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—— 6-[(5E)-4-oxo-5-[4-oxo-3-[6-oxo-6-(pyridin-3-ylamino)hexyl]-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-pyridin-3-ylhexanamide —— C28H30N6O4S4
6-[(5E)-4-oxo-5-[4-oxo-3-[6-oxo-6-(pyridin-3-ylamino)hexyl]-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-pyridin-3-ylhexanamide
—— 6-[(5E)-4-oxo-5-[4-oxo-3-[6-oxo-6-[[5-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-2-yl]amino]hexyl]-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-[5-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-2-yl]hexanamide —— C40H36F6N6O4S6
6-[(5E)-4-oxo-5-[4-oxo-3-[6-oxo-6-[[5-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-2-yl]amino]hexyl]-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-[5-[[3-(trifluoromethyl)phenyl]methyl]-1,3-thiazol-2-yl]hexanamide
—— 6-[(5E)-5-[3-[6-(3-fluoroanilino)-6-oxohexyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-(3-fluorophenyl)hexanamide —— C30H30F2N4O4S4
6-[(5E)-5-[3-[6-(3-fluoroanilino)-6-oxohexyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-(3-fluorophenyl)hexanamide
—— 6-chloro-N-[(3S)-1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]imidazo[1,2-a]pyridine-2-carboxamide —— C19H17ClN4O3
6-chloro-N-[(3S)-1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
—— 6-[(5E)-5-[3-[6-(2-ethylanilino)-6-oxohexyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-(2-ethylphenyl)hexanamide —— C34H40N4O4S4
6-[(5E)-5-[3-[6-(2-ethylanilino)-6-oxohexyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-(2-ethylphenyl)hexanamide
—— 6-[(5E)-4-oxo-5-[4-oxo-3-[6-oxo-6-(4-phenylanilino)hexyl]-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-(4-phenylphenyl)hexanamide —— C42H40N4O4S4
6-[(5E)-4-oxo-5-[4-oxo-3-[6-oxo-6-(4-phenylanilino)hexyl]-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-(4-phenylphenyl)hexanamide
—— 6-[(5E)-5-[3-[6-(4-bromoanilino)-6-oxohexyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-(4-bromophenyl)hexanamide —— C30H30Br2N4O4S4
6-[(5E)-5-[3-[6-(4-bromoanilino)-6-oxohexyl]-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-N-(4-bromophenyl)hexanamide
—— 6-(1-ethylpyrazol-3-yl)-2-methyl-N-[(3R)-1-methylpiperidin-3-yl]pyrimidin-4-amine —— C16H24N6
6-(1-ethylpyrazol-3-yl)-2-methyl-N-[(3R)-1-methylpiperidin-3-yl]pyrimidin-4-amine
—— 6-(4-methoxy-2,5-dimethylphenyl)sulfonyl-N-methyl-2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine —— C22H31N5O3S
6-(4-methoxy-2,5-dimethylphenyl)sulfonyl-N-methyl-2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine
—— 6-[(2S)-1-[4-[2-(dimethylamino)-2-oxoethyl]phenyl]sulfonylpyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide —— C22H28N4O4S
6-[(2S)-1-[4-[2-(dimethylamino)-2-oxoethyl]phenyl]sulfonylpyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide
—— 6-(1-ethylpyrazol-3-yl)-2-methyl-N-[(3S)-1-methylpiperidin-3-yl]pyrimidin-4-amine —— C16H24N6
6-(1-ethylpyrazol-3-yl)-2-methyl-N-[(3S)-1-methylpiperidin-3-yl]pyrimidin-4-amine
—— 6-ethylsulfonyl-N-methyl-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine —— C14H23N5O2S
6-ethylsulfonyl-N-methyl-2-[(2S)-pyrrolidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine
—— 6-(5-fluoro-2-methoxyphenyl)sulfonyl-N-methyl-2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine —— C20H26FN5O3S
6-(5-fluoro-2-methoxyphenyl)sulfonyl-N-methyl-2-piperidin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine
—— 6-[(2S)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C25H30FN5O
6-[(2S)-1-[(1-ethyl-3-methylpyrazol-4-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— 6-[(2R)-1-[2-fluoro-5-(methylsulfamoyl)benzoyl]pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide —— C20H23FN4O4S
6-[(2R)-1-[2-fluoro-5-(methylsulfamoyl)benzoyl]pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide
—— (6-chloro-1H-indol-2-yl)-[4-[7-methyl-4-(methylamino)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-2-yl]piperidin-1-yl]methanone —— C23H27ClN6O
