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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(4-fluorophenyl)-N-[(2R)-4-pyrazol-1-ylbutan-2-yl]imidazo[1,2-a]pyridine-6-carboxamide —— C21H20FN5O
2-(4-fluorophenyl)-N-[(2R)-4-pyrazol-1-ylbutan-2-yl]imidazo[1,2-a]pyridine-6-carboxamide
—— (3S)-3-(1H-imidazol-5-ylmethyl)-4-[4-(1H-pyrazol-5-yl)benzoyl]piperazin-2-one —— C18H18N6O2
(3S)-3-(1H-imidazol-5-ylmethyl)-4-[4-(1H-pyrazol-5-yl)benzoyl]piperazin-2-one
—— (3R)-1-[4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-3,5,5-trimethylhexan-1-one —— C23H33N3O3
(3R)-1-[4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-3,5,5-trimethylhexan-1-one
—— (3S)-1-(furan-2-ylmethyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxamide —— C21H24N4O2
(3S)-1-(furan-2-ylmethyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxamide
—— 3-[[(3R)-1-(4-pyrazol-1-ylbenzoyl)pyrrolidin-3-yl]methyl]benzoic acid —— C22H21N3O3
3-[[(3R)-1-(4-pyrazol-1-ylbenzoyl)pyrrolidin-3-yl]methyl]benzoic acid
—— (3S)-1-[4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-3,5,5-trimethylhexan-1-one —— C23H33N3O3
(3S)-1-[4-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl]-3,5,5-trimethylhexan-1-one
—— (3R)-1-(furan-2-ylmethyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxamide —— C21H24N4O2
(3R)-1-(furan-2-ylmethyl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxamide
—— N-[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-2-(3-methoxyphenyl)sulfanyl-N-methylacetamide —— C17H22N2O2S2
N-[(1R)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-2-(3-methoxyphenyl)sulfanyl-N-methylacetamide
—— (3R)-N-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide —— C18H22N4O2S
(3R)-N-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
—— 3-[[(3S)-1-(4-pyrazol-1-ylbenzoyl)pyrrolidin-3-yl]methyl]benzoic acid —— C22H21N3O3
3-[[(3S)-1-(4-pyrazol-1-ylbenzoyl)pyrrolidin-3-yl]methyl]benzoic acid
—— (2S)-2-[[4-ethyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3-thiazol-2-yl)propanamide —— C16H16FN5OS2
(2S)-2-[[4-ethyl-5-(2-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(1,3-thiazol-2-yl)propanamide
—— (2R)-N-[5-(1,3-benzoxazol-2-yl)-2-methylphenyl]oxolane-2-carboxamide —— C19H18N2O3
(2R)-N-[5-(1,3-benzoxazol-2-yl)-2-methylphenyl]oxolane-2-carboxamide
—— (3R)-3-[1-[[2-(1,2,4-triazol-1-yl)phenyl]methyl]triazol-4-yl]piperidine —— C16H19N7
(3R)-3-[1-[[2-(1,2,4-triazol-1-yl)phenyl]methyl]triazol-4-yl]piperidine
—— 5-cyclobutyl-N-[(1R)-1-(cyclohexen-1-yl)ethyl]-1,3,4-oxadiazol-2-amine —— C14H21N3O
5-cyclobutyl-N-[(1R)-1-(cyclohexen-1-yl)ethyl]-1,3,4-oxadiazol-2-amine
—— (3S)-N-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide —— C18H22N4O2S
(3S)-N-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
—— 4-[3-(3-ethoxy-4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide —— C20H27N3O5
4-[3-(3-ethoxy-4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[[(2R)-oxolan-2-yl]methyl]butanamide
—— N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-2-(3-methoxyphenyl)sulfanyl-N-methylacetamide —— C17H22N2O2S2
N-[(1S)-1-(2,5-dimethyl-1,3-thiazol-4-yl)ethyl]-2-(3-methoxyphenyl)sulfanyl-N-methylacetamide
