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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-6-N-cyclopentyl-5,6-dimethyl-4-oxo-2-N-[3-(2-oxopyrrolidin-1-yl)propyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide —— C22H32N6O4
(6R)-6-N-cyclopentyl-5,6-dimethyl-4-oxo-2-N-[3-(2-oxopyrrolidin-1-yl)propyl]-7H-pyrazolo[1,5-a]pyrazine-2,6-dicarboxamide
—— (6R)-N-cyclohexyl-2-(4-ethoxyphenyl)-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H34N4O3
(6R)-N-cyclohexyl-2-(4-ethoxyphenyl)-6-methyl-4-oxo-5-propyl-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6S)-2-tert-butyl-5-(2-fluorophenyl)-6-methyl-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C23H31FN4O2
(6S)-2-tert-butyl-5-(2-fluorophenyl)-6-methyl-N-(3-methylbutyl)-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6R)-N-cyclohexyl-2-cyclopropyl-6-methyl-5-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C25H32N4O2
(6R)-N-cyclohexyl-2-cyclopropyl-6-methyl-5-[(4-methylphenyl)methyl]-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl (2S,3R)-1-butyl-2-(4-methoxyphenyl)-6-oxopiperidine-3-carboxylate —— C26H30ClNO6
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl (2S,3R)-1-butyl-2-(4-methoxyphenyl)-6-oxopiperidine-3-carboxylate
—— (6R)-6-(cycloheptylcarbamoyl)-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid —— C17H24N4O4
(6R)-6-(cycloheptylcarbamoyl)-5,6-dimethyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2S,3R)-1-butyl-2-(4-methoxyphenyl)-6-oxopiperidine-3-carboxylate —— C26H30N2O8
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2S,3R)-1-butyl-2-(4-methoxyphenyl)-6-oxopiperidine-3-carboxylate
—— 6-[(2R,6S)-2-(4-fluorophenyl)-6-pyridin-3-yl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one —— C21H18FN3O
6-[(2R,6S)-2-(4-fluorophenyl)-6-pyridin-3-yl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[4-[(S)-(3-chlorophenyl)-phenylmethyl]piperazin-1-yl]tetrazolo[5,1-a]phthalazine —— C25H22ClN7
6-[4-[(S)-(3-chlorophenyl)-phenylmethyl]piperazin-1-yl]tetrazolo[5,1-a]phthalazine
—— (6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2S,3S)-1-butyl-2-(4-methoxyphenyl)-6-oxopiperidine-3-carboxylate —— C26H30N2O8
(6-nitro-4H-1,3-benzodioxin-8-yl)methyl (2S,3S)-1-butyl-2-(4-methoxyphenyl)-6-oxopiperidine-3-carboxylate
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl (2R,3S)-1-butyl-2-(4-methoxyphenyl)-6-oxopiperidine-3-carboxylate —— C26H30ClNO6
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl (2R,3S)-1-butyl-2-(4-methoxyphenyl)-6-oxopiperidine-3-carboxylate
—— (6S)-N-(2,5-dimethoxyphenyl)-7-oxo-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C26H25N3O4S
(6S)-N-(2,5-dimethoxyphenyl)-7-oxo-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— (6S)-5-hexanoyl-9,9-dimethyl-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C25H30N2O2S
(6S)-5-hexanoyl-9,9-dimethyl-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R)-N-(2-ethylphenyl)-7-oxo-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C26H25N3O2S
(6R)-N-(2-ethylphenyl)-7-oxo-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— (6S)-6-(2-methoxyphenyl)-9,9-dimethyl-7-oxo-N-phenyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C29H29N3O3
(6S)-6-(2-methoxyphenyl)-9,9-dimethyl-7-oxo-N-phenyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— 6-[(2R,6R)-2-(4-fluorophenyl)-6-pyridin-3-yl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one —— C21H18FN3O
