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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2'R,7S)-5-amino-2,2'-dimethylspiro[4H-[1,3]oxazolo[5,4-b]pyridine-7,3'-oxolane]-6-carbonitrile —— C12H14N4O2
(2'R,7S)-5-amino-2,2'-dimethylspiro[4H-[1,3]oxazolo[5,4-b]pyridine-7,3'-oxolane]-6-carbonitrile
—— (7S)-5-amino-2-phenyl-7-propan-2-yl-4,7-dihydro-[1,3]oxazolo[5,4-b]pyridine-6-carbonitrile —— C16H16N4O
(7S)-5-amino-2-phenyl-7-propan-2-yl-4,7-dihydro-[1,3]oxazolo[5,4-b]pyridine-6-carbonitrile
—— 5-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-[(E)-2-(4-ethoxyphenyl)ethenyl]-1,3-oxazole-4-carbonitrile —— C20H23N3O3
5-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-[(E)-2-(4-ethoxyphenyl)ethenyl]-1,3-oxazole-4-carbonitrile
—— (2R)-2-(3-chlorophenoxy)-N-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]propanamide —— C19H18ClN3O3
(2R)-2-(3-chlorophenoxy)-N-[[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]propanamide
—— (NE)-N-[(6R)-3-ethyl-6-[(2S)-2-ethylsulfanylpropyl]-6,7-dihydro-5H-1,2-benzoxazol-4-ylidene]hydroxylamine —— C14H22N2O2S
(NE)-N-[(6R)-3-ethyl-6-[(2S)-2-ethylsulfanylpropyl]-6,7-dihydro-5H-1,2-benzoxazol-4-ylidene]hydroxylamine
—— (3S)-1-[2-[[1-(4-fluorophenyl)pyrazol-4-yl]methyl-methylamino]pyrimidin-4-yl]pyrrolidin-3-ol —— C19H21FN6O
(3S)-1-[2-[[1-(4-fluorophenyl)pyrazol-4-yl]methyl-methylamino]pyrimidin-4-yl]pyrrolidin-3-ol
—— 1,4,5-triphenyl-3-[[(2R)-thiiran-2-yl]methyl]imidazol-2-one —— C24H20N2OS
1,4,5-triphenyl-3-[[(2R)-thiiran-2-yl]methyl]imidazol-2-one
—— 4-chloro-N-[(2R)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]butan-2-yl]aniline —— C19H22ClN5
4-chloro-N-[(2R)-2-[1-(2,6-dimethylphenyl)tetrazol-5-yl]butan-2-yl]aniline
—— 3-[(3R)-1-methylpiperidin-3-yl]-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]propanamide —— C19H26N4O2
3-[(3R)-1-methylpiperidin-3-yl]-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]propanamide
—— 1-(3-chloro-2-methylphenyl)-5-[(2S)-2-imidazol-1-ylpropyl]-1,2,4-triazole —— C15H16ClN5
1-(3-chloro-2-methylphenyl)-5-[(2S)-2-imidazol-1-ylpropyl]-1,2,4-triazole
—— 3-[(3S)-1-methylpiperidin-3-yl]-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]propanamide —— C19H26N4O2
3-[(3S)-1-methylpiperidin-3-yl]-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]propanamide
—— 1-(3-chloro-2-methylphenyl)-5-[(2R)-2-imidazol-1-ylpropyl]-1,2,4-triazole —— C15H16ClN5
1-(3-chloro-2-methylphenyl)-5-[(2R)-2-imidazol-1-ylpropyl]-1,2,4-triazole
—— [2-(4-fluorophenyl)imidazo[1,2-a]pyridin-6-yl]-[(2S)-2-(hydroxymethyl)piperidin-1-yl]methanone —— C20H20FN3O2
[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-6-yl]-[(2S)-2-(hydroxymethyl)piperidin-1-yl]methanone
—— (2S)-N-(2-imidazo[2,1-b][1,3]thiazol-6-ylethyl)-2-(2-propan-2-ylimidazol-1-yl)propanamide —— C16H21N5OS
(2S)-N-(2-imidazo[2,1-b][1,3]thiazol-6-ylethyl)-2-(2-propan-2-ylimidazol-1-yl)propanamide
—— 5-[(3S)-1-(1,6-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-phenyl-1,2,4-oxadiazole —— C20H21N7O
5-[(3S)-1-(1,6-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(3R)-1-(1,6-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-phenyl-1,2,4-oxadiazole —— C20H21N7O
5-[(3R)-1-(1,6-dimethylpyrazolo[3,4-d]pyrimidin-4-yl)piperidin-3-yl]-3-phenyl-1,2,4-oxadiazole
—— N-(cyclobutylmethyl)-N-[[(2R)-oxolan-2-yl]methyl]-4-(1H-pyrazol-5-yl)benzamide —— C20H25N3O2
