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中文名称 英文名称 CAS号 化学式 结构式图片
—— (4S)-8-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid —— C20H23FN4O3
(4S)-8-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
—— 2-[1-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]triazol-4-yl]-1,3-thiazole —— C15H13N7S
2-[1-[(1R)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]triazol-4-yl]-1,3-thiazole
—— 3-[[5-(2-propoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanoate —— C14H16N3O3S-
3-[[5-(2-propoxyphenyl)-1H-1,2,4-triazol-3-yl]sulfanyl]propanoate
—— 4-tert-butyl-2-[[4-[(3R)-piperidin-3-yl]triazol-1-yl]methyl]-1,3-thiazole —— C15H23N5S
4-tert-butyl-2-[[4-[(3R)-piperidin-3-yl]triazol-1-yl]methyl]-1,3-thiazole
—— (4S)-8-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid —— C21H26N4O3
(4S)-8-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
—— 2-[1-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]triazol-4-yl]-1,3-thiazole —— C15H13N7S
2-[1-[(1S)-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]triazol-4-yl]-1,3-thiazole
—— N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-2-(4-ethyl-3,5-dimethylpyrazol-1-yl)-N-methylacetamide —— C17H26N4OS
N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-2-(4-ethyl-3,5-dimethylpyrazol-1-yl)-N-methylacetamide
—— N-[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-2-(4-ethyl-3,5-dimethylpyrazol-1-yl)-N-methylacetamide —— C17H26N4OS
N-[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-2-(4-ethyl-3,5-dimethylpyrazol-1-yl)-N-methylacetamide
—— 4-tert-butyl-2-[[4-[(3S)-piperidin-3-yl]triazol-1-yl]methyl]-1,3-thiazole —— C15H23N5S
4-tert-butyl-2-[[4-[(3S)-piperidin-3-yl]triazol-1-yl]methyl]-1,3-thiazole
—— [2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] pyridine-4-carboxylate —— C19H18N4O3
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] pyridine-4-carboxylate
—— (4S)-4-[2-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]-1-(2-methoxyethyl)pyrrolidin-2-one —— C15H16Cl2N4O2
(4S)-4-[2-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
—— 2-[3-(3-Chloro-4-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]ethyl-diethylazanium —— C17H22ClN6O+
2-[3-(3-Chloro-4-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]ethyl-diethylazanium
—— (4R)-4-[2-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]-1-(2-methoxyethyl)pyrrolidin-2-one —— C15H16Cl2N4O2
(4R)-4-[2-(2,4-dichlorophenyl)-1,2,4-triazol-3-yl]-1-(2-methoxyethyl)pyrrolidin-2-one
—— 3-amino-N-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-4-phenyl-1H-pyrazole-5-carboxamide —— C21H22N4O3
3-amino-N-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-4-phenyl-1H-pyrazole-5-carboxamide
—— N-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-3-(5-methyltetrazol-1-yl)benzamide —— C20H21N5O3
N-[[(3S)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-3-(5-methyltetrazol-1-yl)benzamide
—— (2R)-2-(furan-2-ylmethyl)-3-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]propan-1-ol —— C13H19N3O3
(2R)-2-(furan-2-ylmethyl)-3-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]propan-1-ol
—— (2R)-2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl-methylamino]-2-(4-pyrazol-1-ylphenyl)acetic acid —— C19H23N5O2
(2R)-2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl-methylamino]-2-(4-pyrazol-1-ylphenyl)acetic acid
—— N-[(2S)-1-imidazol-1-ylbutan-2-yl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide —— C21H21N5O
N-[(2S)-1-imidazol-1-ylbutan-2-yl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
—— [2-[(5-Tert-butyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] pyridine-2-carboxylate —— C21H22N4O3
[2-[(5-Tert-butyl-2-phenylpyrazol-3-yl)amino]-2-oxoethyl] pyridine-2-carboxylate
—— N-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-3-(5-methyltetrazol-1-yl)benzamide —— C20H21N5O3
N-[[(3R)-8-methoxy-3,4-dihydro-2H-chromen-3-yl]methyl]-3-(5-methyltetrazol-1-yl)benzamide
—— 3-(3,4-Dimethoxyphenyl)-6-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]triazolo[4,5-d]pyrimidin-7-one —— C20H24N6O4
3-(3,4-Dimethoxyphenyl)-6-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]triazolo[4,5-d]pyrimidin-7-one
—— N-(2,4-dimethylphenyl)-2-[3-(3,5-dimethylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide —— C22H22N6O2
N-(2,4-dimethylphenyl)-2-[3-(3,5-dimethylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide
—— N-(4-ethylphenyl)-2-[3-(3-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide —— C21H20N6O2
N-(4-ethylphenyl)-2-[3-(3-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide
—— Ethyl 2-[3-(3-chloro-4-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-2-methylpropanoate —— C17H18ClN5O3
Ethyl 2-[3-(3-chloro-4-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-2-methylpropanoate
—— Methyl 5-[[3-(3-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]methyl]furan-2-carboxylate —— C18H15N5O4
Methyl 5-[[3-(3-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]methyl]furan-2-carboxylate
