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—— 6-(trans-3-aminocyclobutyl)-N~4~-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]pyrimidine-2,4-diamine —— C19H25N5O
6-(trans-3-aminocyclobutyl)-N~4~-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]pyrimidine-2,4-diamine
—— (6E)-6-[[4-[2-anilino-5-(1,1,2,2,3,3,3-heptafluoropropylsulfonyl)-3-nitroanilino]anilino]methylidene]-4-bromocyclohexa-2,4-dien-1-one —— C28H18BrF7N4O5S
(6E)-6-[[4-[2-anilino-5-(1,1,2,2,3,3,3-heptafluoropropylsulfonyl)-3-nitroanilino]anilino]methylidene]-4-bromocyclohexa-2,4-dien-1-one
—— 6-(3-aminocyclobutyl)-4-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]pyrimidine-2,4-diamine —— C16H25N7
6-(3-aminocyclobutyl)-4-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]pyrimidine-2,4-diamine
—— (6E)-6-[[4-(1,3-benzoxazol-2-yl)anilino]methylidene]-4,5-dibromo-2-ethoxycyclohexa-2,4-dien-1-one —— C22H16Br2N2O3
(6E)-6-[[4-(1,3-benzoxazol-2-yl)anilino]methylidene]-4,5-dibromo-2-ethoxycyclohexa-2,4-dien-1-one
—— 6-isobutyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-oxo-1,2-dihydropyrimidine-4-carboxamide —— C13H17N5O2S
6-isobutyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-oxo-1,2-dihydropyrimidine-4-carboxamide
—— 6-{[cis-3-(6-Morpholin-4-ylpyrimidin-4-yl)cyclobutyl]amino}pyrimidin-4-ol —— C16H20N6O2
6-{[cis-3-(6-Morpholin-4-ylpyrimidin-4-yl)cyclobutyl]amino}pyrimidin-4-ol
—— 6-[(5Z)-5-[[2-[3-(1H-imidazol-3-ium-3-yl)propylamino]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid —— C25H29N6O4S2+
6-[(5Z)-5-[[2-[3-(1H-imidazol-3-ium-3-yl)propylamino]-9-methyl-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]hexanoic acid
—— 6-(3-aminocyclobutyl)-N~4~-(2,5-dichlorobenzyl)pyrimidine-2,4-diamine —— C15H17Cl2N5
6-(3-aminocyclobutyl)-N~4~-(2,5-dichlorobenzyl)pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N-[(3-pyridin-3-ylisoxazol-5-yl)methyl]pyrimidin-4-amine —— C17H18N6O
6-(3-aminocyclobutyl)-N-[(3-pyridin-3-ylisoxazol-5-yl)methyl]pyrimidin-4-amine
—— 6-{(5Z)-5-[(2-{[3-(1H-imidazol-3-ium-1-yl)propyl]amino}-9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl)methylidene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl}hexanoate —— C25H28N6O4S2
6-{(5Z)-5-[(2-{[3-(1H-imidazol-3-ium-1-yl)propyl]amino}-9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl)methylidene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl}hexanoate
—— 6-{[2-(1-hydroxyethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]sulfonyl}-2H-1,4-benzoxazin-3(4H)-one —— C16H18N4O5S
6-{[2-(1-hydroxyethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]sulfonyl}-2H-1,4-benzoxazin-3(4H)-one
—— 6-{[4-(1,2-benzisothiazol-3-yl)piperazin-1-yl]carbonyl}-4,5-dihydropyridazin-3(2H)-one —— C16H17N5O2S
6-{[4-(1,2-benzisothiazol-3-yl)piperazin-1-yl]carbonyl}-4,5-dihydropyridazin-3(2H)-one
—— 6-{[2-(hydroxymethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]sulfonyl}-2H-1,4-benzoxazin-3(4H)-one —— C16H18N4O5S
6-{[2-(hydroxymethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]sulfonyl}-2H-1,4-benzoxazin-3(4H)-one
—— 6-(cis-3-aminocyclobutyl)-N-[(5-methyl-1H-imidazol-4-yl)methyl]pyrimidin-4-amine —— C13H18N6
6-(cis-3-aminocyclobutyl)-N-[(5-methyl-1H-imidazol-4-yl)methyl]pyrimidin-4-amine
—— 6-amino-N-[trans-3-(cyclobutylmethoxy)tetrahydro-2H-pyran-4-yl]nicotinamide —— C16H23N3O3
6-amino-N-[trans-3-(cyclobutylmethoxy)tetrahydro-2H-pyran-4-yl]nicotinamide
—— 6-methyl-3-sulfanylidene-4-[(Z)-(2,3,4-trimethoxyphenyl)methylideneamino]-2H-1,2,4-triazin-5-one —— C14H16N4O4S
6-methyl-3-sulfanylidene-4-[(Z)-(2,3,4-trimethoxyphenyl)methylideneamino]-2H-1,2,4-triazin-5-one
—— 6-(4-{[2-(Methylthio)pyrimidin-5-yl]methyl}piperazin-1-yl)nicotinonitrile —— C16H18N6S
6-(4-{[2-(Methylthio)pyrimidin-5-yl]methyl}piperazin-1-yl)nicotinonitrile
—— 6-({[6-(cis-3-Aminocyclobutyl)-2-methylpyrimidin-4-yl]amino}methyl)-2-methylpyrimidin-4-ol —— C15H20N6O
6-({[6-(cis-3-Aminocyclobutyl)-2-methylpyrimidin-4-yl]amino}methyl)-2-methylpyrimidin-4-ol
—— 6-(3-aminocyclobutyl)-N-(imidazo[1,2-a]pyridin-2-ylmethyl)pyrimidin-4-amine —— C16H18N6
6-(3-aminocyclobutyl)-N-(imidazo[1,2-a]pyridin-2-ylmethyl)pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)methyl]pyrimidin-4-amine —— C17H22N6OS
6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)methyl]pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N-(1,3-benzodioxol-5-ylmethyl)-2-(methoxymethyl)pyrimidin-4-amine —— C18H22N4O3
6-(cis-3-aminocyclobutyl)-N-(1,3-benzodioxol-5-ylmethyl)-2-(methoxymethyl)pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N-(2,6-dichlorobenzyl)pyrimidin-4-amine —— C15H16Cl2N4
6-(3-aminocyclobutyl)-N-(2,6-dichlorobenzyl)pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N-[(5-methyl-1H-imidazol-4-yl)methyl]-2-pyrrolidin-1-ylpyrimidin-4-amine —— C17H25N7
6-(cis-3-aminocyclobutyl)-N-[(5-methyl-1H-imidazol-4-yl)methyl]-2-pyrrolidin-1-ylpyrimidin-4-amine
—— 6-{1-[(5-amino-4-chloro-1H-pyrazol-3-yl)carbonyl]piperidin-4-yl}-2-methylpyrimidin-4-ol —— C14H17ClN6O2
6-{1-[(5-amino-4-chloro-1H-pyrazol-3-yl)carbonyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
—— 6-(3-aminocyclobutyl)-4-N-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-4-N-methylpyrimidine-2,4-diamine —— C19H22FN7
6-(3-aminocyclobutyl)-4-N-[[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl]-4-N-methylpyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~4~-[2-(4-ethoxyphenyl)ethyl]pyrimidine-2,4-diamine —— C18H25N5O
6-(3-aminocyclobutyl)-N~4~-[2-(4-ethoxyphenyl)ethyl]pyrimidine-2,4-diamine
—— 6-methyl-N-[rac-2-oxabicyclo[3.2.0]hept-6-yl]quinolin-4-amine —— C16H18N2O
6-methyl-N-[rac-2-oxabicyclo[3.2.0]hept-6-yl]quinolin-4-amine
—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-(2,3-dimethylbenzyl)pyrimidin-4-amine —— C20H26N4
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-(2,3-dimethylbenzyl)pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-2-methyl-N-[(4-phenyltetrahydro-2H-pyran-4-yl)methyl]pyrimidin-4-amine —— C21H28N4O
6-(cis-3-aminocyclobutyl)-2-methyl-N-[(4-phenyltetrahydro-2H-pyran-4-yl)methyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)pyrimidin-4-amine —— C15H17N7
6-(3-aminocyclobutyl)-N-(pyrazolo[1,5-a]pyrimidin-3-ylmethyl)pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N-[(2-ethoxypyridin-3-yl)methyl]-2-(methoxymethyl)pyrimidin-4-amine —— C18H25N5O2
6-(trans-3-aminocyclobutyl)-N-[(2-ethoxypyridin-3-yl)methyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[3-(1H-pyrazol-1-yl)propyl]pyrimidine-2,4-diamine —— C15H23N7
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[3-(1H-pyrazol-1-yl)propyl]pyrimidine-2,4-diamine
—— (6Z)-2-cyclohexyl-6-{4-[2-(3,4-dimethylphenoxy)ethoxy]-3-ethoxybenzylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C30H34N4O4S
(6Z)-2-cyclohexyl-6-{4-[2-(3,4-dimethylphenoxy)ethoxy]-3-ethoxybenzylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(3aR,7aS)-5-methyl-1,3,3a,4,7,7a-hexahydroisoindole-2-carbonyl]-1,4-dihydroquinoxaline-2,3-dione —— C18H19N3O3
