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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-(cis-3-aminocyclobutyl)-N~4~-[3-(1H-benzimidazol-2-yl)propyl]pyrimidine-2,4-diamine —— C18H23N7
6-(cis-3-aminocyclobutyl)-N~4~-[3-(1H-benzimidazol-2-yl)propyl]pyrimidine-2,4-diamine
—— 6-(cis-3-aminocyclobutyl)-N~4~-(4-methoxybenzyl)pyrimidine-2,4-diamine —— C16H21N5O
6-(cis-3-aminocyclobutyl)-N~4~-(4-methoxybenzyl)pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~4~-[3-(2-furyl)propyl]pyrimidine-2,4-diamine —— C15H21N5O
6-(3-aminocyclobutyl)-N~4~-[3-(2-furyl)propyl]pyrimidine-2,4-diamine
—— 6-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]carbonyl}-2-methyl-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one —— C19H24FN5O2
6-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]carbonyl}-2-methyl-5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one
—— (6Z)-2-cyclohexyl-6-{[1-(3,5-dichlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H23Cl2N5OS
(6Z)-2-cyclohexyl-6-{[1-(3,5-dichlorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-(1-naphthylmethyl)pyrimidine-2,4-diamine —— C20H23N5
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-(1-naphthylmethyl)pyrimidine-2,4-diamine
—— 6-oxo-N-[1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl]-1,6-dihydropyridine-2-carboxamide —— C16H23N3O3
6-oxo-N-[1-(tetrahydro-2H-pyran-4-yl)piperidin-4-yl]-1,6-dihydropyridine-2-carboxamide
—— 6-[cis-3-(cyclohexylamino)cyclobutyl]-2-pyrrolidin-1-ylpyrimidin-4(3H)-one —— C18H28N4O
6-[cis-3-(cyclohexylamino)cyclobutyl]-2-pyrrolidin-1-ylpyrimidin-4(3H)-one
—— 6-{[2-[hydroxy(phenyl)methyl]-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]methyl}-2-methylpyrimidin-4-ol —— C20H23N5O2
6-{[2-[hydroxy(phenyl)methyl]-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]methyl}-2-methylpyrimidin-4-ol
—— 6-[(Z)-[(3,5-dibromo-4-hydroxyphenyl)hydrazinylidene]methyl]-2,3-dimethoxybenzoic acid —— C16H14Br2N2O5
6-[(Z)-[(3,5-dibromo-4-hydroxyphenyl)hydrazinylidene]methyl]-2,3-dimethoxybenzoic acid
—— (6E)-6-[6-[(4-methoxyphenyl)methyl]-7-phenyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-ylidene]cyclohexa-2,4-dien-1-one —— C25H20N4O2
(6E)-6-[6-[(4-methoxyphenyl)methyl]-7-phenyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-ylidene]cyclohexa-2,4-dien-1-one
—— 6-(cis-3-aminocyclobutyl)-2-methyl-N-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]pyrimidin-4-amine —— C13H18N6S
6-(cis-3-aminocyclobutyl)-2-methyl-N-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]pyrimidin-4-amine
—— (6Z)-4,5-dibromo-6-[(5-butan-2-yl-2-hydroxyanilino)methylidene]-2-ethoxycyclohexa-2,4-dien-1-one —— C19H21Br2NO3
(6Z)-4,5-dibromo-6-[(5-butan-2-yl-2-hydroxyanilino)methylidene]-2-ethoxycyclohexa-2,4-dien-1-one
—— 6-(3-aminocyclobutyl)-N~4~-[2-(2-fluorophenyl)ethyl]pyrimidine-2,4-diamine —— C16H20FN5
6-(3-aminocyclobutyl)-N~4~-[2-(2-fluorophenyl)ethyl]pyrimidine-2,4-diamine
—— (6Z)-6-[[1-[3-(4-chlorophenoxy)propyl]indol-3-yl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C28H21ClN6O2S
(6Z)-6-[[1-[3-(4-chlorophenoxy)propyl]indol-3-yl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-methyl-3-[(E)-3-[4-(3-methylbutoxy)phenyl]prop-2-enoyl]pyran-2,4-dione —— C20H22O5
6-methyl-3-[(E)-3-[4-(3-methylbutoxy)phenyl]prop-2-enoyl]pyran-2,4-dione
—— (6E)-6-(2,4,5-triphenyl-1H-pyrazol-3-ylidene)cyclohexa-2,4-dien-1-one —— C27H20N2O
(6E)-6-(2,4,5-triphenyl-1H-pyrazol-3-ylidene)cyclohexa-2,4-dien-1-one
