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—— (6Z)-6-[[[4-(4-bromophenyl)-2-(oxolan-2-ylmethylimino)-1,3-thiazol-3-yl]amino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C22H22BrN3O3S
(6Z)-6-[[[4-(4-bromophenyl)-2-(oxolan-2-ylmethylimino)-1,3-thiazol-3-yl]amino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— 6-[(2Z)-2-[1-(4-bromophenyl)ethylidene]hydrazinyl]-2,4,5-trichloropyridine-3-carbonitrile —— C14H8BrCl3N4
6-[(2Z)-2-[1-(4-bromophenyl)ethylidene]hydrazinyl]-2,4,5-trichloropyridine-3-carbonitrile
—— (6Z)-2-benzyl-6-{[2,5-dimethyl-1-(2-methylphenyl)-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H23N5OS
(6Z)-2-benzyl-6-{[2,5-dimethyl-1-(2-methylphenyl)-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(cis-3-aminocyclobutyl)-N-[2-(1H-pyrazol-1-yl)benzyl]pyrimidin-4-amine —— C18H20N6
6-(cis-3-aminocyclobutyl)-N-[2-(1H-pyrazol-1-yl)benzyl]pyrimidin-4-amine
—— 6-chloro-N-[(Z)-(2,5-dimethoxyphenyl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide —— C18H17ClN4O3
6-chloro-N-[(Z)-(2,5-dimethoxyphenyl)methylideneamino]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
—— (6Z)-6-[2-amino-5-(2-methoxyphenyl)-1H-pyrimidin-6-ylidene]-3-[(2-methylphenyl)methoxy]cyclohexa-2,4-dien-1-one —— C25H23N3O3
(6Z)-6-[2-amino-5-(2-methoxyphenyl)-1H-pyrimidin-6-ylidene]-3-[(2-methylphenyl)methoxy]cyclohexa-2,4-dien-1-one
—— 6-(3-Aminocyclobutyl)-N-[2-(2,5-dimethylphenoxy)ethyl]pyrimidin-4-amine —— C18H24N4O
6-(3-Aminocyclobutyl)-N-[2-(2,5-dimethylphenoxy)ethyl]pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrimidin-4-amine —— C16H23N7
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N-{2-[(4-fluorophenyl)sulfonyl]ethyl}pyrimidin-4-amine —— C16H19FN4O2S
6-(cis-3-aminocyclobutyl)-N-{2-[(4-fluorophenyl)sulfonyl]ethyl}pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-[2-(1-cyclopentylpiperidin-4-yl)ethyl]pyrimidine-2,4-diamine —— C20H34N6
6-(3-aminocyclobutyl)-N~4~-[2-(1-cyclopentylpiperidin-4-yl)ethyl]pyrimidine-2,4-diamine
—— (6Z)-6-[[1-(1,3-benzodioxol-5-ylmethyl)indol-3-yl]methylidene]-5-imino-2-(2-oxo-2-pyrrolidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H24N6O4S
(6Z)-6-[[1-(1,3-benzodioxol-5-ylmethyl)indol-3-yl]methylidene]-5-imino-2-(2-oxo-2-pyrrolidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-methyl-N-[1-methyl-2-(6-methylpyridin-2-yl)ethyl]-4-oxo-4H-pyran-2-carboxamide —— C16H18N2O3
6-methyl-N-[1-methyl-2-(6-methylpyridin-2-yl)ethyl]-4-oxo-4H-pyran-2-carboxamide
—— (6E)-4-bromo-6-[(3-methoxyanilino)methylidene]-2-nitrocyclohexa-2,4-dien-1-one —— C14H11BrN2O4
(6E)-4-bromo-6-[(3-methoxyanilino)methylidene]-2-nitrocyclohexa-2,4-dien-1-one
—— (6Z)-6-{[1-(2-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H20FN5O2S
(6Z)-6-{[1-(2-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-2-Ethyl-5-imino-6-({1-[2-(4-methoxyphenoxy)ethyl]-1H-indol-3-YL}methylidene)-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C25H23N5O3S
(6Z)-2-Ethyl-5-imino-6-({1-[2-(4-methoxyphenoxy)ethyl]-1H-indol-3-YL}methylidene)-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— 6-tert-butyl-N-(2,4-dimethoxyphenyl)-2-{[(Z)-phenylmethylidene]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C28H32N2O3S
6-tert-butyl-N-(2,4-dimethoxyphenyl)-2-{[(Z)-phenylmethylidene]amino}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6,7-Dihydroxy-4-[[4-(oxolan-2-ylmethyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]sulfanylmethyl]chromen-2-one —— C21H19N3O5S2
6,7-Dihydroxy-4-[[4-(oxolan-2-ylmethyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]sulfanylmethyl]chromen-2-one
—— 6-chloro-3-fluoro-N-[(1S,5S,6R,7S)-7-(methoxymethyl)-2-oxabicyclo[3.2.0]heptan-6-yl]imidazo[1,2-a]pyridine-2-carboxamide —— C16H17ClFN3O3
6-chloro-3-fluoro-N-[(1S,5S,6R,7S)-7-(methoxymethyl)-2-oxabicyclo[3.2.0]heptan-6-yl]imidazo[1,2-a]pyridine-2-carboxamide
—— (6Z)-2-(benzylsulfanyl)-6-(2,4-dimethoxybenzylidene)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C21H18N4O3S2
(6Z)-2-(benzylsulfanyl)-6-(2,4-dimethoxybenzylidene)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3-nitrophenyl)-1-phenyl-5,6-dihydro-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C17H13N5O3
6-(3-nitrophenyl)-1-phenyl-5,6-dihydro-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-(3-aminocyclobutyl)-N~4~-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-2,4-diamine —— C13H19N7
6-(3-aminocyclobutyl)-N~4~-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-2,4-diamine
—— 6-tert-butyl-2-oxo-N-[(3-pyridin-4-yl-1H-1,2,4-triazol-5-yl)methyl]-2,3-dihydropyrimidine-4-carboxamide —— C17H19N7O2
6-tert-butyl-2-oxo-N-[(3-pyridin-4-yl-1H-1,2,4-triazol-5-yl)methyl]-2,3-dihydropyrimidine-4-carboxamide
—— 6-(trans-3-aminocyclobutyl)-N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-(methoxymethyl)pyrimidin-4-amine —— C19H24N4O2
6-(trans-3-aminocyclobutyl)-N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-(methoxymethyl)pyrimidin-4-amine
—— 6-methyl-3-[(2Z)-2-[[3-(trifluoromethyl)phenyl]methylidene]hydrazinyl]-4H-1,2,4-triazin-5-one —— C12H10F3N5O
6-methyl-3-[(2Z)-2-[[3-(trifluoromethyl)phenyl]methylidene]hydrazinyl]-4H-1,2,4-triazin-5-one
—— 6-(3-aminocyclobutyl)-2-(methoxymethyl)-N-[(4-phenyltetrahydro-2H-pyran-4-yl)methyl]pyrimidin-4-amine —— C22H30N4O2
6-(3-aminocyclobutyl)-2-(methoxymethyl)-N-[(4-phenyltetrahydro-2H-pyran-4-yl)methyl]pyrimidin-4-amine
—— (6E)-4-chloro-6-[[[2-(2,5-dichlorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-3,5-dimethylcyclohexa-2,4-dien-1-one —— C22H15Cl3N2O2
(6E)-4-chloro-6-[[[2-(2,5-dichlorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-3,5-dimethylcyclohexa-2,4-dien-1-one
—— (6Z)-2,4-dichloro-6-[[2-[4,6-di(piperidin-1-yl)-1,3,5-triazin-2-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C20H25Cl2N7O
(6Z)-2,4-dichloro-6-[[2-[4,6-di(piperidin-1-yl)-1,3,5-triazin-2-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— 6-{[4-(4H-1,2,4-triazol-3-ylmethyl)piperazin-1-yl]carbonyl}imidazo[1,2-a]pyridine —— C15H17N7O
6-{[4-(4H-1,2,4-triazol-3-ylmethyl)piperazin-1-yl]carbonyl}imidazo[1,2-a]pyridine
—— 6-(3-Aminocyclobutyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-YL]methyl}pyrimidin-4-amine —— C13H18N6O2
6-(3-Aminocyclobutyl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-YL]methyl}pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-[2-(4-methylphenyl)ethyl]pyrimidine-2,4-diamine —— C17H23N5
6-(3-aminocyclobutyl)-N~4~-[2-(4-methylphenyl)ethyl]pyrimidine-2,4-diamine
—— 6-tert-butyl-N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-oxo-2,3-dihydropyrimidine-4-carboxamide —— C18H27N5O2
6-tert-butyl-N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-oxo-2,3-dihydropyrimidine-4-carboxamide
—— 6-{cis-3-[(6-isopropylpyridazin-3-yl)amino]cyclobutyl}-2-pyrrolidin-1-ylpyrimidin-4(3H)-one —— C19H26N6O
6-{cis-3-[(6-isopropylpyridazin-3-yl)amino]cyclobutyl}-2-pyrrolidin-1-ylpyrimidin-4(3H)-one
—— 6-(3-aminocyclobutyl)-2-cyclopropyl-N-(2,4-dimethoxybenzyl)pyrimidin-4-amine —— C20H26N4O2
6-(3-aminocyclobutyl)-2-cyclopropyl-N-(2,4-dimethoxybenzyl)pyrimidin-4-amine
—— (6E)-6-{[1-(3-chlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-pentyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H24ClN5OS
