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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-(4-methylpiperidin-1-yl)sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]-2-pyridin-2-ylquinoline-4-carboxamide —— C26H30N4O4S
6-(4-methylpiperidin-1-yl)sulfonyl-N-[[(2R)-oxolan-2-yl]methyl]-2-pyridin-2-ylquinoline-4-carboxamide
—— (6E)-6-[1-(piperidin-1-ylamino)ethylidene]cyclohexa-2,4-dien-1-one —— C13H18N2O
(6E)-6-[1-(piperidin-1-ylamino)ethylidene]cyclohexa-2,4-dien-1-one
—— (6-bromonaphthalen-2-yl) (E)-3-(3-chlorophenyl)prop-2-enoate —— C19H12BrClO2
(6-bromonaphthalen-2-yl) (E)-3-(3-chlorophenyl)prop-2-enoate
—— 6-[(3R)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(2-phenylethyl)-1H-quinoline-4-carboxamide —— C24H27N3O4S
6-[(3R)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(2-phenylethyl)-1H-quinoline-4-carboxamide
—— 6-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(2-phenylethyl)-1H-quinoline-4-carboxamide —— C24H27N3O4S
6-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(2-phenylethyl)-1H-quinoline-4-carboxamide
—— 6-[(2R)-2-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(3-pyrrolidin-1-ylpropyl)-1H-quinoline-4-carboxamide —— C23H32N4O4S
6-[(2R)-2-methylpiperidin-1-yl]sulfonyl-2-oxo-N-(3-pyrrolidin-1-ylpropyl)-1H-quinoline-4-carboxamide
—— 6-(azepan-1-ylsulfonyl)-N-[(2R)-3-(diethylamino)-2-methylpropyl]-2-oxo-1H-quinoline-4-carboxamide —— C24H36N4O4S
6-(azepan-1-ylsulfonyl)-N-[(2R)-3-(diethylamino)-2-methylpropyl]-2-oxo-1H-quinoline-4-carboxamide
—— 6-[(2S)-2-ethylpiperidin-1-yl]sulfonyl-N-[2-(4-methylphenyl)ethyl]-2-oxo-1H-quinoline-4-carboxamide —— C26H31N3O4S
6-[(2S)-2-ethylpiperidin-1-yl]sulfonyl-N-[2-(4-methylphenyl)ethyl]-2-oxo-1H-quinoline-4-carboxamide
—— 6-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-[(2S)-4-phenylbutan-2-yl]-1H-quinoline-4-carboxamide —— C26H31N3O4S
6-[(3S)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-[(2S)-4-phenylbutan-2-yl]-1H-quinoline-4-carboxamide
—— 6-[2-[(5R)-5-hydroxy-1-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one —— C22H18F3N3O3S
6-[2-[(5R)-5-hydroxy-1-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one
—— (6R,9R)-9-(4-methylphenyl)-6-(4-phenylmethoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C35H29F3N2O3
(6R,9R)-9-(4-methylphenyl)-6-(4-phenylmethoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[2-[(5S)-1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-5-hydroxy-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one —— C21H15F4N3O2S
6-[2-[(5S)-1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-5-hydroxy-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one
—— 6-chloro-3-[(3R)-3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one —— C30H29ClN4O4
6-chloro-3-[(3R)-3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one
—— (6-oxo-7,8,9,10-tetrahydrobenzo[c]chromen-3-yl) (2R)-4-methylsulfanyl-2-(phenylmethoxycarbonylamino)butanoate —— C26H27NO6S
(6-oxo-7,8,9,10-tetrahydrobenzo[c]chromen-3-yl) (2R)-4-methylsulfanyl-2-(phenylmethoxycarbonylamino)butanoate
—— 6-chloro-3-[(3R)-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one —— C31H30ClFN4O2
6-chloro-3-[(3R)-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one
—— 6-[2-[(5S)-5-hydroxy-1-(4-phenyl-1,3-thiazol-2-yl)-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one —— C21H16F3N3O2S
6-[2-[(5S)-5-hydroxy-1-(4-phenyl-1,3-thiazol-2-yl)-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one
—— 6-chloro-3-[(3S)-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one —— C32H33ClN4O3
6-chloro-3-[(3S)-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one
