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—— 6-{cis-3-[(5-isopropyl-1,3,4-thiadiazol-2-yl)amino]cyclobutyl}-2-pyrrolidin-1-ylpyrimidin-4(3H)-one —— C17H24N6OS
6-{cis-3-[(5-isopropyl-1,3,4-thiadiazol-2-yl)amino]cyclobutyl}-2-pyrrolidin-1-ylpyrimidin-4(3H)-one
—— 6-(3-aminocyclobutyl)-N~4~-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]pyrimidine-2,4-diamine —— C17H24N6O
6-(3-aminocyclobutyl)-N~4~-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]pyrimidine-2,4-diamine
—— 6-(cis-3-aminocyclobutyl)-N~4~-[2-(1H-indol-1-yl)ethyl]-N~4~-methylpyrimidine-2,4-diamine —— C19H24N6
6-(cis-3-aminocyclobutyl)-N~4~-[2-(1H-indol-1-yl)ethyl]-N~4~-methylpyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~4~-(3-morpholin-4-ylpropyl)pyrimidine-2,4-diamine —— C15H26N6O
6-(3-aminocyclobutyl)-N~4~-(3-morpholin-4-ylpropyl)pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N-[2-(5-fluoro-1H-benzimidazol-2-yl)ethyl]-N,2-dimethylpyrimidin-4-amine —— C19H23FN6
6-(3-aminocyclobutyl)-N-[2-(5-fluoro-1H-benzimidazol-2-yl)ethyl]-N,2-dimethylpyrimidin-4-amine
—— (6Z)-4-bromo-3-hydroxy-6-[[2-(4-methoxy-6-morpholin-4-yl-1,3,5-triazin-2-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C15H17BrN6O4
(6Z)-4-bromo-3-hydroxy-6-[[2-(4-methoxy-6-morpholin-4-yl-1,3,5-triazin-2-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-6-[[2-[3-[2-[(E)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]hydrazinyl]naphthalen-2-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C24H20N4O2
(6E)-6-[[2-[3-[2-[(E)-(6-oxocyclohexa-2,4-dien-1-ylidene)methyl]hydrazinyl]naphthalen-2-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— 6-{1-[(2-Amino-5,6,7,8-tetrahydroquinazolin-4-yl)carbonyl]piperidin-3-yl}-2-methylpyrimidin-4-ol —— C19H24N6O2
6-{1-[(2-Amino-5,6,7,8-tetrahydroquinazolin-4-yl)carbonyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
—— 6-methyl-N-[(3R,4S)-4-(6-methylpyridin-3-yl)oxyoxan-3-yl]imidazo[2,1-b][1,3]thiazole-5-carboxamide —— C18H20N4O3S
6-methyl-N-[(3R,4S)-4-(6-methylpyridin-3-yl)oxyoxan-3-yl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
—— 6-(cis-3-aminocyclobutyl)-2-cyclopropyl-N-(3,4-dihydro-2H-chromen-6-ylmethyl)pyrimidin-4-amine —— C21H26N4O
6-(cis-3-aminocyclobutyl)-2-cyclopropyl-N-(3,4-dihydro-2H-chromen-6-ylmethyl)pyrimidin-4-amine
—— (6E)-6-[[4-(1H-benzimidazol-2-yl)anilino]methylidene]-4-chloro-2-methoxycyclohexa-2,4-dien-1-one —— C21H16ClN3O2
(6E)-6-[[4-(1H-benzimidazol-2-yl)anilino]methylidene]-4-chloro-2-methoxycyclohexa-2,4-dien-1-one
—— 6-(cis-3-aminocyclobutyl)-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}pyrimidin-4-amine —— C15H19F3N6
6-(cis-3-aminocyclobutyl)-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N-{[4-(1H-benzimidazol-2-yl)cyclohexyl]methyl}pyrimidin-4-amine —— C22H28N6
6-(trans-3-aminocyclobutyl)-N-{[4-(1H-benzimidazol-2-yl)cyclohexyl]methyl}pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N-[3-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-(methoxymethyl)pyrimidin-4-amine —— C17H27N7O
6-(trans-3-aminocyclobutyl)-N-[3-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N~4~-[3-(3,4-dihydroquinolin-1(2H)-yl)propyl]pyrimidine-2,4-diamine —— C20H28N6
6-(cis-3-aminocyclobutyl)-N~4~-[3-(3,4-dihydroquinolin-1(2H)-yl)propyl]pyrimidine-2,4-diamine
