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—— 6-[(2S)-2-(5-methyl-1,2-oxazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione —— C18H20N4O5S
6-[(2S)-2-(5-methyl-1,2-oxazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione
—— (6,7-Dimethylspiro[chromene-2,4'-piperidine]-1'-yl)-morpholin-4-ylmethanone —— C20H26N2O3
(6,7-Dimethylspiro[chromene-2,4'-piperidine]-1'-yl)-morpholin-4-ylmethanone
—— 6-[(2S)-2-(5-methyl-1,2-oxazol-3-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one —— C20H25N3O5S
6-[(2S)-2-(5-methyl-1,2-oxazol-3-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one
—— (6E)-4-bromo-6-[(2-hydroxy-3,5-dimethylanilino)methylidene]-2-nitrocyclohexa-2,4-dien-1-one —— C15H13BrN2O4
(6E)-4-bromo-6-[(2-hydroxy-3,5-dimethylanilino)methylidene]-2-nitrocyclohexa-2,4-dien-1-one
—— (6E)-6-[[2-(2-nitrophenyl)hydrazinyl]methylidene]-3-propoxycyclohexa-2,4-dien-1-one —— C16H17N3O4
(6E)-6-[[2-(2-nitrophenyl)hydrazinyl]methylidene]-3-propoxycyclohexa-2,4-dien-1-one
—— (6Z)-6-{3-chloro-4-[(3-methylbenzyl)oxy]benzylidene}-5-imino-2-[2-(morpholin-4-yl)-2-oxoethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H24ClN5O4S
(6Z)-6-{3-chloro-4-[(3-methylbenzyl)oxy]benzylidene}-5-imino-2-[2-(morpholin-4-yl)-2-oxoethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[2-(2-pyridin-3-yl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C22H19N5OS
(6E)-6-[[2-(2-pyridin-3-yl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-2-bromo-4-tert-butyl-6-[(3,5-dimethylphenyl)hydrazinylidene]cyclohexa-2,4-dien-1-one —— C18H21BrN2O
(6E)-2-bromo-4-tert-butyl-6-[(3,5-dimethylphenyl)hydrazinylidene]cyclohexa-2,4-dien-1-one
—— 6-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one —— C20H25N3O5S
6-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)azepan-1-yl]sulfonyl-3-propan-2-yl-1,3-benzoxazol-2-one
—— 6-[1-(1-methylsulfonylpiperidine-4-carbonyl)piperidine-4-carbonyl]-4H-1,4-benzoxazin-3-one —— C21H27N3O6S
6-[1-(1-methylsulfonylpiperidine-4-carbonyl)piperidine-4-carbonyl]-4H-1,4-benzoxazin-3-one
—— (6E)-6-[(5-ethyl-2-hydroxyanilino)methylidene]-2,4-dinitrocyclohexa-2,4-dien-1-one —— C15H13N3O6
(6E)-6-[(5-ethyl-2-hydroxyanilino)methylidene]-2,4-dinitrocyclohexa-2,4-dien-1-one
—— 6-[1-[2-(4-oxo-3H-phthalazin-1-yl)acetyl]piperidine-4-carbonyl]-4H-1,4-benzoxazin-3-one —— C24H22N4O5
6-[1-[2-(4-oxo-3H-phthalazin-1-yl)acetyl]piperidine-4-carbonyl]-4H-1,4-benzoxazin-3-one
—— 6-[(4-fluorophenyl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H25FN4O
6-[(4-fluorophenyl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-benzyl-2-[(3R)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H26N4O
6-benzyl-2-[(3R)-3-methylpiperidin-1-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6E)-2-bromo-4-nitro-6-[(3-tricyclo[4.3.1.13,8]undecanylmethylamino)methylidene]cyclohexa-2,4-dien-1-one —— C19H23BrN2O3
(6E)-2-bromo-4-nitro-6-[(3-tricyclo[4.3.1.13,8]undecanylmethylamino)methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-6-[[3-bromo-4-(dimethylamino)phenyl]methylidene]-5-imino-2-(2-oxo-2-pyrrolidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C20H21BrN6O2S
(6Z)-6-[[3-bromo-4-(dimethylamino)phenyl]methylidene]-5-imino-2-(2-oxo-2-pyrrolidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-benzyl-2-methyl-4-(4-pyridin-2-ylpiperazin-1-yl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C24H28N6
