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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-(2,3-Dihydro-1-benzofuran-7-YL)-5-methoxypyridine-2-carboxylic acid —— C15H13NO4
6-(2,3-Dihydro-1-benzofuran-7-YL)-5-methoxypyridine-2-carboxylic acid
—— (6E)-4,5-dibromo-6-[[[2-(3-fluorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C21H13Br2FN2O3
(6E)-4,5-dibromo-6-[[[2-(3-fluorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— 6-(4-{[5-(cis-3-aminocyclobutyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperazin-1-yl)nicotinonitrile —— C18H24N8
6-(4-{[5-(cis-3-aminocyclobutyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperazin-1-yl)nicotinonitrile
—— 6-[[2-(5,7-Dihydroxy-4-methyl-2-oxochromen-3-yl)acetyl]amino]hexanoic acid —— C18H21NO7
6-[[2-(5,7-Dihydroxy-4-methyl-2-oxochromen-3-yl)acetyl]amino]hexanoic acid
—— 6-(trans-3-aminocyclobutyl)-N-[(1-isopropyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylpyrimidin-4-amine —— C18H28N6
6-(trans-3-aminocyclobutyl)-N-[(1-isopropyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylpyrimidin-4-amine
—— (6Z)-5-imino-6-{3-methoxy-4-[(2-methylbenzyl)oxy]benzylidene}-2-(pyridin-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H21N5O3S
(6Z)-5-imino-6-{3-methoxy-4-[(2-methylbenzyl)oxy]benzylidene}-2-(pyridin-3-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[2-(1,2-dihydroxyethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]pyridine-2-carbonitrile —— C15H17N5O2
6-[2-(1,2-dihydroxyethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]pyridine-2-carbonitrile
—— 6-(cis-3-aminocyclobutyl)-N-[(1-cyclopentylpiperidin-4-yl)methyl]pyrimidin-4-amine —— C19H31N5
6-(cis-3-aminocyclobutyl)-N-[(1-cyclopentylpiperidin-4-yl)methyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-2-(methoxymethyl)-N-[(8-methylimidazo[1,2-a]pyridin-3-yl)methyl]pyrimidin-4-amine —— C19H24N6O
6-(3-aminocyclobutyl)-2-(methoxymethyl)-N-[(8-methylimidazo[1,2-a]pyridin-3-yl)methyl]pyrimidin-4-amine
—— 6-ethyl-1,5-dimethyl-N-[(3S,4S)-3-(oxan-4-yl)oxan-4-yl]-2-oxopyridine-3-carboxamide —— C20H30N2O4
6-ethyl-1,5-dimethyl-N-[(3S,4S)-3-(oxan-4-yl)oxan-4-yl]-2-oxopyridine-3-carboxamide
—— 6-{[4-(Hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}-2-naphthol —— C22H30N2O2
6-{[4-(Hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}-2-naphthol
—— 6-hydroxy-2-[(E)-2-(4-methoxynaphthalen-1-yl)ethenyl]-5-nitropyrimidin-4(3H)-one —— C17H13N3O5
6-hydroxy-2-[(E)-2-(4-methoxynaphthalen-1-yl)ethenyl]-5-nitropyrimidin-4(3H)-one
—— 6-(3-aminocyclobutyl)-N~4~-[(3-methyl-2-thienyl)methyl]pyrimidine-2,4-diamine —— C14H19N5S
6-(3-aminocyclobutyl)-N~4~-[(3-methyl-2-thienyl)methyl]pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~4~-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidine-2,4-diamine —— C14H22N8O
6-(3-aminocyclobutyl)-N~4~-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidine-2,4-diamine
—— 6-oxo-N-[cis-3-(6-pyrrolidin-1-ylpyrimidin-4-yl)cyclobutyl]-1,6-dihydropyridine-3-carboxamide —— C18H21N5O2
6-oxo-N-[cis-3-(6-pyrrolidin-1-ylpyrimidin-4-yl)cyclobutyl]-1,6-dihydropyridine-3-carboxamide
—— (6Z)-6-{3-chloro-5-ethoxy-4-[2-(4-methylphenoxy)ethoxy]benzylidene}-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C30H27ClN4O5S
(6Z)-6-{3-chloro-5-ethoxy-4-[2-(4-methylphenoxy)ethoxy]benzylidene}-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-cyano-N-{cis-3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]cyclobutyl}nicotinamide —— C15H16N6O2
