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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6E)-2-butyl-6-[[5-(4-chlorophenyl)furan-2-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C20H17ClN4O2S
(6E)-2-butyl-6-[[5-(4-chlorophenyl)furan-2-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6S)-2-[(4-fluorophenyl)methyl]-2,8-diazaspiro[5.5]undecan-1-one —— C16H21FN2O
(6S)-2-[(4-fluorophenyl)methyl]-2,8-diazaspiro[5.5]undecan-1-one
—— (6E)-6-({2,5-dimethyl-1-[2-(2-methylphenoxy)ethyl]-1H-indol-3-yl}methylidene)-5-imino-2-(3-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C32H29N5O2S
(6E)-6-({2,5-dimethyl-1-[2-(2-methylphenoxy)ethyl]-1H-indol-3-yl}methylidene)-5-imino-2-(3-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6R)-2-[(4-bromophenyl)methyl]-2,8-diazaspiro[5.5]undecan-1-one —— C16H21BrN2O
(6R)-2-[(4-bromophenyl)methyl]-2,8-diazaspiro[5.5]undecan-1-one
—— (6S)-2-benzyl-2,8-diazaspiro[5.5]undecan-1-one —— C16H22N2O
(6S)-2-benzyl-2,8-diazaspiro[5.5]undecan-1-one
—— 6-chloro-4-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methylchromen-2-one —— C23H22ClFN4O2S
6-chloro-4-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methylchromen-2-one
—— 6-nitro-2-[(Z)-thiophen-2-ylmethylideneamino]benzo[de]isoquinoline-1,3-dione —— C17H9N3O4S
6-nitro-2-[(Z)-thiophen-2-ylmethylideneamino]benzo[de]isoquinoline-1,3-dione
—— 6-amino-1,3-dimethyl-5-[(2R)-2-[[4-(4-methylphenyl)-1,3-thiazol-2-yl]sulfanyl]propanoyl]pyrimidine-2,4-dione —— C19H20N4O3S2
6-amino-1,3-dimethyl-5-[(2R)-2-[[4-(4-methylphenyl)-1,3-thiazol-2-yl]sulfanyl]propanoyl]pyrimidine-2,4-dione
—— 6-amino-5-[2-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]-1-propylpyrimidine-2,4-dione —— C21H26FN7O3S
6-amino-5-[2-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]-1-propylpyrimidine-2,4-dione
—— 6-amino-5-[2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]-1-propylpyrimidine-2,4-dione —— C21H26FN7O3S
6-amino-5-[2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]-1-propylpyrimidine-2,4-dione
—— 6-amino-5-[(2R)-2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-1,3-dimethylpyrimidine-2,4-dione —— C21H26FN7O3S
6-amino-5-[(2R)-2-[[5-[(1R)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanyl]propanoyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-chloro-4-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methylchromen-2-one —— C23H22ClFN4O2S
6-chloro-4-[[5-[(1S)-1-(dimethylamino)ethyl]-4-(4-fluorophenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-7-methylchromen-2-one
—— (6Z)-6-(3-ethoxy-4-{2-[2-(4-methylphenoxy)ethoxy]ethoxy}benzylidene)-5-imino-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H25F3N4O5S
(6Z)-6-(3-ethoxy-4-{2-[2-(4-methylphenoxy)ethoxy]ethoxy}benzylidene)-5-imino-2-(trifluoromethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6-methoxy-2-oxo-3a,8b-dihydro-1H-furo[2,3-b][1]benzofuran-8-yl) (2Z)-2-(5-oxooxolan-2-ylidene)acetate —— C17H14O8