6-[(2R,6R)-2-(4-fluorophenyl)-6-pyridin-3-yl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one
—— (6R)-N-(3-ethoxypropyl)-6-(furan-2-yl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C25H31N3O4
(6R)-N-(3-ethoxypropyl)-6-(furan-2-yl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6S)-5-[2-(benzenesulfonyl)acetyl]-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C25H22N2O5S
(6S)-5-[2-(benzenesulfonyl)acetyl]-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-N-(4-fluorophenyl)-6-(2-methoxyphenyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C29H28FN3O3
(6S)-N-(4-fluorophenyl)-6-(2-methoxyphenyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R)-6-(furan-2-yl)-N-(2-methoxyethyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C23H27N3O4
(6R)-6-(furan-2-yl)-N-(2-methoxyethyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R)-N-(2-methoxyphenyl)-9,9-dimethyl-7-oxo-6-phenyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C29H29N3O3
(6R)-N-(2-methoxyphenyl)-9,9-dimethyl-7-oxo-6-phenyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R)-N-(5-chloro-2-methoxyphenyl)-7-oxo-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C25H22ClN3O3S
(6R)-N-(5-chloro-2-methoxyphenyl)-7-oxo-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R)-5-(2,5-dimethylphenyl)sulfonyl-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C25H24N2O3S2
(6R)-5-(2,5-dimethylphenyl)sulfonyl-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-5-(4-fluorophenyl)sulfonyl-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C23H19FN2O4S
(6R)-5-(4-fluorophenyl)sulfonyl-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(4-fluorophenyl)-N-(2-methoxyethyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C25H28FN3O3
(6S)-6-(4-fluorophenyl)-N-(2-methoxyethyl)-9,9-dimethyl-7-oxo-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R)-6-(furan-2-yl)-5-(2-morpholin-4-yl-2-oxoethyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C23H25N3O4
(6R)-6-(furan-2-yl)-5-(2-morpholin-4-yl-2-oxoethyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-5-[2-(1H-benzimidazol-2-ylsulfanyl)acetyl]-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C26H22N4O3S
(6R)-5-[2-(1H-benzimidazol-2-ylsulfanyl)acetyl]-6-(furan-2-yl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-6-(furan-2-yl)-5-(4-methylphenyl)sulfonyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C24H22N2O4S
(6R)-6-(furan-2-yl)-5-(4-methylphenyl)sulfonyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-5-(4-fluorobenzoyl)-9,9-dimethyl-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C26H23FN2O2S
(6S)-5-(4-fluorobenzoyl)-9,9-dimethyl-6-thiophen-2-yl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R)-7-oxo-N-propyl-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide —— C21H23N3O2S
(6R)-7-oxo-N-propyl-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R)-5-(4-fluorobenzoyl)-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C24H19FN2O2S
(6R)-5-(4-fluorobenzoyl)-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(furan-2-yl)-9,9-dimethyl-7-oxo-N-propyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C23H27N3O3
(6S)-6-(furan-2-yl)-9,9-dimethyl-7-oxo-N-propyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6S)-5-(4-methylbenzoyl)-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C25H22N2O2S