(6E)-6-{[1-(3-chlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-pentyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3-aminocyclobutyl)-N~4~-[(4-isopropyl-4H-1,2,4-triazol-3-yl)methyl]-N~4~-methylpyrimidine-2,4-diamine —— C15H24N8
6-(3-aminocyclobutyl)-N~4~-[(4-isopropyl-4H-1,2,4-triazol-3-yl)methyl]-N~4~-methylpyrimidine-2,4-diamine
—— (6E)-4-bromo-6-[[3-[3-(4-fluorophenyl)-2-phenyl-3,4-dihydropyrazol-5-yl]anilino]methylidene]cyclohexa-2,4-dien-1-one —— C28H21BrFN3O
(6E)-4-bromo-6-[[3-[3-(4-fluorophenyl)-2-phenyl-3,4-dihydropyrazol-5-yl]anilino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-amino-N-{trans-3-[6-(3-hydroxypyrrolidin-1-yl)pyrimidin-4-yl]cyclobutyl}nicotinamide —— C18H22N6O2
6-amino-N-{trans-3-[6-(3-hydroxypyrrolidin-1-yl)pyrimidin-4-yl]cyclobutyl}nicotinamide
—— 6-(trans-3-aminocyclobutyl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]pyrimidin-4-amine —— C17H19N7
6-(trans-3-aminocyclobutyl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]pyrimidin-4-amine
—— (6E)-6-[[[4-(4-methylphenyl)-5-(4-nitrophenyl)-1,3-thiazol-2-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C23H17N3O3S
(6E)-6-[[[4-(4-methylphenyl)-5-(4-nitrophenyl)-1,3-thiazol-2-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-(cis-3-aminocyclobutyl)-N~4~-[1-(3-methylphenyl)piperidin-4-yl]pyrimidine-2,4-diamine —— C20H28N6
6-(cis-3-aminocyclobutyl)-N~4~-[1-(3-methylphenyl)piperidin-4-yl]pyrimidine-2,4-diamine
—— (6E)-6-[2-amino-5-(morpholin-4-ylmethyl)-1H-pyrimidin-6-ylidene]cyclohexa-2,4-dien-1-one —— C15H18N4O2
(6E)-6-[2-amino-5-(morpholin-4-ylmethyl)-1H-pyrimidin-6-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[[(Z)-(3,4-dipropylphenyl)methylideneamino]-methylamino]-3-methyl-1H-pyrimidine-2,4-dione —— C19H26N4O2
6-[[(Z)-(3,4-dipropylphenyl)methylideneamino]-methylamino]-3-methyl-1H-pyrimidine-2,4-dione
—— (6Z)-2-(furan-2-yl)-6-(4-hydroxy-3-methoxybenzylidene)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C17H12N4O4S
(6Z)-2-(furan-2-yl)-6-(4-hydroxy-3-methoxybenzylidene)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-4-chloro-6-[[2-piperidin-1-yl-5-(trifluoromethyl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C19H18ClF3N2O
(6Z)-4-chloro-6-[[2-piperidin-1-yl-5-(trifluoromethyl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-{[4-(4-Fluorophenyl)-1,4-diazepan-1-yl]carbonyl}imidazo[1,2-a]pyridine —— C19H19FN4O
6-{[4-(4-Fluorophenyl)-1,4-diazepan-1-yl]carbonyl}imidazo[1,2-a]pyridine
—— (6Z)-2-butyl-5-imino-6-{3-[2-(4-methylphenoxy)ethoxy]benzylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H26N4O3S
(6Z)-2-butyl-5-imino-6-{3-[2-(4-methylphenoxy)ethoxy]benzylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[cis-3-(1,3-benzoxazol-2-ylamino)cyclobutyl]-N~4~-methylpyrimidine-2,4-diamine —— C16H18N6O
6-[cis-3-(1,3-benzoxazol-2-ylamino)cyclobutyl]-N~4~-methylpyrimidine-2,4-diamine
—— (6E)-4,5-dibromo-6-[[[2-(3-bromo-4-methoxyphenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-2-ethoxycyclohexa-2,4-dien-1-one —— C23H17Br3N2O4
(6E)-4,5-dibromo-6-[[[2-(3-bromo-4-methoxyphenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-2-ethoxycyclohexa-2,4-dien-1-one
—— 6-(3-Aminocyclobutyl)-N4-((1-ethyl-1H-imidazol-2-yl)methyl)-N4-methylpyrimidine-2,4-diamine —— C15H23N7
6-(3-Aminocyclobutyl)-N4-((1-ethyl-1H-imidazol-2-yl)methyl)-N4-methylpyrimidine-2,4-diamine
—— (6E)-6-[[2-[2-(benzylamino)-6-methylpyrimidin-4-yl]hydrazinyl]methylidene]-3-propoxycyclohexa-2,4-dien-1-one —— C22H25N5O2
(6E)-6-[[2-[2-(benzylamino)-6-methylpyrimidin-4-yl]hydrazinyl]methylidene]-3-propoxycyclohexa-2,4-dien-1-one