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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-3-[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]-2-(4-ethyl-5-methyl-1,3-thiazol-2-yl)-3-oxopropanenitrile —— C19H15Cl2N3O2S
(2R)-3-[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]-2-(4-ethyl-5-methyl-1,3-thiazol-2-yl)-3-oxopropanenitrile
—— (4S)-4-phenyl-1-[(3-pyrazol-1-ylphenyl)methyl]pyrrolidin-2-one —— C20H19N3O
(4S)-4-phenyl-1-[(3-pyrazol-1-ylphenyl)methyl]pyrrolidin-2-one
—— 1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]ethanone —— C19H16F3N5O
1-(3,4-dihydro-1H-isoquinolin-2-yl)-2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]ethanone
—— (3S)-5-(4-chlorophenyl)-3-(4-methoxyphenyl)-2-phenyl-3,4-dihydropyrazole —— C22H19ClN2O
(3S)-5-(4-chlorophenyl)-3-(4-methoxyphenyl)-2-phenyl-3,4-dihydropyrazole
—— (2R)-2-(6-aminopyridin-3-yl)-2-[[1-(3-methoxyphenyl)pyrazol-4-yl]methyl-methylamino]acetic acid —— C19H21N5O3
(2R)-2-(6-aminopyridin-3-yl)-2-[[1-(3-methoxyphenyl)pyrazol-4-yl]methyl-methylamino]acetic acid
—— 2-(2-phenylimidazol-1-yl)-1-[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]ethanone —— C21H25N5O
2-(2-phenylimidazol-1-yl)-1-[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]ethanone
—— (2R)-2-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(4-methylsulfanylphenyl)pyrrolidine-1-carboxamide —— C20H19FN4O2S
(2R)-2-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(4-methylsulfanylphenyl)pyrrolidine-1-carboxamide
—— N-[(1R)-1-cyano-1-cyclopropylethyl]-2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]acetamide —— C16H15F3N6O
N-[(1R)-1-cyano-1-cyclopropylethyl]-2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]acetamide
—— (4-Benzylpiperazin-4-ium-1-yl)-[5-(2,4-dimethoxyphenyl)-2-methylpyrazol-3-yl]methanone —— C24H29N4O3+
(4-Benzylpiperazin-4-ium-1-yl)-[5-(2,4-dimethoxyphenyl)-2-methylpyrazol-3-yl]methanone
—— (3R)-5-(4-chlorophenyl)-3-(4-methoxyphenyl)-2-phenyl-3,4-dihydropyrazole —— C22H19ClN2O
(3R)-5-(4-chlorophenyl)-3-(4-methoxyphenyl)-2-phenyl-3,4-dihydropyrazole
—— ethyl N-[2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]acetyl]carbamate —— C13H12F3N5O3
ethyl N-[2-[5-[3-(trifluoromethyl)phenyl]tetrazol-2-yl]acetyl]carbamate
—— [(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2,5-dimethylfuran-3-carboxylate —— C21H23N3O5
[(2S)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2,5-dimethylfuran-3-carboxylate
—— 1,3-dimethyl-N-[(1R)-1-(1,3-thiazol-2-yl)ethyl]pyrazolo[3,4-d][1,3]thiazol-5-amine —— C11H13N5S2
1,3-dimethyl-N-[(1R)-1-(1,3-thiazol-2-yl)ethyl]pyrazolo[3,4-d][1,3]thiazol-5-amine
—— (2S)-2-chloro-1-[(2S)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-phenylethanone —— C21H19Cl2N3O2
(2S)-2-chloro-1-[(2S)-2-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-2-phenylethanone
—— 1,3-dimethyl-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]pyrazolo[3,4-d][1,3]thiazol-5-amine —— C11H13N5S2
1,3-dimethyl-N-[(1S)-1-(1,3-thiazol-2-yl)ethyl]pyrazolo[3,4-d][1,3]thiazol-5-amine
—— [(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2,5-dimethylfuran-3-carboxylate —— C21H23N3O5
[(2R)-1-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-1-oxopropan-2-yl] 2,5-dimethylfuran-3-carboxylate
—— 5-[1-(3,5-Dimethoxybenzoyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C21H21N3O4
