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—— (6Z)-2-cyclohexyl-6-(3-ethoxy-4-hydroxybenzylidene)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C20H22N4O3S
(6Z)-2-cyclohexyl-6-(3-ethoxy-4-hydroxybenzylidene)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-{3-chloro-5-methoxy-4-[2-(2-methoxyphenoxy)ethoxy]benzylidene}-2-(2-chlorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H22Cl2N4O5S
(6Z)-6-{3-chloro-5-methoxy-4-[2-(2-methoxyphenoxy)ethoxy]benzylidene}-2-(2-chlorophenyl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2-ethoxy-4-nitro-6-[[3-(trifluoromethyl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C16H13F3N2O4
(6E)-2-ethoxy-4-nitro-6-[[3-(trifluoromethyl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-2-Benzyl-6-({3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl}methylidene)-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C28H23FN4O3S
(6Z)-2-Benzyl-6-({3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl}methylidene)-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6Z)-6-[[2-[4-(3,5-dimethylpyrazol-1-yl)-6-(4-methylanilino)-1,3,5-triazin-2-yl]hydrazinyl]methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C23H24N8O2
(6Z)-6-[[2-[4-(3,5-dimethylpyrazol-1-yl)-6-(4-methylanilino)-1,3,5-triazin-2-yl]hydrazinyl]methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— 6-methoxy-N-[(1R)-1-pyridin-3-ylethyl]pyridine-3-carboxamide —— C14H15N3O2
6-methoxy-N-[(1R)-1-pyridin-3-ylethyl]pyridine-3-carboxamide
—— 6-[[(Z)-[7-[(8Z)-8-[(5-carboxypentylamino)methylidene]-1,6-dihydroxy-3-methyl-7-oxo-5-propan-2-ylnaphthalen-2-yl]-3,8-dihydroxy-6-methyl-2-oxo-4-propan-2-ylnaphthalen-1-ylidene]methyl]amino]hexanoic acid —— C42H52N2O10
6-[[(Z)-[7-[(8Z)-8-[(5-carboxypentylamino)methylidene]-1,6-dihydroxy-3-methyl-7-oxo-5-propan-2-ylnaphthalen-2-yl]-3,8-dihydroxy-6-methyl-2-oxo-4-propan-2-ylnaphthalen-1-ylidene]methyl]amino]hexanoic acid
—— (6E)-6-[[2-(7-chloroquinolin-4-yl)hydrazinyl]methylidene]-3-(diethylamino)cyclohexa-2,4-dien-1-one —— C20H21ClN4O
(6E)-6-[[2-(7-chloroquinolin-4-yl)hydrazinyl]methylidene]-3-(diethylamino)cyclohexa-2,4-dien-1-one
—— (6E)-2,4-dichloro-6-[[[(3E)-3-(4-methyl-3H-1,3-benzoxazol-2-ylidene)-4-oxocyclohexa-1,5-dien-1-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C21H14Cl2N2O3
(6E)-2,4-dichloro-6-[[[(3E)-3-(4-methyl-3H-1,3-benzoxazol-2-ylidene)-4-oxocyclohexa-1,5-dien-1-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-2,4-dibromo-6-[[3-(7-methylimidazo[1,2-a]pyridin-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C21H15Br2N3O
(6E)-2,4-dibromo-6-[[3-(7-methylimidazo[1,2-a]pyridin-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-6-[(2,5-dimethylanilino)methylidene]-2-methoxy-4-(morpholin-4-ylmethyl)cyclohexa-2,4-dien-1-one —— C21H26N2O3
(6E)-6-[(2,5-dimethylanilino)methylidene]-2-methoxy-4-(morpholin-4-ylmethyl)cyclohexa-2,4-dien-1-one
—— 6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide —— C26H29N5O3S
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(2R)-2-(dimethylamino)-2-thiophen-2-ylethyl]-1-propan-2-ylpyrazolo[3,4-b]pyridine-4-carboxamide
—— (6Z)-6-[[1-[2-(4-chlorophenoxy)ethyl]indol-3-yl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H20ClN5O2S
(6Z)-6-[[1-[2-(4-chlorophenoxy)ethyl]indol-3-yl]methylidene]-2-ethyl-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-2-Butyl-5-imino-6-(phenylmethylidene)-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C16H16N4OS
(6Z)-2-Butyl-5-imino-6-(phenylmethylidene)-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— 6-{2-[(E)-1-Cyclopropyl-1-phenylmethylidene]hydrazino}-1,3-dimethyl-2,4(1H,3H)-pyrimidinedione —— C16H18N4O2
6-{2-[(E)-1-Cyclopropyl-1-phenylmethylidene]hydrazino}-1,3-dimethyl-2,4(1H,3H)-pyrimidinedione
—— 6-methyl-5-[3-[(2S)-2-methylpiperidin-1-yl]-3-oxopropyl]-2-morpholin-4-yl-1H-pyrimidin-4-one —— C18H28N4O3
