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—— 6-[7-methyl-5-[(3S)-oxolan-3-yl]imidazo[5,1-f][1,2,4]triazin-4-yl]-7,8-dihydro-5H-1,6-naphthyridine —— C18H20N6O
6-[7-methyl-5-[(3S)-oxolan-3-yl]imidazo[5,1-f][1,2,4]triazin-4-yl]-7,8-dihydro-5H-1,6-naphthyridine
—— 6-methoxy-2-[7-methyl-5-[(3S)-oxolan-3-yl]imidazo[5,1-f][1,2,4]triazin-4-yl]-3,4-dihydro-1H-isoquinoline —— C20H23N5O2
6-methoxy-2-[7-methyl-5-[(3S)-oxolan-3-yl]imidazo[5,1-f][1,2,4]triazin-4-yl]-3,4-dihydro-1H-isoquinoline
—— 6-[5-(2-fluorophenyl)-7-methylimidazo[5,1-f][1,2,4]triazin-4-yl]-2-methoxy-7,8-dihydro-5H-1,6-naphthyridine —— C21H19FN6O
6-[5-(2-fluorophenyl)-7-methylimidazo[5,1-f][1,2,4]triazin-4-yl]-2-methoxy-7,8-dihydro-5H-1,6-naphthyridine
—— (6Z)-2-(2-chlorophenyl)-6-{[1-(2-chlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H17Cl2N5OS
(6Z)-2-(2-chlorophenyl)-6-{[1-(2-chlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-2-butyl-6-[[1-(4-fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H22FN5OS
(6Z)-2-butyl-6-[[1-(4-fluorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[(2,4-dichlorophenyl)methylidene]-3-(3,4-dihydroxyphenyl)-[1,3]thiazolo[2,3-b][1,3]thiazol-4-ium-5-one —— C18H10Cl2NO3S2+
(6E)-6-[(2,4-dichlorophenyl)methylidene]-3-(3,4-dihydroxyphenyl)-[1,3]thiazolo[2,3-b][1,3]thiazol-4-ium-5-one
—— 6-chloro-5-(2-(6-(4-cyclopropyl-2-fluorophenyl)-3,4,8,9-tetrahydro-1H-pyrido[4’,3’:4,5]imidazo[2,1-c][1,4]oxazin-7(6H)-yl)-2-oxoethoxy)-N,N-dimethylpicolinamide —— C28H29ClFN5O4
6-chloro-5-(2-(6-(4-cyclopropyl-2-fluorophenyl)-3,4,8,9-tetrahydro-1H-pyrido[4’,3’:4,5]imidazo[2,1-c][1,4]oxazin-7(6H)-yl)-2-oxoethoxy)-N,N-dimethylpicolinamide
—— 6-[(2R)-2-(3-fluorophenyl)pyrrolidin-1-yl]-3-pyridin-2-ylimidazo[1,2-b]pyridazin-1-ium —— C21H19FN5+
6-[(2R)-2-(3-fluorophenyl)pyrrolidin-1-yl]-3-pyridin-2-ylimidazo[1,2-b]pyridazin-1-ium
—— 6-methoxy-2-{7-methyl-5-[(3S)-tetrahydrofuran-3-yl]imidazo[5,1-f][1,2,4]triazin-4-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine —— C19H22N6O2
6-methoxy-2-{7-methyl-5-[(3S)-tetrahydrofuran-3-yl]imidazo[5,1-f][1,2,4]triazin-4-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
—— 6,7-dimethoxy-2-[7-methyl-5-(2-methylphenyl)imidazo[5,1-f][1,2,4]triazin-4-yl]-1,2,3,4-tetrahydroisoquinoline —— C24H25N5O2
6,7-dimethoxy-2-[7-methyl-5-(2-methylphenyl)imidazo[5,1-f][1,2,4]triazin-4-yl]-1,2,3,4-tetrahydroisoquinoline
—— 6-methoxy-2-{7-methyl-5-[(3R)-tetrahydrofuran-3-yl]imidazo[5,1-f][1,2,4]triazin-4-yl}-1,2,3,4-tetrahydroisoquinoline —— C20H23N5O2
6-methoxy-2-{7-methyl-5-[(3R)-tetrahydrofuran-3-yl]imidazo[5,1-f][1,2,4]triazin-4-yl}-1,2,3,4-tetrahydroisoquinoline
—— 6-[5-(2-fluorophenyl)-7-methylimidazo[5,1-f][1,2,4]triazin-4-yl]-N,N-dimethyl-7,8-dihydro-5H-1,6-naphthyridin-2-amine —— C22H22FN7
6-[5-(2-fluorophenyl)-7-methylimidazo[5,1-f][1,2,4]triazin-4-yl]-N,N-dimethyl-7,8-dihydro-5H-1,6-naphthyridin-2-amine