(6-methoxy-2-oxo-3a,8b-dihydro-1H-furo[2,3-b][1]benzofuran-8-yl) (2Z)-2-(5-oxooxolan-2-ylidene)acetate
—— 6-hydroxy-5-nitro-2-{(E)-2-[3-(prop-2-en-1-yloxy)phenyl]ethenyl}pyrimidin-4(3H)-one —— C15H13N3O5
6-hydroxy-5-nitro-2-{(E)-2-[3-(prop-2-en-1-yloxy)phenyl]ethenyl}pyrimidin-4(3H)-one
—— (6E)-4-[(3-bromo-4-methoxyphenyl)methylideneamino]-6-(5-ethyl-3H-1,3-benzoxazol-2-ylidene)cyclohexa-2,4-dien-1-one —— C23H19BrN2O3
(6E)-4-[(3-bromo-4-methoxyphenyl)methylideneamino]-6-(5-ethyl-3H-1,3-benzoxazol-2-ylidene)cyclohexa-2,4-dien-1-one
—— (6Z)-6-[[(1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]methylidene]cyclohexa-2,4-dien-1-one —— C17H23NO
(6Z)-6-[[(1,3,3-trimethyl-2-bicyclo[2.2.1]heptanyl)amino]methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-2-cyclohexyl-6-{3-ethoxy-4-[2-(3-methylphenoxy)ethoxy]benzylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C29H32N4O4S
(6Z)-2-cyclohexyl-6-{3-ethoxy-4-[2-(3-methylphenoxy)ethoxy]benzylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6,7-dimethyl-N-[(2R)-2-phenylpropyl]-2-thiophen-2-ylquinoline-4-carboxamide —— C25H24N2OS
6,7-dimethyl-N-[(2R)-2-phenylpropyl]-2-thiophen-2-ylquinoline-4-carboxamide
—— (6Z)-6-[[1-(2,4-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H28N6O5S
(6Z)-6-[[1-(2,4-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2,4-dibromo-6-[[3-(5,6-dimethyl-1,3-benzoxazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C22H16Br2N2O2
(6E)-2,4-dibromo-6-[[3-(5,6-dimethyl-1,3-benzoxazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-6-(3-ethoxy-4-{2-[2-(prop-2-en-1-yl)phenoxy]ethoxy}benzylidene)-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C32H30N4O5S
(6Z)-6-(3-ethoxy-4-{2-[2-(prop-2-en-1-yl)phenoxy]ethoxy}benzylidene)-5-imino-2-(phenoxymethyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3,4-dimethoxyphenyl)-7-[4-[[(3S)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C24H33N7O2
6-(3,4-dimethoxyphenyl)-7-[4-[[(3S)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— (6E)-4-bromo-2-chloro-6-[[[2-(3,4-dichlorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one —— C20H10BrCl3N2O2
(6E)-4-bromo-2-chloro-6-[[[2-(3,4-dichlorophenyl)-1,3-benzoxazol-5-yl]amino]methylidene]cyclohexa-2,4-dien-1-one
—— (6-chloropyridin-3-yl)-[(1S)-6,7-dimethoxy-1-(4-methoxyphenyl)-3,4-dihydro-1H-isoquinolin-2-yl]methanone —— C24H23ClN2O4
(6-chloropyridin-3-yl)-[(1S)-6,7-dimethoxy-1-(4-methoxyphenyl)-3,4-dihydro-1H-isoquinolin-2-yl]methanone
—— (6Z)-6-{3-bromo-4-[2-(4-bromophenoxy)ethoxy]-5-ethoxybenzylidene}-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H22Br2N4O4S
(6Z)-6-{3-bromo-4-[2-(4-bromophenoxy)ethoxy]-5-ethoxybenzylidene}-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-({3-Bromo-4-[2-(2,4-dimethylphenoxy)ethoxy]-5-methoxyphenyl}methylidene)-5-imino-2-methyl-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C24H23BrN4O4S
