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—— (6,7-dimethyl-2-thiophen-2-ylquinolin-4-yl)-[(3S)-3-methylpiperidin-1-yl]methanone —— C22H24N2OS
(6,7-dimethyl-2-thiophen-2-ylquinolin-4-yl)-[(3S)-3-methylpiperidin-1-yl]methanone
—— (6-chloropyridin-3-yl)-[4-[(R)-(4-methylphenyl)-phenylmethyl]piperazin-1-yl]methanone —— C24H24ClN3O
(6-chloropyridin-3-yl)-[4-[(R)-(4-methylphenyl)-phenylmethyl]piperazin-1-yl]methanone
—— (6Z)-6-(4-{2-[4-(butan-2-yl)phenoxy]ethoxy}benzylidene)-2-(2-chlorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C30H27ClN4O3S
(6Z)-6-(4-{2-[4-(butan-2-yl)phenoxy]ethoxy}benzylidene)-2-(2-chlorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-benzyl-5-methyl-7-[4-[(3S)-3-methylpiperidin-1-yl]piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C24H32N6
6-benzyl-5-methyl-7-[4-[(3S)-3-methylpiperidin-1-yl]piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 6-(3,4-dimethoxyphenyl)-7-[(3S)-3-methylpiperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C19H23N5O2
6-(3,4-dimethoxyphenyl)-7-[(3S)-3-methylpiperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— (6E)-2-ethyl-5-imino-6-({1-[2-(2-methoxyphenoxy)ethyl]-2-methyl-1H-indol-3-yl}methylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H25N5O3S
(6E)-2-ethyl-5-imino-6-({1-[2-(2-methoxyphenoxy)ethyl]-2-methyl-1H-indol-3-yl}methylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-5-imino-6-{3-methoxy-4-[(3-methylbenzyl)oxy]benzylidene}-2-[2-oxo-2-(piperidin-1-yl)ethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H29N5O4S
(6Z)-5-imino-6-{3-methoxy-4-[(3-methylbenzyl)oxy]benzylidene}-2-[2-oxo-2-(piperidin-1-yl)ethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-(aminomethylidene)-4-chlorocyclohexa-2,4-dien-1-one —— C7H6ClNO
(6Z)-6-(aminomethylidene)-4-chlorocyclohexa-2,4-dien-1-one
—— (6Z)-6-{3-chloro-4-[2-(4-cyclohexylphenoxy)ethoxy]-5-methoxybenzylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C30H33ClN4O4S
(6Z)-6-{3-chloro-4-[2-(4-cyclohexylphenoxy)ethoxy]-5-methoxybenzylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2-butyl-6-[[4-[2-(3,4-dimethylphenoxy)ethoxy]phenyl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H28N4O3S
(6E)-2-butyl-6-[[4-[2-(3,4-dimethylphenoxy)ethoxy]phenyl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-chloro-N-[(Z)-2-ethylbutylideneamino]pyridazin-3-amine —— C10H15ClN4
6-chloro-N-[(Z)-2-ethylbutylideneamino]pyridazin-3-amine
—— 6-[(4-benzhydrylpiperazin-1-yl)methyl]-2-oxo-N-[(1S)-1-thiophen-2-ylethyl]-1H-pyridine-3-carboxamide —— C30H32N4O2S
6-[(4-benzhydrylpiperazin-1-yl)methyl]-2-oxo-N-[(1S)-1-thiophen-2-ylethyl]-1H-pyridine-3-carboxamide
—— (6E)-5-imino-2-pentyl-6-[(5-phenylfuran-2-yl)methylidene]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H20N4O2S
(6E)-5-imino-2-pentyl-6-[(5-phenylfuran-2-yl)methylidene]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(5Z)-5-[(2E)-2-(3-ethyl-5-phenyl-1,3-benzoxazol-2-ylidene)ethylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C26H26N2O4S2