—— 6-Ethyl-4,5,6,7-tetrahydro-[1,3]thiazolo[5,4-c]pyridin-2-amine —— C8H13N3S
6-Ethyl-4,5,6,7-tetrahydro-[1,3]thiazolo[5,4-c]pyridin-2-amine
—— (6Z)-4-amino-1-diazenyl-3-(4-nitrophenyl)-5-oxo-6-(phenylhydrazinylidene)naphthalene-2,7-disulfonic acid —— C22H16N6O9S2
(6Z)-4-amino-1-diazenyl-3-(4-nitrophenyl)-5-oxo-6-(phenylhydrazinylidene)naphthalene-2,7-disulfonic acid
—— (6Z)-6-[5-(2-methoxyphenyl)-1H-pyrimidin-6-ylidene]-3-[(2-methylphenyl)methoxy]cyclohexa-2,4-dien-1-one —— C25H22N2O3
(6Z)-6-[5-(2-methoxyphenyl)-1H-pyrimidin-6-ylidene]-3-[(2-methylphenyl)methoxy]cyclohexa-2,4-dien-1-one
—— (6E)-6-{[2,5-dimethyl-1-(naphthalen-2-yl)-1H-pyrrol-3-yl]methylidene}-2-heptyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H31N5OS
(6E)-6-{[2,5-dimethyl-1-(naphthalen-2-yl)-1H-pyrrol-3-yl]methylidene}-2-heptyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-iodo-3-(2-methoxyphenyl)-2-[(E)-2-(pyridin-3-yl)ethenyl]quinazolin-4(3H)-one —— C22H16IN3O2
6-iodo-3-(2-methoxyphenyl)-2-[(E)-2-(pyridin-3-yl)ethenyl]quinazolin-4(3H)-one
—— 6,8,10-Triazatricyclo[5.4.0.02,4]undeca-1,5,7,9-tetraene —— C8H7N3
6,8,10-Triazatricyclo[5.4.0.02,4]undeca-1,5,7,9-tetraene
—— 6-chloro-N-[(Z)-(2-ethoxyphenyl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide —— C18H17ClN4O2
6-chloro-N-[(Z)-(2-ethoxyphenyl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— 6-Methoxy-1-(piperidin-3-yl)-1h-benzo[d]imidazole hydrochloride —— C13H18ClN3O
6-Methoxy-1-(piperidin-3-yl)-1h-benzo[d]imidazole hydrochloride
—— (6E)-2,4-ditert-butyl-6-[[[4-[[(E)-(3,5-ditert-butyl-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]-2,2,3,3-tetramethylbutyl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C38H60N2O2
(6E)-2,4-ditert-butyl-6-[[[4-[[(E)-(3,5-ditert-butyl-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]-2,2,3,3-tetramethylbutyl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-2-benzyl-6-[[1-(2,4-dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H25N5OS
(6Z)-2-benzyl-6-[[1-(2,4-dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[2-(6-methoxypyridin-3-yl)-1,4,6,7-tetrahydro-5H-imidazo[4,5-c]pyridin-5-yl]-N-methylpyridine-2-carboxamide —— C19H20N6O2
6-[2-(6-methoxypyridin-3-yl)-1,4,6,7-tetrahydro-5H-imidazo[4,5-c]pyridin-5-yl]-N-methylpyridine-2-carboxamide
—— 6-(3-aminocyclobutyl)-N~4~-[(1-morpholin-4-ylcycloheptyl)methyl]pyrimidine-2,4-diamine —— C20H34N6O
6-(3-aminocyclobutyl)-N~4~-[(1-morpholin-4-ylcycloheptyl)methyl]pyrimidine-2,4-diamine
—— (6Z)-6-{3-chloro-4-[(4-methylbenzyl)oxy]benzylidene}-5-imino-2-[2-oxo-2-(piperidin-1-yl)ethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H26ClN5O3S
(6Z)-6-{3-chloro-4-[(4-methylbenzyl)oxy]benzylidene}-5-imino-2-[2-oxo-2-(piperidin-1-yl)ethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(4-ethyl-3,3-dimethylpiperazin-1-yl)carbonyl]-2-methyl-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one —— C16H27N5O2
