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—— (6Z)-6-[4-(3,5-dimethylpyrazol-1-yl)-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C16H16N4O
(6Z)-6-[4-(3,5-dimethylpyrazol-1-yl)-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-{trans-3-[(1-isonicotinoylpiperidin-4-yl)amino]cyclobutyl}pyrimidin-4(3H)-one —— C19H23N5O2
6-{trans-3-[(1-isonicotinoylpiperidin-4-yl)amino]cyclobutyl}pyrimidin-4(3H)-one
—— 6-(trans-3-aminocyclobutyl)-N-(imidazo[1,2-a]pyridin-3-ylmethyl)-N-methylpyrimidin-4-amine —— C17H20N6
6-(trans-3-aminocyclobutyl)-N-(imidazo[1,2-a]pyridin-3-ylmethyl)-N-methylpyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidin-4-amine —— C17H24N6
6-(3-aminocyclobutyl)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidin-4-amine
—— 6-cyano-N-[(3R,4R)-3-(6-methylpyridin-3-yl)oxyoxan-4-yl]pyridine-3-carboxamide —— C18H18N4O3
6-cyano-N-[(3R,4R)-3-(6-methylpyridin-3-yl)oxyoxan-4-yl]pyridine-3-carboxamide
—— 6-{cis-3-[(2-amino-6-methoxypyrimidin-4-yl)amino]cyclobutyl}-2-(dimethylamino)pyrimidin-4(3H)-one —— C15H21N7O2
6-{cis-3-[(2-amino-6-methoxypyrimidin-4-yl)amino]cyclobutyl}-2-(dimethylamino)pyrimidin-4(3H)-one
—— 6-(cis-3-aminocyclobutyl)-N-methyl-N-(quinolin-5-ylmethyl)pyrimidin-4-amine —— C19H21N5
6-(cis-3-aminocyclobutyl)-N-methyl-N-(quinolin-5-ylmethyl)pyrimidin-4-amine
—— 6-[2-(2,3-Dihydro-1,4-benzodioxin-2-yl)ethyl]-2-morpholin-4-ylpyrimidin-4-amine —— C18H22N4O3
6-[2-(2,3-Dihydro-1,4-benzodioxin-2-yl)ethyl]-2-morpholin-4-ylpyrimidin-4-amine
—— 6-[2-[(Z)-(5-bromoindol-3-ylidene)methyl]hydrazinyl]-4-[2-[(E)-(5-bromoindol-3-ylidene)methyl]hydrazinyl]-N,N-diphenyl-1,3,5-triazin-2-amine —— C33H24Br2N10
6-[2-[(Z)-(5-bromoindol-3-ylidene)methyl]hydrazinyl]-4-[2-[(E)-(5-bromoindol-3-ylidene)methyl]hydrazinyl]-N,N-diphenyl-1,3,5-triazin-2-amine
—— 6-(3-aminocyclobutyl)-N~4~-[2-(2,5-dimethylphenyl)ethyl]pyrimidine-2,4-diamine —— C18H25N5
6-(3-aminocyclobutyl)-N~4~-[2-(2,5-dimethylphenyl)ethyl]pyrimidine-2,4-diamine
—— 6-methyl-N-[1-(1-methylpiperidin-4-yl)ethyl]-4-oxo-4H-pyran-2-carboxamide —— C15H22N2O3
6-methyl-N-[1-(1-methylpiperidin-4-yl)ethyl]-4-oxo-4H-pyran-2-carboxamide
—— 6-amino-N-[(3S,4S)-3-(oxan-4-yl)oxan-4-yl]pyridine-3-carboxamide —— C16H23N3O3
6-amino-N-[(3S,4S)-3-(oxan-4-yl)oxan-4-yl]pyridine-3-carboxamide
—— 6-(3-aminocyclobutyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(methoxymethyl)-N-methylpyrimidin-4-amine —— C17H26N6O
6-(3-aminocyclobutyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(methoxymethyl)-N-methylpyrimidin-4-amine
—— (6E)-6-[(4-acetylanilino)methylidene]-3-(diethylamino)cyclohexa-2,4-dien-1-one —— C19H22N2O2
(6E)-6-[(4-acetylanilino)methylidene]-3-(diethylamino)cyclohexa-2,4-dien-1-one
—— (6E)-4-benzyl-2-bromo-6-[[4-[4-(furan-2-carbonyl)piperazin-1-yl]anilino]methylidene]cyclohexa-2,4-dien-1-one —— C29H26BrN3O3
(6E)-4-benzyl-2-bromo-6-[[4-[4-(furan-2-carbonyl)piperazin-1-yl]anilino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-({cis-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}amino)pyridine-2-carbonitrile —— C17H18N8
6-({cis-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}amino)pyridine-2-carbonitrile
—— 6-{cis-3-[(5-amino[1,2,4]triazolo[4,3-c]pyrimidin-7-yl)amino]cyclobutyl}-2-cyclopropylpyrimidin-4(3H)-one —— C16H18N8O
6-{cis-3-[(5-amino[1,2,4]triazolo[4,3-c]pyrimidin-7-yl)amino]cyclobutyl}-2-cyclopropylpyrimidin-4(3H)-one
