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—— (6S,7S)-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-7-[[(2S)-2-(4-nitropyrazol-1-yl)propanoyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C16H17N9O6S2
(6S,7S)-3-[(1-methyltetrazol-5-yl)sulfanylmethyl]-7-[[(2S)-2-(4-nitropyrazol-1-yl)propanoyl]amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 6-(4-methoxyphenyl)-7-[(3S)-3-methylpiperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H21N5O
6-(4-methoxyphenyl)-7-[(3S)-3-methylpiperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— (6E)-6-[[2-(cyclohexen-1-yl)ethylamino]methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C15H18N2O3
(6E)-6-[[2-(cyclohexen-1-yl)ethylamino]methylidene]-4-nitrocyclohexa-2,4-dien-1-one
—— 6-benzyl-7-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H25N5
6-benzyl-7-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine
—— 6-(4-methoxyphenyl)-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C19H24N6O
6-(4-methoxyphenyl)-N-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— (6Z)-6-[(1-benzyl-2,5-dimethylpyrrol-3-yl)methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H23N5OS
(6Z)-6-[(1-benzyl-2,5-dimethylpyrrol-3-yl)methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-chloro-N-[[(2S)-5-phenoxy-2,3-dihydro-1-benzofuran-2-yl]methyl]pyridine-3-carboxamide —— C21H17ClN2O3
6-chloro-N-[[(2S)-5-phenoxy-2,3-dihydro-1-benzofuran-2-yl]methyl]pyridine-3-carboxamide
—— (6E)-2-butyl-5-imino-6-[[4-[2-(3-methylphenoxy)ethoxy]phenyl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C25H26N4O3S
(6E)-2-butyl-5-imino-6-[[4-[2-(3-methylphenoxy)ethoxy]phenyl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-4-chloro-6-[[3-(5-chloro-1,3-benzoxazol-2-yl)anilino]methylidene]-3,5-dimethyl-2-nitrocyclohexa-2,4-dien-1-one —— C22H15Cl2N3O4
(6E)-4-chloro-6-[[3-(5-chloro-1,3-benzoxazol-2-yl)anilino]methylidene]-3,5-dimethyl-2-nitrocyclohexa-2,4-dien-1-one
—— (6E)-6-{[1-(3-chloro-4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H22ClN5O2S
(6E)-6-{[1-(3-chloro-4-methoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-2-propyl-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6-bromopyridin-2-yl)-[(2R)-2-[(2,6-dichlorophenyl)methoxymethyl]morpholin-4-yl]methanone —— C18H17BrCl2N2O3
(6-bromopyridin-2-yl)-[(2R)-2-[(2,6-dichlorophenyl)methoxymethyl]morpholin-4-yl]methanone
—— (6Z)-6-(4-fluorobenzylidene)-2-(furan-2-yl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C16H9FN4O2S
(6Z)-6-(4-fluorobenzylidene)-2-(furan-2-yl)-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-benzyl-5-methyl-7-[(3S)-3-methylpiperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C19H23N5
6-benzyl-5-methyl-7-[(3S)-3-methylpiperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 6-benzyl-5-methyl-N-[[(2S)-oxolan-2-yl]methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C18H21N5O
6-benzyl-5-methyl-N-[[(2S)-oxolan-2-yl]methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— (6-bromopyridin-2-yl)-[(2R)-2-[(4-chloro-3-methylphenoxy)methyl]morpholin-4-yl]methanone —— C18H18BrClN2O3
(6-bromopyridin-2-yl)-[(2R)-2-[(4-chloro-3-methylphenoxy)methyl]morpholin-4-yl]methanone
—— (6-chloropyridin-3-yl)-[4-[(2R)-2-(3-methoxyphenyl)-2-prop-2-enoxyethyl]piperazin-1-yl]methanone —— C22H26ClN3O3
(6-chloropyridin-3-yl)-[4-[(2R)-2-(3-methoxyphenyl)-2-prop-2-enoxyethyl]piperazin-1-yl]methanone