—— 6-methyl-4-[(Z)-pyridin-4-ylmethylideneamino]-3-sulfanylidene-2H-1,2,4-triazin-5-one —— C10H9N5OS
6-methyl-4-[(Z)-pyridin-4-ylmethylideneamino]-3-sulfanylidene-2H-1,2,4-triazin-5-one
—— (6Z)-6-[[1-(2,4-dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(furan-2-yl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H21N5O2S
(6Z)-6-[[1-(2,4-dimethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-2-(furan-2-yl)-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— (6E)-2,4-dichloro-6-[[(6-ethoxy-1,3-benzothiazol-2-yl)amino]methylidene]cyclohexa-2,4-dien-1-one —— C16H12Cl2N2O2S
(6E)-2,4-dichloro-6-[[(6-ethoxy-1,3-benzothiazol-2-yl)amino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-methoxy-N-[rac-(1R,5R,6S,7R)-7-pyrrolidin-1-yl-2-oxabicyclo[3.2.0]hept-6-yl]nicotinamide —— C17H23N3O3
6-methoxy-N-[rac-(1R,5R,6S,7R)-7-pyrrolidin-1-yl-2-oxabicyclo[3.2.0]hept-6-yl]nicotinamide
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrimidine-2,4-diamine —— C17H24N6S
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrimidine-2,4-diamine
—— 6-chloro-N-{cis-3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]cyclobutyl}-2H-chromene-3-carboxamide —— C18H19ClN4O3
6-chloro-N-{cis-3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]cyclobutyl}-2H-chromene-3-carboxamide
—— 6-(3-aminocyclobutyl)-N~4~-[2-(5-methoxy-1H-benzimidazol-2-yl)ethyl]-N~4~-methylpyrimidine-2,4-diamine —— C19H25N7O
6-(3-aminocyclobutyl)-N~4~-[2-(5-methoxy-1H-benzimidazol-2-yl)ethyl]-N~4~-methylpyrimidine-2,4-diamine
—— (6-chloroimidazo[1,2-a]pyridin-2-yl)-[(3S,4S)-3-ethoxy-4-hydroxypyrrolidin-1-yl]methanone —— C14H16ClN3O3
(6-chloroimidazo[1,2-a]pyridin-2-yl)-[(3S,4S)-3-ethoxy-4-hydroxypyrrolidin-1-yl]methanone
—— 6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(4-methyl-1H-benzimidazol-2-yl)methyl]pyrimidin-4-amine —— C19H24N6O
6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(4-methyl-1H-benzimidazol-2-yl)methyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-(1H-tetrazol-5-ylmethyl)pyrimidine-2,4-diamine —— C10H15N9
6-(3-aminocyclobutyl)-N~4~-(1H-tetrazol-5-ylmethyl)pyrimidine-2,4-diamine
—— 6-amino-N-{cis-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}nicotinamide —— C17H20N8O
6-amino-N-{cis-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}nicotinamide
—— 6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-(3-morpholin-4-ylpropyl)pyrimidin-4-amine —— C17H29N5O2
6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-(3-morpholin-4-ylpropyl)pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N-[3-(3,5-dimethylisoxazol-4-yl)propyl]-2-(methoxymethyl)pyrimidin-4-amine —— C18H27N5O2
6-(cis-3-aminocyclobutyl)-N-[3-(3,5-dimethylisoxazol-4-yl)propyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N-[3-(2-fluorophenyl)propyl]-2-(methoxymethyl)pyrimidin-4-amine —— C19H25FN4O
6-(cis-3-aminocyclobutyl)-N-[3-(2-fluorophenyl)propyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N-[(2-pyrazin-2-yl-1,3-thiazol-4-yl)methyl]pyrimidin-4-amine —— C16H17N7S
6-(trans-3-aminocyclobutyl)-N-[(2-pyrazin-2-yl-1,3-thiazol-4-yl)methyl]pyrimidin-4-amine
—— 6-{[2-(1,2-dihydroxyethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]carbonyl}-7-methylpyrazolo[1,5-a]pyrimidin-2(1H)-one —— C16H18N6O4
6-{[2-(1,2-dihydroxyethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]carbonyl}-7-methylpyrazolo[1,5-a]pyrimidin-2(1H)-one
