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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[[(2R)-oxolan-2-yl]methyl]-5-phenyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide —— C20H21N3O2S
N-[[(2R)-oxolan-2-yl]methyl]-5-phenyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
—— (5R)-9-[[1-(2-methoxyphenyl)pyrazol-4-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C20H27N3O3
(5R)-9-[[1-(2-methoxyphenyl)pyrazol-4-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— N-[(2S)-5-(diethylamino)pentan-2-yl]-5-(5-methylfuran-2-yl)-2-phenylpyrazole-3-carboxamide —— C24H32N4O2
N-[(2S)-5-(diethylamino)pentan-2-yl]-5-(5-methylfuran-2-yl)-2-phenylpyrazole-3-carboxamide
—— N-[[(2S)-oxolan-2-yl]methyl]-5-phenyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide —— C20H21N3O2S
N-[[(2S)-oxolan-2-yl]methyl]-5-phenyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
—— 4-methyl-5-[[(3S)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methyl]-1,3-thiazole —— C17H23N7S
4-methyl-5-[[(3S)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methyl]-1,3-thiazole
—— 4-methyl-5-[[(3R)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methyl]-1,3-thiazole —— C17H23N7S
4-methyl-5-[[(3R)-3-[4-methyl-5-(pyrazol-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]methyl]-1,3-thiazole
—— 4-(2-methylimidazol-1-yl)-1-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]butan-1-one —— C20H23N5O2
4-(2-methylimidazol-1-yl)-1-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]butan-1-one
—— (5S)-9-[[1-(2-methoxyphenyl)pyrazol-4-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C20H27N3O3
(5S)-9-[[1-(2-methoxyphenyl)pyrazol-4-yl]methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (6S)-6-[(1,3-dimethylpyrazolo[3,4-d][1,3]thiazol-5-yl)amino]-2-methylheptan-2-ol —— C14H24N4OS
(6S)-6-[(1,3-dimethylpyrazolo[3,4-d][1,3]thiazol-5-yl)amino]-2-methylheptan-2-ol
—— (2R)-2-(2-methylphenyl)-N-[2-pyrazol-1-yl-5-(trifluoromethyl)phenyl]pyrrolidine-1-carboxamide —— C22H21F3N4O
(2R)-2-(2-methylphenyl)-N-[2-pyrazol-1-yl-5-(trifluoromethyl)phenyl]pyrrolidine-1-carboxamide
—— [4-[(2R)-2-hydroxy-3,3-dimethylbutyl]piperazin-1-yl]-[3-methyl-5-(methylamino)-1,2-thiazol-4-yl]methanone —— C16H28N4O2S
[4-[(2R)-2-hydroxy-3,3-dimethylbutyl]piperazin-1-yl]-[3-methyl-5-(methylamino)-1,2-thiazol-4-yl]methanone
—— (6R)-6-[(1,3-dimethylpyrazolo[3,4-d][1,3]thiazol-5-yl)amino]-2-methylheptan-2-ol —— C14H24N4OS
(6R)-6-[(1,3-dimethylpyrazolo[3,4-d][1,3]thiazol-5-yl)amino]-2-methylheptan-2-ol
—— (2S)-2-(2-methylphenyl)-N-[2-pyrazol-1-yl-5-(trifluoromethyl)phenyl]pyrrolidine-1-carboxamide —— C22H21F3N4O
(2S)-2-(2-methylphenyl)-N-[2-pyrazol-1-yl-5-(trifluoromethyl)phenyl]pyrrolidine-1-carboxamide
—— [4-[(2S)-2-hydroxy-3,3-dimethylbutyl]piperazin-1-yl]-[3-methyl-5-(methylamino)-1,2-thiazol-4-yl]methanone —— C16H28N4O2S
[4-[(2S)-2-hydroxy-3,3-dimethylbutyl]piperazin-1-yl]-[3-methyl-5-(methylamino)-1,2-thiazol-4-yl]methanone
—— (3R)-1-(6-methylpyridazin-3-yl)-N-[(1-phenylpyrazol-3-yl)methyl]piperidin-3-amine —— C20H24N6
(3R)-1-(6-methylpyridazin-3-yl)-N-[(1-phenylpyrazol-3-yl)methyl]piperidin-3-amine
—— N-[(1-phenylpyrazol-3-yl)methyl]-1-[(2S)-1-pyridazin-3-ylpyrrolidin-2-yl]methanamine —— C19H22N6
N-[(1-phenylpyrazol-3-yl)methyl]-1-[(2S)-1-pyridazin-3-ylpyrrolidin-2-yl]methanamine
—— 4-(2-methylimidazol-1-yl)-1-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]butan-1-one —— C20H23N5O2
