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—— 6-[(3-propan-2-yloxyphenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C21H28N4O
6-[(3-propan-2-yloxyphenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[1-(1-propan-2-ylpiperidine-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C22H30N4O2
6-[1-(1-propan-2-ylpiperidine-4-carbonyl)piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-propan-2-yl-2-[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H24N4O2S
6-propan-2-yl-2-[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-1-(3-methylbutanoyl)-4-prop-2-enyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H31N3O2
(6S)-1-(3-methylbutanoyl)-4-prop-2-enyl-6-[(4-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-propan-2-yl-2-[(2R)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H25N5O2
6-propan-2-yl-2-[(2R)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-(3-methylbutanoyl)-4-prop-2-enyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H31N3O2
(6R)-1-(3-methylbutanoyl)-4-prop-2-enyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(cyclohexylmethyl)-2-[(2S)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H31N5O2
6-(cyclohexylmethyl)-2-[(2S)-1-(pyridine-4-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexanecarbonyl)-2-[(2S)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31N5O3
6-(cyclohexanecarbonyl)-2-[(2S)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexylmethyl)-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H33N5O2
6-(cyclohexylmethyl)-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3-Hydroxyphenyl)methyl]-2-pyridin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C19H18N4O2
6-[(3-Hydroxyphenyl)methyl]-2-pyridin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexylmethyl)-2-[(2R)-1-(2-pyridin-2-ylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C26H35N5O2
6-(cyclohexylmethyl)-2-[(2R)-1-(2-pyridin-2-ylacetyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-cyclohexyl-2-[(2S)-1-(pyrazine-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H30N6O2
6-cyclohexyl-2-[(2S)-1-(pyrazine-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-methyl-1-(3-methylbutanoyl)-1,4-diazepan-5-one —— C25H32N2O3
(6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-methyl-1-(3-methylbutanoyl)-1,4-diazepan-5-one
—— 6-fluoro-2-[(3R)-1-(pyridine-2-carbonyl)piperidin-3-yl]quinoline-3-carboxamide —— C21H19FN4O2
6-fluoro-2-[(3R)-1-(pyridine-2-carbonyl)piperidin-3-yl]quinoline-3-carboxamide
—— 6-(2-cyclopentylacetyl)-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31N5O3
6-(2-cyclopentylacetyl)-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclopentanecarbonyl)-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H29N5O3
6-(cyclopentanecarbonyl)-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3R)-1-[[1-(3-hydroxypropyl)indol-3-yl]methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one —— C25H28N4O2S
6-[(3R)-1-[[1-(3-hydroxypropyl)indol-3-yl]methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one
—— 6-(cyclopropanecarbonyl)-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C22H25N5O3
6-(cyclopropanecarbonyl)-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3S)-1-[[1-(3-hydroxypropyl)indol-3-yl]methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one —— C25H28N4O2S
6-[(3S)-1-[[1-(3-hydroxypropyl)indol-3-yl]methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one
—— (6S)-6-[(4-pyridin-4-ylphenyl)methyl]-1-(quinolin-4-ylmethyl)-1,4-diazepan-5-one —— C27H26N4O
(6S)-6-[(4-pyridin-4-ylphenyl)methyl]-1-(quinolin-4-ylmethyl)-1,4-diazepan-5-one
—— (6R)-1-(cyclopentanecarbonyl)-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N2O2
(6R)-1-(cyclopentanecarbonyl)-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclopentanecarbonyl)-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N2O2
(6S)-1-(cyclopentanecarbonyl)-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-benzoyl-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H24N2O2
(6R)-1-benzoyl-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-[3-(2-oxopyridin-1-yl)propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H27N3O3
(6S)-1-[3-(2-oxopyridin-1-yl)propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[2-(3-fluorophenyl)acetyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H25FN2O2
