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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-1-[(3,4-dimethoxyphenyl)methyl]-4-methyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H31N3O3
(6S)-1-[(3,4-dimethoxyphenyl)methyl]-4-methyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclobutanecarbonyl)-6-[[2-(3-fluorophenyl)phenyl]methyl]-4-methyl-1,4-diazepan-5-one —— C24H27FN2O2
(6S)-1-(cyclobutanecarbonyl)-6-[[2-(3-fluorophenyl)phenyl]methyl]-4-methyl-1,4-diazepan-5-one
—— (6R)-1-[(3-fluorophenyl)methyl]-4-methyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H26FN3O
(6R)-1-[(3-fluorophenyl)methyl]-4-methyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclopentanecarbonyl)-4-methyl-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one —— C25H30N2O2
(6S)-1-(cyclopentanecarbonyl)-4-methyl-6-[(2-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-methyl-1-(pyridin-4-ylmethyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H26N4O
(6S)-4-methyl-1-(pyridin-4-ylmethyl)-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-[(2-methoxyphenyl)methyl]-4-methyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O2
(6R)-1-[(2-methoxyphenyl)methyl]-4-methyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-4-methyl-6-[(4-phenylphenyl)methyl]-1-(pyridin-4-ylmethyl)-1,4-diazepan-5-one —— C25H27N3O
(6S)-4-methyl-6-[(4-phenylphenyl)methyl]-1-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
—— 6-[(2R)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-carbonyl]-1H-pyrimidine-2,4-dione —— C21H26N4O5
6-[(2R)-7-methoxy-1'-methylspiro[3,5-dihydro-1,4-benzoxazepine-2,4'-azepane]-4-carbonyl]-1H-pyrimidine-2,4-dione
—— (6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-methyl-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one —— C27H29N3O3
(6R)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-4-methyl-1-(2-pyridin-3-ylacetyl)-1,4-diazepan-5-one
—— (6R)-1-[(3,4-dimethoxyphenyl)methyl]-4-methyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C27H31N3O3
(6R)-1-[(3,4-dimethoxyphenyl)methyl]-4-methyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclopropylmethyl)-4-methyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C22H27N3O
(6S)-1-(cyclopropylmethyl)-4-methyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-methyl-1-(pyridin-4-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H26N4O
(6R)-4-methyl-1-(pyridin-4-ylmethyl)-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[[3-(4-fluorophenyl)phenyl]methyl]-4-methyl-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C25H26FN3O
(6R)-6-[[3-(4-fluorophenyl)phenyl]methyl]-4-methyl-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6S)-1-benzyl-4-methyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H27N3O
(6S)-1-benzyl-4-methyl-6-[(2-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[[3-(3-methoxyphenyl)phenyl]methyl]-4-methyl-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one —— C24H26N4O3
(6R)-6-[[3-(3-methoxyphenyl)phenyl]methyl]-4-methyl-1-(1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
—— (6S)-1-(cyclopropylmethyl)-4-methyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C22H27N3O
(6S)-1-(cyclopropylmethyl)-4-methyl-6-[(3-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-4-methyl-6-[(4-phenylphenyl)methyl]-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one —— C25H27N3O
(6R)-4-methyl-6-[(4-phenylphenyl)methyl]-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
—— (6R)-4-methyl-6-[(4-phenylphenyl)methyl]-1-(pyridin-4-ylmethyl)-1,4-diazepan-5-one —— C25H27N3O
(6R)-4-methyl-6-[(4-phenylphenyl)methyl]-1-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
—— 6-[[2-methoxy-5-(methoxymethyl)phenyl]methyl]-2-[(2R)-1-methylpiperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C23H32N4O2
6-[[2-methoxy-5-(methoxymethyl)phenyl]methyl]-2-[(2R)-1-methylpiperidin-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6S)-4-methyl-1-(pyridine-2-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C23H23N3O2S
(6S)-4-methyl-1-(pyridine-2-carbonyl)-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(2-methoxyacetyl)-4-methyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C20H24N2O3S
(6R)-1-(2-methoxyacetyl)-4-methyl-6-[(4-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-6-[[4-(4-methoxyphenyl)phenyl]methyl]-4-methyl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one —— C24H27N5O3
(6R)-6-[[4-(4-methoxyphenyl)phenyl]methyl]-4-methyl-1-[2-(1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
—— 6-[1-[2-(dimethylamino)pyrimidine-5-carbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C20H22N6O2
6-[1-[2-(dimethylamino)pyrimidine-5-carbonyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— 6-[(3R)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine —— C23H26FN5
6-[(3R)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine
—— (6R)-1-(1,3-dimethylpyrazole-4-carbonyl)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C25H28N4O3
(6R)-1-(1,3-dimethylpyrazole-4-carbonyl)-6-[[2-(4-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6R)-1-[(4-fluorophenyl)methyl]-4-methyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one —— C25H26FN3O
