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—— 5-(3-chloro-6-oxocyclohexa-2,4-dien-1-ylidene)-N-[2-(phenylcarbamoyl)-1-benzofuran-3-yl]-1,2-dihydropyrazole-3-carboxamide —— C25H17ClN4O4
5-(3-chloro-6-oxocyclohexa-2,4-dien-1-ylidene)-N-[2-(phenylcarbamoyl)-1-benzofuran-3-yl]-1,2-dihydropyrazole-3-carboxamide
—— 5-[1-(3-fluorophenyl)cyclopentyl]-3-[(3R)-oxolan-3-yl]-1,2,4-oxadiazole —— C17H19FN2O2
5-[1-(3-fluorophenyl)cyclopentyl]-3-[(3R)-oxolan-3-yl]-1,2,4-oxadiazole
—— 5-(4-methyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-[2-[(4-methylphenyl)carbamoyl]-1-benzofuran-3-yl]-1,2-dihydropyrazole-3-carboxamide —— C27H22N4O4
5-(4-methyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-[2-[(4-methylphenyl)carbamoyl]-1-benzofuran-3-yl]-1,2-dihydropyrazole-3-carboxamide
—— 5-(4,5-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(6-methoxy-1,3-benzothiazol-2-yl)-1,2-dihydropyrazole-3-carboxamide —— C20H18N4O3S
5-(4,5-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(6-methoxy-1,3-benzothiazol-2-yl)-1,2-dihydropyrazole-3-carboxamide
—— 5-(3-chloro-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-1,2-dihydropyrazole-3-carboxamide —— C21H18ClN5O3
5-(3-chloro-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-1,2-dihydropyrazole-3-carboxamide
—— 5-(3-methyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(5-propyl-1,3,4-thiadiazol-2-yl)-1,2-dihydropyrazole-3-carboxamide —— C16H17N5O2S
5-(3-methyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(5-propyl-1,3,4-thiadiazol-2-yl)-1,2-dihydropyrazole-3-carboxamide
—— 5-methyl-4-[[3-[(3-methyl-1-phenyl-5-sulfanylidenepyrazol-4-ylidene)methylamino]propylamino]methylidene]-2-phenylpyrazole-3-thione —— C25H26N6S2
5-methyl-4-[[3-[(3-methyl-1-phenyl-5-sulfanylidenepyrazol-4-ylidene)methylamino]propylamino]methylidene]-2-phenylpyrazole-3-thione
—— 5-(3,5-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(2,5-dimethylphenyl)-1,2-dihydropyrazole-3-carboxamide —— C20H21N3O2
5-(3,5-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(2,5-dimethylphenyl)-1,2-dihydropyrazole-3-carboxamide
—— 5-(3-methyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(pyridin-4-ylmethyl)-1,2-dihydropyrazole-3-carboxamide —— C17H16N4O2
5-(3-methyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(pyridin-4-ylmethyl)-1,2-dihydropyrazole-3-carboxamide
—— 5-cyclopropyl-2-[(3S)-1,1-dioxothiolan-3-yl]-N-[[3-(trifluoromethyl)phenyl]methyl]pyrazol-3-amine —— C18H20F3N3O2S
5-cyclopropyl-2-[(3S)-1,1-dioxothiolan-3-yl]-N-[[3-(trifluoromethyl)phenyl]methyl]pyrazol-3-amine
—— (5S)-N-[(1R)-2-amino-1-(3-bromophenyl)-2-oxoethyl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H13BrClN3O3S
(5S)-N-[(1R)-2-amino-1-(3-bromophenyl)-2-oxoethyl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-(3,5-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(6-fluoro-1,3-benzothiazol-2-yl)-1,2-dihydropyrazole-3-carboxamide —— C19H15FN4O2S
5-(3,5-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(6-fluoro-1,3-benzothiazol-2-yl)-1,2-dihydropyrazole-3-carboxamide
—— [(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]-[3-(pyrrolidin-1-ylmethyl)phenyl]methanone —— C19H26N2O2
[(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]-[3-(pyrrolidin-1-ylmethyl)phenyl]methanone
—— 5-(4,5-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(3,4-dimethylphenyl)-1,2-dihydropyrazole-3-carboxamide —— C20H21N3O2