4-(2-methylimidazol-1-yl)-1-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]butan-1-one
—— 1-ethyl-1-[(1R)-1-(4-fluorophenyl)ethyl]-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea —— C14H14F4N4OS
1-ethyl-1-[(1R)-1-(4-fluorophenyl)ethyl]-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
—— (3R)-3-[5-cyclobutyl-3-(thiophen-2-ylmethyl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide —— C15H19N3O2S2
(3R)-3-[5-cyclobutyl-3-(thiophen-2-ylmethyl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide
—— 1-ethyl-1-[(1S)-1-(4-fluorophenyl)ethyl]-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea —— C14H14F4N4OS
1-ethyl-1-[(1S)-1-(4-fluorophenyl)ethyl]-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
—— (3S)-3-[5-cyclobutyl-3-(thiophen-2-ylmethyl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide —— C15H19N3O2S2
(3S)-3-[5-cyclobutyl-3-(thiophen-2-ylmethyl)-1,2,4-triazol-1-yl]thiolane 1,1-dioxide
—— 2-[[(2R)-butan-2-yl]-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]amino]acetic acid —— C16H19ClN2O3
2-[[(2R)-butan-2-yl]-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]amino]acetic acid
—— N-[(1-phenylpyrazol-3-yl)methyl]-1-[(2R)-1-pyridazin-3-ylpyrrolidin-2-yl]methanamine —— C19H22N6
N-[(1-phenylpyrazol-3-yl)methyl]-1-[(2R)-1-pyridazin-3-ylpyrrolidin-2-yl]methanamine
—— (3S)-1-(6-methylpyridazin-3-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-3-amine —— C20H23N5O
(3S)-1-(6-methylpyridazin-3-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-3-amine
—— (3S)-1-(6-methylpyridazin-3-yl)-N-[(1-phenylpyrazol-3-yl)methyl]piperidin-3-amine —— C20H24N6
(3S)-1-(6-methylpyridazin-3-yl)-N-[(1-phenylpyrazol-3-yl)methyl]piperidin-3-amine
—— 2-[[(2S)-butan-2-yl]-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]amino]acetic acid —— C16H19ClN2O3
2-[[(2S)-butan-2-yl]-[[2-(3-chlorophenyl)-1,3-oxazol-4-yl]methyl]amino]acetic acid
—— 5-[(1-Phenylpyrazol-3-yl)methyl]furo[3,2-c]pyridin-4-one —— C17H13N3O2
5-[(1-Phenylpyrazol-3-yl)methyl]furo[3,2-c]pyridin-4-one
—— (3R)-1-(6-methylpyridazin-3-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-3-amine —— C20H23N5O
(3R)-1-(6-methylpyridazin-3-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidin-3-amine
—— N-[(1R)-1-(furan-2-yl)ethyl]-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]acetamide —— C18H19N3O2S
N-[(1R)-1-(furan-2-yl)ethyl]-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]acetamide
—— (1S,2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-2-(trifluoromethyl)cyclohexane-1-carboxamide —— C21H19F3N2O2
(1S,2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-2-(trifluoromethyl)cyclohexane-1-carboxamide
—— 2-chloro-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-4-(tetrazol-1-yl)benzamide —— C16H14ClN5O2
2-chloro-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]-4-(tetrazol-1-yl)benzamide
—— (1R,2R)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-2-(trifluoromethyl)cyclohexane-1-carboxamide —— C21H19F3N2O2
(1R,2R)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-2-(trifluoromethyl)cyclohexane-1-carboxamide
—— (2R)-2-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-phenylbutanamide —— C19H19FN4OS
(2R)-2-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-phenylbutanamide
—— (2S)-2-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-phenylbutanamide —— C19H19FN4OS
