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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[[1-(4-fluorophenyl)pyrazol-4-yl]methyl]-5-[(2S)-oxolan-2-yl]thiophene-2-carboxamide —— C19H18FN3O2S
N-[[1-(4-fluorophenyl)pyrazol-4-yl]methyl]-5-[(2S)-oxolan-2-yl]thiophene-2-carboxamide
—— 1-[(3R)-3-[[[5-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl-methylamino]methyl]pyrrolidin-1-yl]ethanone —— C18H23ClN4O
1-[(3R)-3-[[[5-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl-methylamino]methyl]pyrrolidin-1-yl]ethanone
—— [2-[(5-methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] (3R)-3-phenylbutanoate —— C22H23N3O3
[2-[(5-methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] (3R)-3-phenylbutanoate
—— 5-(3-fluorophenyl)-N-[[(3S)-3-hydroxypiperidin-3-yl]methyl]-1H-pyrazole-4-carboxamide —— C16H19FN4O2
5-(3-fluorophenyl)-N-[[(3S)-3-hydroxypiperidin-3-yl]methyl]-1H-pyrazole-4-carboxamide
—— 1-[(4S)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-3-propylurea —— C20H28N4O2
1-[(4S)-1-(4-methoxyphenyl)-6,6-dimethyl-5,7-dihydro-4H-indazol-4-yl]-3-propylurea
—— 4-butyl-N-[2-[2-(4-fluorophenyl)-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-yl]ethyl]benzamide —— C23H23FN4OS
4-butyl-N-[2-[2-(4-fluorophenyl)-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-yl]ethyl]benzamide
—— (3R)-N-[(2R)-butan-2-yl]-1-[4-(tetrazol-1-yl)phenyl]sulfonylpiperidine-3-carboxamide —— C17H24N6O3S
(3R)-N-[(2R)-butan-2-yl]-1-[4-(tetrazol-1-yl)phenyl]sulfonylpiperidine-3-carboxamide
—— N-[(4R)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]morpholine-4-sulfonamide —— C20H28N4O3S
N-[(4R)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]morpholine-4-sulfonamide
—— N-[(4S)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]morpholine-4-sulfonamide —— C20H28N4O3S
N-[(4S)-6,6-dimethyl-1-(2-methylphenyl)-5,7-dihydro-4H-indazol-4-yl]morpholine-4-sulfonamide
—— N-[(1S)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetamide —— C19H20FN5O3
N-[(1S)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetamide
—— (2S)-2-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(4-methylsulfanylphenyl)piperidine-1-carboxamide —— C22H24N4O2S
(2S)-2-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(4-methylsulfanylphenyl)piperidine-1-carboxamide
—— 1-ethyl-N-[(1R)-1-[1-(4-methoxyphenyl)-5-methylpyrazol-4-yl]ethyl]pyrazole-3-carboxamide —— C19H23N5O2
1-ethyl-N-[(1R)-1-[1-(4-methoxyphenyl)-5-methylpyrazol-4-yl]ethyl]pyrazole-3-carboxamide
—— (2S)-2-pyrazol-1-yl-N-[(2-pyrimidin-2-yl-1,3-thiazol-4-yl)methyl]butanamide —— C15H16N6OS
(2S)-2-pyrazol-1-yl-N-[(2-pyrimidin-2-yl-1,3-thiazol-4-yl)methyl]butanamide
—— 1-ethyl-N-[(1S)-1-[1-(4-methoxyphenyl)-5-methylpyrazol-4-yl]ethyl]pyrazole-3-carboxamide —— C19H23N5O2
1-ethyl-N-[(1S)-1-[1-(4-methoxyphenyl)-5-methylpyrazol-4-yl]ethyl]pyrazole-3-carboxamide
—— N-[(1R)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetamide —— C19H20FN5O3
N-[(1R)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-(6-methyl-2,4-dioxo-1H-pyrimidin-5-yl)acetamide
—— (2R)-2-pyrazol-1-yl-N-[(2-pyrimidin-2-yl-1,3-thiazol-4-yl)methyl]butanamide —— C15H16N6OS
(2R)-2-pyrazol-1-yl-N-[(2-pyrimidin-2-yl-1,3-thiazol-4-yl)methyl]butanamide
—— N-[(4S)-1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-4-hydroxy-6-oxo-1H-pyridine-3-carboxamide —— C23H26N4O3
N-[(4S)-1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-4-hydroxy-6-oxo-1H-pyridine-3-carboxamide
