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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-4-ethyl-1-[(2R)-oxolane-2-carbonyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H29N3O3
(6R)-4-ethyl-1-[(2R)-oxolane-2-carbonyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(3-methylpyridine-4-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H27N3O2S
(6R)-4-ethyl-1-(3-methylpyridine-4-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(1-methylimidazole-2-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2
(6S)-4-ethyl-1-(1-methylimidazole-2-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(1H-pyrazole-5-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C22H24N4O2S
(6R)-4-ethyl-1-(1H-pyrazole-5-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N5O2
(6S)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N5O2
(6R)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(1-propan-2-ylpyrazole-4-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O2
(6R)-4-ethyl-1-(1-propan-2-ylpyrazole-4-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(2,4-dimethylpyrimidine-5-carbonyl)-4-ethyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2S
(6S)-1-(2,4-dimethylpyrimidine-5-carbonyl)-4-ethyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H32N2O3S
(6S)-4-ethyl-1-[3-[(2R)-oxolan-2-yl]propanoyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(cyclopropylmethyl)-4-ethyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H29N3O
(6R)-1-(cyclopropylmethyl)-4-ethyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(3R)-1-ethyl-5-oxopyrrolidine-3-carbonyl]-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H31N3O3
(6R)-1-[(3R)-1-ethyl-5-oxopyrrolidine-3-carbonyl]-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(2-methoxyphenyl)methyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H31N3O2
(6R)-4-ethyl-1-[(2-methoxyphenyl)methyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O2
(6S)-4-ethyl-1-(5-propan-2-yl-1H-pyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N5O2
(6S)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-[3-(tetrazol-1-yl)propanoyl]-1,4-diazepan-5-one —— C25H30N6O2
(6R)-4-ethyl-6-[[2-(4-methylphenyl)phenyl]methyl]-1-[3-(tetrazol-1-yl)propanoyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(2R)-2-piperidin-1-ylpropanoyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H36N4O2
(6S)-4-ethyl-1-[(2R)-2-piperidin-1-ylpropanoyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-ethyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H27N3O3S
(6R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-ethyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O2
(6S)-4-ethyl-1-(1-methylimidazole-4-carbonyl)-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(pyridin-2-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O
(6R)-4-ethyl-1-(pyridin-2-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(5-oxo-1,2-dihydro-1,2,4-triazole-3-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C21H23N5O3S
(6R)-4-ethyl-1-(5-oxo-1,2-dihydro-1,2,4-triazole-3-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-ethyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H27N3O3S
(6S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-4-ethyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[2-(4-fluorophenyl)acetyl]-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H28FN3O2
(6S)-4-ethyl-1-[2-(4-fluorophenyl)acetyl]-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(2R)-oxolane-2-carbonyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H30N2O3
(6S)-4-ethyl-1-[(2R)-oxolane-2-carbonyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(2-methylpyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H27N5O2
(6S)-4-ethyl-1-(2-methylpyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[2-(4-methyltriazol-1-yl)acetyl]-1,4-diazepan-5-one —— C26H31N5O2
(6R)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[2-(4-methyltriazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C24H26FN5O2
(6S)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H33N5O2
(6R)-4-ethyl-1-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(2-pyridin-2-yloxyacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H27N3O3S
(6R)-4-ethyl-1-(2-pyridin-2-yloxyacetyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(3-fluorobenzoyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H26FN3O2
(6S)-4-ethyl-1-(3-fluorobenzoyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one —— C26H26FN3O2
(6R)-4-ethyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(pyridin-2-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O
(6R)-4-ethyl-1-(pyridin-2-ylmethyl)-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one —— C26H30N4O3
(6S)-4-ethyl-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[3-(5-methylpyrazol-1-yl)propanoyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H32N4O2
(6R)-4-ethyl-1-[3-(5-methylpyrazol-1-yl)propanoyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[2-(4-methyltriazol-1-yl)acetyl]-1,4-diazepan-5-one —— C26H31N5O2
(6S)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-[2-(4-methyltriazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(3-pyrazol-1-ylpropanoyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6R)-4-ethyl-1-(3-pyrazol-1-ylpropanoyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-[2-(4-methyltriazol-1-yl)acetyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6R)-4-ethyl-1-[2-(4-methyltriazol-1-yl)acetyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one —— C25H28N4O2
(6S)-4-ethyl-6-[[4-(3-methylphenyl)phenyl]methyl]-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(1-methylpyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H27N5O2
(6R)-4-ethyl-1-(1-methylpyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H31N5O2
(6R)-1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-4-ethyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C24H26FN5O2
(6R)-4-ethyl-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(1-methylpyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H27N5O2
(6S)-4-ethyl-1-(1-methylpyrazole-3-carbonyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(pyridin-3-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H28N4O
(6R)-4-ethyl-1-(pyridin-3-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[(3S)-1-ethyl-5-oxopyrrolidine-3-carbonyl]-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C26H31N3O3
(6S)-1-[(3S)-1-ethyl-5-oxopyrrolidine-3-carbonyl]-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[3-(tetrazol-1-yl)propanoyl]-1,4-diazepan-5-one —— C25H30N6O2
(6R)-4-ethyl-6-[[3-(2-methylphenyl)phenyl]methyl]-1-[3-(tetrazol-1-yl)propanoyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[2-(4-methyltriazol-1-yl)acetyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H29N5O2
(6S)-4-ethyl-1-[2-(4-methyltriazol-1-yl)acetyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-(2-phenylacetyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O2
(6S)-4-ethyl-1-(2-phenylacetyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(6-methoxypyridine-3-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H29N3O3
(6R)-4-ethyl-1-(6-methoxypyridine-3-carbonyl)-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[(3R)-1-[(1-ethylpyrazol-4-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one —— C19H23N5OS
6-[(3R)-1-[(1-ethylpyrazol-4-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one
—— (6R)-1-(3,3-dimethylbutanoyl)-4-ethyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H33N3O2
(6R)-1-(3,3-dimethylbutanoyl)-4-ethyl-6-[(3-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-ethyl-1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H29N3O3S
(6S)-4-ethyl-1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one