—— 6-(3-aminocyclobutyl)-N~4~-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyrimidine-2,4-diamine —— C14H20N6S
6-(3-aminocyclobutyl)-N~4~-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyrimidine-2,4-diamine
—— 6-(cis-3-aminocyclobutyl)-N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-2-pyrrolidin-1-ylpyrimidin-4-amine —— C18H27N7
6-(cis-3-aminocyclobutyl)-N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-2-pyrrolidin-1-ylpyrimidin-4-amine
—— 6-amino-N-{trans-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]cyclobutyl}nicotinamide —— C17H20N8O
6-amino-N-{trans-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]cyclobutyl}nicotinamide
—— 6-(trans-3-aminocyclobutyl)-N~4~-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyrimidine-2,4-diamine —— C16H20F3N7
6-(trans-3-aminocyclobutyl)-N~4~-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyrimidine-2,4-diamine
—— 6-{[cis-3-(6-Oxo-2-pyrrolidin-1-yl-1,6-dihydropyrimidin-4-yl)cyclobutyl]amino}nicotinonitrile —— C18H20N6O
6-{[cis-3-(6-Oxo-2-pyrrolidin-1-yl-1,6-dihydropyrimidin-4-yl)cyclobutyl]amino}nicotinonitrile
—— 6-[trans-3-(2,3-dihydro-1H-inden-2-ylamino)cyclobutyl]-2-(methoxymethyl)pyrimidin-4(3H)-one —— C19H23N3O2
6-[trans-3-(2,3-dihydro-1H-inden-2-ylamino)cyclobutyl]-2-(methoxymethyl)pyrimidin-4(3H)-one
—— 6-(cis-3-aminocyclobutyl)-N-[1-(2-furoyl)piperidin-4-yl]-2-methylpyrimidin-4-amine —— C19H25N5O2
6-(cis-3-aminocyclobutyl)-N-[1-(2-furoyl)piperidin-4-yl]-2-methylpyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N~4~-methyl-N~4~-[2-(methylthio)ethyl]pyrimidine-2,4-diamine —— C12H21N5S
6-(cis-3-aminocyclobutyl)-N~4~-methyl-N~4~-[2-(methylthio)ethyl]pyrimidine-2,4-diamine
—— (6E)-6-(1-hydrazinylethylidene)cyclohexa-2,4-dien-1-one —— C8H10N2O
(6E)-6-(1-hydrazinylethylidene)cyclohexa-2,4-dien-1-one
—— 6-methoxy-N'-[(Z)-(4-nitrophenyl)methylideneamino]-1,3-benzothiazole-2-carboximidamide —— C16H13N5O3S
6-methoxy-N'-[(Z)-(4-nitrophenyl)methylideneamino]-1,3-benzothiazole-2-carboximidamide
—— 6-(cis-3-aminocyclobutyl)-N~4~-[(3-isobutyl-1,2,4-oxadiazol-5-yl)methyl]-N~4~-methylpyrimidine-2,4-diamine —— C16H25N7O
6-(cis-3-aminocyclobutyl)-N~4~-[(3-isobutyl-1,2,4-oxadiazol-5-yl)methyl]-N~4~-methylpyrimidine-2,4-diamine
—— 6-[trans-3-(1,3-benzoxazol-2-ylamino)cyclobutyl]-2-cyclopropylpyrimidin-4(3H)-one —— C18H18N4O2
6-[trans-3-(1,3-benzoxazol-2-ylamino)cyclobutyl]-2-cyclopropylpyrimidin-4(3H)-one
—— 6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-[2-(2-methyl-1H-indol-3-yl)ethyl]pyrimidin-4-amine —— C21H27N5O
6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-[2-(2-methyl-1H-indol-3-yl)ethyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N-{2-[(3-chlorobenzyl)thio]ethyl}pyrimidin-4-amine —— C17H21ClN4S
6-(3-aminocyclobutyl)-N-{2-[(3-chlorobenzyl)thio]ethyl}pyrimidin-4-amine
—— (6Z)-6-[[1-(2,5-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H28N6O5S
(6Z)-6-[[1-(2,5-dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-morpholin-4-yl-2-oxoethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[2-(1H-1,2,3-triazol-5-ylthio)ethyl]pyrimidin-4-amine —— C15H21N7S
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[2-(1H-1,2,3-triazol-5-ylthio)ethyl]pyrimidin-4-amine
—— (6Z)-2-cyclohexyl-6-{[1-(4-ethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H29N5O2S
(6Z)-2-cyclohexyl-6-{[1-(4-ethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]methylidene}-5-imino-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one