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—— (6Z)-2-cyclohexyl-6-{[2,5-dimethyl-1-(4-methylphenyl)-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H27N5OS
(6Z)-2-cyclohexyl-6-{[2,5-dimethyl-1-(4-methylphenyl)-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-N-(4-fluorophenyl)-5-N-[(E)-furan-2-ylmethylideneamino]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine —— C15H10FN7O2
6-N-(4-fluorophenyl)-5-N-[(E)-furan-2-ylmethylideneamino]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
—— 6-methyl-3-[(E)-2-oxo-2-(2-thienyl)ethylidene]tetrahydro-2(1H)-pyrazinone —— C11H12N2O2S
6-methyl-3-[(E)-2-oxo-2-(2-thienyl)ethylidene]tetrahydro-2(1H)-pyrazinone
—— (6Z)-5-imino-6-[[1-(4-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H26N6O4S
(6Z)-5-imino-6-[[1-(4-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-benzylidene-3-thiophen-2-yl-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one —— C15H9N3OS2
(6E)-6-benzylidene-3-thiophen-2-yl-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one
—— 6-[(2S,5R)-2,5-dimethylmorpholin-4-yl]-2-methoxypyridin-3-amine —— C12H19N3O2
6-[(2S,5R)-2,5-dimethylmorpholin-4-yl]-2-methoxypyridin-3-amine
—— 6-(4-chlorophenyl)-N-[(2,4-dichlorophenyl)methylideneamino]-4-(trifluoromethyl)pyrimidin-1-ium-2-amine —— C18H11Cl3F3N4+
6-(4-chlorophenyl)-N-[(2,4-dichlorophenyl)methylideneamino]-4-(trifluoromethyl)pyrimidin-1-ium-2-amine
—— 6-[(2R,5R)-2,5-dimethylmorpholin-4-yl]pyridin-3-amine —— C11H17N3O
6-[(2R,5R)-2,5-dimethylmorpholin-4-yl]pyridin-3-amine
—— 6-[(2S,5R)-2,5-dimethylmorpholin-4-yl]pyridine-3-carbothioamide —— C12H17N3OS
6-[(2S,5R)-2,5-dimethylmorpholin-4-yl]pyridine-3-carbothioamide
—— 6-tert-butyl-2-[[(E)-3-(4-methoxyphenyl)prop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H28N2O3S
6-tert-butyl-2-[[(E)-3-(4-methoxyphenyl)prop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-[(2R,5R)-2,5-dimethylmorpholin-4-yl]-2,3-dihydro-1,4-benzodioxin-7-amine —— C14H20N2O3
6-[(2R,5R)-2,5-dimethylmorpholin-4-yl]-2,3-dihydro-1,4-benzodioxin-7-amine
—— (6Z)-6-[[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H26N6O3S
(6Z)-6-[[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-5-imino-2-(2-methylpropyl)-6-[[4-(2-phenoxyethoxy)phenyl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H24N4O3S
(6E)-5-imino-2-(2-methylpropyl)-6-[[4-(2-phenoxyethoxy)phenyl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-2-(2-cyclohexylethyl)-6-[[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H31N5OS
(6Z)-2-(2-cyclohexylethyl)-6-[[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[(1-benzyl-2,5-dimethyl-1H-pyrrol-3-yl)methylidene]-2-heptyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H31N5OS
(6E)-6-[(1-benzyl-2,5-dimethyl-1H-pyrrol-3-yl)methylidene]-2-heptyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-{[1-(4-chlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-heptyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H28ClN5OS
(6E)-6-{[1-(4-chlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-2-heptyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(3R)-3-methylmorpholin-4-yl]-2-propan-2-yloxypyridin-3-amine —— C13H21N3O2
6-[(3R)-3-methylmorpholin-4-yl]-2-propan-2-yloxypyridin-3-amine