—— (6S,9S)-9-(4-methylphenyl)-6-(4-phenylmethoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C35H29F3N2O3
(6S,9S)-9-(4-methylphenyl)-6-(4-phenylmethoxyphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[2-[(5R)-5-hydroxy-1-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one —— C22H18F3N3O2S
6-[2-[(5R)-5-hydroxy-1-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one
—— 6-chloro-3-[(3R)-3-[4-[(2S)-oxolane-2-carbonyl]piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one —— C30H33ClN4O4
6-chloro-3-[(3R)-3-[4-[(2S)-oxolane-2-carbonyl]piperazine-1-carbonyl]piperidin-1-yl]-4-phenyl-1H-quinolin-2-one
—— 6-[2-[(5R)-1-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-5-hydroxy-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one —— C21H15BrF3N3O2S
6-[2-[(5R)-1-[4-(4-bromophenyl)-1,3-thiazol-2-yl]-5-hydroxy-5-(trifluoromethyl)pyrazolidin-3-ylidene]ethylidene]cyclohexa-2,4-dien-1-one
—— (6R)-6-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-9,9-dimethyl-5-(2-methylpropanoyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C34H37ClN2O4
(6R)-6-[4-[(4-chlorophenyl)methoxy]-3-ethoxyphenyl]-9,9-dimethyl-5-(2-methylpropanoyl)-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6E)-2-methoxy-6-[(4-piperidin-1-ylsulfonylanilino)methylidene]cyclohexa-2,4-dien-1-one —— C19H22N2O4S
(6E)-2-methoxy-6-[(4-piperidin-1-ylsulfonylanilino)methylidene]cyclohexa-2,4-dien-1-one
—— (6R,9S)-5-benzoyl-6-(3-chlorophenyl)-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C33H27ClN2O2
(6R,9S)-5-benzoyl-6-(3-chlorophenyl)-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-5-[(6-benzoyl-1H-benzimidazol-2-yl)methyl]-6-(3,4-dichlorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C36H30Cl2N4O2
(6S)-5-[(6-benzoyl-1H-benzimidazol-2-yl)methyl]-6-(3,4-dichlorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S,9R)-N-(3,4-dichlorophenyl)-9-(4-methoxyphenyl)-7-oxo-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C31H25Cl2N3O3S
(6S,9R)-N-(3,4-dichlorophenyl)-9-(4-methoxyphenyl)-7-oxo-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— (6S,9S)-6-(3-chlorophenyl)-9-(4-methylphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H22ClF3N2O2
(6S,9S)-6-(3-chlorophenyl)-9-(4-methylphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9S)-5-(4-chlorobenzoyl)-6-(4-chlorophenyl)-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C32H24Cl2N2O2
(6S,9S)-5-(4-chlorobenzoyl)-6-(4-chlorophenyl)-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6E)-6-[[4-(2,3-dihydroindol-1-ylsulfonyl)anilino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C22H20N2O4S
(6E)-6-[[4-(2,3-dihydroindol-1-ylsulfonyl)anilino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— (6E)-3-(diethylamino)-6-[[4-(2,3-dihydroindol-1-ylsulfonyl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C25H27N3O3S
(6E)-3-(diethylamino)-6-[[4-(2,3-dihydroindol-1-ylsulfonyl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— (6S,9R)-5-benzoyl-6-(3-chlorophenyl)-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C33H27ClN2O2
(6S,9R)-5-benzoyl-6-(3-chlorophenyl)-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6Z)-2,4-dichloro-6-[(heptylamino)methylidene]cyclohexa-2,4-dien-1-one —— C14H19Cl2NO
(6Z)-2,4-dichloro-6-[(heptylamino)methylidene]cyclohexa-2,4-dien-1-one
—— (6R,9R)-6-(3-chlorophenyl)-9-(4-methylphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H22ClF3N2O2
(6R,9R)-6-(3-chlorophenyl)-9-(4-methylphenyl)-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6E)-6-[(heptylamino)methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C14H20N2O3
(6E)-6-[(heptylamino)methylidene]-4-nitrocyclohexa-2,4-dien-1-one
—— (6R,9R)-9-(3,4-dimethoxyphenyl)-5-hexanoyl-6-(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C36H42N2O7
(6R,9R)-9-(3,4-dimethoxyphenyl)-5-hexanoyl-6-(3,4,5-trimethoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9R)-5-benzoyl-6-(3-chlorophenyl)-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C33H27ClN2O2
(6R,9R)-5-benzoyl-6-(3-chlorophenyl)-9-(4-methylphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6E)-6-[(tert-butylamino)methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C11H14N2O3
(6E)-6-[(tert-butylamino)methylidene]-4-nitrocyclohexa-2,4-dien-1-one
—— (6R)-5-benzoyl-6-(4-methoxy-3-phenylmethoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C36H34N2O4
(6R)-5-benzoyl-6-(4-methoxy-3-phenylmethoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R)-2-[(Z)-[(E)-4-[4-(dimethylamino)phenyl]but-3-en-2-ylidene]hydrazinylidene]-4-oxo-N-phenyl-1,3-thiazinane-6-carboxamide —— C23H25N5O2S
(6R)-2-[(Z)-[(E)-4-[4-(dimethylamino)phenyl]but-3-en-2-ylidene]hydrazinylidene]-4-oxo-N-phenyl-1,3-thiazinane-6-carboxamide
—— (6R)-5-[(6-benzoyl-1H-benzimidazol-2-yl)methyl]-6-(3,4-dichlorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C36H30Cl2N4O2
(6R)-5-[(6-benzoyl-1H-benzimidazol-2-yl)methyl]-6-(3,4-dichlorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-5-[2-(4-chlorophenyl)acetyl]-9,9-dimethyl-6-[5-(3-nitrophenyl)furan-2-yl]-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C33H28ClN3O5
(6S)-5-[2-(4-chlorophenyl)acetyl]-9,9-dimethyl-6-[5-(3-nitrophenyl)furan-2-yl]-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R)-5-[2-(4-chlorophenyl)acetyl]-9,9-dimethyl-6-[5-(3-nitrophenyl)furan-2-yl]-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C33H28ClN3O5
(6R)-5-[2-(4-chlorophenyl)acetyl]-9,9-dimethyl-6-[5-(3-nitrophenyl)furan-2-yl]-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-chloro-3-[(5R)-5-(2,5-dimethoxyphenyl)-1-methylsulfonylpyrazolidin-3-ylidene]-4-phenylquinolin-2-one —— C27H24ClN3O5S
6-chloro-3-[(5R)-5-(2,5-dimethoxyphenyl)-1-methylsulfonylpyrazolidin-3-ylidene]-4-phenylquinolin-2-one
—— 6-(3,5-dimethylpyrazol-1-yl)-4-N-phenyl-2-N-[(Z)-(3,4,5-trimethoxyphenyl)methylideneamino]-1,3,5-triazine-2,4-diamine —— C24H26N8O3
6-(3,5-dimethylpyrazol-1-yl)-4-N-phenyl-2-N-[(Z)-(3,4,5-trimethoxyphenyl)methylideneamino]-1,3,5-triazine-2,4-diamine
—— 6-chloro-3-[(5R)-5-(2,3-dimethoxyphenyl)-1-methylsulfonylpyrazolidin-3-ylidene]-4-phenylquinolin-2-one —— C27H24ClN3O5S
6-chloro-3-[(5R)-5-(2,3-dimethoxyphenyl)-1-methylsulfonylpyrazolidin-3-ylidene]-4-phenylquinolin-2-one
—— 6-[6-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-8-oxo-[1,3]dioxolo[4,5-g]quinazolin-7-yl]-N-[(4-methoxyphenyl)methyl]hexanamide —— C29H36N4O6S
6-[6-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]sulfanyl-8-oxo-[1,3]dioxolo[4,5-g]quinazolin-7-yl]-N-[(4-methoxyphenyl)methyl]hexanamide
—— (6R,7S)-6-phenyl-6,7-dihydropyrrolo[2,1-d][1,5]benzothiazepin-7-ol —— C18H15NOS
(6R,7S)-6-phenyl-6,7-dihydropyrrolo[2,1-d][1,5]benzothiazepin-7-ol
—— 6-[(3R)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-[(1S)-1-phenylethyl]-1H-quinoline-4-carboxamide —— C24H27N3O4S
6-[(3R)-3-methylpiperidin-1-yl]sulfonyl-2-oxo-N-[(1S)-1-phenylethyl]-1H-quinoline-4-carboxamide
—— (6S)-6-(3,5-dioxo-4-phenyl-1,2,4-triazolidin-1-yl)-6-methyl-2-phenyl-5H-[1,2,4]triazolo[1,2-a]cinnoline-1,3-dione —— C25H20N6O4
(6S)-6-(3,5-dioxo-4-phenyl-1,2,4-triazolidin-1-yl)-6-methyl-2-phenyl-5H-[1,2,4]triazolo[1,2-a]cinnoline-1,3-dione
—— (6R)-6-(1,3-benzothiazol-2-yl)-6-cyano-N-(2,5-dimethoxyphenyl)-5-oxohexanamide —— C22H21N3O4S
(6R)-6-(1,3-benzothiazol-2-yl)-6-cyano-N-(2,5-dimethoxyphenyl)-5-oxohexanamide