6-[(3aR,7aS)-5-methyl-1,3,3a,4,7,7a-hexahydroisoindole-2-carbonyl]-1,4-dihydroquinoxaline-2,3-dione
—— 6-[2-(2,3-Dihydro-1,4-benzodioxin-2-YL)ethyl]-N,N-dimethylpyridazin-3-amine —— C16H19N3O2
6-[2-(2,3-Dihydro-1,4-benzodioxin-2-YL)ethyl]-N,N-dimethylpyridazin-3-amine
—— 6-isobutyl-2-methyl-N-[trans-3-(1,3-thiazol-4-ylmethoxy)tetrahydro-2H-pyran-4-yl]pyrimidine-4-carboxamide —— C19H26N4O3S
6-isobutyl-2-methyl-N-[trans-3-(1,3-thiazol-4-ylmethoxy)tetrahydro-2H-pyran-4-yl]pyrimidine-4-carboxamide
—— 6-(cis-3-aminocyclobutyl)-N-[2-(1,3-thiazol-4-yl)ethyl]pyrimidin-4-amine —— C13H17N5S
6-(cis-3-aminocyclobutyl)-N-[2-(1,3-thiazol-4-yl)ethyl]pyrimidin-4-amine
—— 6-methyl-N-[2-(5-methyl-2-furyl)ethyl]-4-oxo-4H-pyran-2-carboxamide —— C14H15NO4
6-methyl-N-[2-(5-methyl-2-furyl)ethyl]-4-oxo-4H-pyran-2-carboxamide
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-2,4-diamine —— C14H21N7
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[2-(1H-pyrazol-1-yl)ethyl]pyrimidine-2,4-diamine
—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[(1R)-1-(4-methoxyphenyl)ethyl]pyrimidin-4-amine —— C20H26N4O
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[(1R)-1-(4-methoxyphenyl)ethyl]pyrimidin-4-amine
—— 6-Methyl-N-[3-(4-methyl-1,3-thiazol-2-YL)propyl]pyridine-2-carboxamide —— C14H17N3OS
6-Methyl-N-[3-(4-methyl-1,3-thiazol-2-YL)propyl]pyridine-2-carboxamide
—— 6-(cis-3-aminocyclobutyl)-N~4~-methyl-N~4~-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]pyrimidine-2,4-diamine —— C19H26N6
6-(cis-3-aminocyclobutyl)-N~4~-methyl-N~4~-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]pyrimidine-2,4-diamine
—— (6E)-4,5-dibromo-6-[[2-[4,6-di(piperidin-1-yl)-1,3,5-triazin-2-yl]hydrazinyl]methylidene]-2-ethoxycyclohexa-2,4-dien-1-one —— C22H29Br2N7O2
(6E)-4,5-dibromo-6-[[2-[4,6-di(piperidin-1-yl)-1,3,5-triazin-2-yl]hydrazinyl]methylidene]-2-ethoxycyclohexa-2,4-dien-1-one
—— (6E)-6-[[[2-(2-bromophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-2,4-dinitrocyclohexa-2,4-dien-1-one —— C20H11BrN4O6
(6E)-6-[[[2-(2-bromophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-2,4-dinitrocyclohexa-2,4-dien-1-one
—— 6-(trans-3-aminocyclobutyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylpyrimidin-4-amine —— C15H22N6
6-(trans-3-aminocyclobutyl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylpyrimidin-4-amine
—— (6E)-4,5-dibromo-6-[[4-[[4-[[(Z)-(2,3-dibromo-5-methoxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]phenyl]methyl]anilino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C29H22Br4N2O4
(6E)-4,5-dibromo-6-[[4-[[4-[[(Z)-(2,3-dibromo-5-methoxy-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]phenyl]methyl]anilino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— (6E)-6-[[3-(1,3-benzoxazol-2-yl)-4-chloroanilino]methylidene]-4-bromo-2-ethoxycyclohexa-2,4-dien-1-one —— C22H16BrClN2O3
(6E)-6-[[3-(1,3-benzoxazol-2-yl)-4-chloroanilino]methylidene]-4-bromo-2-ethoxycyclohexa-2,4-dien-1-one
—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-(quinolin-2-ylmethyl)pyrimidin-4-amine —— C22H25N5
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-(quinolin-2-ylmethyl)pyrimidin-4-amine
—— 6-fluoro-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide —— C15H13FN4O4
6-fluoro-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
—— 6-(3-aminocyclobutyl)-N~4~-[2-(6-fluoro-1H-benzimidazol-2-yl)ethyl]pyrimidine-2,4-diamine —— C17H20FN7
6-(3-aminocyclobutyl)-N~4~-[2-(6-fluoro-1H-benzimidazol-2-yl)ethyl]pyrimidine-2,4-diamine