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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[1-[2-[(1S)-cyclopent-2-en-1-yl]acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H23N3O2
6-[1-[2-[(1S)-cyclopent-2-en-1-yl]acetyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-Fluoro-2-[1-(3-morpholin-4-ylpropanoyl)piperidin-4-yl]quinoline-3-carboxamide —— C22H27FN4O3
6-Fluoro-2-[1-(3-morpholin-4-ylpropanoyl)piperidin-4-yl]quinoline-3-carboxamide
—— 6-[(3R)-1-[(2S)-oxolane-2-carbonyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one —— C18H21N3O3
6-[(3R)-1-[(2S)-oxolane-2-carbonyl]piperidin-3-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-(3-pyrazol-1-ylpropanoyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C19H21N5O2
6-[1-(3-pyrazol-1-ylpropanoyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[1-(2-pyridin-3-ylacetyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H20N4O2
6-[1-(2-pyridin-3-ylacetyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— (6-amino-2,3-dihydro-1,4-benzodioxin-7-yl)-[(3R)-3-(5-fluorobenzimidazol-1-yl)piperidin-1-yl]methanone —— C21H21FN4O3
(6-amino-2,3-dihydro-1,4-benzodioxin-7-yl)-[(3R)-3-(5-fluorobenzimidazol-1-yl)piperidin-1-yl]methanone
—— 6-(oxan-4-yl)-2-[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H26N4O3S
6-(oxan-4-yl)-2-[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(thiophene-2-carbonyl)-2-[(3R)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H24N4O2S2
6-(thiophene-2-carbonyl)-2-[(3R)-1-(thiophen-2-ylmethyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(Furan-2-yl)-2-[(4-hydroxypiperidin-4-yl)methyl]pyridazin-3-one —— C14H17N3O3
6-(Furan-2-yl)-2-[(4-hydroxypiperidin-4-yl)methyl]pyridazin-3-one
—— 6-[(2S)-1-cyclopentylpiperidin-2-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one —— C19H24N4O
6-[(2S)-1-cyclopentylpiperidin-2-yl]-2-pyridin-3-yl-1H-pyrimidin-4-one
—— (6S)-4-N-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine —— C19H18ClN5
(6S)-4-N-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine
—— 6-(cyclohexylmethyl)-2-[(2R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H32N4O2S
6-(cyclohexylmethyl)-2-[(2R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-[(2R)-oxane-2-carbonyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H27N3O3
(6R)-1-[(2R)-oxane-2-carbonyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(pyridin-3-ylmethyl)-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H25N5O2S
6-(pyridin-3-ylmethyl)-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6-fluoro-1H-indol-2-yl)-[(3S)-3-(5-thiophen-3-yl-1,3,4-oxadiazol-2-yl)piperidin-1-yl]methanone —— C20H17FN4O2S
(6-fluoro-1H-indol-2-yl)-[(3S)-3-(5-thiophen-3-yl-1,3,4-oxadiazol-2-yl)piperidin-1-yl]methanone
—— (6S)-4-N-(4-chlorophenyl)-2-pyridin-4-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine —— C19H18ClN5
(6S)-4-N-(4-chlorophenyl)-2-pyridin-4-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine
—— 6-(cyclopropanecarbonyl)-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H25N5O3
6-(cyclopropanecarbonyl)-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2-cyclopentylacetyl)-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31N5O3
6-(2-cyclopentylacetyl)-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-4-N-(4-fluorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine —— C19H18FN5
(6R)-4-N-(4-fluorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine
—— (6R)-1-[(3-chlorophenyl)methyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H24ClN3O
(6R)-1-[(3-chlorophenyl)methyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-cyclohexyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H31N5O2
6-cyclohexyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H27FN4O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(4-fluorophenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexylmethyl)-2-[(2R)-1-(4-fluorobenzoyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31FN4O2
6-(cyclohexylmethyl)-2-[(2R)-1-(4-fluorobenzoyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-cyclohexyl-2-[(2S)-1-(4-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31FN4O2
6-cyclohexyl-2-[(2S)-1-(4-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-(pyridin-4-ylmethyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H24N4O
(6R)-1-(pyridin-4-ylmethyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3-fluorobenzoyl)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1,4-diazepan-5-one —— C25H22F2N2O2
(6R)-1-(3-fluorobenzoyl)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-2-pyridin-3-yl-4-N-[3-(trifluoromethyl)phenyl]-5,6,7,8-tetrahydroquinazoline-4,6-diamine —— C20H18F3N5