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[(3-phenylisoxazol-5-yl)methyl]pyrimidine-2,4-diamine —— C19H22N6O
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[(3-phenylisoxazol-5-yl)methyl]pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~4~-[(1S)-2-methoxy-1-methylethyl]pyrimidine-2,4-diamine —— C12H21N5O
6-(3-aminocyclobutyl)-N~4~-[(1S)-2-methoxy-1-methylethyl]pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N-[2-(5-methyl-1H-benzimidazol-2-yl)ethyl]pyrimidin-4-amine —— C18H22N6
6-(3-aminocyclobutyl)-N-[2-(5-methyl-1H-benzimidazol-2-yl)ethyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-2-(methoxymethyl)-N-[(1-piperidin-1-ylcyclopentyl)methyl]pyrimidin-4-amine —— C21H35N5O
6-(3-aminocyclobutyl)-2-(methoxymethyl)-N-[(1-piperidin-1-ylcyclopentyl)methyl]pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N~4~-[2-(2,3-dimethoxyphenyl)ethyl]pyrimidine-2,4-diamine —— C18H25N5O2
6-(cis-3-aminocyclobutyl)-N~4~-[2-(2,3-dimethoxyphenyl)ethyl]pyrimidine-2,4-diamine
—— 6-{[2-(6-chloro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl}pyridine-2-carboxylic acid —— C18H17ClN4O2
6-{[2-(6-chloro-1H-benzimidazol-2-yl)pyrrolidin-1-yl]methyl}pyridine-2-carboxylic acid
—— 6-(3-aminocyclobutyl)-N~4~-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine —— C19H22N6S
6-(3-aminocyclobutyl)-N~4~-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]pyrimidine-2,4-diamine
—— 6-ethyl-N-[rac-(1S,5S,6S,7R)-7-(methoxymethyl)-2-oxabicyclo[3.2.0]hept-6-yl]-2-methylquinoline-4-carboxamide —— C21H26N2O3
6-ethyl-N-[rac-(1S,5S,6S,7R)-7-(methoxymethyl)-2-oxabicyclo[3.2.0]hept-6-yl]-2-methylquinoline-4-carboxamide
—— 6-(3-aminocyclobutyl)-2-cyclopropyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine —— C18H26N6
6-(3-aminocyclobutyl)-2-cyclopropyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
—— 6-(3-Aminocyclobutyl)-N-(1H-imidazol-2-ylmethyl)-N-methylpyrimidin-4-amine —— C13H18N6
6-(3-Aminocyclobutyl)-N-(1H-imidazol-2-ylmethyl)-N-methylpyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N-[3-(1H-imidazol-1-yl)propyl]-2-(methoxymethyl)pyrimidin-4-amine —— C16H24N6O
6-(trans-3-aminocyclobutyl)-N-[3-(1H-imidazol-1-yl)propyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-(3-ethoxy-4-methoxybenzyl)pyrimidine-2,4-diamine —— C18H25N5O2
6-(3-aminocyclobutyl)-N~4~-(3-ethoxy-4-methoxybenzyl)pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~4~-[(2-ethyl-1,3-thiazol-4-yl)methyl]pyrimidine-2,4-diamine —— C14H20N6S
6-(3-aminocyclobutyl)-N~4~-[(2-ethyl-1,3-thiazol-4-yl)methyl]pyrimidine-2,4-diamine
—— 6-(3-Aminocyclobutyl)-N-[2-(4-isopropyl-1,3-thiazol-2-YL)ethyl]pyrimidin-4-amine —— C16H23N5S
6-(3-Aminocyclobutyl)-N-[2-(4-isopropyl-1,3-thiazol-2-YL)ethyl]pyrimidin-4-amine
—— (6Z)-6-[3-bromo-5-ethoxy-4-(2-phenoxyethoxy)benzylidene]-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H23BrN4O4S
(6Z)-6-[3-bromo-5-ethoxy-4-(2-phenoxyethoxy)benzylidene]-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(cis-3-aminocyclobutyl)-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-pyrrolidin-1-ylpyrimidin-4-amine —— C19H29N7
6-(cis-3-aminocyclobutyl)-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-pyrrolidin-1-ylpyrimidin-4-amine
—— (6E)-6-[[(2-methylquinolin-6-yl)amino]methylidene]cyclohexa-2,4-dien-1-one —— C17H14N2O
(6E)-6-[[(2-methylquinolin-6-yl)amino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-[(E)-2-(3,5-dimethoxyphenyl)ethenyl]-5-nitropyrimidine-2,4-diol —— C14H13N3O6