—— N-[(1R)-1-imidazo[1,2-a]pyrimidin-2-ylpropyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C20H20N6O2
N-[(1R)-1-imidazo[1,2-a]pyrimidin-2-ylpropyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— (4aR,6S,8aS)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-6-methoxy-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine —— C19H24FN3O2
(4aR,6S,8aS)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-6-methoxy-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine
—— [2-(2-aminoethyl)-1,3-thiazol-4-yl]-[(3R,4S)-3,4-dimethylpyrrolidin-1-yl]methanone —— C12H19N3OS
[2-(2-aminoethyl)-1,3-thiazol-4-yl]-[(3R,4S)-3,4-dimethylpyrrolidin-1-yl]methanone
—— (4aR,6R,8aR)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-6-methoxy-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine —— C19H24FN3O2
(4aR,6R,8aR)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-6-methoxy-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine
—— 3-(methanesulfonamido)-N-[(1S)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]propanamide —— C16H22N4O3S
3-(methanesulfonamido)-N-[(1S)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]propanamide
—— (2S)-2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-[(2S)-4-phenylbutan-2-yl]propanamide —— C22H26N4OS
(2S)-2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-[(2S)-4-phenylbutan-2-yl]propanamide
—— 3-(methanesulfonamido)-N-[(1R)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]propanamide —— C16H22N4O3S
3-(methanesulfonamido)-N-[(1R)-1-(5-methyl-1-phenylpyrazol-4-yl)ethyl]propanamide
—— 2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-(3-chlorophenyl)acetamide —— C17H15ClN4OS
2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-(3-chlorophenyl)acetamide
—— (4aR,6R,8aS)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-6-methoxy-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine —— C19H24FN3O2
(4aR,6R,8aS)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-6-methoxy-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine
—— methyl 2-[[[(2S)-2-ethylhexanoyl]-(2-methoxyethyl)amino]methyl]-1,3-thiazole-4-carboxylate —— C17H28N2O4S
methyl 2-[[[(2S)-2-ethylhexanoyl]-(2-methoxyethyl)amino]methyl]-1,3-thiazole-4-carboxylate
—— N-[(4R)-1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-4-hydroxy-6-oxo-1H-pyridine-3-carboxamide —— C23H26N4O3
N-[(4R)-1-(4-tert-butylphenyl)-4,5,6,7-tetrahydroindazol-4-yl]-4-hydroxy-6-oxo-1H-pyridine-3-carboxamide
—— 2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-(3,5-dichlorophenyl)acetamide —— C17H14Cl2N4OS
2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-(3,5-dichlorophenyl)acetamide
—— 2-[[5-(2-Chlorophenyl)-2-(4-fluorophenyl)pyrazole-3-carbonyl]amino]ethyl-dimethylazanium —— C20H21ClFN4O+
2-[[5-(2-Chlorophenyl)-2-(4-fluorophenyl)pyrazole-3-carbonyl]amino]ethyl-dimethylazanium
—— [2-(2-aminoethyl)-1,3-thiazol-4-yl]-[(3R,4R)-3,4-dimethylpyrrolidin-1-yl]methanone —— C12H19N3OS
[2-(2-aminoethyl)-1,3-thiazol-4-yl]-[(3R,4R)-3,4-dimethylpyrrolidin-1-yl]methanone
—— N-[(1S)-1-imidazo[1,2-a]pyrimidin-2-ylpropyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide —— C20H20N6O2
N-[(1S)-1-imidazo[1,2-a]pyrimidin-2-ylpropyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
—— (2S)-2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-[4-(trifluoromethyl)phenyl]propanamide —— C19H17F3N4OS
