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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6Z)-6-{3-bromo-4-[2-(4-tert-butylphenoxy)ethoxy]-5-ethoxybenzylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H33BrN4O4S
(6Z)-6-{3-bromo-4-[2-(4-tert-butylphenoxy)ethoxy]-5-ethoxybenzylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[2,5-dimethyl-1-(2-methyl-5-nitrophenyl)pyrrol-3-yl]methylidene]-5-imino-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H27N7O4S
(6Z)-6-[[2,5-dimethyl-1-(2-methyl-5-nitrophenyl)pyrrol-3-yl]methylidene]-5-imino-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z,10E)-9-hydroxy-3,6,10-trimethyl-3a,4,5,8,9,11a-hexahydro-3H-cyclodeca[b]furan-2-one —— C15H22O3
(6Z,10E)-9-hydroxy-3,6,10-trimethyl-3a,4,5,8,9,11a-hexahydro-3H-cyclodeca[b]furan-2-one
—— (6Z)-6-({3-Bromo-4-[2-(4-bromophenoxy)ethoxy]-5-methoxyphenyl}methylidene)-2-ethyl-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C23H20Br2N4O4S
(6Z)-6-({3-Bromo-4-[2-(4-bromophenoxy)ethoxy]-5-methoxyphenyl}methylidene)-2-ethyl-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6Z)-2-(2-chlorophenyl)-6-[3,5-dichloro-4-(2-phenoxyethoxy)benzylidene]-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H17Cl3N4O3S
(6Z)-2-(2-chlorophenyl)-6-[3,5-dichloro-4-(2-phenoxyethoxy)benzylidene]-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-({3-Bromo-5-methoxy-4-[2-(3-methylphenoxy)ethoxy]phenyl}methylidene)-2-ethyl-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C24H23BrN4O4S
(6Z)-6-({3-Bromo-5-methoxy-4-[2-(3-methylphenoxy)ethoxy]phenyl}methylidene)-2-ethyl-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6E)-2-butyl-6-[[2,5-dimethyl-1-(3-methylphenyl)pyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H25N5OS
(6E)-2-butyl-6-[[2,5-dimethyl-1-(3-methylphenyl)pyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[1-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-phenylhexanamide —— C27H34N4O4S
6-[1-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-phenylhexanamide
—— 6-[(5R,10bR)-9-bromo-5-pyridin-4-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C22H18BrN3O2
6-[(5R,10bR)-9-bromo-5-pyridin-4-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— (6S,7R)-6-(4-chlorophenyl)-N-(2-methoxyethyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H20ClN5O2S
(6S,7R)-6-(4-chlorophenyl)-N-(2-methoxyethyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6R,7S)-6-(4-chlorophenyl)-N-(2-methoxyethyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H20ClN5O2S
(6R,7S)-6-(4-chlorophenyl)-N-(2-methoxyethyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]hexanamide —— C26H39N3O5
6-(6,7-diethoxy-2,4-dioxo-1H-quinazolin-3-yl)-N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]hexanamide
—— (6R)-6-methyl-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanyl-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one —— C19H21N3O2S2
(6R)-6-methyl-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanyl-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one
—— (6R)-2-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]sulfanyl-6-methyl-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one —— C23H21N3O2S2
(6R)-2-[2-(2,3-dihydroindol-1-yl)-2-oxoethyl]sulfanyl-6-methyl-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-4-one
—— (6Z)-6-({3-Bromo-4-[2-(3,4-dimethylphenoxy)ethoxy]-5-methoxyphenyl}methylidene)-2-ethyl-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C25H25BrN4O4S
(6Z)-6-({3-Bromo-4-[2-(3,4-dimethylphenoxy)ethoxy]-5-methoxyphenyl}methylidene)-2-ethyl-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6S)-2-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]sulfanyl-6-methyl-3-(4-methylphenyl)-6,7-dihydrothieno[3,2-d]pyrimidin-4-one —— C25H25N3O2S2
(6S)-2-[2-(3,4-dihydro-2H-quinolin-1-yl)-2-oxoethyl]sulfanyl-6-methyl-3-(4-methylphenyl)-6,7-dihydrothieno[3,2-d]pyrimidin-4-one