5-(4,5-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)-N-(3,4-dimethylphenyl)-1,2-dihydropyrazole-3-carboxamide
—— (5S)-N-[(1S)-2-amino-1-(3-bromophenyl)-2-oxoethyl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H13BrClN3O3S
(5S)-N-[(1S)-2-amino-1-(3-bromophenyl)-2-oxoethyl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-cyclopropyl-N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1,2-oxazole-3-carboxamide —— C16H15F3N2O3
5-cyclopropyl-N-[(2S)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1,2-oxazole-3-carboxamide
—— 5-cyclopropyl-2-[(3R)-1,1-dioxothiolan-3-yl]-N-[[3-(trifluoromethyl)phenyl]methyl]pyrazol-3-amine —— C18H20F3N3O2S
5-cyclopropyl-2-[(3R)-1,1-dioxothiolan-3-yl]-N-[[3-(trifluoromethyl)phenyl]methyl]pyrazol-3-amine
—— 5-cyclopropyl-N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1,2-oxazole-3-carboxamide —— C16H15F3N2O3
5-cyclopropyl-N-[(2R)-2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]-1,2-oxazole-3-carboxamide
—— (5R)-N-[(1R)-2-amino-1-(3-bromophenyl)-2-oxoethyl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C16H13BrClN3O3S
(5R)-N-[(1R)-2-amino-1-(3-bromophenyl)-2-oxoethyl]-3-(5-chlorothiophen-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— [(5R)-2-oxa-7-azaspiro[4.4]nonan-7-yl]-[3-(pyrrolidin-1-ylmethyl)phenyl]methanone —— C19H26N2O2
[(5R)-2-oxa-7-azaspiro[4.4]nonan-7-yl]-[3-(pyrrolidin-1-ylmethyl)phenyl]methanone
—— 5,8-difluoro-2-[2-[(2R)-oxolan-2-yl]ethylsulfonyl]-3,4-dihydro-1H-isoquinoline —— C15H19F2NO3S
5,8-difluoro-2-[2-[(2R)-oxolan-2-yl]ethylsulfonyl]-3,4-dihydro-1H-isoquinoline
—— 5,8-difluoro-2-[2-[(2S)-oxolan-2-yl]ethylsulfonyl]-3,4-dihydro-1H-isoquinoline —— C15H19F2NO3S
5,8-difluoro-2-[2-[(2S)-oxolan-2-yl]ethylsulfonyl]-3,4-dihydro-1H-isoquinoline
—— 5-bromo-N-[2-[[(3R)-1-(3,4-difluorophenyl)pyrrolidin-3-yl]methylamino]-2-oxoethyl]thiophene-2-carboxamide —— C18H18BrF2N3O2S
5-bromo-N-[2-[[(3R)-1-(3,4-difluorophenyl)pyrrolidin-3-yl]methylamino]-2-oxoethyl]thiophene-2-carboxamide
—— 5-[[[(3S)-1-(3-chloropyridin-2-yl)pyrrolidin-3-yl]amino]methyl]thiophene-3-carbonitrile —— C15H15ClN4S
5-[[[(3S)-1-(3-chloropyridin-2-yl)pyrrolidin-3-yl]amino]methyl]thiophene-3-carbonitrile
—— (5S,7R)-3-bromo-N-(2-morpholin-4-ylpyridin-3-yl)adamantane-1-carboxamide —— C20H26BrN3O2
(5S,7R)-3-bromo-N-(2-morpholin-4-ylpyridin-3-yl)adamantane-1-carboxamide
—— 5-(2,4-dichlorophenyl)-3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazole —— C12H10Cl2N2O2
5-(2,4-dichlorophenyl)-3-[(3S)-oxolan-3-yl]-1,2,4-oxadiazole
—— 5-[[[(3R)-1-(3-chloropyridin-2-yl)pyrrolidin-3-yl]amino]methyl]thiophene-3-carbonitrile —— C15H15ClN4S
5-[[[(3R)-1-(3-chloropyridin-2-yl)pyrrolidin-3-yl]amino]methyl]thiophene-3-carbonitrile
—— 5-bromo-N-[2-[[(3S)-1-(3,4-difluorophenyl)pyrrolidin-3-yl]methylamino]-2-oxoethyl]thiophene-2-carboxamide —— C18H18BrF2N3O2S
5-bromo-N-[2-[[(3S)-1-(3,4-difluorophenyl)pyrrolidin-3-yl]methylamino]-2-oxoethyl]thiophene-2-carboxamide
—— 5-fluoro-2-[[(3R)-3-[(5-nitropyridin-2-yl)amino]pyrrolidin-1-yl]methyl]benzonitrile —— C17H16FN5O2
5-fluoro-2-[[(3R)-3-[(5-nitropyridin-2-yl)amino]pyrrolidin-1-yl]methyl]benzonitrile
—— 5-fluoro-2-[[(3S)-3-[(5-nitropyridin-2-yl)amino]pyrrolidin-1-yl]methyl]benzonitrile —— C17H16FN5O2
5-fluoro-2-[[(3S)-3-[(5-nitropyridin-2-yl)amino]pyrrolidin-1-yl]methyl]benzonitrile
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2R)-2-(morpholin-4-ylmethyl)piperidin-1-yl]methanone —— C18H26N2O2S