—— (6Z)-5-imino-6-[[1-(3-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H28N6O3S
(6Z)-5-imino-6-[[1-(3-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3-aminocyclobutyl)-N~4~-[2-(4-phenylpiperidin-1-yl)ethyl]pyrimidine-2,4-diamine —— C21H30N6
6-(3-aminocyclobutyl)-N~4~-[2-(4-phenylpiperidin-1-yl)ethyl]pyrimidine-2,4-diamine
—— 6-{[3-(2-hydroxyethyl)-4-isobutylpiperazin-1-yl]carbonyl}pyridin-2(1H)-one —— C16H25N3O3
6-{[3-(2-hydroxyethyl)-4-isobutylpiperazin-1-yl]carbonyl}pyridin-2(1H)-one
—— 6-(3-aminocyclobutyl)-N~4~-[2-fluoro-4-(trifluoromethyl)benzyl]pyrimidine-2,4-diamine —— C16H17F4N5
6-(3-aminocyclobutyl)-N~4~-[2-fluoro-4-(trifluoromethyl)benzyl]pyrimidine-2,4-diamine
—— 6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidin-4-amine —— C15H23N7O
6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-methyl-N-[(3-pyridin-3-ylisoxazol-5-yl)methyl]pyrimidin-4-amine —— C20H24N6O2
6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-methyl-N-[(3-pyridin-3-ylisoxazol-5-yl)methyl]pyrimidin-4-amine
—— 6-(3-Aminocyclobutyl)-N-[1-(pyridin-4-ylmethyl)piperidin-4-YL]pyrimidin-4-amine —— C19H26N6
6-(3-Aminocyclobutyl)-N-[1-(pyridin-4-ylmethyl)piperidin-4-YL]pyrimidin-4-amine
—— 6-(3-Aminocyclobutyl)-N-methyl-N-[2-(4-methylpiperidin-1-YL)ethyl]pyrimidin-4-amine —— C17H29N5
6-(3-Aminocyclobutyl)-N-methyl-N-[2-(4-methylpiperidin-1-YL)ethyl]pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine —— C19H22N6
6-(trans-3-aminocyclobutyl)-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine
—— 6-Methoxy-2-(3-(2-nitrophenyl)-2-propenylidene)-3,4-dihydro-1(2H)-naphthalenone —— C20H17NO4
6-Methoxy-2-(3-(2-nitrophenyl)-2-propenylidene)-3,4-dihydro-1(2H)-naphthalenone
—— 6-Phenyl-3-propyl-6,7-dihydro-5H-benzo[d]isoxazol-4-one oxime —— C16H18N2O2
6-Phenyl-3-propyl-6,7-dihydro-5H-benzo[d]isoxazol-4-one oxime
—— (6E)-6-{[1-(3-chlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H20ClN5OS
(6E)-6-{[1-(3-chlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3-aminocyclobutyl)-N-{[4-(dimethylamino)tetrahydro-2H-pyran-4-yl]methyl}pyrimidin-4-amine —— C16H27N5O
6-(3-aminocyclobutyl)-N-{[4-(dimethylamino)tetrahydro-2H-pyran-4-yl]methyl}pyrimidin-4-amine
—— 6-fluoro-4-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}carbonyl)quinolin-2(1H)-one —— C19H19FN4O3
6-fluoro-4-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}carbonyl)quinolin-2(1H)-one
—— 6-(trans-3-aminocyclobutyl)-N-[2-(3-chlorophenoxy)ethyl]-2-cyclopropyl-N-methylpyrimidin-4-amine —— C20H25ClN4O
6-(trans-3-aminocyclobutyl)-N-[2-(3-chlorophenoxy)ethyl]-2-cyclopropyl-N-methylpyrimidin-4-amine
—— 6-amino-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-methylethyl]nicotinamide —— C14H19N5O
6-amino-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-methylethyl]nicotinamide
—— 6-[(3-piperidin-1-ylazetidin-1-yl)carbonyl]pyridin-2(1H)-one —— C14H19N3O2
6-[(3-piperidin-1-ylazetidin-1-yl)carbonyl]pyridin-2(1H)-one
—— 6-(3-aminocyclobutyl)-N~4~-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrimidine-2,4-diamine —— C13H20N8
6-(3-aminocyclobutyl)-N~4~-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrimidine-2,4-diamine
—— 6-(3-Aminocyclobutyl)-N-[2-(1H-imidazol-4-YL)ethyl]-2-(methoxymethyl)pyrimidin-4-amine —— C15H22N6O