5-[1-(3,5-Dimethoxybenzoyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— 2-(4-fluorophenyl)-N-[(1R)-1-(2H-tetrazol-5-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide —— C17H14FN7O
2-(4-fluorophenyl)-N-[(1R)-1-(2H-tetrazol-5-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
—— (2S)-2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide —— C21H23FN4O
(2S)-2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
—— 2-[[5-(2-methylphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-N-(5-methyl-2-phenylpyrazol-3-yl)acetamide —— C21H19N5O2S
2-[[5-(2-methylphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]-N-(5-methyl-2-phenylpyrazol-3-yl)acetamide
—— (2R)-2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide —— C21H23FN4O
(2R)-2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
—— [2-[2-Cyanoethyl(methyl)amino]-2-oxoethyl] 1,3-diphenylpyrazole-4-carboxylate —— C22H20N4O3
[2-[2-Cyanoethyl(methyl)amino]-2-oxoethyl] 1,3-diphenylpyrazole-4-carboxylate
—— [2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 5-methyl-4-propylthiophene-2-carboxylate —— C22H25N3O3S
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 5-methyl-4-propylthiophene-2-carboxylate
—— 3,3-dimethyl-1-[(2R)-2-methyl-4-[2-[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]acetyl]piperazin-1-yl]butan-1-one —— C22H30N4O3
3,3-dimethyl-1-[(2R)-2-methyl-4-[2-[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]acetyl]piperazin-1-yl]butan-1-one
—— 4-[(4S)-4-(2-fluorophenyl)-6-oxo-3-phenyl-1,4-dihydropyrrolo[3,4-c]pyrazol-5-yl]benzoate —— C24H15FN3O3-
4-[(4S)-4-(2-fluorophenyl)-6-oxo-3-phenyl-1,4-dihydropyrrolo[3,4-c]pyrazol-5-yl]benzoate
—— 1-[(2S)-2-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one —— C22H23N3O3
1-[(2S)-2-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]-3-phenylpropan-1-one
—— 4-[(4S)-4-(4-fluorophenyl)-6-oxo-3-phenyl-1,4-dihydropyrrolo[3,4-c]pyrazol-5-yl]benzoate —— C24H15FN3O3-
4-[(4S)-4-(4-fluorophenyl)-6-oxo-3-phenyl-1,4-dihydropyrrolo[3,4-c]pyrazol-5-yl]benzoate
—— N'-[(2R)-butan-2-yl]-N-[2-(3-fluorophenyl)-5-methyl-4-phenylpyrazol-3-yl]butanediamide —— C24H27FN4O2
N'-[(2R)-butan-2-yl]-N-[2-(3-fluorophenyl)-5-methyl-4-phenylpyrazol-3-yl]butanediamide
—— 2-[[[(2S)-2-ethylhexanoyl]-(3-methoxypropyl)amino]methyl]-N-(3-methoxypropyl)-1,3-thiazole-4-carboxamide —— C21H37N3O4S
2-[[[(2S)-2-ethylhexanoyl]-(3-methoxypropyl)amino]methyl]-N-(3-methoxypropyl)-1,3-thiazole-4-carboxamide
—— [(2R)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]-(4-nitrophenyl)methanone —— C20H18N4O4
[(2R)-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]-(4-nitrophenyl)methanone
—— [2-(Cyclopentylamino)-2-oxoethyl] 1,3-diphenylpyrazole-4-carboxylate —— C23H23N3O3
[2-(Cyclopentylamino)-2-oxoethyl] 1,3-diphenylpyrazole-4-carboxylate
—— 3-cyclopentyl-1-[(2S)-2-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]propan-1-one —— C20H24FN3O2
3-cyclopentyl-1-[(2S)-2-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]propan-1-one
—— [2-[[(1R)-1-cyano-1-cyclopropylethyl]amino]-2-oxoethyl] 1,3-diphenylpyrazole-4-carboxylate —— C24H22N4O3
[2-[[(1R)-1-cyano-1-cyclopropylethyl]amino]-2-oxoethyl] 1,3-diphenylpyrazole-4-carboxylate
—— 2-(4-fluorophenyl)-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide —— C17H14FN7O