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2R)-2-(morpholin-4-ylmethyl)piperidin-1-yl]methanone
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(5R)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone —— C15H19NO2S
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(5R)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone
—— 5-[[(3R)-1-(2,6-difluorophenyl)-2-oxopyrrolidin-3-yl]amino]-3H-1,3-benzoxazol-2-one —— C17H13F2N3O3
5-[[(3R)-1-(2,6-difluorophenyl)-2-oxopyrrolidin-3-yl]amino]-3H-1,3-benzoxazol-2-one
—— 5-chloro-N-[(2-chloro-1,3-thiazol-5-yl)methyl]-2-[[(2S)-oxolan-2-yl]methoxy]aniline —— C15H16Cl2N2O2S
5-chloro-N-[(2-chloro-1,3-thiazol-5-yl)methyl]-2-[[(2S)-oxolan-2-yl]methoxy]aniline
—— 5-chloro-N-[(2-chloro-1,3-thiazol-5-yl)methyl]-2-[[(2R)-oxolan-2-yl]methoxy]aniline —— C15H16Cl2N2O2S
5-chloro-N-[(2-chloro-1,3-thiazol-5-yl)methyl]-2-[[(2R)-oxolan-2-yl]methoxy]aniline
—— 5-(2,4-dichlorophenyl)-3-[(3R)-oxolan-3-yl]-1,2,4-oxadiazole —— C12H10Cl2N2O2
5-(2,4-dichlorophenyl)-3-[(3R)-oxolan-3-yl]-1,2,4-oxadiazole
—— 5-[[(3S)-1-(2,6-difluorophenyl)-2-oxopyrrolidin-3-yl]amino]-3H-1,3-benzoxazol-2-one —— C17H13F2N3O3
5-[[(3S)-1-(2,6-difluorophenyl)-2-oxopyrrolidin-3-yl]amino]-3H-1,3-benzoxazol-2-one
—— 5-methoxy-1-methyl-N'-[(2-oxonaphthalen-1-ylidene)methyl]indole-2-carbohydrazide —— C22H19N3O3
5-methoxy-1-methyl-N'-[(2-oxonaphthalen-1-ylidene)methyl]indole-2-carbohydrazide
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2S)-2-(morpholin-4-ylmethyl)piperidin-1-yl]methanone —— C18H26N2O2S
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(2S)-2-(morpholin-4-ylmethyl)piperidin-1-yl]methanone
—— 5-bromo-6-[4-[(3R)-oxolan-3-yl]piperazin-1-yl]sulfonyl-1,3-dihydrobenzimidazol-2-one —— C15H19BrN4O4S
5-bromo-6-[4-[(3R)-oxolan-3-yl]piperazin-1-yl]sulfonyl-1,3-dihydrobenzimidazol-2-one
—— 5-cyclopropyl-N-[[(3R)-oxolan-3-yl]methyl]-1,2-oxazole-3-carboxamide —— C12H16N2O3
5-cyclopropyl-N-[[(3R)-oxolan-3-yl]methyl]-1,2-oxazole-3-carboxamide
—— 5-bromo-6-[4-[(3S)-oxolan-3-yl]piperazin-1-yl]sulfonyl-1,3-dihydrobenzimidazol-2-one —— C15H19BrN4O4S
5-bromo-6-[4-[(3S)-oxolan-3-yl]piperazin-1-yl]sulfonyl-1,3-dihydrobenzimidazol-2-one
—— 5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone —— C15H19NO2S
5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl-[(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone
—— 5-bromo-2-[(2R)-2-(1H-pyrazol-4-yl)piperidin-1-yl]pyrimidine —— C12H14BrN5
5-bromo-2-[(2R)-2-(1H-pyrazol-4-yl)piperidin-1-yl]pyrimidine
—— (5S)-7-(5-bromopyridin-3-yl)-2-oxa-7-azaspiro[4.4]nonane —— C12H15BrN2O
(5S)-7-(5-bromopyridin-3-yl)-2-oxa-7-azaspiro[4.4]nonane
—— (5-bromothiophen-3-yl)-[(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone —— C12H14BrNO2S
(5-bromothiophen-3-yl)-[(5S)-2-oxa-7-azaspiro[4.4]nonan-7-yl]methanone
—— 5-chloro-N-[(5R,9R)-6-oxa-2-thiaspiro[4.5]decan-9-yl]pyrimidin-2-amine —— C12H16ClN3OS
5-chloro-N-[(5R,9R)-6-oxa-2-thiaspiro[4.5]decan-9-yl]pyrimidin-2-amine
—— 5-cyclopropyl-N-[[(3S)-oxolan-3-yl]methyl]-1,2-oxazole-3-carboxamide —— C12H16N2O3
5-cyclopropyl-N-[[(3S)-oxolan-3-yl]methyl]-1,2-oxazole-3-carboxamide
—— 5-nitro-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]thiophene-3-carboxamide —— C14H18N2O4S2
5-nitro-N-[[(2S)-oxolan-2-yl]methyl]-N-[(3R)-thiolan-3-yl]thiophene-3-carboxamide
—— (5R)-7-(5-bromopyridin-3-yl)-2-oxa-7-azaspiro[4.4]nonane —— C12H15BrN2O
(5R)-7-(5-bromopyridin-3-yl)-2-oxa-7-azaspiro[4.4]nonane