N-(cyclobutylmethyl)-N-[[(2R)-oxolan-2-yl]methyl]-4-(1H-pyrazol-5-yl)benzamide
—— (3S)-5-oxo-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide —— C21H20N4O3
(3S)-5-oxo-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
—— (2R)-N-(2-imidazo[2,1-b][1,3]thiazol-6-ylethyl)-2-(2-propan-2-ylimidazol-1-yl)propanamide —— C16H21N5OS
(2R)-N-(2-imidazo[2,1-b][1,3]thiazol-6-ylethyl)-2-(2-propan-2-ylimidazol-1-yl)propanamide
—— [(4S)-4-[1-(2,6-dimethylphenyl)tetrazol-5-yl]-2,2-dimethyloxan-4-yl]-methylazanium —— C17H26N5O+
[(4S)-4-[1-(2,6-dimethylphenyl)tetrazol-5-yl]-2,2-dimethyloxan-4-yl]-methylazanium
—— 5-cyclopropyl-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]-1,3,4-oxadiazol-2-amine —— C16H17N5O
5-cyclopropyl-N-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]-1,3,4-oxadiazol-2-amine
—— 5-cyclopropyl-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]-1,3,4-oxadiazol-2-amine —— C16H17N5O
5-cyclopropyl-N-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]-1,3,4-oxadiazol-2-amine
—— [2-(4-fluorophenyl)imidazo[1,2-a]pyridin-6-yl]-[(2R)-2-(hydroxymethyl)piperidin-1-yl]methanone —— C20H20FN3O2
[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-6-yl]-[(2R)-2-(hydroxymethyl)piperidin-1-yl]methanone
—— (3R)-5-oxo-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide —— C21H20N4O3
(3R)-5-oxo-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
—— 2-(4-fluorophenyl)-N-[(1S)-1-(5-methyl-1H-imidazol-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide —— C20H18FN5O
2-(4-fluorophenyl)-N-[(1S)-1-(5-methyl-1H-imidazol-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
—— (2-Oxo-2-piperidin-1-ylethyl) 1-(2-chlorophenyl)-3-methylthieno[2,3-c]pyrazole-5-carboxylate —— C20H20ClN3O3S
(2-Oxo-2-piperidin-1-ylethyl) 1-(2-chlorophenyl)-3-methylthieno[2,3-c]pyrazole-5-carboxylate
—— 2-(4-fluorophenyl)-N-[(1R)-1-(5-methyl-1H-imidazol-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide —— C20H18FN5O
2-(4-fluorophenyl)-N-[(1R)-1-(5-methyl-1H-imidazol-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
—— N-(cyclobutylmethyl)-N-[[(2S)-oxolan-2-yl]methyl]-4-(1H-pyrazol-5-yl)benzamide —— C20H25N3O2
N-(cyclobutylmethyl)-N-[[(2S)-oxolan-2-yl]methyl]-4-(1H-pyrazol-5-yl)benzamide
—— (6S)-4-[[1-(4-methoxyphenyl)imidazol-2-yl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one —— C21H29N5O2
(6S)-4-[[1-(4-methoxyphenyl)imidazol-2-yl]methyl]-1-methyl-1,4,10-triazaspiro[5.6]dodecan-9-one
—— (1R)-2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-1-(2,5-difluorophenyl)ethanol —— C17H15F2N3OS
(1R)-2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-1-(2,5-difluorophenyl)ethanol
—— (2R)-N-[[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-1,2,3,4-tetrahydronaphthalen-2-amine —— C22H23F2N3
(2R)-N-[[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-1,2,3,4-tetrahydronaphthalen-2-amine
—— 2-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3H-thieno[3,2-d]pyrimidin-4-one —— C17H15N5O2S2
2-[[5-(4-methoxyphenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-3H-thieno[3,2-d]pyrimidin-4-one
—— (2S)-N-[[3-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-N-methyl-2-(2-propan-2-ylimidazol-1-yl)propanamide —— C22H29N5O
(2S)-N-[[3-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-N-methyl-2-(2-propan-2-ylimidazol-1-yl)propanamide
—— 5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-[(1-phenyltetrazol-5-yl)methyl]-1,2-dihydropyrazole-3-carboxamide —— C18H15N7O2