(6S)-2-pyridin-3-yl-4-N-[3-(trifluoromethyl)phenyl]-5,6,7,8-tetrahydroquinazoline-4,6-diamine
—— 6-[(3-fluorophenyl)methyl]-2-[(3R)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H21FN4
6-[(3-fluorophenyl)methyl]-2-[(3R)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[(3-fluorophenyl)methyl]-2-[(3S)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H21FN4
6-[(3-fluorophenyl)methyl]-2-[(3S)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-cyclohexyl-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31FN4O2
6-cyclohexyl-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2,3-dichlorophenyl)methyl]-2-[(3R)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H20Cl2N4
6-[(2,3-dichlorophenyl)methyl]-2-[(3R)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-chloro-N-[(1-methylimidazol-2-yl)methyl]-1H-indole-2-carboxamide —— C14H13ClN4O
6-chloro-N-[(1-methylimidazol-2-yl)methyl]-1H-indole-2-carboxamide
—— 6-cyclopentyl-2-[(3S)-1-[2-(2,5-difluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H28F2N4O2
6-cyclopentyl-2-[(3S)-1-[2-(2,5-difluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3S)-1-[(3,4-difluorophenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one —— C20H19F2N5O
6-[(3S)-1-[(3,4-difluorophenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one
—— 6-[(3,4-dichlorophenyl)methyl]-2-[(3S)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H20Cl2N4
6-[(3,4-dichlorophenyl)methyl]-2-[(3S)-pyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[(2,3-Dichlorophenyl)methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H15Cl2N5O
6-[(2,3-Dichlorophenyl)methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-(1-methylpyrazole-3-carbonyl)-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H26N4O2S
(6R)-1-(1-methylpyrazole-3-carbonyl)-4-prop-2-enyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(3-Fluorobenzoyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H29FN4O3
6-(3-Fluorobenzoyl)-2-[1-(oxan-4-yl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3,4-Dichlorophenyl)methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H15Cl2N5O
6-[(3,4-Dichlorophenyl)methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3,4-dichlorophenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H20Cl2N4
6-[(3,4-dichlorophenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6S)-4-methyl-1-[(1-methylbenzimidazol-2-yl)methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N5O
(6S)-4-methyl-1-[(1-methylbenzimidazol-2-yl)methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-methyl-1-[(1-methylbenzimidazol-2-yl)methyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N5O
(6S)-4-methyl-1-[(1-methylbenzimidazol-2-yl)methyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6Z)-6-[[[4a-[[(E)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]-1,2,3,4,9,9a-hexahydroxanthen-9-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C27H26N2O3
(6Z)-6-[[[4a-[[(E)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]-1,2,3,4,9,9a-hexahydroxanthen-9-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— (6R)-1-(1-methylpyrazole-3-carbonyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C26H28N4O2
(6R)-1-(1-methylpyrazole-3-carbonyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— 6-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C18H19N5O2
6-[1-(1-methylpyrazole-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— (6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(1-methylpyrazole-4-carbonyl)-1,4-diazepan-5-one —— C24H26N4O3
(6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(1-methylpyrazole-4-carbonyl)-1,4-diazepan-5-one
—— 6-(2-cyclohexylacetyl)-2-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N6O2
6-(2-cyclohexylacetyl)-2-[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6Z)-6-({4-[2-(2,6-Dimethylphenoxy)ethoxy]-3-ethoxyphenyl}methylidene)-5-imino-2-(2-methylpropyl)-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C28H32N4O4S
(6Z)-6-({4-[2-(2,6-Dimethylphenoxy)ethoxy]-3-ethoxyphenyl}methylidene)-5-imino-2-(2-methylpropyl)-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6Z)-4,5-dibromo-6-[(2,5-dimethoxyanilino)methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C16H15Br2NO4
(6Z)-4,5-dibromo-6-[(2,5-dimethoxyanilino)methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— (6S)-1-(1-methylimidazole-2-carbonyl)-6-[(3-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C26H28N4O2
(6S)-1-(1-methylimidazole-2-carbonyl)-6-[(3-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one