—— 3-(3,4-Dimethoxyphenyl)-6-(2-pyrrolidin-1-ium-1-ylethyl)triazolo[4,5-d]pyrimidin-7-one —— C18H23N6O3+
3-(3,4-Dimethoxyphenyl)-6-(2-pyrrolidin-1-ium-1-ylethyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[(2-Chloro-6-fluorophenyl)methyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C18H13ClFN5O
6-[(2-Chloro-6-fluorophenyl)methyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— N-(4-chlorophenyl)-2-[3-(3,5-dimethylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide —— C20H17ClN6O2
N-(4-chlorophenyl)-2-[3-(3,5-dimethylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide
—— 3-(3-Chloro-4-methylphenyl)-6-[(4-nitrophenyl)methyl]triazolo[4,5-d]pyrimidin-7-one —— C18H13ClN6O3
3-(3-Chloro-4-methylphenyl)-6-[(4-nitrophenyl)methyl]triazolo[4,5-d]pyrimidin-7-one
—— N-cyclopentyl-2-[3-(3,5-dimethylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide —— C19H22N6O2
N-cyclopentyl-2-[3-(3,5-dimethylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide
—— (2S)-2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl-methylamino]-2-(4-pyrazol-1-ylphenyl)acetic acid —— C19H23N5O2
(2S)-2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl-methylamino]-2-(4-pyrazol-1-ylphenyl)acetic acid
—— 6-[(4-Methylphenyl)methyl]-3-[4-(trifluoromethoxy)phenyl]triazolo[4,5-d]pyrimidin-7-one —— C19H14F3N5O2
6-[(4-Methylphenyl)methyl]-3-[4-(trifluoromethoxy)phenyl]triazolo[4,5-d]pyrimidin-7-one
—— 3-(4-Bromophenyl)-6-(2-oxo-2-pyrrolidin-1-ylethyl)triazolo[4,5-d]pyrimidin-7-one —— C16H15BrN6O2
3-(4-Bromophenyl)-6-(2-oxo-2-pyrrolidin-1-ylethyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[2-(Azepan-1-yl)-2-oxoethyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C20H24N6O2
6-[2-(Azepan-1-yl)-2-oxoethyl]-3-(3,5-dimethylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 6-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one —— C19H22N6O3
6-[2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]-3-(3-methylphenyl)triazolo[4,5-d]pyrimidin-7-one
—— 2-[3-(3-chloro-4-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-propylacetamide —— C16H17ClN6O2
2-[3-(3-chloro-4-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-propylacetamide
—— 2-[3-(3,5-dimethylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-(4-methoxyphenyl)acetamide —— C21H20N6O3
2-[3-(3,5-dimethylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-(4-methoxyphenyl)acetamide
—— N,N-dimethyl-2-[2-[(3R)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]imidazol-1-yl]ethanamine —— C20H26N6O
N,N-dimethyl-2-[2-[(3R)-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]imidazol-1-yl]ethanamine
—— 6-[(3-Chlorophenyl)methyl]-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one —— C17H10ClF2N5O
6-[(3-Chlorophenyl)methyl]-3-(2,4-difluorophenyl)triazolo[4,5-d]pyrimidin-7-one
—— 2-[3-(4-chlorophenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-(3-methylphenyl)acetamide —— C19H15ClN6O2
2-[3-(4-chlorophenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-(3-methylphenyl)acetamide
—— 2-[3-(4-chlorophenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-(4-methyl-1,3-thiazol-2-yl)acetamide —— C16H12ClN7O2S
2-[3-(4-chlorophenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-(4-methyl-1,3-thiazol-2-yl)acetamide
—— 2-[3-(3-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-phenylacetamide —— C19H16N6O2
2-[3-(3-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-phenylacetamide
—— 3-(3-Chloro-4-methylphenyl)-6-[(2,5-dimethylphenyl)methyl]triazolo[4,5-d]pyrimidin-7-one —— C20H18ClN5O
3-(3-Chloro-4-methylphenyl)-6-[(2,5-dimethylphenyl)methyl]triazolo[4,5-d]pyrimidin-7-one
—— 2-[3-(3-fluorophenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-propylacetamide —— C15H15FN6O2
2-[3-(3-fluorophenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-propylacetamide
—— (4R)-8-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid —— C21H26N4O3
(4R)-8-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
—— 3-(3,5-Dimethylphenyl)-6-(2-piperidin-1-ium-1-ylethyl)triazolo[4,5-d]pyrimidin-7-one —— C19H25N6O+
3-(3,5-Dimethylphenyl)-6-(2-piperidin-1-ium-1-ylethyl)triazolo[4,5-d]pyrimidin-7-one
—— 3-(3-Fluorophenyl)-6-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]triazolo[4,5-d]pyrimidin-7-one —— C18H19FN6O2
3-(3-Fluorophenyl)-6-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]triazolo[4,5-d]pyrimidin-7-one
—— 2-[3-(3,5-dimethylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-(4-ethylphenyl)acetamide —— C22H22N6O2
2-[3-(3,5-dimethylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]-N-(4-ethylphenyl)acetamide
—— N-(3,5-dimethylphenyl)-2-[3-(3-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide —— C21H20N6O2
N-(3,5-dimethylphenyl)-2-[3-(3-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide
—— N-(2-methylphenyl)-2-[3-(3-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide —— C20H18N6O2
N-(2-methylphenyl)-2-[3-(3-methylphenyl)-7-oxotriazolo[4,5-d]pyrimidin-6-yl]acetamide