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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-tert-butyl-N-[(2S)-4-hydroxy-1-methoxybutan-2-yl]-2-methylbenzenesulfonamide —— C16H27NO4S
5-tert-butyl-N-[(2S)-4-hydroxy-1-methoxybutan-2-yl]-2-methylbenzenesulfonamide
—— 5-[(4aR,7aR)-4-methyl-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazine-6-carbonyl]-N-(4-methoxyphenyl)-2-methylbenzenesulfonamide —— C22H27N3O5S
5-[(4aR,7aR)-4-methyl-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazine-6-carbonyl]-N-(4-methoxyphenyl)-2-methylbenzenesulfonamide
—— 5-[(4aS,7aS)-4-methyl-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazine-6-carbonyl]-N-(4-methoxyphenyl)-2-methylbenzenesulfonamide —— C22H27N3O5S
5-[(4aS,7aS)-4-methyl-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazine-6-carbonyl]-N-(4-methoxyphenyl)-2-methylbenzenesulfonamide
—— 5-[(2R)-1-benzylpyrrolidin-2-yl]-3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazole —— C17H21N3O2
5-[(2R)-1-benzylpyrrolidin-2-yl]-3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazole
—— 5-[6-(2,2-difluoroethoxy)pyridin-2-yl]-3-[(3R)-oxolan-3-yl]-1,2,4-oxadiazole —— C13H13F2N3O3
5-[6-(2,2-difluoroethoxy)pyridin-2-yl]-3-[(3R)-oxolan-3-yl]-1,2,4-oxadiazole
—— 5-tert-butyl-N-[(2R)-4-hydroxy-1-methoxybutan-2-yl]-2-methylbenzenesulfonamide —— C16H27NO4S
5-tert-butyl-N-[(2R)-4-hydroxy-1-methoxybutan-2-yl]-2-methylbenzenesulfonamide
—— 5-[6-(2,2-difluoroethoxy)pyridin-2-yl]-3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazole —— C13H13F2N3O3
5-[6-(2,2-difluoroethoxy)pyridin-2-yl]-3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazole
—— 5-[(2R)-1-(2-methyl-5-methylsulfonylphenyl)sulfonylpyrrolidin-2-yl]-3-phenyl-1H-1,2,4-triazole —— C20H22N4O4S2
5-[(2R)-1-(2-methyl-5-methylsulfonylphenyl)sulfonylpyrrolidin-2-yl]-3-phenyl-1H-1,2,4-triazole
—— (5R)-1-(3,4-dimethylphenyl)-5-[3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C19H23N3O3
(5R)-1-(3,4-dimethylphenyl)-5-[3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— 5-[(4aS,7aR)-4-methyl-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazine-6-carbonyl]-N-(4-methoxyphenyl)-2-methylbenzenesulfonamide —— C22H27N3O5S
5-[(4aS,7aR)-4-methyl-2,3,4a,5,7,7a-hexahydropyrrolo[3,4-b][1,4]oxazine-6-carbonyl]-N-(4-methoxyphenyl)-2-methylbenzenesulfonamide
—— (5S)-1-(3,4-dimethylphenyl)-5-[3-[(3R)-oxolan-3-yl]-1,2,4-oxadiazol-5-yl]piperidin-2-one —— C19H23N3O3
(5S)-1-(3,4-dimethylphenyl)-5-[3-[(3R)-oxolan-3-yl]-1,2,4-oxadiazol-5-yl]piperidin-2-one
—— 5-[(2R)-1-benzylpyrrolidin-2-yl]-3-pyrazin-2-yl-1,2,4-oxadiazole —— C17H17N5O
5-[(2R)-1-benzylpyrrolidin-2-yl]-3-pyrazin-2-yl-1,2,4-oxadiazole
—— 5-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]sulfanyl-4-methyl-1,2,4-triazol-3-amine —— C14H15FN6OS
5-[(1S)-1-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]sulfanyl-4-methyl-1,2,4-triazol-3-amine
—— 5-[[(2S)-2,4-dimethylpiperazin-1-yl]methyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole —— C16H21FN4O
5-[[(2S)-2,4-dimethylpiperazin-1-yl]methyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole
—— (5S)-5-tert-butyl-N-(6-methylsulfonylpyridin-3-yl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C19H24N2O3S2
(5S)-5-tert-butyl-N-(6-methylsulfonylpyridin-3-yl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— 5-[3-[(2S)-2,4-dimethylpiperazin-1-yl]propyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole —— C18H25FN4O
5-[3-[(2S)-2,4-dimethylpiperazin-1-yl]propyl]-3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazole
—— 5-(cyclopropylsulfamoyl)-N-[(1R,2S)-2-(hydroxymethyl)cyclohexyl]-2-methylbenzamide —— C18H26N2O4S
