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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-5-butyl-6-N-cyclopentyl-2-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H33N5O5
(6S)-5-butyl-6-N-cyclopentyl-2-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-5-butyl-6-N-cyclopentyl-2-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H33N5O5
(6R)-5-butyl-6-N-cyclopentyl-2-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-2-N-(3,5-dimethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O3
(6S)-5-butyl-6-N-cyclopentyl-2-N-(3,5-dimethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-5-ethyl-2-N-(3-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H31N5O3
(6S)-6-N-cyclopentyl-5-ethyl-2-N-(3-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-5-ethyl-6-methyl-2-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H31N5O3
(6R)-6-N-cyclopentyl-5-ethyl-6-methyl-2-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-6-methyl-2-N-[(4-methylsulfanylphenyl)methyl]-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H33N5O3S
(6R)-6-N-cyclopentyl-6-methyl-2-N-[(4-methylsulfanylphenyl)methyl]-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-5-ethyl-6-methyl-4-oxo-2-N-(pyridin-3-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C22H28N6O3
(6S)-6-N-cyclopentyl-5-ethyl-6-methyl-4-oxo-2-N-(pyridin-3-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5-butyl-N-cyclopentyl-6-methyl-4-oxo-2-(4-pyridin-2-ylpiperazine-1-carbonyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H37N7O3
(6S)-5-butyl-N-cyclopentyl-6-methyl-4-oxo-2-(4-pyridin-2-ylpiperazine-1-carbonyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-2-N-[(3,4-dimethoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C27H37N5O5
(6S)-5-butyl-6-N-cyclopentyl-2-N-[(3,4-dimethoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-2-N-[(2,5-dimethoxyphenyl)methyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O5
(6S)-6-N-cyclopentyl-2-N-[(2,5-dimethoxyphenyl)methyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-6-methyl-2-N-[(3-methylphenyl)methyl]-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H33N5O3
(6R)-6-N-cyclopentyl-6-methyl-2-N-[(3-methylphenyl)methyl]-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-2-N-[(3-fluorophenyl)methyl]-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H23F2N5O3
(6R)-2-N-[(3-fluorophenyl)methyl]-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-5-butyl-6-N-cyclopentyl-2-N-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H32FN5O3
(6R)-5-butyl-6-N-cyclopentyl-2-N-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-N-cyclopentyl-6-methyl-4-oxo-2-(piperidine-1-carbonyl)-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C22H33N5O3
(6S)-N-cyclopentyl-6-methyl-4-oxo-2-(piperidine-1-carbonyl)-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-2-N-[2-(1H-indol-3-yl)ethyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C28H36N6O3
(6S)-5-butyl-6-N-cyclopentyl-2-N-[2-(1H-indol-3-yl)ethyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-6-methyl-4-oxo-2-N-(thiophen-2-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H31N5O3S
(6S)-5-butyl-6-N-cyclopentyl-6-methyl-4-oxo-2-N-(thiophen-2-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5-butyl-2-N-cyclohexyl-6-N-cyclopentyl-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H37N5O3
(6S)-5-butyl-2-N-cyclohexyl-6-N-cyclopentyl-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-N-cyclopentyl-6-methyl-4-oxo-2-(4-phenylpiperazine-1-carbonyl)-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H36N6O3
(6R)-N-cyclopentyl-6-methyl-4-oxo-2-(4-phenylpiperazine-1-carbonyl)-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-2-N-(2-methoxyethyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C21H33N5O4
(6S)-5-butyl-6-N-cyclopentyl-2-N-(2-methoxyethyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-5,6-dimethyl-2-N-[(5-methylfuran-2-yl)methyl]-6-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H27N5O4
(6R)-5,6-dimethyl-2-N-[(5-methylfuran-2-yl)methyl]-6-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-6-methyl-4-oxo-5-propyl-2-N-(pyridin-3-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H30N6O3
(6S)-6-N-cyclopentyl-6-methyl-4-oxo-5-propyl-2-N-(pyridin-3-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-5-butyl-6-N-cyclopentyl-6-methyl-2-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O3
(6R)-5-butyl-6-N-cyclopentyl-6-methyl-2-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-6-methyl-4-oxo-2-N-(4-propan-2-ylphenyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C27H37N5O3
(6S)-5-butyl-6-N-cyclopentyl-6-methyl-4-oxo-2-N-(4-propan-2-ylphenyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-2-N-[(2-ethoxyphenyl)methyl]-5-ethyl-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H33N5O4
(6R)-6-N-cyclopentyl-2-N-[(2-ethoxyphenyl)methyl]-5-ethyl-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-2-N-[[4-(dimethylamino)phenyl]methyl]-5-ethyl-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H34N6O3
(6S)-6-N-cyclopentyl-2-N-[[4-(dimethylamino)phenyl]methyl]-5-ethyl-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-2-N-[2-(2-methylphenyl)ethyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H28FN5O3