6-(3-Aminocyclobutyl)-N-[2-(1H-imidazol-4-YL)ethyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-tert-butyl-N-[(3,5-dimethylisoxazol-4-yl)methyl]-N-methyl-2-oxo-2,3-dihydropyrimidine-4-carboxamide —— C16H22N4O3
6-tert-butyl-N-[(3,5-dimethylisoxazol-4-yl)methyl]-N-methyl-2-oxo-2,3-dihydropyrimidine-4-carboxamide
—— 6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-(2-morpholin-4-ylethyl)pyrimidin-4-amine —— C16H27N5O2
6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-(2-morpholin-4-ylethyl)pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-{2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-2,4-diamine —— C19H23N7O
6-(3-aminocyclobutyl)-N~4~-{2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-2,4-diamine
—— 6-chloro-N'-[(E)-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-2-methylimidazo[1,2-a]pyridine-3-carbohydrazide —— C17H15ClN4O3
6-chloro-N'-[(E)-(3-methoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-2-methylimidazo[1,2-a]pyridine-3-carbohydrazide
—— 6-(cis-3-aminocyclobutyl)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methylpyrimidin-4-amine —— C18H31N5O
6-(cis-3-aminocyclobutyl)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methylpyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-(2,4-dimethylbenzyl)pyrimidine-2,4-diamine —— C17H23N5
6-(3-aminocyclobutyl)-N~4~-(2,4-dimethylbenzyl)pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)thio]propyl}pyrimidin-4-amine —— C14H20N6S2
6-(3-aminocyclobutyl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)thio]propyl}pyrimidin-4-amine
—— 6-(3-Aminocyclobutyl)-N-[2-(3-chlorophenyl)ethyl]pyrimidin-4-amine —— C16H19ClN4
6-(3-Aminocyclobutyl)-N-[2-(3-chlorophenyl)ethyl]pyrimidin-4-amine
—— (6Z)-6-[[[2-(5-bromopyridin-3-yl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C19H12BrN3O2
(6Z)-6-[[[2-(5-bromopyridin-3-yl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-2-bromo-6-[(1,2-dihydroacenaphthylen-5-ylamino)methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C19H13BrN2O3
(6E)-2-bromo-6-[(1,2-dihydroacenaphthylen-5-ylamino)methylidene]-4-nitrocyclohexa-2,4-dien-1-one
—— (6E)-3-ethoxy-6-[[2-(3-methylphenyl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C16H18N2O2
(6E)-3-ethoxy-6-[[2-(3-methylphenyl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— 6-[2-[(Z)-indol-3-ylidenemethyl]hydrazinyl]-5-nitropyrimidin-4-amine —— C13H11N7O2
6-[2-[(Z)-indol-3-ylidenemethyl]hydrazinyl]-5-nitropyrimidin-4-amine
—— 6-fluoro-4-{[4-(tetrahydro-2H-pyran-4-yl)piperazin-1-yl]carbonyl}quinolin-2(1H)-one —— C19H22FN3O3
6-fluoro-4-{[4-(tetrahydro-2H-pyran-4-yl)piperazin-1-yl]carbonyl}quinolin-2(1H)-one
—— (6E)-6-[[(2Z)-2-[(3-nitrophenyl)methylidene]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C14H11N3O3
(6E)-6-[[(2Z)-2-[(3-nitrophenyl)methylidene]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— 6-(cis-3-aminocyclobutyl)-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methylpyrimidin-4-amine —— C16H25N7O
6-(cis-3-aminocyclobutyl)-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methylpyrimidin-4-amine
—— 6-methyl-4-oxo-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-4H-pyran-2-carboxamide —— C16H18N2O3S
6-methyl-4-oxo-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-4H-pyran-2-carboxamide