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—— (6R,7R)-N-(3-methoxyphenyl)-6-(4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H21N5O3S
(6R,7R)-N-(3-methoxyphenyl)-6-(4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— [(6R,7R)-6-(3-chloro-4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone —— C17H20ClN5O3S
[(6R,7R)-6-(3-chloro-4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone
—— 6-[(5R,10bS)-5-(4-hydroxy-3-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-chlorocyclohexa-2,4-dien-1-one —— C23H19ClN2O4
6-[(5R,10bS)-5-(4-hydroxy-3-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-chlorocyclohexa-2,4-dien-1-one
—— (6S,7S)-N-(4-ethylphenyl)-6-(4-fluorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H20FN5OS
(6S,7S)-N-(4-ethylphenyl)-6-(4-fluorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(5R,10bS)-5-(3,4-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-chlorocyclohexa-2,4-dien-1-one —— C24H21ClN2O4
6-[(5R,10bS)-5-(3,4-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]-4-chlorocyclohexa-2,4-dien-1-one
—— (6R)-2-amino-4-(5-bromothiophen-2-yl)-6-methyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile —— C15H14BrN3S
(6R)-2-amino-4-(5-bromothiophen-2-yl)-6-methyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
—— [(6R,7S)-6-(4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-pyrrolidin-1-ylmethanone —— C17H21N5O2S
[(6R,7S)-6-(4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-pyrrolidin-1-ylmethanone
—— (6R,7S)-N-(2,6-dimethylphenyl)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C26H25N5O2S
(6R,7S)-N-(2,6-dimethylphenyl)-6-(4-methoxyphenyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— [(6R,7S)-3,6-diphenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-pyrrolidin-1-ylmethanone —— C21H21N5OS
[(6R,7S)-3,6-diphenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-pyrrolidin-1-ylmethanone
—— (6R,7S)-6-(4-chlorophenyl)-3-methyl-N-(2-methylpropyl)-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C16H20ClN5OS
(6R,7S)-6-(4-chlorophenyl)-3-methyl-N-(2-methylpropyl)-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— [(6R,7R)-6-(3-chloro-4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-pyrrolidin-1-ylmethanone —— C17H20ClN5O2S
[(6R,7R)-6-(3-chloro-4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-pyrrolidin-1-ylmethanone
—— [(6S,7S)-6-(3-chloro-4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone —— C17H20ClN5O3S
[(6S,7S)-6-(3-chloro-4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone
—— (6S,7R)-N-benzyl-6-(4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H21N5O2S
(6S,7R)-N-benzyl-6-(4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6R,7S)-N-(2-methoxyethyl)-6-(4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C16H21N5O3S
(6R,7S)-N-(2-methoxyethyl)-6-(4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,7R)-N-(2-bromo-4-methylphenyl)-6-(4-chlorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C19H17BrClN5OS
(6S,7R)-N-(2-bromo-4-methylphenyl)-6-(4-chlorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— [(6R,7S)-6-(4-fluorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone —— C16H18FN5O2S
[(6R,7S)-6-(4-fluorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone
—— (6R,7R)-6-(4-chlorophenyl)-N-[(4-methoxyphenyl)methyl]-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H20ClN5O2S
(6R,7R)-6-(4-chlorophenyl)-N-[(4-methoxyphenyl)methyl]-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6R,7R)-6-(4-ethoxyphenyl)-3-methyl-N-propyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C17H23N5O2S
(6R,7R)-6-(4-ethoxyphenyl)-3-methyl-N-propyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,7S)-3-methyl-N-[(4-methylphenyl)methyl]-6-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H21N5OS
(6S,7S)-3-methyl-N-[(4-methylphenyl)methyl]-6-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,7S)-6-(4-chlorophenyl)-N-(3-methoxypropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C21H22ClN5O2S
(6S,7S)-6-(4-chlorophenyl)-N-(3-methoxypropyl)-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,7S)-6-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C23H25N5O2S
(6S,7S)-6-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]-3-phenyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6R,7R)-6-(4-ethoxyphenyl)-N-(2-methoxyethyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C17H23N5O3S
(6R,7R)-6-(4-ethoxyphenyl)-N-(2-methoxyethyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,7S)-N-(2-ethylphenyl)-6-(4-fluorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H20FN5OS
(6S,7S)-N-(2-ethylphenyl)-6-(4-fluorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(5S,10bR)-5-(2,5-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C24H22N2O4
6-[(5S,10bR)-5-(2,5-dimethoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— [(6S,7R)-6-(3-chloro-4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone —— C17H20ClN5O3S
[(6S,7R)-6-(3-chloro-4-methoxyphenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl]-morpholin-4-ylmethanone
—— (6S,7S)-6-(4-ethoxyphenyl)-3-methyl-N-propyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C17H23N5O2S