6-[(4-ethyl-3,3-dimethylpiperazin-1-yl)carbonyl]-2-methyl-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one
—— (6E)-2-bromo-4-chloro-6-[[[2-(2,3-dichlorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-3,5-dimethylcyclohexa-2,4-dien-1-one —— C22H14BrCl3N2O2
(6E)-2-bromo-4-chloro-6-[[[2-(2,3-dichlorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-3,5-dimethylcyclohexa-2,4-dien-1-one
—— 6-fluoro-2-methyl-N-{trans-3-[(3-methylbut-2-en-1-yl)oxy]tetrahydro-2H-pyran-4-yl}quinoline-4-carboxamide —— C21H25FN2O3
6-fluoro-2-methyl-N-{trans-3-[(3-methylbut-2-en-1-yl)oxy]tetrahydro-2H-pyran-4-yl}quinoline-4-carboxamide
—— (6Z)-5-imino-6-[[1-[2-(3-methylphenoxy)ethyl]indol-3-yl]methylidene]-2-(2-oxo-2-pyrrolidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H28N6O3S
(6Z)-5-imino-6-[[1-[2-(3-methylphenoxy)ethyl]indol-3-yl]methylidene]-2-(2-oxo-2-pyrrolidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-2-(2-chlorophenyl)-6-({1-[2-(2,4-dimethylphenoxy)ethyl]-1H-indol-3-yl}methylidene)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C30H24ClN5O2S
(6Z)-2-(2-chlorophenyl)-6-({1-[2-(2,4-dimethylphenoxy)ethyl]-1H-indol-3-yl}methylidene)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-{4-[(4-bromobenzyl)oxy]-3-methoxybenzylidene}-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H21BrN4O3S
(6Z)-6-{4-[(4-bromobenzyl)oxy]-3-methoxybenzylidene}-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[(1-propan-2-ylbenzimidazol-2-yl)amino]methylidene]cyclohexa-2,4-dien-1-one —— C17H17N3O
(6E)-6-[[(1-propan-2-ylbenzimidazol-2-yl)amino]methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-6-[2-amino-5-(4-methoxyphenoxy)-1H-pyrimidin-6-ylidene]-3-[(2-fluorophenyl)methoxy]cyclohexa-2,4-dien-1-one —— C24H20FN3O4
(6Z)-6-[2-amino-5-(4-methoxyphenoxy)-1H-pyrimidin-6-ylidene]-3-[(2-fluorophenyl)methoxy]cyclohexa-2,4-dien-1-one
—— (6E)-6-[[[1-hydroxy-2-(hydroxymethyl)butan-2-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C12H17NO3
(6E)-6-[[[1-hydroxy-2-(hydroxymethyl)butan-2-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-methyl-2-morpholin-4-yl-N-[(Z)-(4-pentoxyphenyl)methylideneamino]pyrimidin-4-amine —— C21H29N5O2
6-methyl-2-morpholin-4-yl-N-[(Z)-(4-pentoxyphenyl)methylideneamino]pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(methoxymethyl)pyrimidin-4-amine —— C16H24N6OS
6-(trans-3-aminocyclobutyl)-N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(methoxymethyl)pyrimidin-4-amine
—— 6-[(E)-2-[4-(difluoromethoxy)phenyl]ethenyl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C20H14F2N4O2
6-[(E)-2-[4-(difluoromethoxy)phenyl]ethenyl]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— (6Z)-6-(3-ethoxy-4-{2-[2-(prop-2-en-1-yl)phenoxy]ethoxy}benzylidene)-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H30N4O4S
