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—— 6-tert-butyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-2-oxo-2,3-dihydropyrimidine-4-carboxamide —— C16H20F3N5O2
6-tert-butyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-2-oxo-2,3-dihydropyrimidine-4-carboxamide
—— 6-amino-N-{[1-(methoxymethyl)cyclopentyl]methyl}nicotinamide —— C14H21N3O2
6-amino-N-{[1-(methoxymethyl)cyclopentyl]methyl}nicotinamide
—— 6-methyl-N-[(1S,5R,6S)-2-oxabicyclo[3.2.0]heptan-6-yl]-4-oxo-1H-pyridine-2-carboxamide —— C13H16N2O3
6-methyl-N-[(1S,5R,6S)-2-oxabicyclo[3.2.0]heptan-6-yl]-4-oxo-1H-pyridine-2-carboxamide
—— 6-ethyl 8-isopropyl 5-amino-2-(3-methoxybenzylidene)-7-(3-methoxyphenyl)-3-oxo-2,3-dihydro-7H-[1,3]thiazolo[3,2-a]pyridine-6,8-dicarboxylate —— C29H30N2O7S
6-ethyl 8-isopropyl 5-amino-2-(3-methoxybenzylidene)-7-(3-methoxyphenyl)-3-oxo-2,3-dihydro-7H-[1,3]thiazolo[3,2-a]pyridine-6,8-dicarboxylate
—— 6-(3-Aminocyclobutyl)-N-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-YL]methyl}-N-methylpyrimidin-4-amine —— C19H22N6O2
6-(3-Aminocyclobutyl)-N-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-YL]methyl}-N-methylpyrimidin-4-amine
—— (6E)-4-chloro-6-[[3-(5,7-dimethyl-1,3-benzoxazol-2-yl)-2-methylanilino]methylidene]-2-nitrocyclohexa-2,4-dien-1-one —— C23H18ClN3O4
(6E)-4-chloro-6-[[3-(5,7-dimethyl-1,3-benzoxazol-2-yl)-2-methylanilino]methylidene]-2-nitrocyclohexa-2,4-dien-1-one
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[3-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidine-2,4-diamine —— C16H25N7
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[3-(1-methyl-1H-imidazol-2-yl)propyl]pyrimidine-2,4-diamine
—— 6-ethyl-2-[[(E)-3-(5-methylfuran-2-yl)prop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C19H22N2O3S
6-ethyl-2-[[(E)-3-(5-methylfuran-2-yl)prop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-{[2-(2-Methoxyethyl)morpholin-4-yl]carbonyl}quinoline —— C17H20N2O3
6-{[2-(2-Methoxyethyl)morpholin-4-yl]carbonyl}quinoline
—— 6-{[2-(6-methoxypyridin-3-yl)-1,4,6,7-tetrahydro-5H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-methylpyrimidin-4-ol —— C18H20N6O2
6-{[2-(6-methoxypyridin-3-yl)-1,4,6,7-tetrahydro-5H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-methylpyrimidin-4-ol
—— 6-{[(2R*,6S*)-2,6-dimethylmorpholin-4-yl]methyl}pyridine-2-carboxylic acid —— C13H18N2O3
6-{[(2R*,6S*)-2,6-dimethylmorpholin-4-yl]methyl}pyridine-2-carboxylic acid
—— 6-(trans-3-aminocyclobutyl)-N~4~-[2-(pyridin-3-ylamino)ethyl]pyrimidine-2,4-diamine —— C15H21N7
6-(trans-3-aminocyclobutyl)-N~4~-[2-(pyridin-3-ylamino)ethyl]pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]pyrimidin-4-amine —— C16H24N6
6-(3-aminocyclobutyl)-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]pyrimidin-4-amine
—— 6-methyl-4-oxo-N-{2-[(2-oxopyrrolidin-1-yl)methyl]benzyl}-4H-pyran-2-carboxamide —— C19H20N2O4
6-methyl-4-oxo-N-{2-[(2-oxopyrrolidin-1-yl)methyl]benzyl}-4H-pyran-2-carboxamide
—— 6-(3-aminocyclobutyl)-N~4~-{[1-(dimethylamino)cyclohexyl]methyl}pyrimidine-2,4-diamine —— C17H30N6
6-(3-aminocyclobutyl)-N~4~-{[1-(dimethylamino)cyclohexyl]methyl}pyrimidine-2,4-diamine
—— 6-amino-N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]nicotinamide —— C19H24N4O
6-amino-N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]nicotinamide
—— 6-methyl-N-[rac-2-oxabicyclo[3.2.0]hept-6-yl]pyridazin-3-amine —— C11H15N3O
6-methyl-N-[rac-2-oxabicyclo[3.2.0]hept-6-yl]pyridazin-3-amine