—— (6-fluoro-4H-1,3-benzodioxin-8-yl)-[(2R)-2-(phenylmethoxymethyl)morpholin-4-yl]methanone —— C21H22FNO5
(6-fluoro-4H-1,3-benzodioxin-8-yl)-[(2R)-2-(phenylmethoxymethyl)morpholin-4-yl]methanone
—— (6S,9S)-9-(3-fluorophenyl)-6-(furan-2-yl)-2-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H17FN4O2
(6S,9S)-9-(3-fluorophenyl)-6-(furan-2-yl)-2-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(3-chlorophenyl)-2-ethylsulfanyl-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H19ClN4OS
(6S,9S)-9-(3-chlorophenyl)-2-ethylsulfanyl-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6-bromopyridin-2-yl)-[(2S)-2-[(4-chloro-3-methylphenoxy)methyl]morpholin-4-yl]methanone —— C18H18BrClN2O3
(6-bromopyridin-2-yl)-[(2S)-2-[(4-chloro-3-methylphenoxy)methyl]morpholin-4-yl]methanone
—— (6R,9S)-2,6-dimethyl-9-pyridin-4-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C16H17N5O
(6R,9S)-2,6-dimethyl-9-pyridin-4-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6-bromopyridin-2-yl)-[(2R)-2-[(2-methoxyphenoxy)methyl]morpholin-4-yl]methanone —— C18H19BrN2O4
(6-bromopyridin-2-yl)-[(2R)-2-[(2-methoxyphenoxy)methyl]morpholin-4-yl]methanone
—— (6R,9R)-6-(furan-2-yl)-2-methyl-9-(4-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H17N5O4
(6R,9R)-6-(furan-2-yl)-2-methyl-9-(4-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(2-fluorophenyl)-6-(furan-2-yl)-2-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H17FN4O2
(6S,9S)-9-(2-fluorophenyl)-6-(furan-2-yl)-2-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-2-ethylsulfanyl-9-(3-hydroxyphenyl)-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H20N4O2S
(6R,9R)-2-ethylsulfanyl-9-(3-hydroxyphenyl)-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 6-methyl-2-[[4-[[(2S)-oxolan-2-yl]methyl]-5-pyrrolidin-1-yl-1,2,4-triazol-3-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one —— C21H26N6O2S
6-methyl-2-[[4-[[(2S)-oxolan-2-yl]methyl]-5-pyrrolidin-1-yl-1,2,4-triazol-3-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one
—— (6R,9R)-2-ethylsulfanyl-9-(3-methoxyphenyl)-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C19H22N4O2S
(6R,9R)-2-ethylsulfanyl-9-(3-methoxyphenyl)-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-2,6-dimethyl-9-(2-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C17H17N5O3
(6S,9R)-2,6-dimethyl-9-(2-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(2-chloro-5-nitrophenyl)-2,6-dimethyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C17H16ClN5O3
(6R,9S)-9-(2-chloro-5-nitrophenyl)-2,6-dimethyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 6-methyl-2-[[4-[[(2R)-oxolan-2-yl]methyl]-5-pyrrolidin-1-yl-1,2,4-triazol-3-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one —— C21H26N6O2S
6-methyl-2-[[4-[[(2R)-oxolan-2-yl]methyl]-5-pyrrolidin-1-yl-1,2,4-triazol-3-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one
—— (6R,9R)-9-(3-chlorophenyl)-2-ethylsulfanyl-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H19ClN4OS
(6R,9R)-9-(3-chlorophenyl)-2-ethylsulfanyl-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-2,6-dimethyl-9-(2-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C17H17N5O3
(6R,9S)-2,6-dimethyl-9-(2-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-9-(3-chlorophenyl)-2-ethylsulfanyl-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H19ClN4OS
(6R,9S)-9-(3-chlorophenyl)-2-ethylsulfanyl-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-2-ethylsulfanyl-6-methyl-9-(4-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H19N5O3S