(6R)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-2-N-[2-(2-methylphenyl)ethyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-2-N-[2-(4-ethoxyphenyl)ethyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C27H37N5O4
(6S)-6-N-cyclopentyl-2-N-[2-(4-ethoxyphenyl)ethyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-6-methyl-4-oxo-2-N-(2-phenylethyl)-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H33N5O3
(6S)-6-N-cyclopentyl-6-methyl-4-oxo-2-N-(2-phenylethyl)-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-2-N-[[4-(dimethylamino)phenyl]methyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H36N6O3
(6R)-6-N-cyclopentyl-2-N-[[4-(dimethylamino)phenyl]methyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-2-N-[2-(4-ethoxyphenyl)ethyl]-5,6-dimethyl-6-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C28H33N5O4
(6R)-2-N-[2-(4-ethoxyphenyl)ethyl]-5,6-dimethyl-6-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-5-ethyl-6-methyl-4-oxo-2-N-(pyridin-2-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C22H28N6O3
(6S)-6-N-cyclopentyl-5-ethyl-6-methyl-4-oxo-2-N-(pyridin-2-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5,6-dimethyl-6-N-[(4-methylphenyl)methyl]-4-oxo-2-N-(2-thiophen-2-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H27N5O3S
(6S)-5,6-dimethyl-6-N-[(4-methylphenyl)methyl]-4-oxo-2-N-(2-thiophen-2-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-N-cyclopentyl-6-methyl-2-(4-methylpiperidine-1-carbonyl)-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C23H35N5O3
(6S)-N-cyclopentyl-6-methyl-2-(4-methylpiperidine-1-carbonyl)-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-6-N-cyclopentyl-2-N-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H30FN5O3
(6R)-6-N-cyclopentyl-2-N-[(4-fluorophenyl)methyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-[(4-fluorophenyl)methyl]-2-N-[(4-methoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H26FN5O4
(6S)-6-N-[(4-fluorophenyl)methyl]-2-N-[(4-methoxyphenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-2-N-ethyl-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C19H22FN5O3
(6R)-2-N-ethyl-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-benzyl-2-N-[2-(cyclohexen-1-yl)ethyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H31N5O3
(6R)-6-N-benzyl-2-N-[2-(cyclohexen-1-yl)ethyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-2-N-(3-pyrrolidin-1-ylpropyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H31FN6O3
(6R)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-2-N-(3-pyrrolidin-1-ylpropyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-2-N-[2-(3,4-dimethoxyphenyl)ethyl]-5-ethyl-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O5
(6R)-6-N-cyclopentyl-2-N-[2-(3,4-dimethoxyphenyl)ethyl]-5-ethyl-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-N-cyclopentyl-6-methyl-2-(4-methylpiperidine-1-carbonyl)-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C23H35N5O3
(6R)-N-cyclopentyl-6-methyl-2-(4-methylpiperidine-1-carbonyl)-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-N-cyclopropyl-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C18H27N5O3
(6R)-2-N-cyclopropyl-5,6-dimethyl-6-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-5-ethyl-6-methyl-2-N-[(4-methylsulfanylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H31N5O3S
(6S)-6-N-cyclopentyl-5-ethyl-6-methyl-2-N-[(4-methylsulfanylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-2-N-[(4-ethylphenyl)methyl]-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H28FN5O3
(6R)-2-N-[(4-ethylphenyl)methyl]-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-2-N-(3-propylsulfanylpropyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H30FN5O3S
(6R)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-2-N-(3-propylsulfanylpropyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-2-N-(2-thiophen-2-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C23H24FN5O3S
(6R)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-4-oxo-2-N-(2-thiophen-2-ylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-5-ethyl-2-N-[(4-ethylphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H33N5O3
(6S)-6-N-cyclopentyl-5-ethyl-2-N-[(4-ethylphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-6-N-cyclopentyl-2-N-(3-ethoxypropyl)-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C22H35N5O4
(6S)-6-N-cyclopentyl-2-N-(3-ethoxypropyl)-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-2-(4-methylpiperazine-1-carbonyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C22H27FN6O3
(6R)-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-2-(4-methylpiperazine-1-carbonyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-2-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H26FN5O3
(6S)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-2-N-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-5-butyl-6-N-cyclopentyl-2-N-(2,3-dimethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O3
(6R)-5-butyl-6-N-cyclopentyl-2-N-(2,3-dimethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide