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—— (6R)-1-N-[(4-methoxyphenyl)methyl]-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H35N5O4
(6R)-1-N-[(4-methoxyphenyl)methyl]-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-1-N-[(4-chlorophenyl)methyl]-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H32ClN5O3
(6R)-1-N-[(4-chlorophenyl)methyl]-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-6-N-benzyl-1-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H28FN5O3
(6S)-6-N-benzyl-1-N-[(4-fluorophenyl)methyl]-6-methyl-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-1-N-[(3-bromophenyl)methyl]-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H32BrN5O3
(6S)-1-N-[(3-bromophenyl)methyl]-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-1-N-benzyl-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H33N5O3
(6R)-1-N-benzyl-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6E)-6-[[[(3E)-3-(3H-1,3-benzothiazol-2-ylidene)-4-oxocyclohexa-1,5-dien-1-yl]amino]methylidene]-4,5-dibromo-2-methoxycyclohexa-2,4-dien-1-one —— C21H14Br2N2O3S
(6E)-6-[[[(3E)-3-(3H-1,3-benzothiazol-2-ylidene)-4-oxocyclohexa-1,5-dien-1-yl]amino]methylidene]-4,5-dibromo-2-methoxycyclohexa-2,4-dien-1-one
—— (6S)-1-N-(1,3-benzodioxol-5-ylmethyl)-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H33N5O5
(6S)-1-N-(1,3-benzodioxol-5-ylmethyl)-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-1-N-[(4-fluorophenyl)methyl]-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C24H32FN5O3
(6R)-1-N-[(4-fluorophenyl)methyl]-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6R)-1-N-[2-(4-chlorophenyl)ethyl]-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C25H34ClN5O3
(6R)-1-N-[2-(4-chlorophenyl)ethyl]-6-methyl-6-N-(3-methylbutyl)-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6Z)-2-nitro-6-[(2-quinolin-8-ylhydrazinyl)methylidene]cyclohexa-2,4-dien-1-one —— C16H12N4O3
(6Z)-2-nitro-6-[(2-quinolin-8-ylhydrazinyl)methylidene]cyclohexa-2,4-dien-1-one
—— 6-[(5Z)-5-(2H-chromen-3-ylmethylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]hexanoic acid —— C19H19NO4S2
6-[(5Z)-5-(2H-chromen-3-ylmethylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]hexanoic acid
—— (6S)-6-methyl-6-N-(3-methylbutyl)-1-N-[2-(4-methylphenyl)ethyl]-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C26H37N5O3
(6S)-6-methyl-6-N-(3-methylbutyl)-1-N-[2-(4-methylphenyl)ethyl]-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6Z)-6-[[2,5-dimethyl-1-(4-propan-2-ylphenyl)pyrrol-3-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H30N6O3S
(6Z)-6-[[2,5-dimethyl-1-(4-propan-2-ylphenyl)pyrrol-3-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[(4-ethylphenyl)methylidene]-5-imino-2-[(3-methylphenoxy)methyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H20N4O2S
(6Z)-6-[(4-ethylphenyl)methylidene]-5-imino-2-[(3-methylphenoxy)methyl]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(2-cyclohexyliminopyridine-1-carbonyl)-2-[(3S)-1,1-dioxothiolan-3-yl]-4,5-dihydropyridazin-3-one —— C20H26N4O4S
6-(2-cyclohexyliminopyridine-1-carbonyl)-2-[(3S)-1,1-dioxothiolan-3-yl]-4,5-dihydropyridazin-3-one
—— (6Z)-2-(2-chlorophenyl)-6-(4-{2-[(4-chlorophenyl)sulfanyl]ethoxy}-3-ethoxybenzylidene)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H22Cl2N4O3S2
(6Z)-2-(2-chlorophenyl)-6-(4-{2-[(4-chlorophenyl)sulfanyl]ethoxy}-3-ethoxybenzylidene)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(2-cyclohexyliminopyridine-1-carbonyl)-2-[(3R)-1,1-dioxothiolan-3-yl]-4,5-dihydropyridazin-3-one —— C20H26N4O4S
6-(2-cyclohexyliminopyridine-1-carbonyl)-2-[(3R)-1,1-dioxothiolan-3-yl]-4,5-dihydropyridazin-3-one