6-benzyl-2-methyl-4-(4-pyridin-2-ylpiperazin-1-yl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-benzyl-2-methyl-N-[(5-methylfuran-2-yl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine —— C26H32N4O2
6-benzyl-2-methyl-N-[(5-methylfuran-2-yl)methyl]-N-[[(2S)-oxolan-2-yl]methyl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine
—— (6E)-2,4-dibromo-6-[[[2-(2,5-dichlorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C20H10Br2Cl2N2O2
(6E)-2,4-dibromo-6-[[[2-(2,5-dichlorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-3-benzyl-6-[(2-chloro-6-fluorophenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C18H11ClFN3OS
(6Z)-3-benzyl-6-[(2-chloro-6-fluorophenyl)methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— 6-ethyl-5-methyl-2-[(2R)-1-[2-(3-methyl-6-oxopyridazin-1-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H26N6O3
6-ethyl-5-methyl-2-[(2R)-1-[2-(3-methyl-6-oxopyridazin-1-yl)acetyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-[(2S)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione —— C18H20ClN5O4S
6-[(2S)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione
—— (6,7-dimethyl-2-oxochromen-4-yl)methyl (3S)-3-acetamido-3-thiophen-2-ylpropanoate —— C21H21NO5S
(6,7-dimethyl-2-oxochromen-4-yl)methyl (3S)-3-acetamido-3-thiophen-2-ylpropanoate
—— 6-ethyl-5-methyl-2-[(2R)-1-(1,3-thiazole-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C18H21N5O2S
6-ethyl-5-methyl-2-[(2R)-1-(1,3-thiazole-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-(1-methylsulfonylpiperidine-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C21H31N5O4S
6-ethyl-5-methyl-2-[(2S)-1-(1-methylsulfonylpiperidine-4-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-[(2S)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione —— C18H20ClN5O4S
6-[(2S)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-1H-quinazoline-2,4-dione
—— 6-ethyl-5-methyl-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H23N5O2
6-ethyl-5-methyl-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-[(3S,4R)-4-(4-methoxyphenyl)-1-[(3S)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one —— C24H30N4O4
6-[(3S,4R)-4-(4-methoxyphenyl)-1-[(3S)-5-oxo-1-propan-2-ylpyrrolidine-3-carbonyl]pyrrolidin-3-yl]-2-methyl-1H-pyrimidin-4-one
—— 6-ethyl-5-methyl-2-[(2S)-1-[3-(1,2-oxazol-5-yl)propanoyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H25N5O3
6-ethyl-5-methyl-2-[(2S)-1-[3-(1,2-oxazol-5-yl)propanoyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2S)-1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H31N5O3
6-ethyl-5-methyl-2-[(2S)-1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-[(2S)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-ethyl-1,3-benzoxazol-2-one —— C19H23ClN4O4S
6-[(2S)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3-ethyl-1,3-benzoxazol-2-one
—— 6-ethyl-5-methyl-2-[(2S)-1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C24H32N4O4
6-ethyl-5-methyl-2-[(2S)-1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl (3S)-3-acetamido-3-thiophen-2-ylpropanoate —— C18H18N2O7S
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl (3S)-3-acetamido-3-thiophen-2-ylpropanoate
—— 6-[(2R)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3,4-dihydro-1H-quinolin-2-one —— C19H23ClN4O3S
6-[(2R)-2-(4-chloro-2-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3,4-dihydro-1H-quinolin-2-one
—— 6-[(2S)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3,4-dihydro-1H-quinolin-2-one —— C19H23ClN4O3S
6-[(2S)-2-(4-chloro-1-methylpyrazol-3-yl)azepan-1-yl]sulfonyl-3,4-dihydro-1H-quinolin-2-one