6-[(E)-2-(3,5-dimethoxyphenyl)ethenyl]-5-nitropyrimidine-2,4-diol
—— (6Z)-6-[2-amino-5-(4-methoxyphenoxy)-6-methyl-1H-pyrimidin-4-ylidene]-3-phenylmethoxycyclohexa-2,4-dien-1-one —— C25H23N3O4
(6Z)-6-[2-amino-5-(4-methoxyphenoxy)-6-methyl-1H-pyrimidin-4-ylidene]-3-phenylmethoxycyclohexa-2,4-dien-1-one
—— 6-benzyl-2-[[(E)-(3-chloro-5-methoxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonitrile —— C23H20ClN3O2S
6-benzyl-2-[[(E)-(3-chloro-5-methoxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonitrile
—— 6-(3-aminocyclobutyl)-N~2~,N~2~-dimethyl-N~4~-(3-pyridin-2-ylpropyl)pyrimidine-2,4-diamine —— C18H26N6
6-(3-aminocyclobutyl)-N~2~,N~2~-dimethyl-N~4~-(3-pyridin-2-ylpropyl)pyrimidine-2,4-diamine
—— (6Z)-6-[[1-(2,3-dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-fluorophenyl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H22FN5OS
(6Z)-6-[[1-(2,3-dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-fluorophenyl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-{[2-(5-isopropylisoxazol-3-yl)pyrrolidin-1-yl]carbonyl}-2,3,4,9-tetrahydro-1H-carbazole —— C23H27N3O2
6-{[2-(5-isopropylisoxazol-3-yl)pyrrolidin-1-yl]carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
—— (6Z)-5-imino-6-{[1-(2-methylbenzyl)-1H-indol-3-yl]methylidene}-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H23N5O2S
(6Z)-5-imino-6-{[1-(2-methylbenzyl)-1H-indol-3-yl]methylidene}-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-(pyridin-3-ylmethyl)pyrimidin-4-amine —— C18H23N5
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-(pyridin-3-ylmethyl)pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N~4~-methylpyrimidine-2,4-diamine —— C16H25N7
6-(3-aminocyclobutyl)-N~4~-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N~4~-methylpyrimidine-2,4-diamine
—— (6Z)-2-cyclohexyl-5-imino-6-({1-[2-(4-methylphenoxy)ethyl]-1H-pyrrol-2-yl}methylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H27N5O2S
(6Z)-2-cyclohexyl-5-imino-6-({1-[2-(4-methylphenoxy)ethyl]-1H-pyrrol-2-yl}methylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-(3-ethoxy-4-hydroxybenzylidene)-5-imino-2-(1-phenylpropyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H22N4O3S
(6E)-6-(3-ethoxy-4-hydroxybenzylidene)-5-imino-2-(1-phenylpropyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-5-imino-6-{[1-(2-methoxy-4-nitrophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C20H15F3N6O4S
(6Z)-5-imino-6-{[1-(2-methoxy-4-nitrophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-2-(2-chlorophenyl)-6-{[1-(2,4-dichlorobenzyl)-1H-indol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H16Cl3N5OS
(6Z)-2-(2-chlorophenyl)-6-{[1-(2,4-dichlorobenzyl)-1H-indol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-{3-ethoxy-4-[2-(4-methoxyphenoxy)ethoxy]benzylidene}-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H28N4O5S
(6Z)-6-{3-ethoxy-4-[2-(4-methoxyphenoxy)ethoxy]benzylidene}-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-3-methoxy-6-[1-[2-(2,4,6-trichlorophenyl)hydrazinyl]ethylidene]cyclohexa-2,4-dien-1-one —— C15H13Cl3N2O2
(6Z)-3-methoxy-6-[1-[2-(2,4,6-trichlorophenyl)hydrazinyl]ethylidene]cyclohexa-2,4-dien-1-one
—— 6-(3-aminocyclobutyl)-N~4~-(2,4-dimethoxybenzyl)pyrimidine-2,4-diamine —— C17H23N5O2
6-(3-aminocyclobutyl)-N~4~-(2,4-dimethoxybenzyl)pyrimidine-2,4-diamine