5-(cyclopropylsulfamoyl)-N-[(1R,2S)-2-(hydroxymethyl)cyclohexyl]-2-methylbenzamide
—— 5-(cyclopropylsulfamoyl)-N-[(1R,2R)-2-(hydroxymethyl)cyclohexyl]-2-methylbenzamide —— C18H26N2O4S
5-(cyclopropylsulfamoyl)-N-[(1R,2R)-2-(hydroxymethyl)cyclohexyl]-2-methylbenzamide
—— 5-(cyclopropylsulfamoyl)-N-[(1S,2S)-2-(hydroxymethyl)cyclohexyl]-2-methylbenzamide —— C18H26N2O4S
5-(cyclopropylsulfamoyl)-N-[(1S,2S)-2-(hydroxymethyl)cyclohexyl]-2-methylbenzamide
—— 5-[(3aS,7aS)-2,3,3a,4,5,6,7,7a-octahydroindole-1-carbonyl]-2-(4-methylphenyl)-1H-pyrazol-3-one —— C19H23N3O2
5-[(3aS,7aS)-2,3,3a,4,5,6,7,7a-octahydroindole-1-carbonyl]-2-(4-methylphenyl)-1H-pyrazol-3-one
—— (5-fluoro-2-methylphenyl)-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C16H18FN3O
(5-fluoro-2-methylphenyl)-[(3R)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— (5R)-5-tert-butyl-N-(6-methylsulfonylpyridin-3-yl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C19H24N2O3S2
(5R)-5-tert-butyl-N-(6-methylsulfonylpyridin-3-yl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5-fluoro-2-methylphenyl)-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone —— C16H18FN3O
(5-fluoro-2-methylphenyl)-[(3S)-3-(1H-pyrazol-5-yl)piperidin-1-yl]methanone
—— 5-[(3aR,7aS)-2,3,3a,4,5,6,7,7a-octahydroindole-1-carbonyl]-2-(4-methylphenyl)-1H-pyrazol-3-one —— C19H23N3O2
5-[(3aR,7aS)-2,3,3a,4,5,6,7,7a-octahydroindole-1-carbonyl]-2-(4-methylphenyl)-1H-pyrazol-3-one
—— 5-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]-3-[[5-(4-methylphenyl)tetrazol-2-yl]methyl]-1,2,4-oxadiazole —— C19H16N6O3
5-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]-3-[[5-(4-methylphenyl)tetrazol-2-yl]methyl]-1,2,4-oxadiazole
—— [5-[2-chloro-5-(trifluoromethyl)phenyl]furan-2-yl]-[(2S,5S,6S,13S)-5,13-dihydroxy-5-[[4-(2-hydroxyphenyl)piperazin-1-yl]methyl]-6,10-dimethyl-17-tricyclo[13.2.2.02,6]nonadeca-1(17),9,15,18-tetraenyl]methanone —— C44H48ClF3N2O5
[5-[2-chloro-5-(trifluoromethyl)phenyl]furan-2-yl]-[(2S,5S,6S,13S)-5,13-dihydroxy-5-[[4-(2-hydroxyphenyl)piperazin-1-yl]methyl]-6,10-dimethyl-17-tricyclo[13.2.2.02,6]nonadeca-1(17),9,15,18-tetraenyl]methanone
—— 5-[2-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]ethyl]-1,3,4-thiadiazol-2-amine —— C19H25N7OS
5-[2-[4-[(1S)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]ethyl]-1,3,4-thiadiazol-2-amine
—— 5-[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]-3-[[5-(4-methylphenyl)tetrazol-2-yl]methyl]-1,2,4-oxadiazole —— C19H16N6O3
5-[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]-3-[[5-(4-methylphenyl)tetrazol-2-yl]methyl]-1,2,4-oxadiazole
—— 5-[(3aS,7aR)-2,3,3a,4,5,6,7,7a-octahydroindole-1-carbonyl]-2-(4-methylphenyl)-1H-pyrazol-3-one —— C19H23N3O2
5-[(3aS,7aR)-2,3,3a,4,5,6,7,7a-octahydroindole-1-carbonyl]-2-(4-methylphenyl)-1H-pyrazol-3-one
—— 5-[(3aR,7aR)-2,3,3a,4,5,6,7,7a-octahydroindole-1-carbonyl]-2-(4-methylphenyl)-1H-pyrazol-3-one —— C19H23N3O2
5-[(3aR,7aR)-2,3,3a,4,5,6,7,7a-octahydroindole-1-carbonyl]-2-(4-methylphenyl)-1H-pyrazol-3-one
—— 5-[2-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]ethyl]-1,3,4-thiadiazol-2-amine —— C19H25N7OS
5-[2-[4-[(1R)-1-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]ethyl]-1,3,4-thiadiazol-2-amine
—— [5-(4-methylphenyl)-1,3-oxazol-4-yl]-[(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone —— C18H20N2O3
[5-(4-methylphenyl)-1,3-oxazol-4-yl]-[(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone
—— 5-[(Z)-[(6-chloropyridazin-3-yl)hydrazinylidene]methyl]-1-methyl-N-(4-methylphenyl)sulfonylpyrrole-3-carboxamide —— C18H17ClN6O3S