(6-chloro-1H-indol-2-yl)-[4-[7-methyl-4-(methylamino)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-2-yl]piperidin-1-yl]methanone
—— 6-[(2S)-1-[2-(4-methoxy-3-methylphenyl)acetyl]pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide —— C22H27N3O3
6-[(2S)-1-[2-(4-methoxy-3-methylphenyl)acetyl]pyrrolidin-2-yl]-N,2-dimethylpyridine-3-carboxamide
—— 6-(5-ethyl-2-methylpyrazol-3-yl)-N-[(1S)-1-(2-methoxyphenyl)ethyl]-2-methylpyrimidin-4-amine —— C20H25N5O
6-(5-ethyl-2-methylpyrazol-3-yl)-N-[(1S)-1-(2-methoxyphenyl)ethyl]-2-methylpyrimidin-4-amine
—— (6-ethyl-3-methyl-[1,2]oxazolo[5,4-b]pyridin-4-yl)-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]methanone —— C21H23N3O3
(6-ethyl-3-methyl-[1,2]oxazolo[5,4-b]pyridin-4-yl)-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]methanone
—— 6-[(2S)-1-[(1-ethylimidazol-2-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide —— C24H28FN5O
6-[(2S)-1-[(1-ethylimidazol-2-yl)methyl]pyrrolidin-2-yl]-N-[(4-fluorophenyl)methyl]-2-methylpyridine-3-carboxamide
—— (6-ethyl-3-methyl-[1,2]oxazolo[5,4-b]pyridin-4-yl)-[(3S)-3-(1-methylbenzimidazol-2-yl)piperidin-1-yl]methanone —— C23H25N5O2
(6-ethyl-3-methyl-[1,2]oxazolo[5,4-b]pyridin-4-yl)-[(3S)-3-(1-methylbenzimidazol-2-yl)piperidin-1-yl]methanone
—— 6-[[[4-(2-methoxyphenyl)phenyl]methyl-methylamino]methyl]-N,N-dimethyl-2-piperidin-4-ylpyrimidin-4-amine —— C27H35N5O
6-[[[4-(2-methoxyphenyl)phenyl]methyl-methylamino]methyl]-N,N-dimethyl-2-piperidin-4-ylpyrimidin-4-amine
—— 6-[[[3-(3-methoxyphenyl)phenyl]methyl-methylamino]methyl]-N-methyl-2-piperidin-4-ylpyrimidin-4-amine —— C26H33N5O
6-[[[3-(3-methoxyphenyl)phenyl]methyl-methylamino]methyl]-N-methyl-2-piperidin-4-ylpyrimidin-4-amine
—— 6-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-N-methyl-2-[(3R)-1-methylpiperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine —— C19H28N6O3S
6-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-N-methyl-2-[(3R)-1-methylpiperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine
—— 6-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-N-methyl-2-[(3S)-1-methylpiperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine —— C19H28N6O3S
6-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-N-methyl-2-[(3S)-1-methylpiperidin-3-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-amine
—— 6-[(dimethylamino)methyl]-2-[1-(4-fluoro-3-methylphenyl)sulfonylpiperidin-4-yl]-N-methylpyrimidin-4-amine —— C20H28FN5O2S
6-[(dimethylamino)methyl]-2-[1-(4-fluoro-3-methylphenyl)sulfonylpiperidin-4-yl]-N-methylpyrimidin-4-amine
—— 6-[[(2-fluoro-4-piperidin-1-ylphenyl)methyl-methylamino]methyl]-N,N-dimethyl-2-[(2S)-piperidin-2-yl]pyrimidin-4-amine —— C25H37FN6
6-[[(2-fluoro-4-piperidin-1-ylphenyl)methyl-methylamino]methyl]-N,N-dimethyl-2-[(2S)-piperidin-2-yl]pyrimidin-4-amine
—— [6-[(2R)-1-[(5-fluoro-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]pyridin-3-yl]-morpholin-4-ylmethanone —— C24H27FN4O2
[6-[(2R)-1-[(5-fluoro-1-methylindol-3-yl)methyl]pyrrolidin-2-yl]pyridin-3-yl]-morpholin-4-ylmethanone
—— [6-[(2R)-1-[(1-ethyl-2,3-dihydroindol-5-yl)methyl]pyrrolidin-2-yl]pyridin-3-yl]-morpholin-4-ylmethanone —— C25H32N4O2
[6-[(2R)-1-[(1-ethyl-2,3-dihydroindol-5-yl)methyl]pyrrolidin-2-yl]pyridin-3-yl]-morpholin-4-ylmethanone
—— 6-[(2S)-1-(6-methoxypyridine-3-carbonyl)pyrrolidin-2-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide —— C20H19N5O3S
6-[(2S)-1-(6-methoxypyridine-3-carbonyl)pyrrolidin-2-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide
—— (6-methyl-1H-indol-2-yl)-[3-[(3R)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone —— C22H28N6O
(6-methyl-1H-indol-2-yl)-[3-[(3R)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone
—— [6-[(2R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone —— C22H29N5O3
[6-[(2R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone
—— [6-[1-(2-Methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)piperidin-4-yl]pyridin-3-yl]-morpholin-4-ylmethanone —— C24H31N5O3
[6-[1-(2-Methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)piperidin-4-yl]pyridin-3-yl]-morpholin-4-ylmethanone
—— 6-[(2R)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidin-2-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide —— C19H19N5O2S2
6-[(2R)-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]pyrrolidin-2-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide
—— 6-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-N,N-dimethylpyridine-3-carboxamide —— C20H26N4O3
6-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[1-(pyridine-2-carbonyl)piperidin-4-yl]-N-[2-(1,3,5-trimethylpyrazol-4-yl)ethyl]pyridine-3-carboxamide —— C25H30N6O2
6-[1-(pyridine-2-carbonyl)piperidin-4-yl]-N-[2-(1,3,5-trimethylpyrazol-4-yl)ethyl]pyridine-3-carboxamide
—— [6-[1-(3-Ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]pyridin-3-yl]-piperidin-1-ylmethanone —— C23H30N4O3
[6-[1-(3-Ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]pyridin-3-yl]-piperidin-1-ylmethanone
—— (6-methoxy-2-methylquinolin-3-yl)-[4-(methylamino)-2-[(2S)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]methanone —— C25H30N6O2
(6-methoxy-2-methylquinolin-3-yl)-[4-(methylamino)-2-[(2S)-1-methylpyrrolidin-2-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]methanone
—— 6-(1-methylsulfonylpiperidin-4-yl)-N-[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]pyridine-3-carboxamide —— C20H26N4O3S2
6-(1-methylsulfonylpiperidin-4-yl)-N-[(6R)-6-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]pyridine-3-carboxamide
—— [6-[(2S)-1-(1,3-dimethylpyrazole-4-carbonyl)pyrrolidin-2-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone —— C21H28N6O2
[6-[(2S)-1-(1,3-dimethylpyrazole-4-carbonyl)pyrrolidin-2-yl]pyridin-3-yl]-(4-methylpiperazin-1-yl)methanone
—— 6-[1-[3-(4-methoxy-3-methylphenyl)propanoyl]piperidin-4-yl]-N,N-dimethylpyridine-3-carboxamide —— C24H31N3O3
6-[1-[3-(4-methoxy-3-methylphenyl)propanoyl]piperidin-4-yl]-N,N-dimethylpyridine-3-carboxamide
—— [6-[1-(2-Methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)piperidin-4-yl]pyridin-3-yl]-piperidin-1-ylmethanone —— C25H33N5O2
[6-[1-(2-Methyl-4,5,6,7-tetrahydroindazole-3-carbonyl)piperidin-4-yl]pyridin-3-yl]-piperidin-1-ylmethanone
—— 6-(1-acetylpiperidin-4-yl)-N-methyl-N-[(2S)-2-phenylpropyl]pyridine-3-carboxamide —— C23H29N3O2
6-(1-acetylpiperidin-4-yl)-N-methyl-N-[(2S)-2-phenylpropyl]pyridine-3-carboxamide
—— 6-(1-acetylpiperidin-4-yl)-N-methyl-N-(quinolin-6-ylmethyl)pyridine-3-carboxamide —— C24H26N4O2
6-(1-acetylpiperidin-4-yl)-N-methyl-N-(quinolin-6-ylmethyl)pyridine-3-carboxamide
—— 6-[1-[2-[(2R)-2-methylpiperidin-1-yl]acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide —— C22H29N5O2S
6-[1-[2-[(2R)-2-methylpiperidin-1-yl]acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide
—— 6-[1-[2-(4-methylpyrazol-1-yl)acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide —— C20H22N6O2S
6-[1-[2-(4-methylpyrazol-1-yl)acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide
—— 6-[(3R)-1-[3-(4-methoxy-3-methylphenyl)propanoyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide —— C24H31N3O3
6-[(3R)-1-[3-(4-methoxy-3-methylphenyl)propanoyl]piperidin-3-yl]-N,N-dimethylpyridine-3-carboxamide
—— 6-[1-(2,4-dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide —— C23H23FN4O2S
6-[1-(2,4-dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-N-(4-fluorophenyl)pyridine-3-carboxamide
—— 6-[1-[2-[(2S)-2-methylpiperidin-1-yl]acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide —— C22H29N5O2S
6-[1-[2-[(2S)-2-methylpiperidin-1-yl]acetyl]piperidin-4-yl]-N-(1,3-thiazol-2-yl)pyridine-3-carboxamide
—— (6Z)-6-[[5-(1,3-benzoxazol-2-yl)-2-methylanilino]methylidene]-2-ethoxy-4-nitrocyclohexa-2,4-dien-1-one —— C23H19N3O5
(6Z)-6-[[5-(1,3-benzoxazol-2-yl)-2-methylanilino]methylidene]-2-ethoxy-4-nitrocyclohexa-2,4-dien-1-one