(6S)-5-(4-methylbenzoyl)-6-thiophen-2-yl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(furan-2-yl)-9,9-dimethyl-7-oxo-N-[[(2R)-oxolan-2-yl]methyl]-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C25H29N3O4
(6S)-6-(furan-2-yl)-9,9-dimethyl-7-oxo-N-[[(2R)-oxolan-2-yl]methyl]-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— (6R)-6-(furan-2-yl)-9,9-dimethyl-7-oxo-N-[[(2S)-oxolan-2-yl]methyl]-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide —— C25H29N3O4
(6R)-6-(furan-2-yl)-9,9-dimethyl-7-oxo-N-[[(2S)-oxolan-2-yl]methyl]-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepine-5-carboxamide
—— 6-[(2S,6S)-2-(4-fluorophenyl)-6-pyridin-2-yl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one —— C21H18FN3O
6-[(2S,6S)-2-(4-fluorophenyl)-6-pyridin-2-yl-1,3-diazinan-4-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(R)-amino(1,3-benzodioxol-5-yl)methyl]-3,4-dihydro-1H-quinolin-2-one —— C17H16N2O3
6-[(R)-amino(1,3-benzodioxol-5-yl)methyl]-3,4-dihydro-1H-quinolin-2-one
—— 6-[(1S)-1-amino-2-(3-methoxyphenyl)ethyl]-3,4-dihydro-1H-quinolin-2-one —— C18H20N2O2
6-[(1S)-1-amino-2-(3-methoxyphenyl)ethyl]-3,4-dihydro-1H-quinolin-2-one
—— 6-[(R)-amino-(3-methoxy-4-methylphenyl)methyl]-3,4-dihydro-1H-quinolin-2-one —— C18H20N2O2
6-[(R)-amino-(3-methoxy-4-methylphenyl)methyl]-3,4-dihydro-1H-quinolin-2-one
—— 6-[(1R,2S)-1-amino-2-phenylbutyl]-3,4-dihydro-1H-quinolin-2-one —— C19H22N2O
6-[(1R,2S)-1-amino-2-phenylbutyl]-3,4-dihydro-1H-quinolin-2-one
—— 6-[(R)-amino-(4-propan-2-ylphenyl)methyl]-3,4-dihydro-1H-quinolin-2-one —— C19H22N2O
6-[(R)-amino-(4-propan-2-ylphenyl)methyl]-3,4-dihydro-1H-quinolin-2-one
—— 6-[(S)-amino-(2-ethoxyphenyl)methyl]-3,4-dihydro-1H-quinolin-2-one —— C18H20N2O2
6-[(S)-amino-(2-ethoxyphenyl)methyl]-3,4-dihydro-1H-quinolin-2-one
—— 6-[(S)-amino(1,3-benzodioxol-5-yl)methyl]-3,4-dihydro-1H-quinolin-2-one —— C17H16N2O3
6-[(S)-amino(1,3-benzodioxol-5-yl)methyl]-3,4-dihydro-1H-quinolin-2-one
—— 6-[(S)-amino(2,3-dihydro-1H-inden-5-yl)methyl]-3,4-dihydro-1H-quinolin-2-one —— C19H20N2O
6-[(S)-amino(2,3-dihydro-1H-inden-5-yl)methyl]-3,4-dihydro-1H-quinolin-2-one
—— 6-[(1R)-1-amino-2-methyl-2-phenylpropyl]-3,4-dihydro-1H-quinolin-2-one —— C19H22N2O
6-[(1R)-1-amino-2-methyl-2-phenylpropyl]-3,4-dihydro-1H-quinolin-2-one
—— 6-methoxy-4-[[4-[(2R)-2-phenylbutanoyl]piperazin-1-yl]methyl]chromen-2-one —— C25H28N2O4
6-methoxy-4-[[4-[(2R)-2-phenylbutanoyl]piperazin-1-yl]methyl]chromen-2-one
—— (6S)-5-[(2-chlorophenyl)methyl]-N-cycloheptyl-2-(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide —— C30H35ClN4O2
(6S)-5-[(2-chlorophenyl)methyl]-N-cycloheptyl-2-(4-ethylphenyl)-6-methyl-4-oxo-7H-pyrazolo[1,5-a]pyrazine-6-carboxamide
—— 6-[2-[(2S)-3-acetyl-2-(2,4-dimethoxyphenyl)-2H-1,3,4-oxadiazol-5-yl]ethylamino]-2H-1,2,4-triazine-3,5-dione —— C17H20N6O6
6-[2-[(2S)-3-acetyl-2-(2,4-dimethoxyphenyl)-2H-1,3,4-oxadiazol-5-yl]ethylamino]-2H-1,2,4-triazine-3,5-dione
—— 6-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-5-[(4-methylphenyl)sulfonylamino]pyridine-3-carboxylic acid —— C25H28N4O4S
6-[(3R)-3-methyl-4-(3-methylphenyl)piperazin-1-yl]-5-[(4-methylphenyl)sulfonylamino]pyridine-3-carboxylic acid
—— (6R)-1,3-dimethyl-6-(4-methylphenyl)sulfonyl-6H-pyrrolo[2,3-d]pyrimidine-2,4-dione —— C15H15N3O4S
(6R)-1,3-dimethyl-6-(4-methylphenyl)sulfonyl-6H-pyrrolo[2,3-d]pyrimidine-2,4-dione