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—— (6R)-2-tert-butyl-N-cycloheptyl-5-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H36N4O3
(6R)-2-tert-butyl-N-cycloheptyl-5-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-(4-methoxyphenyl)-N-(3-methoxypropyl)-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H28N4O4
(6S)-5-(4-methoxyphenyl)-N-(3-methoxypropyl)-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-benzyl-5-(3-ethylphenyl)-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C30H30N4O3
(6S)-N-benzyl-5-(3-ethylphenyl)-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-benzyl-5-cyclopropyl-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H24N4O2
(6S)-N-benzyl-5-cyclopropyl-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-[(4-ethoxyphenyl)methyl]-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C31H32N4O4
(6S)-5-[(4-ethoxyphenyl)methyl]-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-(4-ethoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C30H30N4O4
(6S)-5-(4-ethoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-(3-methoxypropyl)-6-methyl-4-oxo-2-phenyl-5-(4-propan-2-ylphenyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O3
(6R)-N-(3-methoxypropyl)-6-methyl-4-oxo-2-phenyl-5-(4-propan-2-ylphenyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-benzyl-5-(2,5-dimethylphenyl)-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C30H30N4O3
(6R)-N-benzyl-5-(2,5-dimethylphenyl)-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-benzyl-5-(2,3-dimethylphenyl)-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H28N4O2
(6R)-N-benzyl-5-(2,3-dimethylphenyl)-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-tert-butyl-N-cyclohexyl-5-[(3-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H33FN4O2
(6S)-2-tert-butyl-N-cyclohexyl-5-[(3-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-[(3-chlorophenyl)methyl]-N-cyclohexyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H31ClN4O2
(6R)-5-[(3-chlorophenyl)methyl]-N-cyclohexyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-benzyl-5-[(4-fluorophenyl)methyl]-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H27FN4O3
(6R)-N-benzyl-5-[(4-fluorophenyl)methyl]-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6Z)-6-[[1-[2-(4-butan-2-ylphenoxy)ethyl]indol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H25N5O2S
(6Z)-6-[[1-[2-(4-butan-2-ylphenoxy)ethyl]indol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-N-cyclohexyl-2-(4-methoxyphenyl)-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H32N4O3
(6S)-N-cyclohexyl-2-(4-methoxyphenyl)-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-5-(2-phenylethyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C31H32N4O4
(6R)-2-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-5-(2-phenylethyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-(4-chlorophenyl)-N-cycloheptyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H31ClN4O2
(6R)-5-(4-chlorophenyl)-N-cycloheptyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-benzyl-5-(2,3-dimethylphenyl)-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C30H30N4O3
(6R)-N-benzyl-5-(2,3-dimethylphenyl)-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-5-[2-(diethylamino)ethyl]-2-(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H41N5O2
(6R)-N-cyclohexyl-5-[2-(diethylamino)ethyl]-2-(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-cycloheptyl-N-cyclohexyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H38N4O2
(6S)-5-cycloheptyl-N-cyclohexyl-6-methyl-4-oxo-2-propan-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O4
(6S)-2-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-(4-fluoro-2-methylphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H27FN4O3
(6S)-5-(4-fluoro-2-methylphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-[2-(furan-2-yl)ethyl]-2-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H30N4O5
(6R)-5-[2-(furan-2-yl)ethyl]-2-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cycloheptyl-2-cyclopropyl-5-(4-ethoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H34N4O3
(6S)-N-cycloheptyl-2-cyclopropyl-5-(4-ethoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-(3,5-dimethylphenyl)-N-(3-methoxypropyl)-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O3
(6S)-5-(3,5-dimethylphenyl)-N-(3-methoxypropyl)-6-methyl-4-oxo-2-phenyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-5-[(3-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C31H32N4O4
(6R)-2-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-5-[(3-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-2-tert-butyl-N-cycloheptyl-5-(4-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H33FN4O2
(6R)-2-tert-butyl-N-cycloheptyl-5-(4-fluorophenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-5-[2-(furan-2-yl)ethyl]-2-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C29H30N4O5
(6S)-5-[2-(furan-2-yl)ethyl]-2-(4-methoxyphenyl)-N-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-2-cyclopropyl-5-[(2-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H31FN4O2
(6R)-N-cycloheptyl-2-cyclopropyl-5-[(2-fluorophenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-2-(4-methoxyphenyl)-6-methyl-4-oxo-5-(pyridin-3-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H31N5O3
(6R)-N-cyclohexyl-2-(4-methoxyphenyl)-6-methyl-4-oxo-5-(pyridin-3-ylmethyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-5-[(2-fluorophenyl)methyl]-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H31FN4O3
(6R)-N-cyclohexyl-5-[(2-fluorophenyl)methyl]-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-5-(3,4-dimethylphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O2S
(6S)-N-cyclohexyl-5-(3,4-dimethylphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-5-(3-methylsulfanylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O3S
(6R)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-5-(3-methylsulfanylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-5-(2-fluorophenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H27FN4O2S
(6R)-N-cycloheptyl-5-(2-fluorophenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-5-[(2R)-2-phenylpropyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H34N4O3
(6S)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-5-[(2R)-2-phenylpropyl]-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-5-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H34N4O3
(6R)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-5-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-6-methyl-5-[(2-methylphenyl)methyl]-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O2S
(6R)-N-cyclohexyl-6-methyl-5-[(2-methylphenyl)methyl]-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-tert-butyl-5-(3-fluorophenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C22H23FN4O3
(6S)-N-tert-butyl-5-(3-fluorophenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(4-propan-2-ylphenyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H34N4O3
(6S)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(4-propan-2-ylphenyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-2-(furan-2-yl)-5-[(4-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H32N4O4
(6R)-N-cycloheptyl-2-(furan-2-yl)-5-[(4-methoxyphenyl)methyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cycloheptyl-5-(4-methoxyphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O3S
(6S)-N-cycloheptyl-5-(4-methoxyphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-(4-chlorophenyl)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H27ClN4O3
(6R)-5-(4-chlorophenyl)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-(1,3-benzodioxol-5-ylmethyl)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H28N4O5
(6R)-5-(1,3-benzodioxol-5-ylmethyl)-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-5-[(4-fluorophenyl)methyl]-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H31FN4O3
(6R)-N-cyclohexyl-5-[(4-fluorophenyl)methyl]-2-(4-methoxyphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-5-[2-(4-chlorophenyl)ethyl]-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H29ClN4O3
(6R)-5-[2-(4-chlorophenyl)ethyl]-N-cyclohexyl-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-5-(4-ethoxyphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O3S
(6R)-N-cyclohexyl-5-(4-ethoxyphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-5-(4-fluorophenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H25FN4O2S
(6R)-N-cyclohexyl-5-(4-fluorophenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-5-(2,4-difluorophenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H24F2N4O3
(6R)-N-cyclohexyl-5-(2,4-difluorophenyl)-2-(furan-2-yl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cyclohexyl-6-methyl-4-oxo-5-(3-propylsulfanylpropyl)-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C24H34N4O2S2
(6S)-N-cyclohexyl-6-methyl-4-oxo-5-(3-propylsulfanylpropyl)-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-N-cycloheptyl-5-(3-methoxyphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C26H30N4O3S
(6S)-N-cycloheptyl-5-(3-methoxyphenyl)-6-methyl-4-oxo-2-thiophen-2-yl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(3-phenylpropyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C28H34N4O3
(6R)-N-cycloheptyl-2-(furan-2-yl)-6-methyl-4-oxo-5-(3-phenylpropyl)-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide