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—— (6E)-6-[4-(2,4-dimethyl-1,3-thiazol-5-yl)-1,2-dihydropyrazol-3-ylidene]-5-hydroxy-3-methylcyclohexa-2,4-dien-1-one —— C15H15N3O2S
(6E)-6-[4-(2,4-dimethyl-1,3-thiazol-5-yl)-1,2-dihydropyrazol-3-ylidene]-5-hydroxy-3-methylcyclohexa-2,4-dien-1-one
—— (6R)-1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C25H29N3O3
(6R)-1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-(cyclopentanecarbonyl)-2-[(2R)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H32N4O3
6-(cyclopentanecarbonyl)-2-[(2R)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-1-[(3S)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C25H29N3O3
(6S)-1-[(3S)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-(2-methoxyacetyl)-2-[(2R)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H28N4O4
6-(2-methoxyacetyl)-2-[(2R)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-methyl-1'-[1-(pyridin-2-ylmethyl)piperidine-4-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C26H31N3O3
6-methyl-1'-[1-(pyridin-2-ylmethyl)piperidine-4-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— (6R)-1-(3-methoxypropanoyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C23H28N2O3
(6R)-1-(3-methoxypropanoyl)-6-[[4-(3-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-(4-methylcyclohexyl)-2-[(2S)-1-[2-(3-methylphenyl)acetyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C27H36N4O2
6-(4-methylcyclohexyl)-2-[(2S)-1-[2-(3-methylphenyl)acetyl]pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-methyl-3-[[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]chromen-4-one —— C23H22N4O2
6-methyl-3-[[(1R,12S)-7-methyl-4,8,9,15-tetrazatetracyclo[10.2.1.02,10.05,9]pentadeca-2(10),3,5,7-tetraen-15-yl]methyl]chromen-4-one
—— (6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one —— C25H25N3O2
(6S)-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
—— 6-methyl-1'-(3-pyrimidin-2-yloxybenzoyl)spiro[3H-chromene-2,4'-piperidine]-4-one —— C25H23N3O4
6-methyl-1'-(3-pyrimidin-2-yloxybenzoyl)spiro[3H-chromene-2,4'-piperidine]-4-one
—— (6Z)-2-(2-chlorophenyl)-6-[[1-[(4-chlorophenyl)methyl]-2-methylindol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H19Cl2N5OS
(6Z)-2-(2-chlorophenyl)-6-[[1-[(4-chlorophenyl)methyl]-2-methylindol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-1-(5-methylthiophene-2-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C24H24N2O2S
(6S)-1-(5-methylthiophene-2-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-methyl-1'-[(2S)-2-(4-oxoquinazolin-3-yl)propanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C25H25N3O4
6-methyl-1'-[(2S)-2-(4-oxoquinazolin-3-yl)propanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 6-(5-methylthiophene-2-carbonyl)-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H23N5O3S
6-(5-methylthiophene-2-carbonyl)-2-[(2R)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-1-(5-methylthiophene-2-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C24H24N2O2S
(6S)-1-(5-methylthiophene-2-carbonyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-methyl-1-[[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one —— C21H23F3N4O
6-methyl-1-[[(2S)-1-[(1-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]methyl]-2-(trifluoromethyl)quinolin-4-one
—— (6Z)-4-chloro-6-[5-(1,1,2,2-tetrafluoroethyl)-1,2-oxazol-3-ylidene]cyclohexa-2,4-dien-1-one —— C11H6ClF4NO2
(6Z)-4-chloro-6-[5-(1,1,2,2-tetrafluoroethyl)-1,2-oxazol-3-ylidene]cyclohexa-2,4-dien-1-one
—— (6S)-6-[[4-(4-methoxyphenyl)phenyl]methyl]-1-(5-methylthiophene-2-carbonyl)-1,4-diazepan-5-one —— C25H26N2O3S
(6S)-6-[[4-(4-methoxyphenyl)phenyl]methyl]-1-(5-methylthiophene-2-carbonyl)-1,4-diazepan-5-one
—— (6E)-6-{[1-(2-ethylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-hexyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H31N5OS
(6E)-6-{[1-(2-ethylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-hexyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6R)-1-[2-(4-methoxyphenyl)acetyl]-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C28H30N2O3
(6R)-1-[2-(4-methoxyphenyl)acetyl]-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-1-(3-methylbutanoyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C24H30N2O2
(6S)-1-(3-methylbutanoyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-6-[[2-(4-methylphenyl)phenyl]methyl]-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)-1,4-diazepan-5-one —— C26H30N4O2
(6R)-6-[[2-(4-methylphenyl)phenyl]methyl]-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)-1,4-diazepan-5-one
—— 6-methyl-N-[(1S,5S,6R,7S)-7-phenyl-6-bicyclo[3.2.0]heptanyl]pyridine-3-carboxamide —— C20H22N2O
6-methyl-N-[(1S,5S,6R,7S)-7-phenyl-6-bicyclo[3.2.0]heptanyl]pyridine-3-carboxamide
—— 6-(3-fluoro-4-methylphenyl)sulfonyl-2-[(3S)-1-methylpyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H23FN4O2S
6-(3-fluoro-4-methylphenyl)sulfonyl-2-[(3S)-1-methylpyrrolidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-(3-fluoro-4-methylphenyl)sulfonyl-2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H23FN4O2S
