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—— 6-methylsulfonyl-2-[(2R)-1-(thiophene-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H22N4O4S2
6-methylsulfonyl-2-[(2R)-1-(thiophene-3-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2-methoxyphenyl)methyl]-2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H26N4O
6-[(2-methoxyphenyl)methyl]-2-[(2R)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6R)-1-(cyclopropanecarbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C23H26N2O3
(6R)-1-(cyclopropanecarbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one —— C19H21N5O2S
6-[(3S)-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-3-yl]-2-thiophen-2-yl-1H-pyrimidin-4-one
—— 6-methylsulfonyl-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C18H22N4O4S2
6-methylsulfonyl-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(2-methoxyphenyl)methyl]-2-[(2S)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H26N4O
6-[(2-methoxyphenyl)methyl]-2-[(2S)-piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(2-pyridin-2-ylacetyl)-1,4-diazepan-5-one —— C26H27N3O3
(6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(2-pyridin-2-ylacetyl)-1,4-diazepan-5-one
—— (6S)-6-[[2-(4-fluoro-2-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C19H21FN2O
(6S)-6-[[2-(4-fluoro-2-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-fluoro-N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1H-indole-2-carboxamide —— C22H20FN5O2S
6-fluoro-N-[(1S)-3-methylsulfanyl-1-(6-oxo-2-pyridin-2-yl-1H-pyrimidin-4-yl)propyl]-1H-indole-2-carboxamide
—— 6-[(2-methoxyphenyl)methyl]-2-[(3S)-1-(pyridine-4-carbonyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H27N5O3
6-[(2-methoxyphenyl)methyl]-2-[(3S)-1-(pyridine-4-carbonyl)pyrrolidin-3-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(2-pyridin-2-ylacetyl)-1,4-diazepan-5-one —— C26H27N3O3
(6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(2-pyridin-2-ylacetyl)-1,4-diazepan-5-one
—— 6-[(5Z)-5-[[5-(3-nitrophenyl)-1H-pyrazol-4-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C19H18N4O5S2
6-[(5Z)-5-[[5-(3-nitrophenyl)-1H-pyrazol-4-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— 6-[(5Z)-5-[[1-(4-nitrophenyl)pyrrol-2-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C20H19N3O5S2
6-[(5Z)-5-[[1-(4-nitrophenyl)pyrrol-2-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— 6-[(5Z)-4-oxo-5-[(3-phenyl-2,1-benzoxazol-5-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C23H20N2O4S2
6-[(5Z)-4-oxo-5-[(3-phenyl-2,1-benzoxazol-5-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— (6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C19H22N2O2
(6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-6-[[2-(3,5-dimethylphenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one —— C25H28N4O2
(6S)-6-[[2-(3,5-dimethylphenyl)phenyl]methyl]-1-(2-methylpyrazole-3-carbonyl)-1,4-diazepan-5-one
—— (6S)-1-[2-(2-methoxyphenyl)acetyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H28N2O3
(6S)-1-[2-(2-methoxyphenyl)acetyl]-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[(3R)-1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one —— C22H25N5O3
6-[(3R)-1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one
—— 6-methyl-3-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C19H19F3N4O
6-methyl-3-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— (6S)-6-[[2-(3,5-dimethylphenyl)phenyl]methyl]-1-(pyridine-3-carbonyl)-1,4-diazepan-5-one —— C26H27N3O2
(6S)-6-[[2-(3,5-dimethylphenyl)phenyl]methyl]-1-(pyridine-3-carbonyl)-1,4-diazepan-5-one
—— (6R)-1-(2-methoxybenzoyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H26N2O3
(6R)-1-(2-methoxybenzoyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(2,3-dimethoxyphenyl)methyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O3
(6R)-1-[(2,3-dimethoxyphenyl)methyl]-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-6-[[4-(3,5-dimethylphenyl)phenyl]methyl]-4-methyl-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one —— C25H28N4O2
(6S)-6-[[4-(3,5-dimethylphenyl)phenyl]methyl]-4-methyl-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
—— (6R)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(2-methoxybenzoyl)-1,4-diazepan-5-one —— C26H25FN2O3
(6R)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(2-methoxybenzoyl)-1,4-diazepan-5-one
—— (6S)-1-(2,6-dimethoxybenzoyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C27H28N2O4
(6S)-1-(2,6-dimethoxybenzoyl)-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[(2,6-Dimethoxyphenyl)methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C20H21N5O3
6-[(2,6-Dimethoxyphenyl)methyl]-2-pyrazin-2-yl-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-methyl-2-[(2S)-1-[(3-methyl-1-benzofuran-2-yl)methyl]piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C23H28N4O
6-methyl-2-[(2S)-1-[(3-methyl-1-benzofuran-2-yl)methyl]piperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6R)-1-[2-(4-fluorophenyl)acetyl]-6-[[3-(3-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H27FN2O3
(6R)-1-[2-(4-fluorophenyl)acetyl]-6-[[3-(3-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-[(2,3-dimethoxyphenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C20H26N4O2
6-[(2,3-dimethoxyphenyl)methyl]-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6R)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(2-methoxybenzoyl)-1,4-diazepan-5-one —— C26H25FN2O3
(6R)-6-[[3-(4-fluorophenyl)phenyl]methyl]-1-(2-methoxybenzoyl)-1,4-diazepan-5-one
—— (6R)-6-[[3-(3-methoxyphenyl)phenyl]methyl]-1-(3-phenylpropanoyl)-1,4-diazepan-5-one —— C28H30N2O3
(6R)-6-[[3-(3-methoxyphenyl)phenyl]methyl]-1-(3-phenylpropanoyl)-1,4-diazepan-5-one
—— 6-[(5Z)-5-[[5-(3,5-dichlorophenyl)furan-2-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C20H17Cl2NO4S2
6-[(5Z)-5-[[5-(3,5-dichlorophenyl)furan-2-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— 6-[(3S)-1-[(2,6-dimethoxyphenyl)methyl]pyrrolidin-3-yl]-2-morpholin-4-yl-1H-pyrimidin-4-one —— C21H28N4O4
6-[(3S)-1-[(2,6-dimethoxyphenyl)methyl]pyrrolidin-3-yl]-2-morpholin-4-yl-1H-pyrimidin-4-one
—— (6S)-6-[[3-(3-methoxyphenyl)phenyl]methyl]-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one —— C26H27N3O3
(6S)-6-[[3-(3-methoxyphenyl)phenyl]methyl]-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one
—— 6-[1-[(2-Methoxyphenyl)methyl]piperidin-4-yl]-3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C21H22F3N3O2
6-[1-[(2-Methoxyphenyl)methyl]piperidin-4-yl]-3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine
—— (6-methoxy-3-methyl-1-benzofuran-2-yl)-[(4S)-4-(4-methoxyphenyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methanone —— C24H23N3O4
(6-methoxy-3-methyl-1-benzofuran-2-yl)-[(4S)-4-(4-methoxyphenyl)-1,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]methanone
—— 6-[(3R)-1-[(3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one —— C21H23N5O2
6-[(3R)-1-[(3-methoxyphenyl)methyl]piperidin-3-yl]-2-pyrazin-2-yl-1H-pyrimidin-4-one
—— 6-methoxy-N-[1-[[2-methyl-5-(4-methyl-1,3-thiazol-5-yl)pyrazol-3-yl]methyl]piperidin-4-yl]pyridine-3-carboxamide —— C21H26N6O2S
6-methoxy-N-[1-[[2-methyl-5-(4-methyl-1,3-thiazol-5-yl)pyrazol-3-yl]methyl]piperidin-4-yl]pyridine-3-carboxamide
—— 6-[1-(Cyclohexylmethyl)piperidin-4-yl]-4-(difluoromethyl)-3-methyl-[1,2]oxazolo[5,4-b]pyridine —— C20H27F2N3O
6-[1-(Cyclohexylmethyl)piperidin-4-yl]-4-(difluoromethyl)-3-methyl-[1,2]oxazolo[5,4-b]pyridine
—— (6R)-1-(3-methoxybenzoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H24N2O3S
(6R)-1-(3-methoxybenzoyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(3-methoxybenzoyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H28N2O4
(6S)-1-(3-methoxybenzoyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-1-(3-methoxybenzoyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H25N3O3
(6R)-1-(3-methoxybenzoyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6-methoxy-1H-indol-2-yl)-[(3S)-3-(1H-pyrrolo[3,2-b]pyridin-2-yl)piperidin-1-yl]methanone —— C22H22N4O2
(6-methoxy-1H-indol-2-yl)-[(3S)-3-(1H-pyrrolo[3,2-b]pyridin-2-yl)piperidin-1-yl]methanone
—— 6-[(3R)-1-[(5-tert-butyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl]-4-(difluoromethyl)-3-methyl-[1,2]oxazolo[5,4-b]pyridine —— C21H27F2N5O
6-[(3R)-1-[(5-tert-butyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl]-4-(difluoromethyl)-3-methyl-[1,2]oxazolo[5,4-b]pyridine
—— (6-methoxy-1H-indol-2-yl)-[(3S)-3-[5-(trifluoromethyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methanone —— C23H21F3N4O2
(6-methoxy-1H-indol-2-yl)-[(3S)-3-[5-(trifluoromethyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methanone
—— (6S)-1-(3-methoxybenzoyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H25N3O3
(6S)-1-(3-methoxybenzoyl)-6-[(2-pyridin-4-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-methoxy-N-[(1S)-2-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)-1-phenylethyl]pyridine-3-carboxamide —— C24H21N5O3
6-methoxy-N-[(1S)-2-(6-oxo-2-pyridin-3-yl-1H-pyrimidin-4-yl)-1-phenylethyl]pyridine-3-carboxamide
—— (6R)-1-[2-(3-methoxyphenyl)acetyl]-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H26N2O3S
(6R)-1-[2-(3-methoxyphenyl)acetyl]-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[(3S)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-3-yl]-4-(difluoromethyl)-3-methyl-[1,2]oxazolo[5,4-b]pyridine —— C20H25F2N3O
6-[(3S)-1-[[(1R)-cyclohex-3-en-1-yl]methyl]piperidin-3-yl]-4-(difluoromethyl)-3-methyl-[1,2]oxazolo[5,4-b]pyridine
—— 6-[(3R)-1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl]-3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine —— C22H24F3N3O3
6-[(3R)-1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl]-3-methyl-4-(trifluoromethyl)-[1,2]oxazolo[5,4-b]pyridine