6-cyano-N-{cis-3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]cyclobutyl}nicotinamide
—— (6Z)-6-[(pyridin-3-ylamino)methylidene]cyclohexa-2,4-dien-1-one —— C12H10N2O
(6Z)-6-[(pyridin-3-ylamino)methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-6-[(4-chlorophenyl)methylene]-3-(4-nitrophenyl)-7aH-thiazolo[2,3-b]thiazol-5-one —— C18H11ClN2O3S2
(6Z)-6-[(4-chlorophenyl)methylene]-3-(4-nitrophenyl)-7aH-thiazolo[2,3-b]thiazol-5-one
—— (6Z)-6-{[5-(2-chlorophenyl)furan-2-yl]methylidene}-5-imino-2-[2-oxo-2-(piperidin-1-yl)ethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H20ClN5O3S
(6Z)-6-{[5-(2-chlorophenyl)furan-2-yl]methylidene}-5-imino-2-[2-oxo-2-(piperidin-1-yl)ethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-{trans-3-[(2-amino-5-chloro-6-methylpyrimidin-4-yl)amino]cyclobutyl}pyrimidin-4(3H)-one —— C13H15ClN6O
6-{trans-3-[(2-amino-5-chloro-6-methylpyrimidin-4-yl)amino]cyclobutyl}pyrimidin-4(3H)-one
—— (6Z)-5-Imino-6-[(4-methylphenyl)methylidene]-3-(methylsulfanyl)-5H,6H,7H-[1,2,4]thiadiazolo[4,5-A]pyrimidin-7-one —— C14H12N4OS2
(6Z)-5-Imino-6-[(4-methylphenyl)methylidene]-3-(methylsulfanyl)-5H,6H,7H-[1,2,4]thiadiazolo[4,5-A]pyrimidin-7-one
—— 6-(3-aminocyclobutyl)-N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]pyrimidin-4-amine —— C12H17N7S
6-(3-aminocyclobutyl)-N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-[2-(2-chlorophenoxy)ethyl]pyrimidine-2,4-diamine —— C16H20ClN5O
6-(3-aminocyclobutyl)-N~4~-[2-(2-chlorophenoxy)ethyl]pyrimidine-2,4-diamine
—— (6Z)-5-imino-6-{4-[2-(3-methylphenoxy)ethoxy]benzylidene}-2-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H27N5O4S
(6Z)-5-imino-6-{4-[2-(3-methylphenoxy)ethoxy]benzylidene}-2-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-methyl-N-[rac-2-oxabicyclo[3.2.0]hept-6-yl]thieno[2,3-d]pyrimidin-4-amine —— C13H15N3OS
6-methyl-N-[rac-2-oxabicyclo[3.2.0]hept-6-yl]thieno[2,3-d]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N-{[5-(2-chlorophenyl)-2-furyl]methyl}pyrimidin-4-amine —— C19H19ClN4O
6-(3-aminocyclobutyl)-N-{[5-(2-chlorophenyl)-2-furyl]methyl}pyrimidin-4-amine
—— (6Z)-6-{[2,5-dimethyl-1-(naphthalen-1-yl)-1H-pyrrol-3-yl]methylidene}-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H23N5OS
(6Z)-6-{[2,5-dimethyl-1-(naphthalen-1-yl)-1H-pyrrol-3-yl]methylidene}-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3-aminocyclobutyl)-N~4~-[(3,5-dimethylisoxazol-4-yl)methyl]pyrimidine-2,4-diamine —— C14H20N6O
6-(3-aminocyclobutyl)-N~4~-[(3,5-dimethylisoxazol-4-yl)methyl]pyrimidine-2,4-diamine
—— 6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidin-4-amine —— C18H26N6O
6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidin-4-amine
—— 6-(3-Aminocyclobutyl)-2-cyclopropyl-N-[2-(3-methoxyphenyl)ethyl]pyrimidin-4-amine —— C20H26N4O
6-(3-Aminocyclobutyl)-2-cyclopropyl-N-[2-(3-methoxyphenyl)ethyl]pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N-[2-(2-fluorophenyl)ethyl]pyrimidin-4-amine —— C16H19FN4
6-(trans-3-aminocyclobutyl)-N-[2-(2-fluorophenyl)ethyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-{2-[3-(trifluoromethyl)phenyl]ethyl}pyrimidine-2,4-diamine —— C17H20F3N5
6-(3-aminocyclobutyl)-N~4~-{2-[3-(trifluoromethyl)phenyl]ethyl}pyrimidine-2,4-diamine