(6S,7S)-6-(4-ethoxyphenyl)-3-methyl-N-propyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,7R)-6-(4-fluorophenyl)-N-(2-methoxyethyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C15H18FN5O2S
(6S,7R)-6-(4-fluorophenyl)-N-(2-methoxyethyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(5R,10bR)-5-(2-fluorophenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C22H17FN2O2
6-[(5R,10bR)-5-(2-fluorophenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6S)-9,9-dimethyl-6-(2-nitrophenyl)-6,8,10,11-tetrahydro-5H-pyrido[3,2-b][1,4]benzodiazepin-7-one —— C20H20N4O3
(6S)-9,9-dimethyl-6-(2-nitrophenyl)-6,8,10,11-tetrahydro-5H-pyrido[3,2-b][1,4]benzodiazepin-7-one
—— (6S,7R)-N-(4-ethylphenyl)-6-(4-fluorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H20FN5OS
(6S,7R)-N-(4-ethylphenyl)-6-(4-fluorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— 6-[(5S,10bR)-9-chloro-5-(3-hydroxy-4-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C23H19ClN2O4
6-[(5S,10bR)-9-chloro-5-(3-hydroxy-4-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— 6-[(5S,10bS)-9-chloro-5-(4-hydroxy-3-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one —— C23H19ClN2O4
6-[(5S,10bS)-9-chloro-5-(4-hydroxy-3-methoxyphenyl)-1,3,5,10b-tetrahydropyrazolo[1,5-c][1,3]benzoxazin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6S,7R)-N-(2-ethylphenyl)-6-(4-fluorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide —— C20H20FN5OS
(6S,7R)-N-(2-ethylphenyl)-6-(4-fluorophenyl)-3-methyl-6,7-dihydro-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine-7-carboxamide
—— (6S,9R)-9-(3-hydroxyphenyl)-2,6-dimethyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C17H18N4O2
(6S,9R)-9-(3-hydroxyphenyl)-2,6-dimethyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6E)-6-[[2-[3-[(3,4-dichlorophenyl)methylsulfanyl]-1H-1,2,4-triazol-5-yl]hydrazinyl]methylidene]-2-prop-2-enylcyclohexa-2,4-dien-1-one —— C19H17Cl2N5OS
(6E)-6-[[2-[3-[(3,4-dichlorophenyl)methylsulfanyl]-1H-1,2,4-triazol-5-yl]hydrazinyl]methylidene]-2-prop-2-enylcyclohexa-2,4-dien-1-one
—— (6E)-4-chloro-6-[(3,6-dimethyl-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl)methylidene]cyclohexa-2,4-dien-1-one —— C13H11ClN4OS
(6E)-4-chloro-6-[(3,6-dimethyl-5H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-7-yl)methylidene]cyclohexa-2,4-dien-1-one
—— (6Z)-2,4-dibromo-6-[[2-(5-sulfanylidene-1,2-dihydro-1,2,4-triazol-3-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C9H7Br2N5OS
(6Z)-2,4-dibromo-6-[[2-(5-sulfanylidene-1,2-dihydro-1,2,4-triazol-3-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6E)-2-prop-2-enyl-6-[[2-(3-prop-2-enylsulfanyl-1H-1,2,4-triazol-5-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C15H17N5OS
(6E)-2-prop-2-enyl-6-[[2-(3-prop-2-enylsulfanyl-1H-1,2,4-triazol-5-yl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6S,9R)-6-(furan-2-yl)-2-methyl-9-thiophen-2-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H16N4O2S
(6S,9R)-6-(furan-2-yl)-2-methyl-9-thiophen-2-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-6-(furan-2-yl)-2-methylsulfanyl-9-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H18N4O2S
(6R,9R)-6-(furan-2-yl)-2-methylsulfanyl-9-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-6-(furan-2-yl)-2-methyl-9-thiophen-2-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H16N4O2S
(6R,9S)-6-(furan-2-yl)-2-methyl-9-thiophen-2-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-6-(furan-2-yl)-2-methyl-9-(2-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H17N5O4
(6S,9S)-6-(furan-2-yl)-2-methyl-9-(2-nitrophenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-6-(furan-2-yl)-2-methyl-9-(4-methylsulfanylphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C21H20N4O2S
(6S,9R)-6-(furan-2-yl)-2-methyl-9-(4-methylsulfanylphenyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9R)-2-ethylsulfanyl-6-methyl-9-thiophen-2-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C16H18N4OS2
(6S,9R)-2-ethylsulfanyl-6-methyl-9-thiophen-2-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-6-(furan-2-yl)-2-methylsulfanyl-9-thiophen-2-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C18H16N4O2S2
(6R,9S)-6-(furan-2-yl)-2-methylsulfanyl-9-thiophen-2-yl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-[4-(dimethylamino)phenyl]-6-(furan-2-yl)-2-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C22H23N5O2
(6R,9R)-9-[4-(dimethylamino)phenyl]-6-(furan-2-yl)-2-methyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9R)-9-(4-fluorophenyl)-6-(furan-2-yl)-2-methylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H17FN4O2S
(6R,9R)-9-(4-fluorophenyl)-6-(furan-2-yl)-2-methylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(4-chlorophenyl)-6-(furan-2-yl)-2-methylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H17ClN4O2S
(6S,9S)-9-(4-chlorophenyl)-6-(furan-2-yl)-2-methylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6R,9S)-6-(furan-2-yl)-2-methylsulfanyl-9-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H18N4O2S
(6R,9S)-6-(furan-2-yl)-2-methylsulfanyl-9-phenyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— (6S,9S)-9-(4-fluorophenyl)-6-(furan-2-yl)-2-methylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C20H17FN4O2S
(6S,9S)-9-(4-fluorophenyl)-6-(furan-2-yl)-2-methylsulfanyl-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one