—— 6-bromo-3-[2-[(2Z)-2-[(4-nitrophenyl)methylidene]hydrazinyl]-1,3-thiazol-5-yl]chromen-2-one —— C19H11BrN4O4S
6-bromo-3-[2-[(2Z)-2-[(4-nitrophenyl)methylidene]hydrazinyl]-1,3-thiazol-5-yl]chromen-2-one
—— 6-tert-butyl-2-[[(Z)-(5-methoxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonitrile —— C21H24N2O2S
6-tert-butyl-2-[[(Z)-(5-methoxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonitrile
—— (6S,10S)-N-[(4-chlorophenyl)methyl]-10-methyl-1,4-diazaspiro[5.5]undec-4-en-5-amine —— C17H24ClN3
(6S,10S)-N-[(4-chlorophenyl)methyl]-10-methyl-1,4-diazaspiro[5.5]undec-4-en-5-amine
—— (6Z)-4-hexyl-6-[1-(hydroxyamino)decylidene]-3-methoxycyclohexa-2,4-dien-1-one —— C23H39NO3
(6Z)-4-hexyl-6-[1-(hydroxyamino)decylidene]-3-methoxycyclohexa-2,4-dien-1-one
—— (6S)-N-cyclohexyl-6-phenyl-1,2,3,6-tetrahydropyrazin-5-amine —— C16H23N3
(6S)-N-cyclohexyl-6-phenyl-1,2,3,6-tetrahydropyrazin-5-amine
—— (6E)-2,4-dichloro-6-[[2-[2-nitro-4-(trifluoromethyl)phenyl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C14H8Cl2F3N3O3
(6E)-2,4-dichloro-6-[[2-[2-nitro-4-(trifluoromethyl)phenyl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— 6-[4-[(3S)-1-(3,4-dimethylphenyl)-5-oxopyrrolidine-3-carbonyl]piperazin-1-yl]sulfonyl-4H-1,4-benzoxazin-3-one —— C25H28N4O6S
6-[4-[(3S)-1-(3,4-dimethylphenyl)-5-oxopyrrolidine-3-carbonyl]piperazin-1-yl]sulfonyl-4H-1,4-benzoxazin-3-one
—— (6Z)-6-[[1-(4-butan-2-ylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-methylsulfanyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H25N5OS2
(6Z)-6-[[1-(4-butan-2-ylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-methylsulfanyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[4-[(3S)-5-oxo-1-phenylpyrrolidine-3-carbonyl]piperazin-1-yl]sulfonyl-4H-1,4-benzoxazin-3-one —— C23H24N4O6S
6-[4-[(3S)-5-oxo-1-phenylpyrrolidine-3-carbonyl]piperazin-1-yl]sulfonyl-4H-1,4-benzoxazin-3-one
—— (6Z)-6-[[2-(6-chloro-2-methylpyrimidin-4-yl)hydrazinyl]methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C13H13ClN4O2
(6Z)-6-[[2-(6-chloro-2-methylpyrimidin-4-yl)hydrazinyl]methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— (6Z)-5-imino-6-[[1-(2-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H20N6O2S
(6Z)-5-imino-6-[[1-(2-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-4-methoxy-6-[(3-methoxyanilino)methylidene]cyclohexa-2,4-dien-1-one —— C15H15NO3
(6E)-4-methoxy-6-[(3-methoxyanilino)methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-5-imino-6-{4-[2-(4-methylphenoxy)ethoxy]benzylidene}-2-(2-methylpropyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H26N4O3S
(6Z)-5-imino-6-{4-[2-(4-methylphenoxy)ethoxy]benzylidene}-2-(2-methylpropyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-N-cyclohexyl-6-(4-methylphenyl)-1,6-dihydro-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine —— C17H21N5O
(6S)-N-cyclohexyl-6-(4-methylphenyl)-1,6-dihydro-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
—— (6E)-6-({1-[2-(2-chlorophenoxy)ethyl]-1H-pyrrol-2-yl}methylidene)-5-imino-3-phenyl-5,6-dihydro-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C25H19ClN4O2S
(6E)-6-({1-[2-(2-chlorophenoxy)ethyl]-1H-pyrrol-2-yl}methylidene)-5-imino-3-phenyl-5,6-dihydro-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (6S,10R)-N-[(4-chlorophenyl)methyl]-10-methyl-1,4-diazaspiro[5.5]undec-4-en-5-amine —— C17H24ClN3
(6S,10R)-N-[(4-chlorophenyl)methyl]-10-methyl-1,4-diazaspiro[5.5]undec-4-en-5-amine
—— (6Z)-6-{3-chloro-5-ethoxy-4-[2-(4-methylphenoxy)ethoxy]benzylidene}-5-imino-2-(4-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C30H27ClN4O4S
