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中文名称 英文名称 CAS号 化学式 结构式图片
—— [(2R)-3-methyl-1-oxo-1-[[(2R)-oxolan-2-yl]methylamino]butan-2-yl] 4,5-dichloro-1,2-thiazole-3-carboxylate —— C14H18Cl2N2O4S
[(2R)-3-methyl-1-oxo-1-[[(2R)-oxolan-2-yl]methylamino]butan-2-yl] 4,5-dichloro-1,2-thiazole-3-carboxylate
—— [(2S)-3-methyl-1-oxo-1-(2-phenylethylamino)butan-2-yl] 4,5-dichloro-1,2-thiazole-3-carboxylate —— C17H18Cl2N2O3S
[(2S)-3-methyl-1-oxo-1-(2-phenylethylamino)butan-2-yl] 4,5-dichloro-1,2-thiazole-3-carboxylate
—— (3R)-3-(furan-2-yl)-5-(4-methoxyphenyl)-2-phenyl-3,4-dihydropyrazole —— C20H18N2O2
(3R)-3-(furan-2-yl)-5-(4-methoxyphenyl)-2-phenyl-3,4-dihydropyrazole
—— N-[[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-[(2R)-1-methylpiperidin-2-yl]propanamide —— C18H23FN4O2
N-[[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-[(2R)-1-methylpiperidin-2-yl]propanamide
—— (7S)-2-(2,3-difluorophenyl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C20H17F2N3O2
(7S)-2-(2,3-difluorophenyl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— (7R)-2-(2,3-difluorophenyl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one —— C20H17F2N3O2
(7R)-2-(2,3-difluorophenyl)-7-(2-methoxyphenyl)-5,6,7,8-tetrahydro-1H-imidazo[4,5-c]azepin-4-one
—— N-[[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-[(2S)-1-methylpiperidin-2-yl]propanamide —— C18H23FN4O2
N-[[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-[(2S)-1-methylpiperidin-2-yl]propanamide
—— (2S)-2-[3-(1H-pyrazol-5-yl)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid —— C21H23N5O2
(2S)-2-[3-(1H-pyrazol-5-yl)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
—— 2-[1-[(1R)-1-(4,5-dimethyl-1,3-thiazol-2-yl)propyl]triazol-4-yl]benzoic acid —— C17H18N4O2S
2-[1-[(1R)-1-(4,5-dimethyl-1,3-thiazol-2-yl)propyl]triazol-4-yl]benzoic acid
—— (5S)-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C17H21N3O3
(5S)-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (2R)-2-[3-(1H-pyrazol-5-yl)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid —— C21H23N5O2
(2R)-2-[3-(1H-pyrazol-5-yl)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
—— (5R)-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol —— C17H21N3O3
(5R)-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
—— (2R)-1-amino-3-[2-(3-chloro-4-fluorophenyl)-1,2,4-triazol-3-yl]propan-2-ol —— C11H12ClFN4O
(2R)-1-amino-3-[2-(3-chloro-4-fluorophenyl)-1,2,4-triazol-3-yl]propan-2-ol
—— (2S)-2-[methyl(2-morpholin-4-ylethyl)amino]-2-[4-(1H-pyrazol-5-yl)phenyl]acetic acid —— C18H24N4O3
(2S)-2-[methyl(2-morpholin-4-ylethyl)amino]-2-[4-(1H-pyrazol-5-yl)phenyl]acetic acid
—— (4R)-6-amino-3-(4-ethoxyphenyl)-4-[(E)-1-(furan-2-yl)prop-1-en-2-yl]-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C22H20N4O3
(4R)-6-amino-3-(4-ethoxyphenyl)-4-[(E)-1-(furan-2-yl)prop-1-en-2-yl]-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— N-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-2-(1,2,4-triazol-1-yl)benzamide —— C20H20N4O3
N-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-2-(1,2,4-triazol-1-yl)benzamide
—— (4S)-6-amino-3-(4-ethoxyphenyl)-4-[(E)-1-(furan-2-yl)prop-1-en-2-yl]-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C22H20N4O3
