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—— (5S)-5-[(5,6-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]-1-methylpiperidin-2-one —— C13H18N6O
(5S)-5-[(5,6-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]-1-methylpiperidin-2-one
—— 5-[(1S)-1-[5-(4-chlorophenyl)-4-methyl-1,3-oxazol-2-yl]ethyl]sulfanyl-4-methyl-1,2,4-triazol-3-amine —— C15H16ClN5OS
5-[(1S)-1-[5-(4-chlorophenyl)-4-methyl-1,3-oxazol-2-yl]ethyl]sulfanyl-4-methyl-1,2,4-triazol-3-amine
—— 5-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid —— C30H33NO6S
5-[4-[(2S,4R,5R,6S)-4-[4-(hydroxymethyl)phenyl]-5-methyl-6-(phenylsulfanylmethyl)-1,3-dioxan-2-yl]anilino]-5-oxopentanoic acid
—— (5S)-7-[(1R)-1-[5-(4-chlorophenyl)-4-methyl-1,3-oxazol-2-yl]ethyl]-2-oxa-7-azaspiro[4.4]nonane —— C19H23ClN2O2
(5S)-7-[(1R)-1-[5-(4-chlorophenyl)-4-methyl-1,3-oxazol-2-yl]ethyl]-2-oxa-7-azaspiro[4.4]nonane
—— 5,6-dimethyl-N-[(5S,9S)-6-oxa-2-thiaspiro[4.5]decan-9-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H21N5OS
5,6-dimethyl-N-[(5S,9S)-6-oxa-2-thiaspiro[4.5]decan-9-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— [(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]-(2,4,5-trimethylfuran-3-yl)methanone —— C15H21NO3
[(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]-(2,4,5-trimethylfuran-3-yl)methanone
—— 5-methyl-N-[(2R)-4-methylpentan-2-yl]-1-quinolin-8-yltriazole-4-carboxamide —— C19H23N5O
5-methyl-N-[(2R)-4-methylpentan-2-yl]-1-quinolin-8-yltriazole-4-carboxamide
—— (5S)-7-[(1S)-1-[5-(4-chlorophenyl)-4-methyl-1,3-oxazol-2-yl]ethyl]-2-oxa-7-azaspiro[4.4]nonane —— C19H23ClN2O2
(5S)-7-[(1S)-1-[5-(4-chlorophenyl)-4-methyl-1,3-oxazol-2-yl]ethyl]-2-oxa-7-azaspiro[4.4]nonane
—— 5,6-dimethyl-N-[(5R,9R)-6-oxa-2-thiaspiro[4.5]decan-9-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H21N5OS
5,6-dimethyl-N-[(5R,9R)-6-oxa-2-thiaspiro[4.5]decan-9-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-(1-isoquinolin-5-yl-5-methyltriazol-4-yl)-3-[(3R)-oxolan-3-yl]-1,2,4-oxadiazole —— C18H16N6O2
5-(1-isoquinolin-5-yl-5-methyltriazol-4-yl)-3-[(3R)-oxolan-3-yl]-1,2,4-oxadiazole
—— 5,6-dimethyl-N-[(5R,9S)-6-oxa-2-thiaspiro[4.5]decan-9-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H21N5OS
5,6-dimethyl-N-[(5R,9S)-6-oxa-2-thiaspiro[4.5]decan-9-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5,6-dimethyl-N-[(5S,9R)-6-oxa-2-thiaspiro[4.5]decan-9-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C15H21N5OS
5,6-dimethyl-N-[(5S,9R)-6-oxa-2-thiaspiro[4.5]decan-9-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-(4-chlorophenyl)-4-methyl-2-[(1R)-1-(1-methyltetrazol-5-yl)sulfanylethyl]-1,3-oxazole —— C14H14ClN5OS
5-(4-chlorophenyl)-4-methyl-2-[(1R)-1-(1-methyltetrazol-5-yl)sulfanylethyl]-1,3-oxazole
—— (5R)-5-[(5,6-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]-1-methylpiperidin-2-one —— C13H18N6O
(5R)-5-[(5,6-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)amino]-1-methylpiperidin-2-one
—— 5-methyl-N-[(2S)-4-methylpentan-2-yl]-1-quinolin-8-yltriazole-4-carboxamide —— C19H23N5O
5-methyl-N-[(2S)-4-methylpentan-2-yl]-1-quinolin-8-yltriazole-4-carboxamide
—— 5-(4-chlorophenyl)-4-methyl-2-[(1S)-1-(1-methyltetrazol-5-yl)sulfanylethyl]-1,3-oxazole —— C14H14ClN5OS
5-(4-chlorophenyl)-4-methyl-2-[(1S)-1-(1-methyltetrazol-5-yl)sulfanylethyl]-1,3-oxazole
—— [(5R)-2-oxa-7-azaspiro[4.4]nonan-7-yl]-(2,4,5-trimethylfuran-3-yl)methanone —— C15H21NO3