6-methyl-5-[3-[(2S)-2-methylpiperidin-1-yl]-3-oxopropyl]-2-morpholin-4-yl-1H-pyrimidin-4-one
—— (6E)-2-butyl-6-[[1-(3-chloro-4-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H24ClN5O2S
(6E)-2-butyl-6-[[1-(3-chloro-4-methoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-6-[[2-(1H-benzimidazol-2-yl)hydrazinyl]methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C15H14N4O2
(6E)-6-[[2-(1H-benzimidazol-2-yl)hydrazinyl]methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— 6-(2,5-dimethylfuran-3-yl)-3-methyl-N-[(2S)-pentan-2-yl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C19H23N3O3
6-(2,5-dimethylfuran-3-yl)-3-methyl-N-[(2S)-pentan-2-yl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-(2,5-dimethylfuran-3-yl)-N-[(2S)-1-methoxypropan-2-yl]-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C18H21N3O4
6-(2,5-dimethylfuran-3-yl)-N-[(2S)-1-methoxypropan-2-yl]-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-(2,5-dimethylfuran-3-yl)-3-methyl-N-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C24H26N4O3S
6-(2,5-dimethylfuran-3-yl)-3-methyl-N-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— (6Z)-6-[[1-(2,5-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(furan-2-yl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H21N5O4S
(6Z)-6-[[1-(2,5-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(furan-2-yl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(2,5-dimethylfuran-3-yl)-3-methyl-N-[(2R)-pentan-2-yl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide —— C19H23N3O3
6-(2,5-dimethylfuran-3-yl)-3-methyl-N-[(2R)-pentan-2-yl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
—— 6-(4-chlorophenyl)-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-5-methylsulfonylpyridine-3-carbonitrile —— C19H20ClN3O3S
6-(4-chlorophenyl)-2-[(2S,6S)-2,6-dimethylmorpholin-4-yl]-5-methylsulfonylpyridine-3-carbonitrile
—— (6R)-2-amino-4-cyclopropyl-6-thiophen-2-ylcyclohexa-2,4-diene-1,1,3-tricarbonitrile —— C16H12N4S
(6R)-2-amino-4-cyclopropyl-6-thiophen-2-ylcyclohexa-2,4-diene-1,1,3-tricarbonitrile
—— (6Z)-5-Imino-2-methyl-6-({1-[(4-methylphenyl)methyl]-1H-indol-3-YL}methylidene)-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C23H19N5OS
(6Z)-5-Imino-2-methyl-6-({1-[(4-methylphenyl)methyl]-1H-indol-3-YL}methylidene)-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6Z)-5-Imino-2-(2-methylpropyl)-6-(phenylmethylidene)-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C16H16N4OS
(6Z)-5-Imino-2-(2-methylpropyl)-6-(phenylmethylidene)-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6Z)-6-({4-[2-(4-Bromophenoxy)ethoxy]phenyl}methylidene)-5-imino-2-propyl-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C23H21BrN4O3S
(6Z)-6-({4-[2-(4-Bromophenoxy)ethoxy]phenyl}methylidene)-5-imino-2-propyl-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6Z)-6-[1-(hydroxyamino)decylidene]-4-methylcyclohexa-2,4-dien-1-one —— C17H27NO2
(6Z)-6-[1-(hydroxyamino)decylidene]-4-methylcyclohexa-2,4-dien-1-one
—— (6Z)-4-chloro-6-[[4-(5,6-dimethyl-1,3-benzoxazol-2-yl)anilino]methylidene]-3,5-dimethyl-2-nitrocyclohexa-2,4-dien-1-one —— C24H20ClN3O4
(6Z)-4-chloro-6-[[4-(5,6-dimethyl-1,3-benzoxazol-2-yl)anilino]methylidene]-3,5-dimethyl-2-nitrocyclohexa-2,4-dien-1-one
—— (6Z)-3-methoxy-6-[1-[(2E)-2-(3-methyl-1,3-benzothiazol-2-ylidene)hydrazinyl]ethylidene]cyclohexa-2,4-dien-1-one —— C17H17N3O2S
(6Z)-3-methoxy-6-[1-[(2E)-2-(3-methyl-1,3-benzothiazol-2-ylidene)hydrazinyl]ethylidene]cyclohexa-2,4-dien-1-one
—— (6E)-4-nitro-6-[(1-phenylethylamino)methylidene]cyclohexa-2,4-dien-1-one —— C15H14N2O3
(6E)-4-nitro-6-[(1-phenylethylamino)methylidene]cyclohexa-2,4-dien-1-one
—— 6-[(2R)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]sulfonyl-1,4-dihydroquinoxaline-2,3-dione —— C20H21N3O6S