(6Z)-6-{3-chloro-5-ethoxy-4-[2-(4-methylphenoxy)ethoxy]benzylidene}-5-imino-2-(4-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(3R)-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-5-[(2,4,5-trimethylphenyl)sulfonylamino]pyridine-3-carboxylic acid —— C25H34N4O4S
6-[(3R)-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-5-[(2,4,5-trimethylphenyl)sulfonylamino]pyridine-3-carboxylic acid
—— (6Z)-4,5-dibromo-2-ethoxy-6-[[3-(5-ethyl-1,3-benzoxazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C24H20Br2N2O3
(6Z)-4,5-dibromo-2-ethoxy-6-[[3-(5-ethyl-1,3-benzoxazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-Ethyl-7-hydroxy-4-methyl-8-[(4-methylpiperidin-1-ium-1-yl)methyl]chromen-2-one —— C19H26NO3+
6-Ethyl-7-hydroxy-4-methyl-8-[(4-methylpiperidin-1-ium-1-yl)methyl]chromen-2-one
—— (6Z)-2-(2-chlorophenyl)-5-imino-6-(3-methoxy-4-{2-[(4-methylphenyl)sulfanyl]ethoxy}benzylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H23ClN4O3S2
(6Z)-2-(2-chlorophenyl)-5-imino-6-(3-methoxy-4-{2-[(4-methylphenyl)sulfanyl]ethoxy}benzylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[(5-benzyl-1,3,4-thiadiazol-2-yl)amino]methylidene]-4-chloro-2-nitrocyclohexa-2,4-dien-1-one —— C16H11ClN4O3S
(6E)-6-[[(5-benzyl-1,3,4-thiadiazol-2-yl)amino]methylidene]-4-chloro-2-nitrocyclohexa-2,4-dien-1-one
—— (6Z)-5-imino-6-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methylidene)-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C20H18N4O2S2
(6Z)-5-imino-6-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methylidene)-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[5-(4-chlorophenyl)sulfanylfuran-2-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H18ClN5O4S2
(6Z)-6-[[5-(4-chlorophenyl)sulfanylfuran-2-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6,8-dimethyl-N-[4-[2-[(2S)-2-methylpiperidin-1-yl]ethylcarbamoyl]phenyl]-2,3-dihydropyrido[2,3-b][1,4]thiazine-1-carboxamide —— C25H33N5O2S
6,8-dimethyl-N-[4-[2-[(2S)-2-methylpiperidin-1-yl]ethylcarbamoyl]phenyl]-2,3-dihydropyrido[2,3-b][1,4]thiazine-1-carboxamide
—— (6R)-6-N-cyclopentyl-5-ethyl-2-N-(3-methoxypropyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C20H31N5O4
(6R)-6-N-cyclopentyl-5-ethyl-2-N-(3-methoxypropyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-cyclopentyl-2-N-[(2-ethoxyphenyl)methyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H35N5O4
(6R)-6-N-cyclopentyl-2-N-[(2-ethoxyphenyl)methyl]-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-2-N-(3-fluoro-4-methylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H32FN5O3
(6S)-5-butyl-6-N-cyclopentyl-2-N-(3-fluoro-4-methylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-5-butyl-6-N-cyclopentyl-6-methyl-2-N-(2-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H33N5O3
(6R)-5-butyl-6-N-cyclopentyl-6-methyl-2-N-(2-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-2-N-[2-(3-methylphenyl)ethyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C26H28FN5O3
(6R)-6-N-[(4-fluorophenyl)methyl]-5,6-dimethyl-2-N-[2-(3-methylphenyl)ethyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-N-cyclopentyl-5-ethyl-2-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C27H36N6O4
(6S)-N-cyclopentyl-5-ethyl-2-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-6-N-cyclopentyl-5-ethyl-6-methyl-4-oxo-2-N-(2-phenylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C24H31N5O3
(6S)-6-N-cyclopentyl-5-ethyl-6-methyl-4-oxo-2-N-(2-phenylethyl)-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6S)-5-butyl-6-N-cyclopentyl-6-methyl-2-N-(4-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C25H33N5O3
(6S)-5-butyl-6-N-cyclopentyl-6-methyl-2-N-(4-methylphenyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide