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—— 6-[(1S,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(1,3,4-thiadiazol-2-yl)hexanamide —— C17H20N4O3S
6-[(1S,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(1,3,4-thiadiazol-2-yl)hexanamide
—— 6-[(1S,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(3-hydroxypyridin-2-yl)hexanamide —— C20H23N3O4
6-[(1S,2R,6S,7R)-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl]-N-(3-hydroxypyridin-2-yl)hexanamide
—— (6S,7S)-6-(4-methylphenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C22H25N5OS
(6S,7S)-6-(4-methylphenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(10bR)-7-methoxyspiro[3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclopentane]-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C22H24N2O4
6-[(10bR)-7-methoxyspiro[3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclopentane]-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-5-(3-hydroxyphenyl)-7-methoxy-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C24H22N2O4
6-[(5R,10bS)-5-(3-hydroxyphenyl)-7-methoxy-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-5-(2,4-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C25H24N2O4
6-[(5R,10bS)-5-(2,4-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-5-(2,3-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C25H24N2O4
6-[(5R,10bS)-5-(2,3-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-5-(2-methylpropyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C21H24N2O2
6-[(5R,10bS)-5-(2-methylpropyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— 6-(3-ethoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-3-(4-methylphenyl)-1,2-dihydropyrazolo[3,4-b]pyridine-4-carboxylic acid —— C22H19N3O4
6-(3-ethoxy-4-oxocyclohexa-2,5-dien-1-ylidene)-3-(4-methylphenyl)-1,2-dihydropyrazolo[3,4-b]pyridine-4-carboxylic acid
—— 6-[(10bS)-7-methoxy-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C19H20N2O3
6-[(10bS)-7-methoxy-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(10bR)-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C18H18N2O2
6-[(10bR)-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(10bR)-9-bromo-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C19H19BrN2O3
6-[(10bR)-9-bromo-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— 6-[(5S,10bS)-5-(2-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C23H20N2O2
6-[(5S,10bS)-5-(2-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6R,7S)-6-(4-methoxyphenyl)-3-methyl-N-[[(2S)-oxolan-2-yl]methyl]-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C18H23N5O3S
(6R,7S)-6-(4-methoxyphenyl)-3-methyl-N-[[(2S)-oxolan-2-yl]methyl]-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6R,7R)-6-(4-fluorophenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C21H22FN5OS
(6R,7R)-6-(4-fluorophenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(5R,10bS)-5-(4-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C23H20N2O2
6-[(5R,10bS)-5-(4-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(10bS)-7-methoxy-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C20H22N2O4
6-[(10bS)-7-methoxy-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-7-methoxy-5-(2-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C24H22N2O3
6-[(5R,10bS)-7-methoxy-5-(2-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6R,7S)-6-(4-methoxyphenyl)-3-phenyl-N-propyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C21H23N5O2S
(6R,7S)-6-(4-methoxyphenyl)-3-phenyl-N-propyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(5R,10bS)-7-methoxy-5-(2-methylpropyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C21H24N2O3
6-[(5R,10bS)-7-methoxy-5-(2-methylpropyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-5-(3-hydroxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C23H20N2O3
6-[(5R,10bS)-5-(3-hydroxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-5-(4-ethoxy-3-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C25H24N2O4
6-[(5R,10bS)-5-(4-ethoxy-3-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(5S,10bS)-7-methoxy-5-(4-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C24H22N2O3
6-[(5S,10bS)-7-methoxy-5-(4-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6R,7S)-6-(4-methoxyphenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C22H25N5O2S
(6R,7S)-6-(4-methoxyphenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,7R)-6-(4-methylphenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C22H25N5OS
(6S,7R)-6-(4-methylphenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(5S,10bR)-5-(4-hydroxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C22H18N2O3
6-[(5S,10bR)-5-(4-hydroxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(10bS)-spiro[3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclopentane]-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C21H22N2O3
6-[(10bS)-spiro[3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine-5,1'-cyclopentane]-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— (6S,7R)-N-(3-methoxypropyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C22H25N5O2S
(6S,7R)-N-(3-methoxypropyl)-6-(4-methylphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(5R,10bR)-5-thiophen-3-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C21H18N2O3S
6-[(5R,10bR)-5-thiophen-3-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— 6-[(10bS)-9-chloro-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C19H19ClN2O3
6-[(10bS)-9-chloro-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— 6-[(5R,10bR)-5-(2,5-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C25H24N2O4
6-[(5R,10bR)-5-(2,5-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— (6S)-6-[4-(diethylamino)phenyl]-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C26H31N3O2
(6S)-6-[4-(diethylamino)phenyl]-5-propanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[(5R,10bS)-7-methoxy-5-pyridin-3-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C23H21N3O4
6-[(5R,10bS)-7-methoxy-5-pyridin-3-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— 6-[(5S,10bS)-5-(2,3-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C24H22N2O4
6-[(5S,10bS)-5-(2,3-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(5S,10bS)-7-methoxy-5-(2-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C25H24N2O4
6-[(5S,10bS)-7-methoxy-5-(2-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-5-(3-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C23H20N2O3
6-[(5R,10bS)-5-(3-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-5-(4-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C23H20N2O3
6-[(5R,10bS)-5-(4-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(10bS)-7-methoxy-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-chlorocyclohexa-2,4-dien-1-one —— C19H19ClN2O3
6-[(10bS)-7-methoxy-5,5-dimethyl-3,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-chlorocyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-9-chloro-5-(2-methylsulfanylethyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C20H21ClN2O2S
6-[(5R,10bS)-9-chloro-5-(2-methylsulfanylethyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-7-methoxy-5-(3-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C24H22N2O3
6-[(5R,10bS)-7-methoxy-5-(3-methylphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-5-(3,4-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C25H24N2O4
6-[(5R,10bS)-5-(3,4-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— 6-[(5S,10bS)-5-(3-hydroxy-4-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C23H20N2O4
6-[(5S,10bS)-5-(3-hydroxy-4-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(5S,10bR)-5-(4-hydroxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-chlorocyclohexa-2,4-dien-1-one —— C22H17ClN2O3
6-[(5S,10bR)-5-(4-hydroxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-chlorocyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-5-(2,5-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C25H24N2O4
6-[(5R,10bS)-5-(2,5-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— 6-[(5R,10bS)-7-methoxy-5-propan-2-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C21H24N2O3
6-[(5R,10bS)-7-methoxy-5-propan-2-yl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— (6R)-6-(4-methylsulfanylphenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C25H28N2O2S
(6R)-6-(4-methylsulfanylphenyl)-5-pentanoyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6-[(5R,10bR)-5-(4-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one —— C24H22N2O3
6-[(5R,10bR)-5-(4-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methylcyclohexa-2,4-dien-1-one
—— (6R,7R)-6-(4-methylphenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C22H25N5OS
(6R,7R)-6-(4-methylphenyl)-N-(2-methylpropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6R)-2-benzoyl-6-(4-ethylphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one —— C28H26N2O2
(6R)-2-benzoyl-6-(4-ethylphenyl)-5,6,8,9,10,11-hexahydrobenzo[b][1,4]benzodiazepin-7-one
—— 6-[(5R,10bS)-7-methoxy-5-phenyl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C24H22N2O4
6-[(5R,10bS)-7-methoxy-5-phenyl-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-methoxycyclohexa-2,4-dien-1-one