6-[(5Z)-5-[(2E)-2-(3-ethyl-5-phenyl-1,3-benzoxazol-2-ylidene)ethylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— (6Z)-6-[[2,5-dimethyl-1-(4-propan-2-ylphenyl)pyrrol-3-yl]methylidene]-2-(4-fluorophenyl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H24FN5OS
(6Z)-6-[[2,5-dimethyl-1-(4-propan-2-ylphenyl)pyrrol-3-yl]methylidene]-2-(4-fluorophenyl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-{4-[2-(4-cyclohexylphenoxy)ethoxy]benzylidene}-2-heptyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C33H40N4O3S
(6Z)-6-{4-[2-(4-cyclohexylphenoxy)ethoxy]benzylidene}-2-heptyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(S)-(4-hydroxyphenyl)-piperazin-1-ylmethyl]-1,3-benzodioxol-5-ol —— C18H20N2O4
6-[(S)-(4-hydroxyphenyl)-piperazin-1-ylmethyl]-1,3-benzodioxol-5-ol
—— (6Z)-4-chloro-6-[[3-(2-chloro-6-nitroanilino)propylamino]methylidene]cyclohexa-2,4-dien-1-one —— C16H15Cl2N3O3
(6Z)-4-chloro-6-[[3-(2-chloro-6-nitroanilino)propylamino]methylidene]cyclohexa-2,4-dien-1-one
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl (E)-3-(3-chlorophenyl)prop-2-enoate —— C18H14ClNO6
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl (E)-3-(3-chlorophenyl)prop-2-enoate
—— (6R)-8-chloro-6-(4-methylpiperazin-1-yl)-5,6-dihydro-[1]benzothiepino[2,3-b]pyridine —— C18H20ClN3S
(6R)-8-chloro-6-(4-methylpiperazin-1-yl)-5,6-dihydro-[1]benzothiepino[2,3-b]pyridine
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3R)-3-acetamido-3-(4-chlorophenyl)propanoate —— C21H20ClN3O4
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3R)-3-acetamido-3-(4-chlorophenyl)propanoate
—— (6S)-6-(4-methylpiperazin-1-yl)-5,6-dihydro-[1]benzothiepino[2,3-b]pyridine —— C18H21N3S
(6S)-6-(4-methylpiperazin-1-yl)-5,6-dihydro-[1]benzothiepino[2,3-b]pyridine
—— (6E)-2-bromo-4-chloro-6-[[3-(5-ethyl-1,3-benzoxazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C22H16BrClN2O2
(6E)-2-bromo-4-chloro-6-[[3-(5-ethyl-1,3-benzoxazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-6-[(2,4-dimethylphenyl)hydrazinylidene]-5-oxonaphthalene-1-sulfonic acid —— C18H16N2O4S
(6E)-6-[(2,4-dimethylphenyl)hydrazinylidene]-5-oxonaphthalene-1-sulfonic acid
—— 6-[[(Z)-[3-methyl-1-(4-methylphenyl)-5-oxopyrazol-4-ylidene]methyl]amino]-6-azatetracyclo[6.5.2.04,15.011,14]pentadeca-1(14),2,4(15),8,10-pentaene-5,7-dione —— C26H20N4O3
6-[[(Z)-[3-methyl-1-(4-methylphenyl)-5-oxopyrazol-4-ylidene]methyl]amino]-6-azatetracyclo[6.5.2.04,15.011,14]pentadeca-1(14),2,4(15),8,10-pentaene-5,7-dione
—— (6E)-6-[[2-bis(4-tert-butylphenoxy)phosphinothioylhydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C27H33N2O3PS
(6E)-6-[[2-bis(4-tert-butylphenoxy)phosphinothioylhydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-2-methoxy-6-[[2-methyl-2-(6-nitro-1,1-dioxo-1,2-benzothiazol-3-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C16H14N4O6S