(2S)-2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-[4-(trifluoromethyl)phenyl]propanamide
—— 2-[2-(4-Bromophenoxy)ethylsulfanyl]-4-phenylimidazol-1-amine —— C17H16BrN3OS
2-[2-(4-Bromophenoxy)ethylsulfanyl]-4-phenylimidazol-1-amine
—— (4aR,6S,8aR)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-6-methoxy-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine —— C19H24FN3O2
(4aR,6S,8aR)-4-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-6-methoxy-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazine
—— 2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-[(1S)-1-cyclopropylethyl]-N-(2,2,2-trifluoroethyl)acetamide —— C18H21F3N4OS
2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-[(1S)-1-cyclopropylethyl]-N-(2,2,2-trifluoroethyl)acetamide
—— [2-(2-aminoethyl)-1,3-thiazol-4-yl]-[(3S,4S)-3,4-dimethylpyrrolidin-1-yl]methanone —— C12H19N3OS
[2-(2-aminoethyl)-1,3-thiazol-4-yl]-[(3S,4S)-3,4-dimethylpyrrolidin-1-yl]methanone
—— (3S)-1-[2-[[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]amino]ethyl]piperidine-3-carboxamide —— C18H22FN5O2
(3S)-1-[2-[[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]amino]ethyl]piperidine-3-carboxamide
—— (2R)-1-[[1-(4-methylphenyl)pyrazolo[3,4-d]pyrimidin-4-yl]amino]propan-2-ol —— C15H17N5O
(2R)-1-[[1-(4-methylphenyl)pyrazolo[3,4-d]pyrimidin-4-yl]amino]propan-2-ol
—— (3R)-1-[2-[[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]amino]ethyl]piperidine-3-carboxamide —— C18H22FN5O2
(3R)-1-[2-[[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]amino]ethyl]piperidine-3-carboxamide
—— 5-cyclohexyl-N-[(1R)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide —— C17H25N5O2
5-cyclohexyl-N-[(1R)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
—— N-[[(2S)-oxolan-2-yl]methyl]-2-(2-phenylimidazol-1-yl)acetamide —— C16H19N3O2
N-[[(2S)-oxolan-2-yl]methyl]-2-(2-phenylimidazol-1-yl)acetamide
—— 2-(3-methylphenyl)-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-5-phenylpyrazole-3-carboxamide —— C26H32N4O
2-(3-methylphenyl)-N-[3-[(2R)-2-methylpiperidin-1-yl]propyl]-5-phenylpyrazole-3-carboxamide
—— 5-cyclohexyl-N-[(1S)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide —— C17H25N5O2
5-cyclohexyl-N-[(1S)-2-methoxy-1-(2-methylpyrazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
—— 2-propyl-N-[(1S)-2,2,2-trifluoro-1-pyridin-2-ylethyl]-1,3-thiazole-4-carboxamide —— C14H14F3N3OS
2-propyl-N-[(1S)-2,2,2-trifluoro-1-pyridin-2-ylethyl]-1,3-thiazole-4-carboxamide
—— 2-(3-methylphenyl)-N-[3-[(2R)-2-methylpiperidin-1-ium-1-yl]propyl]-5-phenylpyrazole-3-carboxamide —— C26H33N4O+
2-(3-methylphenyl)-N-[3-[(2R)-2-methylpiperidin-1-ium-1-yl]propyl]-5-phenylpyrazole-3-carboxamide
—— N-[(1S)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-methyl-1-propylpyrazole-4-carboxamide —— C20H24FN5O
N-[(1S)-1-[1-(3-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-3-methyl-1-propylpyrazole-4-carboxamide
—— (2R)-2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-(3,5-dichlorophenyl)propanamide —— C18H16Cl2N4OS
(2R)-2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-N-(3,5-dichlorophenyl)propanamide
—— N-[[(2R)-oxolan-2-yl]methyl]-2-(2-phenylimidazol-1-yl)acetamide —— C16H19N3O2
N-[[(2R)-oxolan-2-yl]methyl]-2-(2-phenylimidazol-1-yl)acetamide
—— 2-[(3,4-Dichlorophenyl)methylsulfanyl]-4-phenylimidazol-1-amine —— C16H13Cl2N3S
2-[(3,4-Dichlorophenyl)methylsulfanyl]-4-phenylimidazol-1-amine