—— 6-[(3S)-3-methylmorpholin-4-yl]imidazo[2,1-b][1,3]thiazole-5-carbaldehyde —— C11H13N3O2S
6-[(3S)-3-methylmorpholin-4-yl]imidazo[2,1-b][1,3]thiazole-5-carbaldehyde
—— 6-[(3R)-3-methylmorpholin-4-yl]-2-[(2-methylpropan-2-yl)oxy]pyridin-3-amine —— C14H23N3O2
6-[(3R)-3-methylmorpholin-4-yl]-2-[(2-methylpropan-2-yl)oxy]pyridin-3-amine
—— 6-amino-7-[(3R)-3-methylmorpholin-4-yl]-1H-quinazolin-4-one —— C13H16N4O2
6-amino-7-[(3R)-3-methylmorpholin-4-yl]-1H-quinazolin-4-one
—— (6E)-2-heptyl-5-imino-6-{[1-(4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H31N5O2S
(6E)-2-heptyl-5-imino-6-{[1-(4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2-hexyl-5-imino-6-{[1-(4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H29N5O2S
(6E)-2-hexyl-5-imino-6-{[1-(4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2-ethyl-6-{[1-(4-fluorobenzyl)-2,5-dimethyl-1H-indol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H22FN5OS
(6E)-2-ethyl-6-{[1-(4-fluorobenzyl)-2,5-dimethyl-1H-indol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-ethyl 8-methyl (2Z)-5-amino-2-(4-methylbenzylidene)-7-(4-methylphenyl)-3-oxo-2,3-dihydro-7H-[1,3]thiazolo[3,2-a]pyridine-6,8-dicarboxylate —— C27H26N2O5S
6-ethyl 8-methyl (2Z)-5-amino-2-(4-methylbenzylidene)-7-(4-methylphenyl)-3-oxo-2,3-dihydro-7H-[1,3]thiazolo[3,2-a]pyridine-6,8-dicarboxylate
—— (6E)-6-{[1-(4-Bromophenyl)-2,5-dimethyl-1H-pyrrol-3-YL]methylidene}-2-ethyl-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C20H18BrN5OS
(6E)-6-{[1-(4-Bromophenyl)-2,5-dimethyl-1H-pyrrol-3-YL]methylidene}-2-ethyl-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6E)-5-imino-6-[[4-(3-phenoxypropoxy)phenyl]methylidene]-3-phenyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C28H23N3O3S
(6E)-5-imino-6-[[4-(3-phenoxypropoxy)phenyl]methylidene]-3-phenyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[(2,5-dimethyl-1-phenylpyrrol-3-yl)methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C20H19N5OS
(6E)-6-[(2,5-dimethyl-1-phenylpyrrol-3-yl)methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2-heptyl-5-imino-6-[[1-[2-(4-methoxyphenoxy)ethyl]indol-3-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C30H33N5O3S
(6E)-2-heptyl-5-imino-6-[[1-[2-(4-methoxyphenoxy)ethyl]indol-3-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-{[2,5-Dimethyl-1-(4-methylphenyl)-1H-pyrrol-3-YL]methylidene}-5-imino-2-methyl-5H,6H,7H-[1,3]thiazolo[3,2-A]pyrimidin-7-one —— C21H20N4OS
(6Z)-6-{[2,5-Dimethyl-1-(4-methylphenyl)-1H-pyrrol-3-YL]methylidene}-5-imino-2-methyl-5H,6H,7H-[1,3]thiazolo[3,2-A]pyrimidin-7-one
—— 6-(4-chlorophenyl)-N-[(2,4-dimethoxyphenyl)methylideneamino]-4-(trifluoromethyl)pyrimidin-1-ium-2-amine —— C20H17ClF3N4O2+
6-(4-chlorophenyl)-N-[(2,4-dimethoxyphenyl)methylideneamino]-4-(trifluoromethyl)pyrimidin-1-ium-2-amine
—— (6E)-6-[[1-[(4-chlorophenyl)methyl]indol-3-yl]methylidene]-2-heptyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H28ClN5OS
(6E)-6-[[1-[(4-chlorophenyl)methyl]indol-3-yl]methylidene]-2-heptyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6R)-6-[4-[[(2R)-2-ethylhexanoyl]amino]phenyl]-8-methyl-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C29H36N4O2S