—— (3S)-3-[1-[[2-(1,2,4-triazol-1-yl)phenyl]methyl]triazol-4-yl]piperidine —— C16H19N7
(3S)-3-[1-[[2-(1,2,4-triazol-1-yl)phenyl]methyl]triazol-4-yl]piperidine
—— (2R)-N-cyclopropyl-2-(dimethylamino)-2-(3-fluorophenyl)-N-[(1-phenylpyrazol-4-yl)methyl]acetamide —— C23H25FN4O
(2R)-N-cyclopropyl-2-(dimethylamino)-2-(3-fluorophenyl)-N-[(1-phenylpyrazol-4-yl)methyl]acetamide
—— 1,3-Benzodioxol-5-ylmethyl-[2-(1-phenyltetrazol-5-yl)sulfanylethyl]azanium —— C17H18N5O2S+
1,3-Benzodioxol-5-ylmethyl-[2-(1-phenyltetrazol-5-yl)sulfanylethyl]azanium
—— (2S)-2-(4-chloro-3-methylphenoxy)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide —— C19H18ClN3O3
(2S)-2-(4-chloro-3-methylphenoxy)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
—— (3R)-1-cyclopentyl-N-[(1-phenyltetrazol-5-yl)methyl]piperidine-3-carboxamide —— C19H26N6O
(3R)-1-cyclopentyl-N-[(1-phenyltetrazol-5-yl)methyl]piperidine-3-carboxamide
—— (3S)-1-cyclopentyl-N-[(1-phenyltetrazol-5-yl)methyl]piperidine-3-carboxamide —— C19H26N6O
(3S)-1-cyclopentyl-N-[(1-phenyltetrazol-5-yl)methyl]piperidine-3-carboxamide
—— (2S)-N-cyclopropyl-2-(dimethylamino)-2-(3-fluorophenyl)-N-[(1-phenylpyrazol-4-yl)methyl]acetamide —— C23H25FN4O
(2S)-N-cyclopropyl-2-(dimethylamino)-2-(3-fluorophenyl)-N-[(1-phenylpyrazol-4-yl)methyl]acetamide
—— (2S)-N-[[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-phenoxypropanamide —— C19H19N3O4
(2S)-N-[[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-phenoxypropanamide
—— (2S)-N-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-phenoxypropanamide —— C18H16ClN3O3
(2S)-N-[[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-phenoxypropanamide
—— 5-cyclobutyl-N-[(1S)-1-(cyclohexen-1-yl)ethyl]-1,3,4-oxadiazol-2-amine —— C14H21N3O
5-cyclobutyl-N-[(1S)-1-(cyclohexen-1-yl)ethyl]-1,3,4-oxadiazol-2-amine
—— 5-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-[(E)-2-thiophen-2-ylethenyl]-1,3-oxazole-4-carbonitrile —— C16H17N3O2S
5-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-[(E)-2-thiophen-2-ylethenyl]-1,3-oxazole-4-carbonitrile
—— (3R)-5-oxo-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide —— C21H21N5O2
(3R)-5-oxo-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
—— (2S)-2-[3-(hydroxymethyl)phenyl]-2-[methyl-[(4-pyrazol-1-ylphenyl)methyl]amino]acetic acid —— C20H21N3O3
(2S)-2-[3-(hydroxymethyl)phenyl]-2-[methyl-[(4-pyrazol-1-ylphenyl)methyl]amino]acetic acid
—— (2S)-2-[methyl(oxan-4-ylmethyl)amino]-2-(4-methyl-2-pyrazol-1-ylphenyl)acetic acid —— C19H25N3O3
(2S)-2-[methyl(oxan-4-ylmethyl)amino]-2-(4-methyl-2-pyrazol-1-ylphenyl)acetic acid
—— (3S)-5-oxo-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide —— C21H21N5O2
(3S)-5-oxo-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
—— (2R)-2-[methyl(oxan-4-ylmethyl)amino]-2-(4-methyl-2-pyrazol-1-ylphenyl)acetic acid —— C19H25N3O3
(2R)-2-[methyl(oxan-4-ylmethyl)amino]-2-(4-methyl-2-pyrazol-1-ylphenyl)acetic acid
—— (2R)-1-[5-(2-chlorophenyl)-3-propan-2-yl-1,2,4-triazol-1-yl]butan-2-ol —— C15H20ClN3O
(2R)-1-[5-(2-chlorophenyl)-3-propan-2-yl-1,2,4-triazol-1-yl]butan-2-ol
—— (2S)-1-[5-(2-chlorophenyl)-3-propan-2-yl-1,2,4-triazol-1-yl]butan-2-ol —— C15H20ClN3O
(2S)-1-[5-(2-chlorophenyl)-3-propan-2-yl-1,2,4-triazol-1-yl]butan-2-ol