(6R)-1-[2-(3-fluorophenyl)acetyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-Benzyl-2-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H29N5O
6-Benzyl-2-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[[(3S)-1-benzylpiperidin-3-yl]methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H28N6O
6-[[(3S)-1-benzylpiperidin-3-yl]methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-6-[(2-phenylphenyl)methyl]-1-(3-phenylpropanoyl)-1,4-diazepan-5-one —— C27H28N2O2
(6R)-6-[(2-phenylphenyl)methyl]-1-(3-phenylpropanoyl)-1,4-diazepan-5-one
—— 6-cyclopentyl-2-[(3R)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H32N4O2
6-cyclopentyl-2-[(3R)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-(3-phenylpropyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O
(6R)-1-(3-phenylpropyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-1,4-diazepan-5-one —— C21H20FN5O3
(6R)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(5-oxo-1,4-dihydro-1,2,4-triazole-3-carbonyl)-1,4-diazepan-5-one
—— (6S)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one —— C24H22FN3O2
(6S)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(pyridine-2-carbonyl)-1,4-diazepan-5-one
—— (6R)-6-(4-chlorophenyl)-1,2,3,4,5,6-hexahydro-2,5-benzodiazocine —— C16H17ClN2
(6R)-6-(4-chlorophenyl)-1,2,3,4,5,6-hexahydro-2,5-benzodiazocine
—— (6S)-3-chloro-6-(4-methylpiperazin-1-yl)-5,6-dihydrobenzo[b][1]benzothiepin-8-ol —— C19H21ClN2OS
(6S)-3-chloro-6-(4-methylpiperazin-1-yl)-5,6-dihydrobenzo[b][1]benzothiepin-8-ol
—— (6R)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(2-phenylacetyl)-1,4-diazepan-5-one —— C26H25FN2O2
(6R)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(2-phenylacetyl)-1,4-diazepan-5-one
—— (6R)-1-benzoyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1,4-diazepan-5-one —— C25H23FN2O2
(6R)-1-benzoyl-6-[[3-(4-fluorophenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-1-benzoyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H22N2O2S
(6R)-1-benzoyl-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[(2-fluorophenyl)methyl]-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H24FN5O2
6-[(2-fluorophenyl)methyl]-2-[(2S)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2-chlorophenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C18H21ClN4
6-[(2-chlorophenyl)methyl]-2-[(2R)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[(2-chlorophenyl)methyl]-2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H23ClN4
6-[(2-chlorophenyl)methyl]-2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6S)-6-(4-chlorophenyl)-1,2,3,4,5,6-hexahydro-2,5-benzodiazocine —— C16H17ClN2
(6S)-6-(4-chlorophenyl)-1,2,3,4,5,6-hexahydro-2,5-benzodiazocine
—— (6R)-1-(3-fluorobenzoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H21FN2O2S
(6R)-1-(3-fluorobenzoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[(2-fluorophenyl)methyl]-2-[(2S)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H23FN4O2S
6-[(2-fluorophenyl)methyl]-2-[(2S)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-(cyclohexylmethyl)-2-[(2S)-1-(2-fluorobenzoyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H31FN4O2
6-(cyclohexylmethyl)-2-[(2S)-1-(2-fluorobenzoyl)pyrrolidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-1-[(2-chlorophenyl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H24ClN3O
(6R)-1-[(2-chlorophenyl)methyl]-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(cyclopropanecarbonyl)-2-[(3S)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C23H27FN4O2
6-(cyclopropanecarbonyl)-2-[(3S)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-Fluoro-2-[1-(pyridin-4-ylmethyl)piperidin-4-yl]quinolin-3-amine —— C20H21FN4
6-Fluoro-2-[1-(pyridin-4-ylmethyl)piperidin-4-yl]quinolin-3-amine
—— (6R)-4-N-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine —— C19H18ClN5
(6R)-4-N-(4-chlorophenyl)-2-pyridin-3-yl-5,6,7,8-tetrahydroquinazoline-4,6-diamine
—— (6R)-1-[(2S)-oxane-2-carbonyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H27N3O3
(6R)-1-[(2S)-oxane-2-carbonyl]-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-(cyclopropanecarbonyl)-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C21H24N4O3S
6-(cyclopropanecarbonyl)-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one