[(5R)-2-oxa-7-azaspiro[4.4]nonan-7-yl]-(2,4,5-trimethylfuran-3-yl)methanone
—— (5S)-2-[(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione —— C16H16N2O3S2
(5S)-2-[(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione
—— 5-(1-isoquinolin-5-yl-5-methyltriazol-4-yl)-3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazole —— C18H16N6O2
5-(1-isoquinolin-5-yl-5-methyltriazol-4-yl)-3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazole
—— (5R)-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione —— C18H18N2O3S
(5R)-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione
—— (5S)-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione —— C18H18N2O3S
(5S)-2-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione
—— (5R)-2-[(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione —— C16H16N2O3S2
(5R)-2-[(5-methyl-2-thiophen-3-yl-1,3-oxazol-4-yl)methyl]-7-thia-2-azaspiro[4.4]nonane-1,3-dione
—— 5-methyl-1-[4-[(2R)-2-phenylazetidine-1-carbonyl]phenyl]pyrazole-4-carboxylic acid —— C21H19N3O3
5-methyl-1-[4-[(2R)-2-phenylazetidine-1-carbonyl]phenyl]pyrazole-4-carboxylic acid
—— 5-methyl-1-[4-[(2S)-2-phenylazetidine-1-carbonyl]phenyl]pyrazole-4-carboxylic acid —— C21H19N3O3
5-methyl-1-[4-[(2S)-2-phenylazetidine-1-carbonyl]phenyl]pyrazole-4-carboxylic acid
—— (5-methyl-1H-pyrazol-4-yl)-[(2S)-2-thiophen-2-ylmorpholin-4-yl]methanone —— C13H15N3O2S
(5-methyl-1H-pyrazol-4-yl)-[(2S)-2-thiophen-2-ylmorpholin-4-yl]methanone
—— 5-methyl-N-[(3S,4R)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]-1H-pyrazole-4-carboxamide —— C16H23N5OS
5-methyl-N-[(3S,4R)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]-1H-pyrazole-4-carboxamide
—— (5-methyl-1H-pyrazol-4-yl)-[(2R)-2-thiophen-2-ylmorpholin-4-yl]methanone —— C13H15N3O2S
(5-methyl-1H-pyrazol-4-yl)-[(2R)-2-thiophen-2-ylmorpholin-4-yl]methanone
—— 5-methyl-N-[(2S)-1-morpholin-4-yl-3-phenylpropan-2-yl]-1H-pyrazole-4-carboxamide —— C18H24N4O2
5-methyl-N-[(2S)-1-morpholin-4-yl-3-phenylpropan-2-yl]-1H-pyrazole-4-carboxamide
—— 5-methyl-N-[(3S,4S)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]-1H-pyrazole-4-carboxamide —— C16H23N5OS
5-methyl-N-[(3S,4S)-3-methyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl]-1H-pyrazole-4-carboxamide
—— 5-methyl-N-[(2R)-1-morpholin-4-yl-3-phenylpropan-2-yl]-1H-pyrazole-4-carboxamide —— C18H24N4O2
5-methyl-N-[(2R)-1-morpholin-4-yl-3-phenylpropan-2-yl]-1H-pyrazole-4-carboxamide
—— 5-[(3S,4S)-3-(dimethylamino)-4-methylpyrrolidine-1-carbonyl]-3,6-dimethylfuro[2,3-d]pyrimidin-4-one —— C16H22N4O3
5-[(3S,4S)-3-(dimethylamino)-4-methylpyrrolidine-1-carbonyl]-3,6-dimethylfuro[2,3-d]pyrimidin-4-one
—— 5-[(2R)-2,4-dimethylpiperazine-1-carbonyl]-6-methyl-3H-furo[2,3-d]pyrimidin-4-one —— C14H18N4O3
5-[(2R)-2,4-dimethylpiperazine-1-carbonyl]-6-methyl-3H-furo[2,3-d]pyrimidin-4-one
—— 5-[(3S,4R)-3-(dimethylamino)-4-methylpyrrolidine-1-carbonyl]-3,6-dimethylfuro[2,3-d]pyrimidin-4-one —— C16H22N4O3
5-[(3S,4R)-3-(dimethylamino)-4-methylpyrrolidine-1-carbonyl]-3,6-dimethylfuro[2,3-d]pyrimidin-4-one
—— 5-[(3R,4R)-3-(dimethylamino)-4-methylpyrrolidine-1-carbonyl]-3,6-dimethylfuro[2,3-d]pyrimidin-4-one —— C16H22N4O3
5-[(3R,4R)-3-(dimethylamino)-4-methylpyrrolidine-1-carbonyl]-3,6-dimethylfuro[2,3-d]pyrimidin-4-one
—— 5-[(3R,4S)-3-(dimethylamino)-4-methylpyrrolidine-1-carbonyl]-3,6-dimethylfuro[2,3-d]pyrimidin-4-one —— C16H22N4O3