6-(3-fluoro-4-methylphenyl)sulfonyl-2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6-methylpyridin-3-yl)-[(2R)-2-[5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone —— C21H22F3N5O
(6-methylpyridin-3-yl)-[(2R)-2-[5-propan-2-yl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]pyrrolidin-1-yl]methanone
—— 6-methyl-2-[(3S)-1-(4-methylphenyl)sulfonylpiperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H26N4O2S
6-methyl-2-[(3S)-1-(4-methylphenyl)sulfonylpiperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6R)-1-benzoyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H26N2O2
(6R)-1-benzoyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-[(3,4-dimethylphenyl)methyl]-2-[(2S)-1-methylpiperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C22H30N4
6-[(3,4-dimethylphenyl)methyl]-2-[(2S)-1-methylpiperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6R)-1-(cyclobutanecarbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C24H28N2O2
(6R)-1-(cyclobutanecarbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-1-[2-(4-methoxyphenyl)acetyl]-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C28H30N2O3
(6S)-1-[2-(4-methoxyphenyl)acetyl]-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-chloro-N-[(1S,5R,6S)-3-(4-methylphenyl)sulfonyl-3-azabicyclo[3.2.0]heptan-6-yl]-1H-indole-2-carboxamide —— C22H22ClN3O3S
6-chloro-N-[(1S,5R,6S)-3-(4-methylphenyl)sulfonyl-3-azabicyclo[3.2.0]heptan-6-yl]-1H-indole-2-carboxamide
—— (6S)-1-(2-methoxyacetyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C22H26N2O3
(6S)-1-(2-methoxyacetyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-(4-methylcyclohexyl)-2-[(3R)-1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H35N5O2
6-(4-methylcyclohexyl)-2-[(3R)-1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopentanecarbonyl)-2-[(2S)-1-(6-methylpyridine-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31N5O3
6-(cyclopentanecarbonyl)-2-[(2S)-1-(6-methylpyridine-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(2-methoxyacetyl)-2-[(2S)-1-[2-(4-methylphenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H30N4O4
6-(2-methoxyacetyl)-2-[(2S)-1-[2-(4-methylphenyl)acetyl]piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— [(6S,7S,8R)-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-yl]hydrazine —— C20H24N2O6
[(6S,7S,8R)-7-methyl-8-(3,4,5-trimethoxyphenyl)-7,8-dihydro-6H-[1,3]dioxolo[4,5-g]chromen-6-yl]hydrazine
—— (6S)-1-[2-(2-methoxy-5-methylphenyl)acetyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O3
(6S)-1-[2-(2-methoxy-5-methylphenyl)acetyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-methyl-2-[2-[(3R)-3-[3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-6-yl]piperidin-1-yl]-2-oxoethyl]pyridazin-3-one —— C20H20F3N5O3
6-methyl-2-[2-[(3R)-3-[3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-6-yl]piperidin-1-yl]-2-oxoethyl]pyridazin-3-one
—— (6R)-6-[[2-(2,4-dimethylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C20H24N2O
(6R)-6-[[2-(2,4-dimethylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-methyl-3-[(3R)-3-[3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-6-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C20H19F3N4O3
6-methyl-3-[(3R)-3-[3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-6-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— 6-chloro-3-[3-[(4S)-2-(2-ethoxyphenyl)imino-4-methyl-1,3-thiazolidin-3-yl]-3-oxopropyl]-1,3-benzoxazol-2-one —— C22H22ClN3O4S
6-chloro-3-[3-[(4S)-2-(2-ethoxyphenyl)imino-4-methyl-1,3-thiazolidin-3-yl]-3-oxopropyl]-1,3-benzoxazol-2-one
—— (6-methoxy-2-methylquinolin-3-yl)-[(2R)-2-(2-methylpyrazolo[1,5-a]pyrimidin-7-yl)pyrrolidin-1-yl]methanone —— C23H23N5O2
(6-methoxy-2-methylquinolin-3-yl)-[(2R)-2-(2-methylpyrazolo[1,5-a]pyrimidin-7-yl)pyrrolidin-1-yl]methanone
—— 6-[1-[(2-methoxy-4-methylphenyl)methyl]piperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C24H29N5O
6-[1-[(2-methoxy-4-methylphenyl)methyl]piperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— (6R)-6-[[2-(2,4-dimethylphenyl)phenyl]methyl]-1-propan-2-ylsulfonyl-1,4-diazepan-5-one —— C23H30N2O3S
(6R)-6-[[2-(2,4-dimethylphenyl)phenyl]methyl]-1-propan-2-ylsulfonyl-1,4-diazepan-5-one
—— 6-[1-(2-fluoro-5-methylphenyl)sulfonylpiperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine —— C22H24FN5O2S
6-[1-(2-fluoro-5-methylphenyl)sulfonylpiperidin-4-yl]-N-methyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-(4-methoxyphenyl)-3-[(2S)-2-(2-methylpyrazolo[1,5-a]pyrimidin-7-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one —— C24H23N5O3
6-(4-methoxyphenyl)-3-[(2S)-2-(2-methylpyrazolo[1,5-a]pyrimidin-7-yl)pyrrolidine-1-carbonyl]-1H-pyridin-2-one
—— 6-methyl-3-[(3R)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidine-1-carbonyl]-1H-pyridin-2-one —— C22H23F3N4O3
6-methyl-3-[(3R)-3-[6-propan-2-yl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridin-3-yl]piperidine-1-carbonyl]-1H-pyridin-2-one
—— 6-(cyclopropanecarbonyl)-2-[(2S)-1-(4-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H28N4O3
6-(cyclopropanecarbonyl)-2-[(2S)-1-(4-methylbenzoyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one