—— 6-amino-N-[3-(4,5-dimethyl-1,3-thiazol-2-yl)propyl]nicotinamide —— C14H18N4OS
6-amino-N-[3-(4,5-dimethyl-1,3-thiazol-2-yl)propyl]nicotinamide
—— 6-(cis-3-aminocyclobutyl)-N-(2-chloro-6-fluorobenzyl)pyrimidin-4-amine —— C15H16ClFN4
6-(cis-3-aminocyclobutyl)-N-(2-chloro-6-fluorobenzyl)pyrimidin-4-amine
—— 6-cyano-N-[cis-4-(3-fluorophenoxy)tetrahydro-2H-pyran-3-yl]nicotinamide —— C18H16FN3O3
6-cyano-N-[cis-4-(3-fluorophenoxy)tetrahydro-2H-pyran-3-yl]nicotinamide
—— 6-Amino-N-(isoquinolin-5-ylmethyl)-N-methylpyridine-2-carboxamide —— C17H16N4O
6-Amino-N-(isoquinolin-5-ylmethyl)-N-methylpyridine-2-carboxamide
—— 6-(3-Aminocyclobutyl)-N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(methoxymethyl)-N-methylpyrimidin-4-amine —— C18H22N6O2
6-(3-Aminocyclobutyl)-N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(methoxymethyl)-N-methylpyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N-{[1-(cyclopropylcarbonyl)piperidin-4-yl]methyl}-2-methylpyrimidin-4-amine —— C19H29N5O
6-(cis-3-aminocyclobutyl)-N-{[1-(cyclopropylcarbonyl)piperidin-4-yl]methyl}-2-methylpyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)pyrimidin-4-amine —— C17H21N7O
6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)pyrimidin-4-amine
—— (6Z)-5-imino-6-[[3-methoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H26N4O4S
(6Z)-5-imino-6-[[3-methoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl]methylidene]-2-propan-2-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3-aminocyclobutyl)-N~4~-(isoxazol-3-ylmethyl)-N~4~-methylpyrimidine-2,4-diamine —— C13H18N6O
6-(3-aminocyclobutyl)-N~4~-(isoxazol-3-ylmethyl)-N~4~-methylpyrimidine-2,4-diamine
—— 6-bromo-N-[(Z)-(6-nitro-1,3-benzodioxol-5-yl)methylideneamino]-4-phenylquinolin-2-amine —— C23H15BrN4O4
6-bromo-N-[(Z)-(6-nitro-1,3-benzodioxol-5-yl)methylideneamino]-4-phenylquinolin-2-amine
—— 6-(3-aminocyclobutyl)-N~4~-(3-ethoxybenzyl)-N~4~-methylpyrimidine-2,4-diamine —— C18H25N5O
6-(3-aminocyclobutyl)-N~4~-(3-ethoxybenzyl)-N~4~-methylpyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~4~-({1-[ethyl(methyl)amino]cyclohexyl}methyl)pyrimidine-2,4-diamine —— C18H32N6
6-(3-aminocyclobutyl)-N~4~-({1-[ethyl(methyl)amino]cyclohexyl}methyl)pyrimidine-2,4-diamine
—— 6-(3-Aminocyclobutyl)-N-{[1-(4-chlorophenyl)cyclopropyl]methyl}pyrimidin-4-amine —— C18H21ClN4
6-(3-Aminocyclobutyl)-N-{[1-(4-chlorophenyl)cyclopropyl]methyl}pyrimidin-4-amine
—— (6E)-4-(chloromethyl)-6-[[3-[[(E)-[3-(chloromethyl)-6-oxocyclohexa-2,4-dien-1-ylidene]methyl]amino]anilino]methylidene]cyclohexa-2,4-dien-1-one —— C22H18Cl2N2O2
(6E)-4-(chloromethyl)-6-[[3-[[(E)-[3-(chloromethyl)-6-oxocyclohexa-2,4-dien-1-ylidene]methyl]amino]anilino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-(4-chlorophenyl)-8-(2-phenylvinyl)-3,4a,7a,8-tetrahydropyrrolo[3',4':5,6]thiopyrano[2,3-d][1,3]thiazole-2,5,7(6H)-trione —— C22H15ClN2O3S2
6-(4-chlorophenyl)-8-(2-phenylvinyl)-3,4a,7a,8-tetrahydropyrrolo[3',4':5,6]thiopyrano[2,3-d][1,3]thiazole-2,5,7(6H)-trione
—— (6Z)-6-[[2-morpholin-4-yl-5-(trifluoromethyl)anilino]methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C18H16F3N3O4
(6Z)-6-[[2-morpholin-4-yl-5-(trifluoromethyl)anilino]methylidene]-4-nitrocyclohexa-2,4-dien-1-one
—— (6E)-4-chloro-6-[(3-hydroxy-4-methylanilino)methylidene]cyclohexa-2,4-dien-1-one —— C14H12ClNO2
(6E)-4-chloro-6-[(3-hydroxy-4-methylanilino)methylidene]cyclohexa-2,4-dien-1-one