5-[(3R,4S)-3-(dimethylamino)-4-methylpyrrolidine-1-carbonyl]-3,6-dimethylfuro[2,3-d]pyrimidin-4-one
—— 5-[[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-1,4-diazepan-1-yl]methyl]-3-[(1R)-1-methoxyethyl]-1,2,4-oxadiazole —— C17H27N5O3
5-[[4-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-1,4-diazepan-1-yl]methyl]-3-[(1R)-1-methoxyethyl]-1,2,4-oxadiazole
—— 5-[(1S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsulfonyl]ethyl]-3-methyl-1,2,4-oxadiazole —— C11H15N3O4S
5-[(1S)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsulfonyl]ethyl]-3-methyl-1,2,4-oxadiazole
—— 5-[(2S)-2,4-dimethylpiperazine-1-carbonyl]-6-methyl-3H-furo[2,3-d]pyrimidin-4-one —— C14H18N4O3
5-[(2S)-2,4-dimethylpiperazine-1-carbonyl]-6-methyl-3H-furo[2,3-d]pyrimidin-4-one
—— 5-[(1R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsulfonyl]ethyl]-3-methyl-1,2,4-oxadiazole —— C11H15N3O4S
5-[(1R)-1-[(3,5-dimethyl-1,2-oxazol-4-yl)methylsulfonyl]ethyl]-3-methyl-1,2,4-oxadiazole
—— (5R)-7-[7,8-dimethyl-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]-2-oxa-7-azaspiro[4.4]nonane —— C15H18F3N5O
(5R)-7-[7,8-dimethyl-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]-2-oxa-7-azaspiro[4.4]nonane
—— 5-[[(4R)-4-methyl-4,5-dihydro-1,3-thiazol-2-yl]sulfanylmethyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carbonitrile —— C12H11N5OS2
5-[[(4R)-4-methyl-4,5-dihydro-1,3-thiazol-2-yl]sulfanylmethyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carbonitrile
—— 5-[[(4S)-4-methyl-4,5-dihydro-1,3-thiazol-2-yl]sulfanylmethyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carbonitrile —— C12H11N5OS2
5-[[(4S)-4-methyl-4,5-dihydro-1,3-thiazol-2-yl]sulfanylmethyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidine-3-carbonitrile
—— 5-bromo-N-[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]pyridin-2-amine —— C13H16BrN3O
5-bromo-N-[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]pyridin-2-amine
—— (5S)-7-[7,8-dimethyl-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]-2-oxa-7-azaspiro[4.4]nonane —— C15H18F3N5O
(5S)-7-[7,8-dimethyl-3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]-2-oxa-7-azaspiro[4.4]nonane
—— 5-bromo-N-[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]pyridin-2-amine —— C13H16BrN3O
5-bromo-N-[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propyl]pyridin-2-amine
—— 5-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-1-phenyltetrazole —— C15H18N6O
5-[[2-[(1R)-1-ethoxyethyl]imidazol-1-yl]methyl]-1-phenyltetrazole
—— [5-chloro-1-[(4-fluorophenyl)methyl]-3-methylpyrazol-4-yl]-[(2R,5S)-2-(hydroxymethyl)-5-methylmorpholin-4-yl]methanone —— C18H21ClFN3O3
[5-chloro-1-[(4-fluorophenyl)methyl]-3-methylpyrazol-4-yl]-[(2R,5S)-2-(hydroxymethyl)-5-methylmorpholin-4-yl]methanone
—— 5-[[2-[(1S)-1-ethoxyethyl]imidazol-1-yl]methyl]-1-phenyltetrazole —— C15H18N6O
5-[[2-[(1S)-1-ethoxyethyl]imidazol-1-yl]methyl]-1-phenyltetrazole
—— [5-chloro-1-[(4-fluorophenyl)methyl]-3-methylpyrazol-4-yl]-[(2R,5R)-2-(hydroxymethyl)-5-methylmorpholin-4-yl]methanone —— C18H21ClFN3O3
[5-chloro-1-[(4-fluorophenyl)methyl]-3-methylpyrazol-4-yl]-[(2R,5R)-2-(hydroxymethyl)-5-methylmorpholin-4-yl]methanone
—— [5-chloro-1-[(4-fluorophenyl)methyl]-3-methylpyrazol-4-yl]-[(2S,5R)-2-(hydroxymethyl)-5-methylmorpholin-4-yl]methanone —— C18H21ClFN3O3
[5-chloro-1-[(4-fluorophenyl)methyl]-3-methylpyrazol-4-yl]-[(2S,5R)-2-(hydroxymethyl)-5-methylmorpholin-4-yl]methanone