5-[(Z)-[(6-chloropyridazin-3-yl)hydrazinylidene]methyl]-1-methyl-N-(4-methylphenyl)sulfonylpyrrole-3-carboxamide
—— 5-[[[(1S)-2,3-dihydro-1H-inden-1-yl]-methylamino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide —— C22H24N4OS
5-[[[(1S)-2,3-dihydro-1H-inden-1-yl]-methylamino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide
—— (5R)-7,9-dimethyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C16H25NO3S
(5R)-7,9-dimethyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— 5-[[(R)-(4-methylphenyl)methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine —— C17H18O3S
5-[[(R)-(4-methylphenyl)methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine
—— (5S)-7,9-dimethyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C16H25NO3S
(5S)-7,9-dimethyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— 5-[[cyclopropyl-[(1S)-2,3-dihydro-1H-inden-1-yl]amino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide —— C24H26N4OS
5-[[cyclopropyl-[(1S)-2,3-dihydro-1H-inden-1-yl]amino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide
—— 5-[[[(1S)-2,3-dihydro-1H-inden-1-yl]-prop-2-ynylamino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide —— C24H24N4OS
5-[[[(1S)-2,3-dihydro-1H-inden-1-yl]-prop-2-ynylamino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide
—— 5-[[(S)-(4-methylphenyl)methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine —— C17H18O3S
5-[[(S)-(4-methylphenyl)methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine
—— (5R)-7,9-dimethyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C16H25NO3S
(5R)-7,9-dimethyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— [5-(4-methylphenyl)-1,3-oxazol-4-yl]-[(5R)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone —— C18H20N2O3
[5-(4-methylphenyl)-1,3-oxazol-4-yl]-[(5R)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone
—— 5-[[cyclopropyl-[(1R)-2,3-dihydro-1H-inden-1-yl]amino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide —— C24H26N4OS
5-[[cyclopropyl-[(1R)-2,3-dihydro-1H-inden-1-yl]amino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide
—— 5-[[[(1R)-2,3-dihydro-1H-inden-1-yl]-methylamino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide —— C22H24N4OS
5-[[[(1R)-2,3-dihydro-1H-inden-1-yl]-methylamino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide
—— (5S)-7,9-dimethyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C16H25NO3S
(5S)-7,9-dimethyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— 5-[[[(1R)-2,3-dihydro-1H-inden-1-yl]-prop-2-ynylamino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide —— C24H24N4OS
5-[[[(1R)-2,3-dihydro-1H-inden-1-yl]-prop-2-ynylamino]methyl]-N-[(4-methylphenyl)methyl]-1,3,4-thiadiazole-2-carboxamide
—— 5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2R)-2-hydroxy-2-(4-methylphenyl)ethyl]thiophene-2-carboxamide —— C22H21NO4S
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2R)-2-hydroxy-2-(4-methylphenyl)ethyl]thiophene-2-carboxamide
—— (5S)-N-(2-tert-butylsulfonylethyl)-1,2,4,5-tetrahydro-3-benzothiepin-5-amine —— C16H25NO2S2
(5S)-N-(2-tert-butylsulfonylethyl)-1,2,4,5-tetrahydro-3-benzothiepin-5-amine
—— (5S,7R)-N-methyl-3-(4-methylphenyl)-N-(3,3,3-trifluoropropyl)adamantane-1-carboxamide —— C22H28F3NO
(5S,7R)-N-methyl-3-(4-methylphenyl)-N-(3,3,3-trifluoropropyl)adamantane-1-carboxamide
—— 5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2S)-2-hydroxy-2-(4-methylphenyl)ethyl]thiophene-2-carboxamide —— C22H21NO4S
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2S)-2-hydroxy-2-(4-methylphenyl)ethyl]thiophene-2-carboxamide