6-[(2R)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]sulfonyl-1,4-dihydroquinoxaline-2,3-dione
—— (6Z)-2-butyl-5-imino-6-{4-[2-(4-methoxyphenoxy)ethoxy]benzylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H26N4O4S
(6Z)-2-butyl-5-imino-6-{4-[2-(4-methoxyphenoxy)ethoxy]benzylidene}-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-[(2S)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]sulfonyl-1,4-dihydroquinoxaline-2,3-dione —— C20H21N3O6S
6-[(2S)-2-(3,4-dimethoxyphenyl)pyrrolidin-1-yl]sulfonyl-1,4-dihydroquinoxaline-2,3-dione
—— 6-chloro-2-[[(2R)-oxolan-2-yl]methylsulfanyl]-1H-benzimidazole —— C12H13ClN2OS
6-chloro-2-[[(2R)-oxolan-2-yl]methylsulfanyl]-1H-benzimidazole
—— (6Z)-6-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2-dihydropyrazol-3-ylidene]-3,4-dimethylcyclohexa-2,4-dien-1-one —— C19H18N2O3
(6Z)-6-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2-dihydropyrazol-3-ylidene]-3,4-dimethylcyclohexa-2,4-dien-1-one
—— (6Z)-4-chloro-6-[[3-(5,6-dimethyl-1,3-benzoxazol-2-yl)anilino]methylidene]-3,5-dimethyl-2-nitrocyclohexa-2,4-dien-1-one —— C24H20ClN3O4
(6Z)-4-chloro-6-[[3-(5,6-dimethyl-1,3-benzoxazol-2-yl)anilino]methylidene]-3,5-dimethyl-2-nitrocyclohexa-2,4-dien-1-one
—— 6-[2-(2,3-dihydro-1,4-benzodioxin-6-ylimino)-3-[[(2R)-oxolan-2-yl]methyl]-1,3-thiazol-4-yl]-4H-1,4-benzoxazin-3-one —— C24H23N3O5S
6-[2-(2,3-dihydro-1,4-benzodioxin-6-ylimino)-3-[[(2R)-oxolan-2-yl]methyl]-1,3-thiazol-4-yl]-4H-1,4-benzoxazin-3-one
—— (6Z)-6-{3-chloro-5-ethoxy-4-[(2-nitrobenzyl)oxy]benzylidene}-5-imino-2-methyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H18ClN5O5S
(6Z)-6-{3-chloro-5-ethoxy-4-[(2-nitrobenzyl)oxy]benzylidene}-5-imino-2-methyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-4-bromo-6-[[[2-(3,4-dichlorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-2-nitrocyclohexa-2,4-dien-1-one —— C20H10BrCl2N3O4
(6E)-4-bromo-6-[[[2-(3,4-dichlorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-2-nitrocyclohexa-2,4-dien-1-one
—— 6-(3,5-dimethylpyrazol-1-yl)-2-N-[(Z)-1-(4-fluorophenyl)ethylideneamino]-4-N-(4-methylphenyl)-1,3,5-triazine-2,4-diamine —— C23H23FN8
6-(3,5-dimethylpyrazol-1-yl)-2-N-[(Z)-1-(4-fluorophenyl)ethylideneamino]-4-N-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
—— (6Z)-6-[1-(hydroxyamino)hexylidene]-3-methylcyclohexa-2,4-dien-1-one —— C13H19NO2
(6Z)-6-[1-(hydroxyamino)hexylidene]-3-methylcyclohexa-2,4-dien-1-one
—— (6E)-4-bromo-6-[(2-sulfanylethylamino)methylidene]cyclohexa-2,4-dien-1-one —— C9H10BrNOS
(6E)-4-bromo-6-[(2-sulfanylethylamino)methylidene]cyclohexa-2,4-dien-1-one
—— 6-[(2S)-2-benzylpyrrolidin-1-yl]sulfonyl-1,4-dihydroquinoxaline-2,3-dione —— C19H19N3O4S
6-[(2S)-2-benzylpyrrolidin-1-yl]sulfonyl-1,4-dihydroquinoxaline-2,3-dione
—— 6-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonylamino)-N-[(1R)-2-methyl-1-phenylpropyl]hexanamide —— C24H32N2O5S
6-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonylamino)-N-[(1R)-2-methyl-1-phenylpropyl]hexanamide
—— (6Z)-3-(benzylsulfanyl)-6-{4-[(4-chlorobenzyl)oxy]-3-ethoxybenzylidene}-5-imino-5,6-dihydro-7H-[1,2,4]thiadiazolo[4,5-a]pyrimidin-7-one —— C28H23ClN4O3S2
(6Z)-3-(benzylsulfanyl)-6-{4-[(4-chlorobenzyl)oxy]-3-ethoxybenzylidene}-5-imino-5,6-dihydro-7H-[1,2,4]thiadiazolo[4,5-a]pyrimidin-7-one
—— (6Z)-6-[(3,4-dichlorophenyl)hydrazinylidene]-4-phenylcyclohexa-2,4-dien-1-one —— C18H12Cl2N2O
(6Z)-6-[(3,4-dichlorophenyl)hydrazinylidene]-4-phenylcyclohexa-2,4-dien-1-one
—— 6-chloro-N-[(R)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]-2H-chromene-3-carboxamide —— C23H22ClN3O4
6-chloro-N-[(R)-(3,5-dimethoxyphenyl)-(1-methylimidazol-2-yl)methyl]-2H-chromene-3-carboxamide
—— (6Z)-6-{[1-(2,4-dimethylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H25N5O2S
(6Z)-6-{[1-(2,4-dimethylphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one