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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-hydroxy-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]-1-[2-(trifluoromethyl)phenyl]pyrazole-3-carboxamide —— C17H18F3N3O3
4-hydroxy-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]-1-[2-(trifluoromethyl)phenyl]pyrazole-3-carboxamide
—— (5R)-7-(2-methoxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H28N4O3
(5R)-7-(2-methoxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— 4-hydroxy-N-[(1R)-1-[(2R)-oxolan-2-yl]ethyl]-1-[2-(trifluoromethyl)phenyl]pyrazole-3-carboxamide —— C17H18F3N3O3
4-hydroxy-N-[(1R)-1-[(2R)-oxolan-2-yl]ethyl]-1-[2-(trifluoromethyl)phenyl]pyrazole-3-carboxamide
—— (5S)-7-(2-methoxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one —— C21H28N4O3
(5S)-7-(2-methoxyethyl)-2-[[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl]-2,7-diazaspiro[4.5]decan-6-one
—— (3S)-1-[2-[methyl-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino]pyrimidin-4-yl]pyrrolidin-3-ol —— C18H20N6O2
(3S)-1-[2-[methyl-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino]pyrimidin-4-yl]pyrrolidin-3-ol
—— 4-hydroxy-N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]-1-[2-(trifluoromethyl)phenyl]pyrazole-3-carboxamide —— C17H18F3N3O3
4-hydroxy-N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]-1-[2-(trifluoromethyl)phenyl]pyrazole-3-carboxamide
—— 2-[[5-(4-Bromophenyl)-4-(2-methylprop-2-enyl)-1,2,4-triazol-3-yl]sulfanyl]acetate —— C14H13BrN3O2S-
2-[[5-(4-Bromophenyl)-4-(2-methylprop-2-enyl)-1,2,4-triazol-3-yl]sulfanyl]acetate
—— 5-phenyl-N-[[(3S)-1-pyridin-2-ylpiperidin-3-yl]methyl]-1H-pyrazole-4-carboxamide —— C21H23N5O
5-phenyl-N-[[(3S)-1-pyridin-2-ylpiperidin-3-yl]methyl]-1H-pyrazole-4-carboxamide
—— 6-tert-butyl-N-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C17H28N4OS
6-tert-butyl-N-[2-[(1S,2S)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— 5-phenyl-N-[[(3R)-1-pyridin-2-ylpiperidin-3-yl]methyl]-1H-pyrazole-4-carboxamide —— C21H23N5O
5-phenyl-N-[[(3R)-1-pyridin-2-ylpiperidin-3-yl]methyl]-1H-pyrazole-4-carboxamide
—— 6-tert-butyl-N-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C17H28N4OS
6-tert-butyl-N-[2-[(1R,2S)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— (4R)-7-amino-4-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3,4-dihydro-1H-1,8-naphthyridin-2-one —— C19H19N5O
(4R)-7-amino-4-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3,4-dihydro-1H-1,8-naphthyridin-2-one
—— [4-(1H-pyrazol-5-yl)phenyl]-[(2R)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone —— C17H16N4OS
[4-(1H-pyrazol-5-yl)phenyl]-[(2R)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone
—— (4S)-7-amino-4-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3,4-dihydro-1H-1,8-naphthyridin-2-one —— C19H19N5O
(4S)-7-amino-4-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3,4-dihydro-1H-1,8-naphthyridin-2-one
—— 6-tert-butyl-N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C17H28N4OS
6-tert-butyl-N-[2-[(1R,2R)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— N-[[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]methyl]-N-methyl-1-[(2R)-oxolan-2-yl]methanamine —— C15H18ClN3O2
N-[[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]methyl]-N-methyl-1-[(2R)-oxolan-2-yl]methanamine