—— 6-methyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C22H19N5O3
6-methyl-N-[[4-[5-(3-methyl-1,2-oxazol-5-yl)pyrimidin-4-yl]phenyl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— 6,7-dimethoxy-2-[[2-(4-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]methyl]-3,4-dihydro-1H-isoquinoline —— C26H27N3O3
6,7-dimethoxy-2-[[2-(4-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]methyl]-3,4-dihydro-1H-isoquinoline
—— 6-ethyl-2-[(2S)-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidin-2-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H24N4O4
6-ethyl-2-[(2S)-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidin-2-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-5-methyl-2-[(2R)-1-(1-methylsulfonylpiperidine-4-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H29N5O4S
6-ethyl-5-methyl-2-[(2R)-1-(1-methylsulfonylpiperidine-4-carbonyl)pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-N-[(1R)-1-(2-methoxyphenyl)ethyl]-5-methyl-2-(oxan-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine —— C23H30N4O2
6-ethyl-N-[(1R)-1-(2-methoxyphenyl)ethyl]-5-methyl-2-(oxan-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
—— 6-ethyl-5-methyl-2-[(2S)-1-[3-(1,3,5-trimethylpyrazol-4-yl)propanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C22H30N6O2
6-ethyl-5-methyl-2-[(2S)-1-[3-(1,3,5-trimethylpyrazol-4-yl)propanoyl]pyrrolidin-2-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— 6-ethyl-2-[(2R)-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidin-2-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C20H24N4O4
6-ethyl-2-[(2R)-1-[5-(methoxymethyl)furan-2-carbonyl]pyrrolidin-2-yl]-5-methyl-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (6R)-6-(3,4-dimethoxyphenyl)-3,4,6,7-tetrahydro-2H-pyrimido[1,2-c]quinazoline —— C19H21N3O2
(6R)-6-(3,4-dimethoxyphenyl)-3,4,6,7-tetrahydro-2H-pyrimido[1,2-c]quinazoline
—— 6-ethyl-5-methyl-2-[(3R)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C19H22N6O2
6-ethyl-5-methyl-2-[(3R)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (6E)-6-[(2-hydroxy-5-phenylanilino)methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C20H17NO3
(6E)-6-[(2-hydroxy-5-phenylanilino)methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— (6Z)-6-[[2-(1,3-benzoxazol-2-yl)anilino]methylidene]-4-chloro-2-nitrocyclohexa-2,4-dien-1-one —— C20H12ClN3O4
(6Z)-6-[[2-(1,3-benzoxazol-2-yl)anilino]methylidene]-4-chloro-2-nitrocyclohexa-2,4-dien-1-one
—— (6E)-4-benzyl-2-chloro-6-[(4-methoxyanilino)methylidene]cyclohexa-2,4-dien-1-one —— C21H18ClNO2
(6E)-4-benzyl-2-chloro-6-[(4-methoxyanilino)methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-2-bromo-4-[(2-chlorophenyl)methyl]-6-[(3-morpholin-4-ylpropylamino)methylidene]cyclohexa-2,4-dien-1-one —— C21H24BrClN2O2
(6E)-2-bromo-4-[(2-chlorophenyl)methyl]-6-[(3-morpholin-4-ylpropylamino)methylidene]cyclohexa-2,4-dien-1-one
—— 6-[(3S)-3-(5-ethyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-2-yl)piperidine-1-carbonyl]-5-methyl-3H-thieno[2,3-d]pyrimidin-4-one —— C21H22N6O3S
6-[(3S)-3-(5-ethyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-2-yl)piperidine-1-carbonyl]-5-methyl-3H-thieno[2,3-d]pyrimidin-4-one
—— (6Z)-2-[(4-chlorophenyl)methyl]-6-[[2,5-dimethyl-1-(3-methylphenyl)pyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H22ClN5OS
(6Z)-2-[(4-chlorophenyl)methyl]-6-[[2,5-dimethyl-1-(3-methylphenyl)pyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one