(2S)-2-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanyl]-N-phenylbutanamide
—— (2S)-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-phenylbutanamide —— C21H24N4O2S
(2S)-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-phenylbutanamide
—— (6E)-6-[(5-methylfuran-2-yl)methylidene]-3-(2-methylphenyl)[1,3]thiazolo[2,3-c][1,2,4]triazol-5(6H)-one —— C17H13N3O2S
(6E)-6-[(5-methylfuran-2-yl)methylidene]-3-(2-methylphenyl)[1,3]thiazolo[2,3-c][1,2,4]triazol-5(6H)-one
—— (2R)-N-[5-(2,6-difluorophenyl)-1H-pyrazol-3-yl]-2-pyrazol-1-ylpropanamide —— C15H13F2N5O
(2R)-N-[5-(2,6-difluorophenyl)-1H-pyrazol-3-yl]-2-pyrazol-1-ylpropanamide
—— (2S)-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[[4-methyl-5-[(1S)-1-phenoxyethyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C19H23N5O2S2
(2S)-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[[4-methyl-5-[(1S)-1-phenoxyethyl]-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— 3-Phenyl-5-(3,4,5-triethoxyphenyl)-1,2,4-oxadiazole —— C20H22N2O4
3-Phenyl-5-(3,4,5-triethoxyphenyl)-1,2,4-oxadiazole
—— (2R)-N-(1,3-benzodioxol-5-yl)-2-[[4-ethyl-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide —— C21H22N4O3S
(2R)-N-(1,3-benzodioxol-5-yl)-2-[[4-ethyl-5-(4-methylphenyl)-1,2,4-triazol-3-yl]sulfanyl]propanamide
—— N-[(4S)-2,2-dimethyl-4-[1-(2-methylphenyl)tetrazol-5-yl]oxan-4-yl]-N-methylacetamide —— C18H25N5O2
N-[(4S)-2,2-dimethyl-4-[1-(2-methylphenyl)tetrazol-5-yl]oxan-4-yl]-N-methylacetamide
—— 3-(2-methylsulfanylimidazol-1-yl)-N-[(1R,2R)-2-(trifluoromethyl)cyclohexyl]benzamide —— C18H20F3N3OS
3-(2-methylsulfanylimidazol-1-yl)-N-[(1R,2R)-2-(trifluoromethyl)cyclohexyl]benzamide
—— (1R,2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-2-(trifluoromethyl)cyclohexane-1-carboxamide —— C21H19F3N2O2
(1R,2S)-N-[4-(1,3-benzoxazol-2-yl)phenyl]-2-(trifluoromethyl)cyclohexane-1-carboxamide
—— (2S)-N-[5-(2,6-difluorophenyl)-1H-pyrazol-3-yl]-2-pyrazol-1-ylpropanamide —— C15H13F2N5O
(2S)-N-[5-(2,6-difluorophenyl)-1H-pyrazol-3-yl]-2-pyrazol-1-ylpropanamide
—— (2S)-2-[[5-(3-methylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methyl-1,3-thiazol-2-yl)propanamide —— C19H21N5OS2
(2S)-2-[[5-(3-methylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-(4-methyl-1,3-thiazol-2-yl)propanamide
—— (6Z)-3-(2-chlorophenyl)-6-(3,4-dimethoxybenzylidene)[1,3]thiazolo[2,3-c][1,2,4]triazol-5(6H)-one —— C19H14ClN3O3S
(6Z)-3-(2-chlorophenyl)-6-(3,4-dimethoxybenzylidene)[1,3]thiazolo[2,3-c][1,2,4]triazol-5(6H)-one
—— N-[(1S)-1-(furan-2-yl)ethyl]-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]acetamide —— C18H19N3O2S
N-[(1S)-1-(furan-2-yl)ethyl]-2-[(1-phenylpyrazol-3-yl)methylsulfanyl]acetamide
—— (2S)-2-[[5-(3-methylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3-thiazol-2-yl)propanamide —— C18H19N5OS2
(2S)-2-[[5-(3-methylphenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3-thiazol-2-yl)propanamide
—— (2R)-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3-thiazol-2-yl)propanamide —— C17H19N5O2S2
(2R)-2-[[4-ethyl-5-(4-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3-thiazol-2-yl)propanamide
—— (2S)-2-[[5-(2-fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3-thiazol-2-yl)propanamide —— C17H16FN5OS2
(2S)-2-[[5-(2-fluorophenyl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3-thiazol-2-yl)propanamide