(6Z)-2-methoxy-6-[[2-methyl-2-(6-nitro-1,1-dioxo-1,2-benzothiazol-3-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3S)-3-acetamido-3-(4-chlorophenyl)propanoate —— C21H20ClN3O4
(6-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (3S)-3-acetamido-3-(4-chlorophenyl)propanoate
—— 6-ethyl-3-[(S)-[4-[(2-methoxyphenyl)methyl]piperazin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C30H37N7O3
6-ethyl-3-[(S)-[4-[(2-methoxyphenyl)methyl]piperazin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-ethyl-3-[(R)-[4-[(2-methoxyphenyl)methyl]piperazin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C30H37N7O3
6-ethyl-3-[(R)-[4-[(2-methoxyphenyl)methyl]piperazin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-acetyl-2-[(3R)-3-(4-aminophenyl)sulfanyl-2,5-dioxopyrrolidin-1-yl]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonitrile —— C20H18N4O3S2
6-acetyl-2-[(3R)-3-(4-aminophenyl)sulfanyl-2,5-dioxopyrrolidin-1-yl]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonitrile
—— (6Z)-6-[(4-bromophenyl)hydrazinylidene]-3,4-dimethylcyclohexa-2,4-dien-1-one —— C14H13BrN2O
(6Z)-6-[(4-bromophenyl)hydrazinylidene]-3,4-dimethylcyclohexa-2,4-dien-1-one
—— (6Z)-6-{4-[2-(4-bromophenoxy)ethoxy]-3-chloro-5-methoxybenzylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H22BrClN4O4S
(6Z)-6-{4-[2-(4-bromophenoxy)ethoxy]-3-chloro-5-methoxybenzylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[4-(5,6-dimethyl-1,3-benzoxazol-2-yl)anilino]methylidene]-2-methylcyclohexa-2,4-dien-1-one —— C23H20N2O2
(6E)-6-[[4-(5,6-dimethyl-1,3-benzoxazol-2-yl)anilino]methylidene]-2-methylcyclohexa-2,4-dien-1-one
—— 6-[(S)-[4-[(R)-(6-hydroxy-1,3-benzodioxol-5-yl)-(3-hydroxy-4-methoxyphenyl)methyl]piperazin-1-yl]-(3-hydroxy-4-methoxyphenyl)methyl]-1,3-benzodioxol-5-ol —— C34H34N2O10
6-[(S)-[4-[(R)-(6-hydroxy-1,3-benzodioxol-5-yl)-(3-hydroxy-4-methoxyphenyl)methyl]piperazin-1-yl]-(3-hydroxy-4-methoxyphenyl)methyl]-1,3-benzodioxol-5-ol
—— 6-[(R)-[4-[(S)-(6-hydroxy-1,3-benzodioxol-5-yl)-(2-hydroxy-3-methoxyphenyl)methyl]piperazin-1-yl]-(2-hydroxy-3-methoxyphenyl)methyl]-1,3-benzodioxol-5-ol —— C34H34N2O10
6-[(R)-[4-[(S)-(6-hydroxy-1,3-benzodioxol-5-yl)-(2-hydroxy-3-methoxyphenyl)methyl]piperazin-1-yl]-(2-hydroxy-3-methoxyphenyl)methyl]-1,3-benzodioxol-5-ol
—— 6-[(R)-[4-[(R)-(6-hydroxy-1,3-benzodioxol-5-yl)-(4-hydroxy-3-methoxyphenyl)methyl]piperazin-1-yl]-(4-hydroxy-3-methoxyphenyl)methyl]-1,3-benzodioxol-5-ol —— C34H34N2O10
6-[(R)-[4-[(R)-(6-hydroxy-1,3-benzodioxol-5-yl)-(4-hydroxy-3-methoxyphenyl)methyl]piperazin-1-yl]-(4-hydroxy-3-methoxyphenyl)methyl]-1,3-benzodioxol-5-ol
—— 6-[(R)-(4-chlorophenyl)-[4-[(R)-(4-chlorophenyl)-(6-hydroxy-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl]methyl]-1,3-benzodioxol-5-ol —— C32H28Cl2N2O6
6-[(R)-(4-chlorophenyl)-[4-[(R)-(4-chlorophenyl)-(6-hydroxy-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl]methyl]-1,3-benzodioxol-5-ol
—— 6-[(R)-[4-(dimethylamino)phenyl]-[4-[(R)-[4-(dimethylamino)phenyl]-(6-hydroxy-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl]methyl]-1,3-benzodioxol-5-ol —— C36H40N4O6