(6Z)-6-({3-Bromo-4-[2-(2,4-dimethylphenoxy)ethoxy]-5-methoxyphenyl}methylidene)-5-imino-2-methyl-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6E)-2-bromo-6-[[5-[[3-[[(E)-(5-bromo-3-chloro-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]-4-hydroxyphenyl]methyl]-2-hydroxyanilino]methylidene]-4-chlorocyclohexa-2,4-dien-1-one —— C27H18Br2Cl2N2O4
(6E)-2-bromo-6-[[5-[[3-[[(E)-(5-bromo-3-chloro-6-oxocyclohexa-2,4-dien-1-ylidene)methyl]amino]-4-hydroxyphenyl]methyl]-2-hydroxyanilino]methylidene]-4-chlorocyclohexa-2,4-dien-1-one
—— (6E)-6-[[(5-chloropyridin-2-yl)amino]methylidene]-3-(diethylamino)cyclohexa-2,4-dien-1-one —— C16H18ClN3O
(6E)-6-[[(5-chloropyridin-2-yl)amino]methylidene]-3-(diethylamino)cyclohexa-2,4-dien-1-one
—— [6-[2-(3,7-dimethylocta-1,6-dien-3-yloxy)-4,5-dihydroxy-6-(hydroxymethyl)oxan-3-yl]oxy-4,5-dihydroxy-2-methyloxan-3-yl] (2E)-6-[3,5-dihydroxy-6-(hydroxymethyl)-4-oxooxan-2-yl]oxy-2,6-dimethylocta-2,7-dienoate —— C38H60O17
[6-[2-(3,7-dimethylocta-1,6-dien-3-yloxy)-4,5-dihydroxy-6-(hydroxymethyl)oxan-3-yl]oxy-4,5-dihydroxy-2-methyloxan-3-yl] (2E)-6-[3,5-dihydroxy-6-(hydroxymethyl)-4-oxooxan-2-yl]oxy-2,6-dimethylocta-2,7-dienoate
—— 6-[4-(2-Phenylethenesulfonyl)piperazine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one —— C17H20N4O4S
6-[4-(2-Phenylethenesulfonyl)piperazine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
—— 6-Benzyl-7-(4-butylsulfonylpiperazin-1-yl)-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine —— C21H28N6O2S
6-Benzyl-7-(4-butylsulfonylpiperazin-1-yl)-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine
—— 6-(4-methoxyphenyl)-7-(4-methylsulfonyl-1,4-diazepan-1-yl)-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H22N6O3S
6-(4-methoxyphenyl)-7-(4-methylsulfonyl-1,4-diazepan-1-yl)-[1,2,4]triazolo[1,5-a]pyrimidine
—— 6-(3,4-dimethoxyphenyl)-N-[[(3S)-3-(dimethylamino)thiolan-3-yl]methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C20H26N6O2S
6-(3,4-dimethoxyphenyl)-N-[[(3S)-3-(dimethylamino)thiolan-3-yl]methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 6-bromo-N-[(Z)-(4-chlorophenyl)methylideneamino]-2-methylquinolin-4-amine —— C17H13BrClN3
6-bromo-N-[(Z)-(4-chlorophenyl)methylideneamino]-2-methylquinolin-4-amine
—— (6Z)-2-Benzyl-6-({3-ethoxy-4-[2-(2-methylphenoxy)ethoxy]phenyl}methylidene)-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one —— C30H28N4O4S
(6Z)-2-Benzyl-6-({3-ethoxy-4-[2-(2-methylphenoxy)ethoxy]phenyl}methylidene)-5-imino-5H,6H,7H-[1,3,4]thiadiazolo[3,2-A]pyrimidin-7-one
—— (6E)-6-[[3-(5,7-dimethyl-1,3-benzoxazol-2-yl)anilino]methylidene]-2,4-dinitrocyclohexa-2,4-dien-1-one —— C22H16N4O6
(6E)-6-[[3-(5,7-dimethyl-1,3-benzoxazol-2-yl)anilino]methylidene]-2,4-dinitrocyclohexa-2,4-dien-1-one
—— 6-(4-methoxyphenyl)-7-[4-[[(3R)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C23H31N7O