—— 6-[(4-ethyl-2-methyl-3-oxopiperazin-1-yl)carbonyl]-3,4-dihydro[1]benzothieno[2,3-c]pyridin-1(2H)-one —— C19H21N3O3S
6-[(4-ethyl-2-methyl-3-oxopiperazin-1-yl)carbonyl]-3,4-dihydro[1]benzothieno[2,3-c]pyridin-1(2H)-one
—— (6E)-6-{[1-(2,5-dichlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(pentan-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H23Cl2N5OS
(6E)-6-{[1-(2,5-dichlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(pentan-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(cis-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-[(3-phenylisoxazol-5-yl)methyl]pyrimidin-4-amine —— C22H25N5O
6-(cis-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-[(3-phenylisoxazol-5-yl)methyl]pyrimidin-4-amine
—— 6-(3-Aminocyclobutyl)-N-[(2-isopropyl-4-methyl-1,3-thiazol-5-YL)methyl]pyrimidin-4-amine —— C16H23N5S
6-(3-Aminocyclobutyl)-N-[(2-isopropyl-4-methyl-1,3-thiazol-5-YL)methyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N-(2-azepan-1-ylethyl)-2-(methoxymethyl)-N-methylpyrimidin-4-amine —— C19H33N5O
6-(3-aminocyclobutyl)-N-(2-azepan-1-ylethyl)-2-(methoxymethyl)-N-methylpyrimidin-4-amine
—— 6-fluoro-N-{[4-(hydroxymethyl)tetrahydro-2H-pyran-4-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide —— C17H19FN2O4
6-fluoro-N-{[4-(hydroxymethyl)tetrahydro-2H-pyran-4-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
—— (6Z)-3-(4-tert-butylphenyl)-6-[(3,4-dimethoxyphenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C23H23N3O3S
(6Z)-3-(4-tert-butylphenyl)-6-[(3,4-dimethoxyphenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— 6-[2-(2,3-Dihydro-1,4-benzodioxin-2-YL)ethyl]-N-isopropylpyridazin-3-amine —— C17H21N3O2
6-[2-(2,3-Dihydro-1,4-benzodioxin-2-YL)ethyl]-N-isopropylpyridazin-3-amine
—— 6-cyano-N-[rac-(1R,5R,6S,7R)-7-pyrrolidin-1-yl-2-oxabicyclo[3.2.0]hept-6-yl]nicotinamide —— C17H20N4O2
6-cyano-N-[rac-(1R,5R,6S,7R)-7-pyrrolidin-1-yl-2-oxabicyclo[3.2.0]hept-6-yl]nicotinamide
—— 6-[2-[2-(dimethylamino)-1-hydroxyethyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]-2,4-dimethylnicotinonitrile —— C18H24N6O
6-[2-[2-(dimethylamino)-1-hydroxyethyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]-2,4-dimethylnicotinonitrile
—— 6-(3-Aminocyclobutyl)-2-cyclopropyl-N-[2-(2-fluorophenyl)ethyl]pyrimidin-4-amine —— C19H23FN4
6-(3-Aminocyclobutyl)-2-cyclopropyl-N-[2-(2-fluorophenyl)ethyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(methoxymethyl)-N-methylpyrimidin-4-amine —— C19H30N6O
6-(3-aminocyclobutyl)-N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(methoxymethyl)-N-methylpyrimidin-4-amine
—— (6E)-6-[(2Z)-2-[(4E)-6-amino-4-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-1,3,5-triazin-2-ylidene]ethylidene]-4-bromocyclohexa-2,4-dien-1-one —— C17H13BrN4O2
(6E)-6-[(2Z)-2-[(4E)-6-amino-4-(6-oxocyclohexa-2,4-dien-1-ylidene)-1H-1,3,5-triazin-2-ylidene]ethylidene]-4-bromocyclohexa-2,4-dien-1-one
—— 6-(cis-3-aminocyclobutyl)-N~4~-(2,3-dimethoxybenzyl)pyrimidine-2,4-diamine —— C17H23N5O2
6-(cis-3-aminocyclobutyl)-N~4~-(2,3-dimethoxybenzyl)pyrimidine-2,4-diamine
—— (6Z)-6-[[1-(4-ethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H30N6O3S
(6Z)-6-[[1-(4-ethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-(quinolin-3-ylmethyl)pyrimidine-2,4-diamine —— C19H22N6
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-(quinolin-3-ylmethyl)pyrimidine-2,4-diamine
—— 6-(cis-3-aminocyclobutyl)-N-[(3S)-1-benzylpiperidin-3-yl]pyrimidin-4-amine —— C20H27N5
6-(cis-3-aminocyclobutyl)-N-[(3S)-1-benzylpiperidin-3-yl]pyrimidin-4-amine