—— (2R)-1-[5-(methoxymethyl)-3-(2-methyl-1,3-thiazol-4-yl)-1,2,4-triazol-1-yl]butan-2-ol —— C12H18N4O2S
(2R)-1-[5-(methoxymethyl)-3-(2-methyl-1,3-thiazol-4-yl)-1,2,4-triazol-1-yl]butan-2-ol
—— N-[[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]methyl]-N-methyl-1-[(2S)-oxolan-2-yl]methanamine —— C15H18ClN3O2
N-[[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]methyl]-N-methyl-1-[(2S)-oxolan-2-yl]methanamine
—— 6-tert-butyl-N-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine —— C17H28N4OS
6-tert-butyl-N-[2-[(1S,2R)-2-methylcyclohexyl]oxyethyl]imidazo[2,1-b][1,3,4]thiadiazol-2-amine
—— [4-(1H-pyrazol-5-yl)phenyl]-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone —— C17H16N4OS
[4-(1H-pyrazol-5-yl)phenyl]-[(2S)-2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methanone
—— N-[(2R)-butan-2-yl]-2-[[4-(4-fluorophenyl)-5-(2-methylfuran-3-yl)-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C19H21FN4O2S
N-[(2R)-butan-2-yl]-2-[[4-(4-fluorophenyl)-5-(2-methylfuran-3-yl)-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— (2S)-1-[5-(methoxymethyl)-3-(2-methyl-1,3-thiazol-4-yl)-1,2,4-triazol-1-yl]butan-2-ol —— C12H18N4O2S
(2S)-1-[5-(methoxymethyl)-3-(2-methyl-1,3-thiazol-4-yl)-1,2,4-triazol-1-yl]butan-2-ol
—— 2-[[5-(cyclohexylcarbamoylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]-N-(furan-2-ylmethyl)acetamide —— C16H21N5O3S2
2-[[5-(cyclohexylcarbamoylamino)-1,3,4-thiadiazol-2-yl]sulfanyl]-N-(furan-2-ylmethyl)acetamide
—— (3R)-5-oxo-1-(pyridin-3-ylmethyl)-N-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]pyrrolidine-3-carboxamide —— C20H20N6O2
(3R)-5-oxo-1-(pyridin-3-ylmethyl)-N-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]pyrrolidine-3-carboxamide
—— (3S)-5-oxo-1-(pyridin-3-ylmethyl)-N-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]pyrrolidine-3-carboxamide —— C20H20N6O2
(3S)-5-oxo-1-(pyridin-3-ylmethyl)-N-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]pyrrolidine-3-carboxamide
—— 5-(morpholin-4-ylmethyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]furan-3-carboxamide —— C20H23N5O3
5-(morpholin-4-ylmethyl)-N-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]furan-3-carboxamide
—— 5-tert-butyl-N-[(1S)-1-(2-methylpyrazol-3-yl)propyl]-1,3,4-oxadiazol-2-amine —— C13H21N5O
5-tert-butyl-N-[(1S)-1-(2-methylpyrazol-3-yl)propyl]-1,3,4-oxadiazol-2-amine
—— 2-((5-(3-(tert-butyl)ureido)-1,3,4-thiadiazol-2-yl)thio)-N-isopropylacetamide —— C12H21N5O2S2
2-((5-(3-(tert-butyl)ureido)-1,3,4-thiadiazol-2-yl)thio)-N-isopropylacetamide
—— 1-Cyclohexyl-3-(5-((2-morpholino-2-oxoethyl)thio)-1,3,4-thiadiazol-2-yl)urea —— C15H23N5O3S2
1-Cyclohexyl-3-(5-((2-morpholino-2-oxoethyl)thio)-1,3,4-thiadiazol-2-yl)urea
—— 1-(Tert-butyl)-3-(5-((2-morpholino-2-oxoethyl)thio)-1,3,4-thiadiazol-2-yl)urea —— C13H21N5O3S2
1-(Tert-butyl)-3-(5-((2-morpholino-2-oxoethyl)thio)-1,3,4-thiadiazol-2-yl)urea
—— 1-(Tert-butyl)-3-(5-((2-oxo-2-(pyrrolidin-1-yl)ethyl)thio)-1,3,4-thiadiazol-2-yl)urea —— C13H21N5O2S2
1-(Tert-butyl)-3-(5-((2-oxo-2-(pyrrolidin-1-yl)ethyl)thio)-1,3,4-thiadiazol-2-yl)urea
—— 2-[(E)-2-(2-methoxyphenyl)ethenyl]-5-[[(2S)-oxolan-2-yl]methylamino]-1,3-oxazole-4-carbonitrile —— C18H19N3O3
2-[(E)-2-(2-methoxyphenyl)ethenyl]-5-[[(2S)-oxolan-2-yl]methylamino]-1,3-oxazole-4-carbonitrile