(6R)-6-[4-[[(2R)-2-ethylhexanoyl]amino]phenyl]-8-methyl-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— 6-tert-butyl-2-[[(E)-3-(4-tert-butylphenyl)prop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C26H34N2O2S
6-tert-butyl-2-[[(E)-3-(4-tert-butylphenyl)prop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— (6R)-6-[3-[(3-methoxyphenyl)carbamoylamino]phenyl]-8-methyl-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C29H29N5O3S
(6R)-6-[3-[(3-methoxyphenyl)carbamoylamino]phenyl]-8-methyl-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— (6R)-6-[4-[(2,3-dimethylphenyl)carbamoylamino]phenyl]-N,8-dimethyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C25H29N5O2S
(6R)-6-[4-[(2,3-dimethylphenyl)carbamoylamino]phenyl]-N,8-dimethyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— (6R)-N,N,8-trimethyl-6-[4-(naphthalen-1-ylcarbamoylamino)phenyl]-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C28H29N5O2S
(6R)-N,N,8-trimethyl-6-[4-(naphthalen-1-ylcarbamoylamino)phenyl]-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— (6S)-6-[3-[(2-fluorobenzoyl)amino]phenyl]-8-methyl-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C28H25FN4O2S
(6S)-6-[3-[(2-fluorobenzoyl)amino]phenyl]-8-methyl-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— 6-ethoxy-2-N-[(1R)-1-(furan-2-yl)ethyl]pyridine-2,5-diamine —— C13H17N3O2
6-ethoxy-2-N-[(1R)-1-(furan-2-yl)ethyl]pyridine-2,5-diamine
—— 6-propan-2-yloxy-2-N-[(1S)-1-thiophen-2-ylethyl]pyridine-2,5-diamine —— C14H19N3OS
6-propan-2-yloxy-2-N-[(1S)-1-thiophen-2-ylethyl]pyridine-2,5-diamine
—— 6-ethoxy-2-N-[(1R)-1-thiophen-2-ylethyl]pyridine-2,5-diamine —— C13H17N3OS
6-ethoxy-2-N-[(1R)-1-thiophen-2-ylethyl]pyridine-2,5-diamine
—— 6-amino-1-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]pyrimidine-2,4-dione —— C10H15N3O3
6-amino-1-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]pyrimidine-2,4-dione
—— 6-amino-1-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]pyrimidine-2,4-dione —— C10H15N3O3
6-amino-1-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]pyrimidine-2,4-dione
—— 6-ethoxy-2-N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]pyridine-2,5-diamine —— C13H21N3O2
6-ethoxy-2-N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]pyridine-2,5-diamine
—— 6-amino-1-[(1S)-1-cyclopropylethyl]pyrimidine-2,4-dione —— C9H13N3O2
6-amino-1-[(1S)-1-cyclopropylethyl]pyrimidine-2,4-dione
—— 6-N-[(1R)-1-cyclopropylethyl]-2,3-dihydro-1,4-benzodioxine-6,7-diamine —— C13H18N2O2
6-N-[(1R)-1-cyclopropylethyl]-2,3-dihydro-1,4-benzodioxine-6,7-diamine
—— 6-[[(1S)-1-cyclopropylethyl]amino]-5-nitro-1,3-dihydroindol-2-one —— C13H15N3O3
6-[[(1S)-1-cyclopropylethyl]amino]-5-nitro-1,3-dihydroindol-2-one
—— 6-[[(1S)-1-cyclopropylethyl]amino]pyridine-3-carboxylic acid —— C11H14N2O2
6-[[(1S)-1-cyclopropylethyl]amino]pyridine-3-carboxylic acid
—— 6-amino-1-[(1R)-1-cyclopropylethyl]pyrimidine-2,4-dione —— C9H13N3O2
6-amino-1-[(1R)-1-cyclopropylethyl]pyrimidine-2,4-dione
—— 6-methoxy-2-N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]pyridine-2,5-diamine —— C12H19N3O2
6-methoxy-2-N-[(1S)-1-[(2R)-oxolan-2-yl]ethyl]pyridine-2,5-diamine
—— 6-ethoxy-2-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]pyridine-2,5-diamine —— C13H21N3O2
6-ethoxy-2-N-[(1R)-1-[(2S)-oxolan-2-yl]ethyl]pyridine-2,5-diamine