2-(4-fluorophenyl)-N-[(1S)-1-(2H-tetrazol-5-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
—— (2S)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-(3,4-difluorophenyl)pyrrolidine-1-carboxamide —— C19H15ClF2N4O2
(2S)-2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-(3,4-difluorophenyl)pyrrolidine-1-carboxamide
—— N-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-[[5-(3-methylphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide —— C22H21N5O2S
N-(3,5-dimethyl-1-phenylpyrazol-4-yl)-2-[[5-(3-methylphenyl)-1,3,4-oxadiazol-2-yl]sulfanyl]acetamide
—— (4R)-8-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid —— C21H25N3O4
(4R)-8-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
—— (2S)-2-(4-chloropyrazol-1-yl)-N-methyl-N-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]propanamide —— C14H19ClN4OS
(2S)-2-(4-chloropyrazol-1-yl)-N-methyl-N-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]propanamide
—— (2S)-2-(6-aminopyridin-3-yl)-2-[[1-(3-methoxyphenyl)pyrazol-4-yl]methyl-methylamino]acetic acid —— C19H21N5O3
(2S)-2-(6-aminopyridin-3-yl)-2-[[1-(3-methoxyphenyl)pyrazol-4-yl]methyl-methylamino]acetic acid
—— (4S)-8-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid —— C21H25N3O4
(4S)-8-[[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
—— (2R)-1-(2-methoxyacetyl)-N,4-dimethyl-N-[(1-phenylpyrazol-4-yl)methyl]piperazine-2-carboxamide —— C20H27N5O3
(2R)-1-(2-methoxyacetyl)-N,4-dimethyl-N-[(1-phenylpyrazol-4-yl)methyl]piperazine-2-carboxamide
—— (2R)-2-(4-chloropyrazol-1-yl)-N-methyl-N-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]propanamide —— C14H19ClN4OS
(2R)-2-(4-chloropyrazol-1-yl)-N-methyl-N-[(2-propan-2-yl-1,3-thiazol-4-yl)methyl]propanamide
—— (2S)-1-(2-methoxyacetyl)-N,4-dimethyl-N-[(1-phenylpyrazol-4-yl)methyl]piperazine-2-carboxamide —— C20H27N5O3
(2S)-1-(2-methoxyacetyl)-N,4-dimethyl-N-[(1-phenylpyrazol-4-yl)methyl]piperazine-2-carboxamide
—— [(2S)-1-(cyclopropylamino)-1-oxopropan-2-yl] 1-phenyl-3-thiophen-2-ylpyrazole-4-carboxylate —— C20H19N3O3S
[(2S)-1-(cyclopropylamino)-1-oxopropan-2-yl] 1-phenyl-3-thiophen-2-ylpyrazole-4-carboxylate
—— 2-(4-fluorophenyl)-N-methyl-N-[(1S)-1-pyridin-3-ylethyl]imidazo[1,2-a]pyridine-6-carboxamide —— C22H19FN4O
2-(4-fluorophenyl)-N-methyl-N-[(1S)-1-pyridin-3-ylethyl]imidazo[1,2-a]pyridine-6-carboxamide
—— 2-(3-chlorophenyl)-5-phenyl-N-(2-pyrrolidin-1-ium-1-ylethyl)pyrazole-3-carboxamide —— C22H24ClN4O+
2-(3-chlorophenyl)-5-phenyl-N-(2-pyrrolidin-1-ium-1-ylethyl)pyrazole-3-carboxamide
—— 2-(4-fluorophenyl)-N-methyl-N-[(1R)-1-pyridin-3-ylethyl]imidazo[1,2-a]pyridine-6-carboxamide —— C22H19FN4O
2-(4-fluorophenyl)-N-methyl-N-[(1R)-1-pyridin-3-ylethyl]imidazo[1,2-a]pyridine-6-carboxamide
—— 3-[(2Z)-2-[[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]hydrazinyl]benzoate —— C24H19N4O3-
3-[(2Z)-2-[[3-(4-methoxyphenyl)-1-phenylpyrazol-4-yl]methylidene]hydrazinyl]benzoate
—— [2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 4-ethoxy-3-methoxybenzoate —— C22H23N3O5
[2-[(5-Methyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] 4-ethoxy-3-methoxybenzoate
—— (2S)-2-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methylphenyl)pyrrolidine-1-carboxamide —— C20H19FN4O2
(2S)-2-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methylphenyl)pyrrolidine-1-carboxamide