—— (6Z)-4-phenyl-6-[(4-piperidin-1-ylsulfonylphenyl)hydrazinylidene]cyclohexa-2,4-dien-1-one —— C23H23N3O3S
(6Z)-4-phenyl-6-[(4-piperidin-1-ylsulfonylphenyl)hydrazinylidene]cyclohexa-2,4-dien-1-one
—— (6E)-6-{[2,5-dimethyl-1-(naphthalen-2-yl)-1H-pyrrol-3-yl]methylidene}-5-imino-2-(3-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H23N5OS
(6E)-6-{[2,5-dimethyl-1-(naphthalen-2-yl)-1H-pyrrol-3-yl]methylidene}-5-imino-2-(3-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2-hydroxy-6-[[4-nitro-2-(trifluoromethyl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C14H9F3N2O4
(6E)-2-hydroxy-6-[[4-nitro-2-(trifluoromethyl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-6-[[[(4Z)-4-(3H-1,3-benzoxazol-2-ylidene)-3-oxocyclohexa-1,5-dien-1-yl]amino]methylidene]-2,4-dichlorocyclohexa-2,4-dien-1-one —— C20H12Cl2N2O3
(6E)-6-[[[(4Z)-4-(3H-1,3-benzoxazol-2-ylidene)-3-oxocyclohexa-1,5-dien-1-yl]amino]methylidene]-2,4-dichlorocyclohexa-2,4-dien-1-one
—— (6Z)-6-{3-chloro-4-[(2-fluorobenzyl)oxy]-5-methoxybenzylidene}-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H20ClFN4O4S
(6Z)-6-{3-chloro-4-[(2-fluorobenzyl)oxy]-5-methoxybenzylidene}-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-{[1-(2-fluorobenzyl)-1H-pyrrol-2-yl]methylidene}-5-imino-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C18H11F4N5OS
(6Z)-6-{[1-(2-fluorobenzyl)-1H-pyrrol-2-yl]methylidene}-5-imino-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-{3-bromo-5-ethoxy-4-[2-(2-methylphenoxy)ethoxy]benzylidene}-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H25BrN4O4S
(6Z)-6-{3-bromo-5-ethoxy-4-[2-(2-methylphenoxy)ethoxy]benzylidene}-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-[[3-bromo-5-methoxy-4-[2-(2-methylphenoxy)ethoxy]phenyl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H25BrN4O4S
(6Z)-6-[[3-bromo-5-methoxy-4-[2-(2-methylphenoxy)ethoxy]phenyl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-({3-Bromo-5-methoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl}methylidene)-2-ethyl-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C24H23BrN4O4S
(6Z)-6-({3-Bromo-5-methoxy-4-[2-(4-methylphenoxy)ethoxy]phenyl}methylidene)-2-ethyl-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6Z)-6-{[1-(2-ethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H25N5O2S
(6Z)-6-{[1-(2-ethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6aS)-N-[(4-ethylphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C23H27N3O2
(6aS)-N-[(4-ethylphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aR)-N-[(3-bromophenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C21H22BrN3O2
(6aR)-N-[(3-bromophenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6Z)-3-pentoxy-6-[(4-pentylanilino)methylidene]cyclohexa-2,4-dien-1-one —— C23H31NO2
(6Z)-3-pentoxy-6-[(4-pentylanilino)methylidene]cyclohexa-2,4-dien-1-one
—— (6aR)-5-methyl-6-oxo-N-[2-(4-sulfamoylphenyl)ethyl]-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C22H26N4O4S
(6aR)-5-methyl-6-oxo-N-[2-(4-sulfamoylphenyl)ethyl]-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aR)-N-[[1-[(4-methylphenyl)methyl]piperidin-4-yl]methyl]-6-oxo-5,6a,7,8,9,10-hexahydropyrido[1,2-a]quinoxaline-3-carboxamide —— C27H34N4O2
(6aR)-N-[[1-[(4-methylphenyl)methyl]piperidin-4-yl]methyl]-6-oxo-5,6a,7,8,9,10-hexahydropyrido[1,2-a]quinoxaline-3-carboxamide
—— (6E)-4-bromo-6-[[2-phenoxy-5-(trifluoromethyl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C20H13BrF3NO2
(6E)-4-bromo-6-[[2-phenoxy-5-(trifluoromethyl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-2-methoxy-4-nitro-6-[[3-[2-nitro-4-(trifluoromethyl)anilino]propylamino]methylidene]cyclohexa-2,4-dien-1-one —— C18H17F3N4O6
(6Z)-2-methoxy-4-nitro-6-[[3-[2-nitro-4-(trifluoromethyl)anilino]propylamino]methylidene]cyclohexa-2,4-dien-1-one
—— (6aS)-N-[(2-methoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C22H25N3O3
(6aS)-N-[(2-methoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6Z)-6-{3-[2-(4-bromophenoxy)ethoxy]benzylidene}-2-(2-chlorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H18BrClN4O3S
(6Z)-6-{3-[2-(4-bromophenoxy)ethoxy]benzylidene}-2-(2-chlorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6aR)-N-[(4-ethoxy-3-methoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C24H29N3O4
(6aR)-N-[(4-ethoxy-3-methoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6Z)-2-cyclohexyl-5-imino-6-[(1-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}-1H-pyrrol-2-yl)methylidene]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H29N5O2S
(6Z)-2-cyclohexyl-5-imino-6-[(1-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}-1H-pyrrol-2-yl)methylidene]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-4-benzyl-6-[[[2-(4-fluorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C27H19FN2O2
(6Z)-4-benzyl-6-[[[2-(4-fluorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-[(3S,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(3-methoxypropyl)-4-oxo-1H-quinoline-3-carboxamide —— C21H29N3O5S
6-[(3S,5R)-3,5-dimethylpiperidin-1-yl]sulfonyl-N-(3-methoxypropyl)-4-oxo-1H-quinoline-3-carboxamide
—— 6-[[5-[(3R)-3-phenylpyrrolidin-1-yl]sulfonylthiophen-2-yl]methyl]pyrrolo[3,4-b]pyridine-5,7-dione —— C22H19N3O4S2
6-[[5-[(3R)-3-phenylpyrrolidin-1-yl]sulfonylthiophen-2-yl]methyl]pyrrolo[3,4-b]pyridine-5,7-dione
—— 6-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-[(4-methoxyphenyl)methyl]-[1,3]dioxolo[4,5-g]quinazolin-8-one —— C26H29N3O5S
6-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]sulfanyl-7-[(4-methoxyphenyl)methyl]-[1,3]dioxolo[4,5-g]quinazolin-8-one
—— (6aR)-N-(3-methoxypropyl)-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C18H25N3O3
(6aR)-N-(3-methoxypropyl)-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aR)-N-[(2,4-dimethoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C23H27N3O4
(6aR)-N-[(2,4-dimethoxyphenyl)methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— 6-[2-[(2S)-1-(2,6-diethylanilino)-1-oxobutan-2-yl]sulfanyl-4-oxothieno[3,2-d]pyrimidin-3-yl]hexanoic acid —— C26H33N3O4S2
6-[2-[(2S)-1-(2,6-diethylanilino)-1-oxobutan-2-yl]sulfanyl-4-oxothieno[3,2-d]pyrimidin-3-yl]hexanoic acid
—— 6-methoxy-1-[(4-methylphenyl)methyl]-3-[[[(2R)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid —— C28H30N2O3
6-methoxy-1-[(4-methylphenyl)methyl]-3-[[[(2R)-2-phenylpropyl]amino]methyl]indole-2-carboxylic acid
—— 6-(4-benzylpiperidine-1-carbonyl)-5-methyl-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one —— C28H34N4O3S
6-(4-benzylpiperidine-1-carbonyl)-5-methyl-3-[2-[(2S)-2-methylpiperidin-1-yl]-2-oxoethyl]thieno[2,3-d]pyrimidin-4-one
—— (6E)-4-bromo-6-[[2-[4-morpholin-4-yl-6-(N-phenylanilino)-1,3,5-triazin-2-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C26H24BrN7O2
(6E)-4-bromo-6-[[2-[4-morpholin-4-yl-6-(N-phenylanilino)-1,3,5-triazin-2-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6aR)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6a,7,8,9,10-hexahydropyrido[1,2-a]quinoxalin-6-one —— C20H25N3O4
(6aR)-3-(1,4-dioxa-8-azaspiro[4.5]decane-8-carbonyl)-5,6a,7,8,9,10-hexahydropyrido[1,2-a]quinoxalin-6-one
—— (6aS)-N-[[1-[(4-chlorophenyl)methyl]piperidin-4-yl]methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C27H33ClN4O2
(6aS)-N-[[1-[(4-chlorophenyl)methyl]piperidin-4-yl]methyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide
—— (6aS)-N-[3-[4-(4-methoxyphenyl)piperazin-1-yl]propyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide —— C28H37N5O3
(6aS)-N-[3-[4-(4-methoxyphenyl)piperazin-1-yl]propyl]-5-methyl-6-oxo-7,8,9,10-tetrahydro-6aH-pyrido[1,2-a]quinoxaline-3-carboxamide