5-(6-oxocyclohexa-2,4-dien-1-ylidene)-N-[(1-phenyltetrazol-5-yl)methyl]-1,2-dihydropyrazole-3-carboxamide
—— 3-(3-bromophenyl)-5-[(1S)-1-(3-methylphenoxy)ethyl]-1,2,4-oxadiazole —— C17H15BrN2O2
3-(3-bromophenyl)-5-[(1S)-1-(3-methylphenoxy)ethyl]-1,2,4-oxadiazole
—— (1S)-2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-1-(2,5-difluorophenyl)ethanol —— C17H15F2N3OS
(1S)-2-(1-amino-4-phenylimidazol-2-yl)sulfanyl-1-(2,5-difluorophenyl)ethanol
—— (3S,4R)-N,N-dimethyl-1-[3-(2-methylimidazol-1-yl)propyl]-4-propan-2-ylpyrrolidin-3-amine —— C16H30N4
(3S,4R)-N,N-dimethyl-1-[3-(2-methylimidazol-1-yl)propyl]-4-propan-2-ylpyrrolidin-3-amine
—— (3R)-1-(furan-2-ylmethyl)-N-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]piperidine-3-carboxamide —— C20H23N5O2
(3R)-1-(furan-2-ylmethyl)-N-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]piperidine-3-carboxamide
—— 5,6-dimethyl-2-[(1S)-1-[(4-phenyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C18H17N5OS2
5,6-dimethyl-2-[(1S)-1-[(4-phenyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (3S)-1-(furan-2-ylmethyl)-N-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]piperidine-3-carboxamide —— C20H23N5O2
(3S)-1-(furan-2-ylmethyl)-N-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]piperidine-3-carboxamide
—— (2R)-N-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-2-(2-propan-2-ylimidazol-1-yl)propanamide —— C15H22N6O
(2R)-N-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-2-(2-propan-2-ylimidazol-1-yl)propanamide
—— 2-[1-[(2R)-2-methoxy-2-thiophen-2-ylethyl]triazol-4-yl]-1,3-thiazole —— C12H12N4OS2
2-[1-[(2R)-2-methoxy-2-thiophen-2-ylethyl]triazol-4-yl]-1,3-thiazole
—— (2S)-N-[[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-1,2,3,4-tetrahydronaphthalen-2-amine —— C22H23F2N3
(2S)-N-[[1-(2,4-difluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-1,2,3,4-tetrahydronaphthalen-2-amine
—— 5,6-dimethyl-2-[(1R)-1-[(4-phenyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one —— C18H17N5OS2
5,6-dimethyl-2-[(1R)-1-[(4-phenyl-1,2,4-triazol-3-yl)sulfanyl]ethyl]-3H-thieno[2,3-d]pyrimidin-4-one
—— (2R)-N-[[3-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-N-methyl-2-(2-propan-2-ylimidazol-1-yl)propanamide —— C22H29N5O
(2R)-N-[[3-(3,5-dimethylpyrazol-1-yl)phenyl]methyl]-N-methyl-2-(2-propan-2-ylimidazol-1-yl)propanamide
—— (2S)-N-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-2-(2-propan-2-ylimidazol-1-yl)propanamide —— C15H22N6O
(2S)-N-(6,7-dihydro-5H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl)-2-(2-propan-2-ylimidazol-1-yl)propanamide
—— 4-[[5-(4-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-2-ethanimidoyl-3-oxobutanenitrile —— C19H20ClN5O2S
4-[[5-(4-chlorophenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-2-ethanimidoyl-3-oxobutanenitrile
—— 4-[(1S)-1-[4-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)phenyl]ethyl]morpholine —— C18H24N4O
4-[(1S)-1-[4-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)phenyl]ethyl]morpholine
—— 2-[1-[(2S)-2-methoxy-2-thiophen-2-ylethyl]triazol-4-yl]-1,3-thiazole —— C12H12N4OS2
2-[1-[(2S)-2-methoxy-2-thiophen-2-ylethyl]triazol-4-yl]-1,3-thiazole
—— 4-[(1R)-1-[4-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)phenyl]ethyl]morpholine —— C18H24N4O
4-[(1R)-1-[4-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)phenyl]ethyl]morpholine