(4S)-6-amino-3-(4-ethoxyphenyl)-4-[(E)-1-(furan-2-yl)prop-1-en-2-yl]-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— (3S)-3-(2-chlorophenyl)-2,5-diphenyl-3,4-dihydropyrazole —— C21H17ClN2
(3S)-3-(2-chlorophenyl)-2,5-diphenyl-3,4-dihydropyrazole
—— (2R)-2-[[4-(1,3-diphenylpyrazol-4-yl)triazol-1-yl]methyl]morpholine —— C22H22N6O
(2R)-2-[[4-(1,3-diphenylpyrazol-4-yl)triazol-1-yl]methyl]morpholine
—— N-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-4-(1H-pyrazol-5-yl)benzamide —— C18H21N5O
N-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-4-(1H-pyrazol-5-yl)benzamide
—— (2R)-2-(4-methoxy-2-pyrazol-1-ylphenyl)-2-[methyl(2-methylpropyl)amino]acetic acid —— C17H23N3O3
(2R)-2-(4-methoxy-2-pyrazol-1-ylphenyl)-2-[methyl(2-methylpropyl)amino]acetic acid
—— (2S)-2-[[4-(1,3-diphenylpyrazol-4-yl)triazol-1-yl]methyl]morpholine —— C22H22N6O
(2S)-2-[[4-(1,3-diphenylpyrazol-4-yl)triazol-1-yl]methyl]morpholine
—— 2-(4-fluorophenyl)-N-methyl-N-[[(2S)-oxan-2-yl]methyl]imidazo[1,2-a]pyridine-6-carboxamide —— C21H22FN3O2
2-(4-fluorophenyl)-N-methyl-N-[[(2S)-oxan-2-yl]methyl]imidazo[1,2-a]pyridine-6-carboxamide
—— N-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-4-(1H-pyrazol-5-yl)benzamide —— C18H21N5O
N-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-4-(1H-pyrazol-5-yl)benzamide
—— N-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-2-(1,2,4-triazol-1-yl)benzamide —— C20H20N4O3
N-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-2-(1,2,4-triazol-1-yl)benzamide
—— (2S)-1-amino-3-[2-(3-chloro-4-fluorophenyl)-1,2,4-triazol-3-yl]propan-2-ol —— C11H12ClFN4O
(2S)-1-amino-3-[2-(3-chloro-4-fluorophenyl)-1,2,4-triazol-3-yl]propan-2-ol
—— (2S)-2-(4-methoxy-2-pyrazol-1-ylphenyl)-2-[methyl(2-methylpropyl)amino]acetic acid —— C17H23N3O3
(2S)-2-(4-methoxy-2-pyrazol-1-ylphenyl)-2-[methyl(2-methylpropyl)amino]acetic acid
—— (2R)-2-[methyl(2-morpholin-4-ylethyl)amino]-2-[4-(1H-pyrazol-5-yl)phenyl]acetic acid —— C18H24N4O3
(2R)-2-[methyl(2-morpholin-4-ylethyl)amino]-2-[4-(1H-pyrazol-5-yl)phenyl]acetic acid
—— 2-(4-fluorophenyl)-N-methyl-N-[[(2R)-oxan-2-yl]methyl]imidazo[1,2-a]pyridine-6-carboxamide —— C21H22FN3O2
2-(4-fluorophenyl)-N-methyl-N-[[(2R)-oxan-2-yl]methyl]imidazo[1,2-a]pyridine-6-carboxamide
—— N-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-3-[(2S)-1-methylpiperidin-2-yl]propanamide —— C21H29FN4O
N-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-3-[(2S)-1-methylpiperidin-2-yl]propanamide
—— (2S)-2-(4-ethoxycarbonylpiperazin-1-yl)-2-[3-(1H-pyrazol-5-yl)phenyl]acetic acid —— C18H22N4O4
(2S)-2-(4-ethoxycarbonylpiperazin-1-yl)-2-[3-(1H-pyrazol-5-yl)phenyl]acetic acid
—— (3R)-1-(oxan-4-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-3-carboxamide —— C20H27N5O2
(3R)-1-(oxan-4-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-3-carboxamide
—— [(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(1-phenyltriazol-4-yl)methanone —— C18H22N4O3
[(5S)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(1-phenyltriazol-4-yl)methanone
—— N-[(2S)-2-(2-fluorophenyl)-2-pyrrolidin-1-ylethyl]-4-(1H-pyrazol-5-yl)benzamide —— C22H23FN4O
