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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N3O3
(6R)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(cyclohexanecarbonyl)-2-[(2R)-1-(cyclopropanecarbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N4O3
6-(cyclohexanecarbonyl)-2-[(2R)-1-(cyclopropanecarbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-1-(cyclopentanecarbonyl)-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N3O2
(6S)-1-(cyclopentanecarbonyl)-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-chloro-N-[(Z)-(3,5-ditert-butylphenyl)methylideneamino]-4-phenylquinazolin-2-amine —— C29H31ClN4
6-chloro-N-[(Z)-(3,5-ditert-butylphenyl)methylideneamino]-4-phenylquinazolin-2-amine
—— (6R)-1-(6-oxo-1H-pyridazine-3-carbonyl)-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H25N5O3
(6R)-1-(6-oxo-1H-pyridazine-3-carbonyl)-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(cyclopentanecarbonyl)-2-[(2R)-1-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H34N4O3
6-(cyclopentanecarbonyl)-2-[(2R)-1-[2-[(1R)-cyclopent-2-en-1-yl]acetyl]piperidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N3O3
(6S)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N3O3
(6R)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-[(2R)-oxolane-2-carbonyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C26H29FN2O3
(6S)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-[(2R)-oxolane-2-carbonyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— (6Z)-2-bromo-4-chloro-3,5-dimethyl-6-[[3-(4-methyl-1,3-benzoxazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C23H18BrClN2O2
(6Z)-2-bromo-4-chloro-3,5-dimethyl-6-[[3-(4-methyl-1,3-benzoxazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— (6S)-1-(3-fluorobenzoyl)-4-prop-2-enyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H26FN3O2
(6S)-1-(3-fluorobenzoyl)-4-prop-2-enyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-[(2S)-5-oxopyrrolidine-2-carbonyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C26H28FN3O3
(6R)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-[(2S)-5-oxopyrrolidine-2-carbonyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— (6S)-6-[[2-(3-fluorophenyl)phenyl]methyl]-4-prop-2-enyl-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one —— C27H26FN3O2
(6S)-6-[[2-(3-fluorophenyl)phenyl]methyl]-4-prop-2-enyl-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
—— (6S)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N3O3
(6S)-1-[(2S)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-benzoyl-4-prop-2-enyl-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H27N3O2
(6R)-1-benzoyl-4-prop-2-enyl-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6Z)-6-[[1-[(2-chlorophenyl)methyl]indol-3-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H23ClN6O3S
(6Z)-6-[[1-[(2-chlorophenyl)methyl]indol-3-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6R)-4-prop-2-enyl-1-(pyridine-4-carbonyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H26N4O2
(6R)-4-prop-2-enyl-1-(pyridine-4-carbonyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-methyl-2-[(2R)-1-[(E)-2-methyl-3-phenylprop-2-enyl]piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C23H30N4
6-methyl-2-[(2R)-1-[(E)-2-methyl-3-phenylprop-2-enyl]piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6Z)-6-[(4-ethylphenyl)methylidene]-5-imino-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H23N5O2S
(6Z)-6-[(4-ethylphenyl)methylidene]-5-imino-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(cyclohexylmethyl)-2-[(2R)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H34N4O3
6-(cyclohexylmethyl)-2-[(2R)-1-[(3R)-oxolane-3-carbonyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-1-(2-phenylacetyl)-4-prop-2-enyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C28H29N3O2
(6S)-1-(2-phenylacetyl)-4-prop-2-enyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-prop-2-enyl-1-(pyridin-4-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H28N4O
(6S)-4-prop-2-enyl-1-(pyridin-4-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(3-fluorobenzoyl)-4-prop-2-enyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H26FN3O2
(6S)-1-(3-fluorobenzoyl)-4-prop-2-enyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6E)-4-chloro-6-[[4-[4-[[(E)-(3-chloro-2,4-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]phenyl]anilino]methylidene]-2,5-dimethylcyclohexa-2,4-dien-1-one —— C30H26Cl2N2O2
(6E)-4-chloro-6-[[4-[4-[[(E)-(3-chloro-2,4-dimethyl-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]phenyl]anilino]methylidene]-2,5-dimethylcyclohexa-2,4-dien-1-one
—— (6R)-1-(cyclopropylmethyl)-4-prop-2-enyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H29N3O