—— (3S)-N-[3-(4,5-dimethyl-1,3-thiazol-2-yl)propyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide —— C15H23N3O2S
(3S)-N-[3-(4,5-dimethyl-1,3-thiazol-2-yl)propyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
—— (4S)-1-ethyl-4-(3-phenyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl)pyrrolidin-2-one —— C19H23N5O2
(4S)-1-ethyl-4-(3-phenyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl)pyrrolidin-2-one
—— (3R)-1-(furan-2-ylmethyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine-3-carboxamide —— C21H23N3O3
(3R)-1-(furan-2-ylmethyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine-3-carboxamide
—— (4R)-1-ethyl-4-(3-phenyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl)pyrrolidin-2-one —— C19H23N5O2
(4R)-1-ethyl-4-(3-phenyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl)pyrrolidin-2-one
—— (3S)-1-(furan-2-ylmethyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine-3-carboxamide —— C21H23N3O3
(3S)-1-(furan-2-ylmethyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine-3-carboxamide
—— (3R)-N-[3-(4,5-dimethyl-1,3-thiazol-2-yl)propyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide —— C15H23N3O2S
(3R)-N-[3-(4,5-dimethyl-1,3-thiazol-2-yl)propyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
—— (6S)-5-[4-(3,5-dimethylpyrazol-1-yl)benzoyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C19H19N5O3
(6S)-5-[4-(3,5-dimethylpyrazol-1-yl)benzoyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (2S)-2-(4-pyrazol-1-ylphenyl)-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]acetic acid —— C20H22N4O2S
(2S)-2-(4-pyrazol-1-ylphenyl)-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]acetic acid
—— (6R)-5-[4-(3,5-dimethylpyrazol-1-yl)benzoyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid —— C19H19N5O3
(6R)-5-[4-(3,5-dimethylpyrazol-1-yl)benzoyl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridine-6-carboxylic acid
—— (2R)-2-(4-pyrazol-1-ylphenyl)-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]acetic acid —— C20H22N4O2S
(2R)-2-(4-pyrazol-1-ylphenyl)-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]acetic acid
—— (2R)-2-[3-(hydroxymethyl)phenyl]-2-[methyl-[(4-pyrazol-1-ylphenyl)methyl]amino]acetic acid —— C20H21N3O3
(2R)-2-[3-(hydroxymethyl)phenyl]-2-[methyl-[(4-pyrazol-1-ylphenyl)methyl]amino]acetic acid
—— (2R)-N-[[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-phenoxypropanamide —— C19H19N3O3
(2R)-N-[[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-phenoxypropanamide
—— 5-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-[(E)-2-(3-methoxyphenyl)ethenyl]-1,3-oxazole-4-carbonitrile —— C19H21N3O3
5-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-[(E)-2-(3-methoxyphenyl)ethenyl]-1,3-oxazole-4-carbonitrile
—— (2R)-2-[4-[2-(2-phenylethynyl)phenyl]triazol-1-yl]propanoic acid —— C19H15N3O2
(2R)-2-[4-[2-(2-phenylethynyl)phenyl]triazol-1-yl]propanoic acid
—— 5-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-[(E)-2-(3-methoxyphenyl)ethenyl]-1,3-oxazole-4-carbonitrile —— C19H21N3O3
5-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-2-[(E)-2-(3-methoxyphenyl)ethenyl]-1,3-oxazole-4-carbonitrile