(6R)-1-[(4-fluorophenyl)methyl]-4-methyl-6-[(4-pyridin-3-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-cyclohexyl-2-[(2R)-1-(1,3-dimethylpyrazole-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N6O2
6-cyclohexyl-2-[(2R)-1-(1,3-dimethylpyrazole-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3R)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-4-ylpyrimidin-4-amine —— C24H28FN5O
6-[(3R)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-4-ylpyrimidin-4-amine
—— 6-cyclohexyl-2-[(2S)-1-(1,3-dimethylpyrazole-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C24H34N6O2
6-cyclohexyl-2-[(2S)-1-(1,3-dimethylpyrazole-4-carbonyl)piperidin-2-yl]-3,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— 6-[(3R)-1-[(2-methoxyphenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine —— C24H29N5O
6-[(3R)-1-[(2-methoxyphenyl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl]-N,N-dimethyl-2-pyridin-4-ylpyrimidin-4-amine —— C25H31N5O2
6-[1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl]-N,N-dimethyl-2-pyridin-4-ylpyrimidin-4-amine
—— 6-[(3R)-1-[(7-methoxy-1-benzofuran-2-yl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine —— C26H29N5O2
6-[(3R)-1-[(7-methoxy-1-benzofuran-2-yl)methyl]piperidin-3-yl]-N,N-dimethyl-2-pyridin-3-ylpyrimidin-4-amine
—— 6-methoxy-2-methyl-N-(1-methylpiperidin-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]quinoline-3-carboxamide —— C23H31N3O3
6-methoxy-2-methyl-N-(1-methylpiperidin-4-yl)-N-[[(2S)-oxolan-2-yl]methyl]quinoline-3-carboxamide
—— 6-(4-methylcyclohexyl)-2-[(2R)-1-(2-methylpyridine-3-carbonyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one —— C25H33N5O2
6-(4-methylcyclohexyl)-2-[(2R)-1-(2-methylpyridine-3-carbonyl)pyrrolidin-2-yl]-1,5,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-one
—— (6R)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(5-methyl-1H-pyrazole-4-carbonyl)-4-prop-2-enyl-1,4-diazepan-5-one —— C26H27FN4O2
(6R)-6-[[4-(2-fluorophenyl)phenyl]methyl]-1-(5-methyl-1H-pyrazole-4-carbonyl)-4-prop-2-enyl-1,4-diazepan-5-one
—— 6-[1-[(1,3-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-5H-pyrrolo[2,3-b]pyrazine —— C17H22N6
6-[1-[(1,3-dimethylpyrazol-4-yl)methyl]piperidin-4-yl]-5H-pyrrolo[2,3-b]pyrazine
—— (6S)-1-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O3
(6S)-1-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]-6-[(3-phenylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[1-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one —— C21H24N4O3
6-[1-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]piperidin-4-yl]-7H-1,7-naphthyridin-8-one
—— (6S)-1-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one —— C26H29N3O3
(6S)-1-[3-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]-6-[(4-phenylphenyl)methyl]-1,4-diazepan-5-one
—— (6R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one —— C27H29N3O3
(6R)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)-6-[(4-phenylphenyl)methyl]-4-prop-2-enyl-1,4-diazepan-5-one
—— (6R)-1-[(1-ethylimidazol-2-yl)methyl]-6-[[3-(4-fluorophenyl)phenyl]methyl]-4-methyl-1,4-diazepan-5-one —— C25H29FN4O
(6R)-1-[(1-ethylimidazol-2-yl)methyl]-6-[[3-(4-fluorophenyl)phenyl]methyl]-4-methyl-1,4-diazepan-5-one
—— (6R)-4-ethyl-1-(3-ethylimidazole-4-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one —— C24H28N4O2S
(6R)-4-ethyl-1-(3-ethylimidazole-4-carbonyl)-6-[(2-thiophen-2-ylphenyl)methyl]-1,4-diazepan-5-one
—— 6-[(3R)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]pyrrolidin-3-yl]-2-morpholin-4-yl-1H-pyrimidin-4-one —— C22H30N4O3
6-[(3R)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]pyrrolidin-3-yl]-2-morpholin-4-yl-1H-pyrimidin-4-one
—— (6R)-4-ethyl-1-(3-ethylimidazole-4-carbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H32N4O2
(6R)-4-ethyl-1-(3-ethylimidazole-4-carbonyl)-6-[[2-(4-methylphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— 6-fluoro-N-[(2R)-1-[(3S)-3-(2-methylsulfonylacetyl)piperidin-1-yl]-1-oxopropan-2-yl]-1H-indole-2-carboxamide —— C20H24FN3O5S
6-fluoro-N-[(2R)-1-[(3S)-3-(2-methylsulfonylacetyl)piperidin-1-yl]-1-oxopropan-2-yl]-1H-indole-2-carboxamide
—— (6S)-1-[2-(4-fluorophenyl)acetyl]-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H27FN2O3
(6S)-1-[2-(4-fluorophenyl)acetyl]-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-1-(cyclopropanecarbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C23H26N2O3
(6S)-1-(cyclopropanecarbonyl)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-6-[[4-(3,5-dimethylphenyl)phenyl]methyl]-4-methyl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one —— C26H28N4O2
(6S)-6-[[4-(3,5-dimethylphenyl)phenyl]methyl]-4-methyl-1-(pyrazine-2-carbonyl)-1,4-diazepan-5-one
—— (6R)-1-[2-(3-fluorophenyl)acetyl]-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one —— C27H27FN2O3
(6R)-1-[2-(3-fluorophenyl)acetyl]-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1,4-diazepan-5-one
—— (6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(3-phenylpropanoyl)-1,4-diazepan-5-one —— C28H30N2O3
(6S)-6-[[2-(2-methoxyphenyl)phenyl]methyl]-1-(3-phenylpropanoyl)-1,4-diazepan-5-one