6-[(R)-[4-(dimethylamino)phenyl]-[4-[(R)-[4-(dimethylamino)phenyl]-(6-hydroxy-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl]methyl]-1,3-benzodioxol-5-ol
—— 6-[(S)-[4-[(S)-(6-hydroxy-1,3-benzodioxol-5-yl)-(2-hydroxy-3-methoxyphenyl)methyl]piperazin-1-yl]-(2-hydroxy-3-methoxyphenyl)methyl]-1,3-benzodioxol-5-ol —— C34H34N2O10
6-[(S)-[4-[(S)-(6-hydroxy-1,3-benzodioxol-5-yl)-(2-hydroxy-3-methoxyphenyl)methyl]piperazin-1-yl]-(2-hydroxy-3-methoxyphenyl)methyl]-1,3-benzodioxol-5-ol
—— 6-chloro-3-[(5R)-1-[2-(4-methylpiperazin-1-yl)acetyl]-5-phenylpyrazolidin-3-ylidene]-4-phenylquinolin-2-one —— C31H30ClN5O2
6-chloro-3-[(5R)-1-[2-(4-methylpiperazin-1-yl)acetyl]-5-phenylpyrazolidin-3-ylidene]-4-phenylquinolin-2-one
—— (6E)-3-benzyl-6-[[[2-(2-fluorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C27H19FN2O2
(6E)-3-benzyl-6-[[[2-(2-fluorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-ethyl 8-methyl 5-amino-2-(3-bromobenzylidene)-7-(3-bromophenyl)-3-oxo-2,3-dihydro-7H-[1,3]thiazolo[3,2-a]pyridine-6,8-dicarboxylate —— C25H20Br2N2O5S
6-ethyl 8-methyl 5-amino-2-(3-bromobenzylidene)-7-(3-bromophenyl)-3-oxo-2,3-dihydro-7H-[1,3]thiazolo[3,2-a]pyridine-6,8-dicarboxylate
—— (6E)-4-bromo-6-[[(3-chloro-1-adamantyl)methylamino]methylidene]cyclohexa-2,4-dien-1-one —— C18H21BrClNO
(6E)-4-bromo-6-[[(3-chloro-1-adamantyl)methylamino]methylidene]cyclohexa-2,4-dien-1-one
—— (6S,7R)-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-7-[[(2R)-2-(4-nitropyrazol-1-yl)propanoyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C16H17N9O6S2
(6S,7R)-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-7-[[(2R)-2-(4-nitropyrazol-1-yl)propanoyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,7S)-7-[[(2R)-2-(5-methyl-3-nitropyrazol-1-yl)propanoyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C17H19N9O6S2
(6S,7S)-7-[[(2R)-2-(5-methyl-3-nitropyrazol-1-yl)propanoyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— (6S,7R)-7-[[(2R)-2-(5-methyl-3-nitropyrazol-1-yl)propanoyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C17H19N9O6S2
(6S,7R)-7-[[(2R)-2-(5-methyl-3-nitropyrazol-1-yl)propanoyl]amino]-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 6-(4-methoxyphenyl)-N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C19H24N6O
6-(4-methoxyphenyl)-N-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— (6E)-4-bromo-6-[[4-[4-[(6-nitro-1,3-benzodioxol-5-yl)methylideneamino]phenyl]sulfonylanilino]methylidene]cyclohexa-2,4-dien-1-one —— C27H18BrN3O7S
(6E)-4-bromo-6-[[4-[4-[(6-nitro-1,3-benzodioxol-5-yl)methylideneamino]phenyl]sulfonylanilino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-(trifluoromethyl)-3-[(2S)-2-[[3-(trifluoromethyl)phenoxy]methyl]morpholine-4-carbonyl]-1H-pyridin-2-one —— C19H16F6N2O4
6-(trifluoromethyl)-3-[(2S)-2-[[3-(trifluoromethyl)phenoxy]methyl]morpholine-4-carbonyl]-1H-pyridin-2-one