(6Z)-6-(3-ethoxy-4-{2-[2-(prop-2-en-1-yl)phenoxy]ethoxy}benzylidene)-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6,8-dibromo-2-oxo-N'-[(E)-(2-oxonaphthalen-1-ylidene)methyl]chromene-3-carbohydrazide —— C21H12Br2N2O4
6,8-dibromo-2-oxo-N'-[(E)-(2-oxonaphthalen-1-ylidene)methyl]chromene-3-carbohydrazide
—— 6-(3-aminocyclobutyl)-N-[1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl]pyrimidin-4-amine —— C18H29N5O
6-(3-aminocyclobutyl)-N-[1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N-(1,3-benzodioxol-5-ylmethyl)-2-methylpyrimidin-4-amine —— C17H20N4O2
6-(3-aminocyclobutyl)-N-(1,3-benzodioxol-5-ylmethyl)-2-methylpyrimidin-4-amine
—— 6-{[4-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]carbonyl}-2-methyl-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one —— C19H31N5O3
6-{[4-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]carbonyl}-2-methyl-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one
—— (6E)-2,4-dibromo-6-[[(2E)-2-(3-methyl-1,3-benzothiazol-2-ylidene)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C15H11Br2N3OS
(6E)-2,4-dibromo-6-[[(2E)-2-(3-methyl-1,3-benzothiazol-2-ylidene)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— 6-(3-aminocyclobutyl)-N-{[3-(4-methoxyphenyl)isoxazol-5-yl]methyl}pyrimidin-4-amine —— C19H21N5O2
6-(3-aminocyclobutyl)-N-{[3-(4-methoxyphenyl)isoxazol-5-yl]methyl}pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N-[3-(4,5-dimethyl-1H-benzimidazol-2-yl)propyl]pyrimidin-4-amine —— C20H26N6
6-(cis-3-aminocyclobutyl)-N-[3-(4,5-dimethyl-1H-benzimidazol-2-yl)propyl]pyrimidin-4-amine
—— (6Z)-6-[(2-chloro-6-fluorophenyl)methylidene]-3-(5-chloro-2-methoxyphenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C18H10Cl2FN3O2S
(6Z)-6-[(2-chloro-6-fluorophenyl)methylidene]-3-(5-chloro-2-methoxyphenyl)-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— (6Z)-6-{3-chloro-4-[2-(3,4-dimethylphenoxy)ethoxy]benzylidene}-5-imino-2-(4-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H25ClN4O3S
(6Z)-6-{3-chloro-4-[2-(3,4-dimethylphenoxy)ethoxy]benzylidene}-5-imino-2-(4-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-5-imino-6-{[1-(2-methoxy-5-methylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(2-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H25N5O2S
(6Z)-5-imino-6-{[1-(2-methoxy-5-methylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(2-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-isobutyl-N-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-2-oxo-1,2-dihydropyrimidine-4-carboxamide —— C15H21N5O2
6-isobutyl-N-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-2-oxo-1,2-dihydropyrimidine-4-carboxamide
—— 6-(3-aminocyclobutyl)-N~4~-{3-[cyclopentyl(methyl)amino]propyl}pyrimidine-2,4-diamine —— C17H30N6
6-(3-aminocyclobutyl)-N~4~-{3-[cyclopentyl(methyl)amino]propyl}pyrimidine-2,4-diamine