N-[(2S)-2-(2-fluorophenyl)-2-pyrrolidin-1-ylethyl]-4-(1H-pyrazol-5-yl)benzamide
—— N-[(1S)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-piperidin-1-ylbutanamide —— C13H23N5OS
N-[(1S)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-piperidin-1-ylbutanamide
—— (2R)-2-(4-ethoxycarbonylpiperazin-1-yl)-2-[3-(1H-pyrazol-5-yl)phenyl]acetic acid —— C18H22N4O4
(2R)-2-(4-ethoxycarbonylpiperazin-1-yl)-2-[3-(1H-pyrazol-5-yl)phenyl]acetic acid
—— N-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-3-[(2R)-1-methylpiperidin-2-yl]propanamide —— C21H29FN4O
N-[[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]methyl]-3-[(2R)-1-methylpiperidin-2-yl]propanamide
—— (3S)-1-(oxan-4-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-3-carboxamide —— C20H27N5O2
(3S)-1-(oxan-4-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-3-carboxamide
—— N-[(1R)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-piperidin-1-ylbutanamide —— C13H23N5OS
N-[(1R)-1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-piperidin-1-ylbutanamide
—— N-[[1-(3-fluorophenyl)pyrazol-4-yl]methyl]-3-[(2S)-1-methylpiperidin-2-yl]propanamide —— C19H25FN4O
N-[[1-(3-fluorophenyl)pyrazol-4-yl]methyl]-3-[(2S)-1-methylpiperidin-2-yl]propanamide
—— 5-[(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]-1-(4-methylsulfanylphenyl)-1,2,4-triazole —— C16H22N4OS
5-[(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]-1-(4-methylsulfanylphenyl)-1,2,4-triazole
—— (2S)-1-chloro-3-[3-[(4-chlorophenyl)methyl]-2-methyl-5-nitroimidazol-4-yl]sulfanylpropan-2-ol —— C14H15Cl2N3O3S
(2S)-1-chloro-3-[3-[(4-chlorophenyl)methyl]-2-methyl-5-nitroimidazol-4-yl]sulfanylpropan-2-ol
—— [(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(1-phenyltriazol-4-yl)methanone —— C18H22N4O3
[(5R)-5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl]-(1-phenyltriazol-4-yl)methanone
—— N-[[1-(3-fluorophenyl)pyrazol-4-yl]methyl]-3-[(2R)-1-methylpiperidin-2-yl]propanamide —— C19H25FN4O
N-[[1-(3-fluorophenyl)pyrazol-4-yl]methyl]-3-[(2R)-1-methylpiperidin-2-yl]propanamide
—— N-[(2R)-2-(2-fluorophenyl)-2-pyrrolidin-1-ylethyl]-4-(1H-pyrazol-5-yl)benzamide —— C22H23FN4O
N-[(2R)-2-(2-fluorophenyl)-2-pyrrolidin-1-ylethyl]-4-(1H-pyrazol-5-yl)benzamide
—— [(4R)-4-[(2,7-dimethyl-3-phenylpyrazolo[1,5-a]pyrimidine-6-carbonyl)amino]pentyl]-diethylazanium —— C24H34N5O+
[(4R)-4-[(2,7-dimethyl-3-phenylpyrazolo[1,5-a]pyrimidine-6-carbonyl)amino]pentyl]-diethylazanium
—— 1-[(3S)-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]heptan-1-one —— C20H26FN3O2
1-[(3S)-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]heptan-1-one
—— (2R)-N-(3,4-dimethylphenyl)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide —— C21H22N4O2
(2R)-N-(3,4-dimethylphenyl)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxamide
—— [(2R)-1-(tert-butylamino)-1-oxopropan-2-yl] 4,5-dichloro-1,2-thiazole-3-carboxylate —— C11H14Cl2N2O3S
[(2R)-1-(tert-butylamino)-1-oxopropan-2-yl] 4,5-dichloro-1,2-thiazole-3-carboxylate
—— cyclobutyl-[(3S)-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]methanone —— C21H27N3O2
cyclobutyl-[(3S)-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]methanone