—— 1-Tert-butyl-3-(5-butylsulfanyl-1,3,4-thiadiazol-2-yl)urea —— C11H20N4OS2
1-Tert-butyl-3-(5-butylsulfanyl-1,3,4-thiadiazol-2-yl)urea
—— 2-({5-[(Tert-butylcarbamoyl)amino]-1,3,4-thiadiazol-2-YL}sulfanyl)-N-propylacetamide —— C12H21N5O2S2
2-({5-[(Tert-butylcarbamoyl)amino]-1,3,4-thiadiazol-2-YL}sulfanyl)-N-propylacetamide
—— (3R)-1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperidine-3-carboxamide —— C20H19FN4O2
(3R)-1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperidine-3-carboxamide
—— 5-tert-butyl-N-[(1R)-1-(2-methylpyrazol-3-yl)propyl]-1,3,4-oxadiazol-2-amine —— C13H21N5O
5-tert-butyl-N-[(1R)-1-(2-methylpyrazol-3-yl)propyl]-1,3,4-oxadiazol-2-amine
—— (3S)-1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperidine-3-carboxamide —— C20H19FN4O2
(3S)-1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperidine-3-carboxamide
—— 5-(morpholin-4-ylmethyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]furan-3-carboxamide —— C20H23N5O3
5-(morpholin-4-ylmethyl)-N-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]furan-3-carboxamide
—— N-[(1S)-1-[1-(4-methoxyphenyl)pyrazol-4-yl]ethyl]-4-methylpyrimidin-2-amine —— C17H19N5O
N-[(1S)-1-[1-(4-methoxyphenyl)pyrazol-4-yl]ethyl]-4-methylpyrimidin-2-amine
—— (2-cyclopropylpyrimidin-5-yl)-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C20H19N5O2
(2-cyclopropylpyrimidin-5-yl)-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— (2-cyclopropylpyrimidin-5-yl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone —— C20H19N5O2
(2-cyclopropylpyrimidin-5-yl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methanone
—— N-[(1R)-1-[1-(4-methoxyphenyl)pyrazol-4-yl]ethyl]-4-methylpyrimidin-2-amine —— C17H19N5O
N-[(1R)-1-[1-(4-methoxyphenyl)pyrazol-4-yl]ethyl]-4-methylpyrimidin-2-amine
—— 2-[[5-(4-chlorophenyl)-1H-imidazol-2-yl]sulfanyl]-1-[(3S)-3-methylpiperidin-1-yl]ethanone —— C17H20ClN3OS
2-[[5-(4-chlorophenyl)-1H-imidazol-2-yl]sulfanyl]-1-[(3S)-3-methylpiperidin-1-yl]ethanone
—— (3S)-1-(furan-2-ylmethyl)-N-[(2-pyrazol-1-ylphenyl)methyl]piperidine-3-carboxamide —— C21H24N4O2
(3S)-1-(furan-2-ylmethyl)-N-[(2-pyrazol-1-ylphenyl)methyl]piperidine-3-carboxamide
—— (3R)-3-[3-(ethoxymethyl)-5-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide —— C16H23N5O3S
(3R)-3-[3-(ethoxymethyl)-5-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide
—— (3S)-3-[3-(ethoxymethyl)-5-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide —— C16H23N5O3S
(3S)-3-[3-(ethoxymethyl)-5-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide
—— (3R)-1-(furan-2-ylmethyl)-N-[(2-pyrazol-1-ylphenyl)methyl]piperidine-3-carboxamide —— C21H24N4O2
(3R)-1-(furan-2-ylmethyl)-N-[(2-pyrazol-1-ylphenyl)methyl]piperidine-3-carboxamide
—— (2S)-2-[[4-(5-methoxy-2-pyrazol-1-ylphenyl)triazol-1-yl]methyl]morpholine —— C17H20N6O2
(2S)-2-[[4-(5-methoxy-2-pyrazol-1-ylphenyl)triazol-1-yl]methyl]morpholine
—— [(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-(2-pyrazol-1-ylphenyl)methanone —— C21H28N4O3
[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-(2-pyrazol-1-ylphenyl)methanone
—— (6R)-1,10-dimethyl-4-[(3-pyrazol-1-ylphenyl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H29N5O
(6R)-1,10-dimethyl-4-[(3-pyrazol-1-ylphenyl)methyl]-1,4,10-triazaspiro[5.6]dodecan-9-one