(6S,9R)-2-ethylsulfanyl-6-methyl-9-(4-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-2-ethylsulfanyl-9-(3-hydroxyphenyl)-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H20N4O2S
(6R,9S)-2-ethylsulfanyl-9-(3-hydroxyphenyl)-6-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-9-(3-fluorophenyl)-6-(furan-2-yl)-2-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H17FN4O2
(6S,9R)-9-(3-fluorophenyl)-6-(furan-2-yl)-2-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-2,6-dimethyl-9-pyridin-4-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C16H17N5O
(6S,9S)-2,6-dimethyl-9-pyridin-4-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6-bromopyridin-2-yl)-[(2S)-2-[(2-methoxyphenoxy)methyl]morpholin-4-yl]methanone —— C18H19BrN2O4
(6-bromopyridin-2-yl)-[(2S)-2-[(2-methoxyphenoxy)methyl]morpholin-4-yl]methanone
—— (6R)-6-tert-butyl-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonitrile —— C25H31N5O2S
(6R)-6-tert-butyl-2-[[2-(4-methylpiperazin-1-yl)-5-nitrophenyl]methylideneamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonitrile
—— (6R,9S)-2-ethylsulfanyl-6-methyl-9-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C21H26N4OS
(6R,9S)-2-ethylsulfanyl-6-methyl-9-(4-propan-2-ylphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(2-chloro-5-nitrophenyl)-2,6-dimethyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C17H16ClN5O3
(6R,9R)-9-(2-chloro-5-nitrophenyl)-2,6-dimethyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-2-ethylsulfanyl-6-methyl-9-(4-methylsulfanylphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C19H22N4OS2
(6S,9R)-2-ethylsulfanyl-6-methyl-9-(4-methylsulfanylphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-2-ethylsulfanyl-6-methyl-9-(4-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H19N5O3S
(6S,9S)-2-ethylsulfanyl-6-methyl-9-(4-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6Z)-2-methoxy-6-[[2-[6-(3-methyl-5-phenylpyrazol-1-yl)pyrimidin-4-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C22H20N6O2
(6Z)-2-methoxy-6-[[2-[6-(3-methyl-5-phenylpyrazol-1-yl)pyrimidin-4-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6-bromopyridin-2-yl)-[(2S)-2-[(2-fluorophenyl)methoxymethyl]morpholin-4-yl]methanone —— C18H18BrFN2O3
(6-bromopyridin-2-yl)-[(2S)-2-[(2-fluorophenyl)methoxymethyl]morpholin-4-yl]methanone
—— (6-bromopyridin-2-yl)-[(2S)-2-[(3-methylphenyl)methoxymethyl]morpholin-4-yl]methanone —— C19H21BrN2O3
(6-bromopyridin-2-yl)-[(2S)-2-[(3-methylphenyl)methoxymethyl]morpholin-4-yl]methanone
—— (6E)-6-[[2-(2-morpholin-4-ylsulfonyl-4-nitrophenyl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C17H18N4O6S
(6E)-6-[[2-(2-morpholin-4-ylsulfonyl-4-nitrophenyl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-2-heptyl-5-imino-6-[[5-(4-nitrophenyl)furan-2-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H23N5O4S
(6E)-2-heptyl-5-imino-6-[[5-(4-nitrophenyl)furan-2-yl]methylidene]-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2,4-dichloro-6-(1-hydrazinylethylidene)-5-methylcyclohexa-2,4-dien-1-one —— C9H10Cl2N2O
(6E)-2,4-dichloro-6-(1-hydrazinylethylidene)-5-methylcyclohexa-2,4-dien-1-one
—— (6Z)-6-[4-(benzyloxy)-3-chloro-5-methoxybenzylidene]-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C23H21ClN4O3S
(6Z)-6-[4-(benzyloxy)-3-chloro-5-methoxybenzylidene]-5-imino-2-(propan-2-yl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one