6-(4-methoxyphenyl)-7-[4-[[(3R)-1-methylpiperidin-3-yl]methyl]piperazin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— (6E)-6-[[[2-(4-tert-butylphenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-4-chloro-3,5-dimethylcyclohexa-2,4-dien-1-one —— C26H25ClN2O2
(6E)-6-[[[2-(4-tert-butylphenyl)-1,3-benzoxazol-5-yl]amino]methylidene]-4-chloro-3,5-dimethylcyclohexa-2,4-dien-1-one
—— (6Z)-5-imino-6-{2-[(2-methylbenzyl)oxy]benzylidene}-2-[(2-methylphenoxy)methyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H24N4O3S
(6Z)-5-imino-6-{2-[(2-methylbenzyl)oxy]benzylidene}-2-[(2-methylphenoxy)methyl]-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3,4-dimethoxyphenyl)-N-[[(3R)-3-(dimethylamino)thiolan-3-yl]methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C20H26N6O2S
6-(3,4-dimethoxyphenyl)-N-[[(3R)-3-(dimethylamino)thiolan-3-yl]methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— (6-chloropyridin-3-yl)-[4-[(2S)-2-(3-methoxyphenyl)-2-[(4-methylphenyl)methoxy]ethyl]piperazin-1-yl]methanone —— C27H30ClN3O3
(6-chloropyridin-3-yl)-[4-[(2S)-2-(3-methoxyphenyl)-2-[(4-methylphenyl)methoxy]ethyl]piperazin-1-yl]methanone
—— 6-bromo-3-[2-[(2Z)-2-[(2-chlorophenyl)methylidene]hydrazinyl]-1,3-thiazol-5-yl]chromen-2-one —— C19H11BrClN3O2S
6-bromo-3-[2-[(2Z)-2-[(2-chlorophenyl)methylidene]hydrazinyl]-1,3-thiazol-5-yl]chromen-2-one
—— (6Z)-6-{3-bromo-5-methoxy-4-[2-(2-methylphenoxy)ethoxy]benzylidene}-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H23BrN4O4S
(6Z)-6-{3-bromo-5-methoxy-4-[2-(2-methylphenoxy)ethoxy]benzylidene}-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-2-cyclohexyl-5-imino-6-(4-{2-[2-methoxy-4-(prop-2-en-1-yl)phenoxy]ethoxy}benzylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C30H32N4O4S
(6Z)-2-cyclohexyl-5-imino-6-(4-{2-[2-methoxy-4-(prop-2-en-1-yl)phenoxy]ethoxy}benzylidene)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-2-butyl-6-{4-[(2-chlorobenzyl)oxy]-3-methoxybenzylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H23ClN4O3S
(6Z)-2-butyl-6-{4-[(2-chlorobenzyl)oxy]-3-methoxybenzylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6Z)-6-(3-bromo-4-{2-[4-(butan-2-yl)phenoxy]ethoxy}-5-methoxybenzylidene)-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H29BrN4O4S
(6Z)-6-(3-bromo-4-{2-[4-(butan-2-yl)phenoxy]ethoxy}-5-methoxybenzylidene)-2-ethyl-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(4-methoxyphenyl)-7-[(3S)-3-(trifluoromethyl)piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H18F3N5O
6-(4-methoxyphenyl)-7-[(3S)-3-(trifluoromethyl)piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 6-[(E)-2-(3,4-dimethylphenyl)ethenyl]-3-(4-methoxybenzyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C21H20N4OS
6-[(E)-2-(3,4-dimethylphenyl)ethenyl]-3-(4-methoxybenzyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— (6,7-dimethyl-2-thiophen-2-ylquinolin-4-yl)-[(3R)-3-methylpiperidin-1-yl]methanone —— C22H24N2OS
(6,7-dimethyl-2-thiophen-2-ylquinolin-4-yl)-[(3R)-3-methylpiperidin-1-yl]methanone