-ethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-one —— C14H17F2N3OS
(6S)-3-[[1-(difluoromethyl)imidazol-2-yl]methyl]-6-ethyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-one
—— [(3S,4R)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-[1-ethyl-5-(trifluoromethyl)pyrazol-4-yl]methanone —— C15H23F3N4O
[(3S,4R)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-[1-ethyl-5-(trifluoromethyl)pyrazol-4-yl]methanone
—— N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-[(3R)-1,1-dioxothiolan-3-yl]acetamide —— C17H20BrN3O4S
N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-[(3R)-1,1-dioxothiolan-3-yl]acetamide
—— 2-[3-[(3S,4R)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C17H25N5O2
2-[3-[(3S,4R)-3-(dimethylamino)-4-ethylpyrrolidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-3-(2-chlorophenyl)propanamide —— C20H19BrClN3O2
N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-3-(2-chlorophenyl)propanamide
—— 1-phenyl-4-[[(S)-[(1S)-1-phenylpropyl]sulfinyl]methyl]pyrazole —— C19H20N2OS
1-phenyl-4-[[(S)-[(1S)-1-phenylpropyl]sulfinyl]methyl]pyrazole
—— 1-phenyl-4-[[(R)-[(1S)-1-phenylpropyl]sulfinyl]methyl]pyrazole —— C19H20N2OS
1-phenyl-4-[[(R)-[(1S)-1-phenylpropyl]sulfinyl]methyl]pyrazole
—— N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-[(3S)-1,1-dioxothiolan-3-yl]acetamide —— C17H20BrN3O4S
N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-[(3S)-1,1-dioxothiolan-3-yl]acetamide
—— N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-methyl-5-methylsulfanylbenzamide —— C20H20BrN3O2S
N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-methyl-5-methylsulfanylbenzamide
—— N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-1H-indazole-7-carboxamide —— C19H16BrN5O2
N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-1H-indazole-7-carboxamide
—— N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-methyl-5-methylsulfanylbenzamide —— C20H20BrN3O2S
N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-methyl-5-methylsulfanylbenzamide
—— 1-[(1S,3S)-3-[(S)-ethylsulfinyl]cyclohexyl]-3-[(1R)-1-(1,3-thiazol-2-yl)propyl]urea —— C15H25N3O2S2
1-[(1S,3S)-3-[(S)-ethylsulfinyl]cyclohexyl]-3-[(1R)-1-(1,3-thiazol-2-yl)propyl]urea
—— N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-4-chlorobenzamide —— C18H15BrClN3O2
N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-4-chlorobenzamide
—— 1-[(1R,3S)-3-[(S)-ethylsulfinyl]cyclohexyl]-3-[(1R)-1-(1,3-thiazol-2-yl)propyl]urea —— C15H25N3O2S2
1-[(1R,3S)-3-[(S)-ethylsulfinyl]cyclohexyl]-3-[(1R)-1-(1,3-thiazol-2-yl)propyl]urea
—— N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-(4-methylphenyl)sulfanylacetamide —— C20H20BrN3O2S
N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-(4-methylphenyl)sulfanylacetamide
—— N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-[(3R)-1,1-dioxothiolan-3-yl]acetamide —— C17H20BrN3O4S
N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-[(3R)-1,1-dioxothiolan-3-yl]acetamide
—— N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-3-(2-chlorophenyl)propanamide —— C20H19BrClN3O2
N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-3-(2-chlorophenyl)propanamide
—— 1-[(1R,3S)-3-[(S)-ethylsulfinyl]cyclohexyl]-3-[(1S)-1-(1,3-thiazol-2-yl)propyl]urea —— C15H25N3O2S2
1-[(1R,3S)-3-[(S)-ethylsulfinyl]cyclohexyl]-3-[(1S)-1-(1,3-thiazol-2-yl)propyl]urea
—— 1-phenyl-4-[[(R)-[(1R)-1-phenylpropyl]sulfinyl]methyl]pyrazole —— C19H20N2OS
1-phenyl-4-[[(R)-[(1R)-1-phenylpropyl]sulfinyl]methyl]pyrazole
—— N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-3-(4-chlorophenyl)propanamide —— C20H19BrClN3O2
N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-3-(4-chlorophenyl)propanamide
—— N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-1H-indazole-7-carboxamide —— C19H16BrN5O2
N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-1H-indazole-7-carboxamide
—— N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-4-chlorobenzamide —— C18H15BrClN3O2
N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-4-chlorobenzamide
—— N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-6-methylpyridine-2-carboxamide —— C18H17BrN4O2
N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-6-methylpyridine-2-carboxamide
—— N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-[(3S)-1,1-dioxothiolan-3-yl]acetamide —— C17H20BrN3O4S
N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-[(3S)-1,1-dioxothiolan-3-yl]acetamide
—— N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-3-(4-chlorophenyl)propanamide —— C20H19BrClN3O2
N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-3-(4-chlorophenyl)propanamide
—— 1-phenyl-4-[[(S)-[(1R)-1-phenylpropyl]sulfinyl]methyl]pyrazole —— C19H20N2OS
1-phenyl-4-[[(S)-[(1R)-1-phenylpropyl]sulfinyl]methyl]pyrazole
—— N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-(4-methylphenyl)sulfanylacetamide —— C20H20BrN3O2S
N-[(1S)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-2-(4-methylphenyl)sulfanylacetamide
—— methyl 3-[2-[2-[[(1S)-1-(4-chlorophenyl)propyl]amino]-2-oxoethyl]tetrazol-5-yl]benzoate —— C20H20ClN5O3
methyl 3-[2-[2-[[(1S)-1-(4-chlorophenyl)propyl]amino]-2-oxoethyl]tetrazol-5-yl]benzoate
—— 1-[(1S,3S)-3-[(S)-ethylsulfinyl]cyclohexyl]-3-[(1S)-1-(1,3-thiazol-2-yl)propyl]urea —— C15H25N3O2S2
1-[(1S,3S)-3-[(S)-ethylsulfinyl]cyclohexyl]-3-[(1S)-1-(1,3-thiazol-2-yl)propyl]urea
—— N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-6-methylpyridine-2-carboxamide —— C18H17BrN4O2
N-[(1R)-1-[5-(3-bromophenyl)-1,2,4-oxadiazol-3-yl]propyl]-6-methylpyridine-2-carboxamide
—— 1-[1-(2-fluorophenyl)pyrazol-4-yl]-3-[(2R)-1-hydroxybutan-2-yl]urea —— C14H17FN4O2
1-[1-(2-fluorophenyl)pyrazol-4-yl]-3-[(2R)-1-hydroxybutan-2-yl]urea
—— methyl 3-[2-[2-[[(1R)-1-(4-chlorophenyl)propyl]amino]-2-oxoethyl]tetrazol-5-yl]benzoate —— C20H20ClN5O3
methyl 3-[2-[2-[[(1R)-1-(4-chlorophenyl)propyl]amino]-2-oxoethyl]tetrazol-5-yl]benzoate
—— 1-[1-(2-fluorophenyl)pyrazol-4-yl]-3-[(2S)-1-hydroxybutan-2-yl]urea —— C14H17FN4O2
1-[1-(2-fluorophenyl)pyrazol-4-yl]-3-[(2S)-1-hydroxybutan-2-yl]urea
—— (3R)-3-[[(2-tert-butyl-1,3-thiazol-5-yl)methylamino]methyl]pentan-1-ol —— C14H26N2OS
(3R)-3-[[(2-tert-butyl-1,3-thiazol-5-yl)methylamino]methyl]pentan-1-ol