(6R)-1-(cyclopropylmethyl)-4-prop-2-enyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-prop-2-enyl-1-(pyridine-4-carbonyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H26N4O2
(6R)-4-prop-2-enyl-1-(pyridine-4-carbonyl)-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-bromo-3-(2-methoxyphenyl)-2-[(E)-2-(3-nitrophenyl)ethenyl]quinazolin-4(3H)-one —— C23H16BrN3O4
6-bromo-3-(2-methoxyphenyl)-2-[(E)-2-(3-nitrophenyl)ethenyl]quinazolin-4(3H)-one
—— (6S)-1-(2-phenylacetyl)-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C28H29N3O2
(6S)-1-(2-phenylacetyl)-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(Cyclopentanecarbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H34N4O3
6-(Cyclopentanecarbonyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-4-prop-2-enyl-1-(2-pyridin-3-ylacetyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H28N4O2
(6S)-4-prop-2-enyl-1-(2-pyridin-3-ylacetyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(1H-imidazol-2-ylmethyl)-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H26N4OS
(6R)-1-(1H-imidazol-2-ylmethyl)-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-methyl-2-[(2S)-1-[(E)-2-methyl-3-phenylprop-2-enyl]piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C23H30N4
6-methyl-2-[(2S)-1-[(E)-2-methyl-3-phenylprop-2-enyl]piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[(2S)-oxolane-2-carbonyl]-2-pyrrolidin-1-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C16H22N4O3
6-[(2S)-oxolane-2-carbonyl]-2-pyrrolidin-1-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-4-prop-2-enyl-1-(pyridin-2-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H28N4O
(6R)-4-prop-2-enyl-1-(pyridin-2-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6Z)-6-(4-{2-[4-(butan-2-yl)phenoxy]ethoxy}-3-methoxybenzylidene)-5-imino-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H25F3N4O4S
(6Z)-6-(4-{2-[4-(butan-2-yl)phenoxy]ethoxy}-3-methoxybenzylidene)-5-imino-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z,21Z)-1,16-diazatetracyclo[27.3.1.112,16.014,30]tetratriaconta-6,21-diene —— C32H56N2
(6Z,21Z)-1,16-diazatetracyclo[27.3.1.112,16.014,30]tetratriaconta-6,21-diene
—— (6S)-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-4-prop-2-enyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O3
(6S)-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-4-prop-2-enyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one —— C27H27N3O2
(6R)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
—— (6R)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C26H28FN3O3
(6R)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-[(2R)-5-oxopyrrolidine-2-carbonyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— (6S)-1-[(2R)-oxolane-2-carbonyl]-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C26H30N2O3
(6S)-1-[(2R)-oxolane-2-carbonyl]-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— (6R)-1-(3-fluorobenzoyl)-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H26FN3O2
(6R)-1-(3-fluorobenzoyl)-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(2R)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N2O3S
(6R)-1-[(2R)-oxolane-2-carbonyl]-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(6-oxo-1H-pyridazine-3-carbonyl)-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H25N5O3
(6S)-1-(6-oxo-1H-pyridazine-3-carbonyl)-4-prop-2-enyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(cyclopentanecarbonyl)-2-[(2R)-1-[(2S)-oxolane-2-carbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H32N4O4
6-(cyclopentanecarbonyl)-2-[(2R)-1-[(2S)-oxolane-2-carbonyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-(3-fluorobenzoyl)-4-prop-2-enyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H26FN3O2
(6R)-1-(3-fluorobenzoyl)-4-prop-2-enyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1-(3-pyrazol-1-ylpropanoyl)-1,4-diazepan-5-one —— C27H30N4O2
(6R)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1-(3-pyrazol-1-ylpropanoyl)-1,4-diazepan-5-one
—— 6-chloro-4-phenyl-2-[(2Z)-2-(quinoxalin-6-ylmethylidene)hydrazinyl]quinazoline —— C23H15ClN6
6-chloro-4-phenyl-2-[(2Z)-2-(quinoxalin-6-ylmethylidene)hydrazinyl]quinazoline
—— (6R)-6-[(3-phenylphenyl)methyl]-4-prop-2-enyl-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one —— C27H27N3O2
(6R)-6-[(3-phenylphenyl)methyl]-4-prop-2-enyl-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
—— 6-cyclohexyl-2-[(2S)-1-(oxane-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H36N4O3
6-cyclohexyl-2-[(2S)-1-(oxane-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6H-furo[2,3-b]pyrrol-2-ylmethanamine —— C7H8N2O
6H-furo[2,3-b]pyrrol-2-ylmethanamine