—— 6-{[2-(5-methylisoxazol-3-yl)piperidin-1-yl]carbonyl}pyridin-2(1H)-one —— C15H17N3O3
6-{[2-(5-methylisoxazol-3-yl)piperidin-1-yl]carbonyl}pyridin-2(1H)-one
—— 6-(cis-3-aminocyclobutyl)-N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)pyrimidin-4-amine —— C18H31N5
6-(cis-3-aminocyclobutyl)-N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)pyrimidin-4-amine
—— (6Z)-3-butoxy-6-[1-(hydroxyamino)-2-phenylethylidene]cyclohexa-2,4-dien-1-one —— C18H21NO3
(6Z)-3-butoxy-6-[1-(hydroxyamino)-2-phenylethylidene]cyclohexa-2,4-dien-1-one
—— 6-methyl-3-[(2Z)-2-[(1-methyl-2-phenylindol-3-yl)methylidene]hydrazinyl]-4H-1,2,4-triazin-5-one —— C20H18N6O
6-methyl-3-[(2Z)-2-[(1-methyl-2-phenylindol-3-yl)methylidene]hydrazinyl]-4H-1,2,4-triazin-5-one
—— 6-{cis-3-[(1-benzylpiperidin-4-yl)amino]cyclobutyl}pyrimidin-4(3H)-one —— C20H26N4O
6-{cis-3-[(1-benzylpiperidin-4-yl)amino]cyclobutyl}pyrimidin-4(3H)-one
—— 6-(3-aminocyclobutyl)-N~4~-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidine-2,4-diamine —— C15H23N7
6-(3-aminocyclobutyl)-N~4~-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidine-2,4-diamine
—— (6Z)-4-amino-6-[[4-[4-[(2Z)-2-(8-amino-1-oxo-5,7-disulfonatonaphthalen-2-ylidene)hydrazinyl]-3-methylphenyl]-2-methylphenyl]hydrazinylidene]-5-oxonaphthalene-1,3-disulfonate —— C34H24N6O14S4-4
(6Z)-4-amino-6-[[4-[4-[(2Z)-2-(8-amino-1-oxo-5,7-disulfonatonaphthalen-2-ylidene)hydrazinyl]-3-methylphenyl]-2-methylphenyl]hydrazinylidene]-5-oxonaphthalene-1,3-disulfonate
—— 6-amino-N-[1-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)ethyl]pyridine-2-carboxamide —— C15H14N6O2
6-amino-N-[1-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)ethyl]pyridine-2-carboxamide
—— (6Z)-3-butoxy-6-[1-(hydroxyamino)tetradecylidene]cyclohexa-2,4-dien-1-one —— C24H41NO3
(6Z)-3-butoxy-6-[1-(hydroxyamino)tetradecylidene]cyclohexa-2,4-dien-1-one
—— 6-(3-Aminocyclobutyl)-N-{[1-(dimethylamino)cyclohexyl]methyl}-2-(methoxymethyl)pyrimidin-4-amine —— C19H33N5O
6-(3-Aminocyclobutyl)-N-{[1-(dimethylamino)cyclohexyl]methyl}-2-(methoxymethyl)pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-pyrrolidin-1-ylpyrimidin-4-amine —— C19H27N7
6-(cis-3-aminocyclobutyl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-pyrrolidin-1-ylpyrimidin-4-amine
—— 6-N-[(Z)-[1-[2-(4-cyclohexylphenoxy)ethyl]indol-3-yl]methylideneamino]-4-N,4-N-dimethyl-2-propan-2-ylpyrimidine-4,6-diamine —— C32H40N6O
6-N-[(Z)-[1-[2-(4-cyclohexylphenoxy)ethyl]indol-3-yl]methylideneamino]-4-N,4-N-dimethyl-2-propan-2-ylpyrimidine-4,6-diamine
—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-[(3-methyl-2-thienyl)methyl]pyrimidin-4-amine —— C18H24N4S
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-[(3-methyl-2-thienyl)methyl]pyrimidin-4-amine
—— 6-{[3-(2,3-Dimethoxyphenyl)pyrrolidin-1-yl]carbonyl}-2-methylimidazo[1,2-a]pyridine —— C21H23N3O3
6-{[3-(2,3-Dimethoxyphenyl)pyrrolidin-1-yl]carbonyl}-2-methylimidazo[1,2-a]pyridine
—— 6-(3-aminocyclobutyl)-N~2~,N~2~,N~4~-trimethyl-N~4~-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-2,4-diamine —— C20H27N5
6-(3-aminocyclobutyl)-N~2~,N~2~,N~4~-trimethyl-N~4~-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-2,4-diamine
—— (6E)-6-(4-methyl-3H-1,3-benzoxazol-2-ylidene)-4-[[(E)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]cyclohexa-2,4-dien-1-one —— C21H16N2O3
(6E)-6-(4-methyl-3H-1,3-benzoxazol-2-ylidene)-4-[[(E)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]cyclohexa-2,4-dien-1-one