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—— (6E)-2,4-dichloro-6-[[(3-hydroxypyridin-2-yl)amino]methylidene]cyclohexa-2,4-dien-1-one —— C12H8Cl2N2O2
(6E)-2,4-dichloro-6-[[(3-hydroxypyridin-2-yl)amino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-(3-aminocyclobutyl)-N~4~-[2-(1-methylpiperidin-4-yl)ethyl]pyrimidine-2,4-diamine —— C16H28N6
6-(3-aminocyclobutyl)-N~4~-[2-(1-methylpiperidin-4-yl)ethyl]pyrimidine-2,4-diamine
—— 6-hydroxy-2,5,7,8-tetramethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]chromane-2-carboxamide —— C18H23N3O3S
6-hydroxy-2,5,7,8-tetramethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]chromane-2-carboxamide
—— (6E)-4-chloro-2-methoxy-6-[[4-(6-methyl-1,3-benzothiazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one —— C22H17ClN2O2S
(6E)-4-chloro-2-methoxy-6-[[4-(6-methyl-1,3-benzothiazol-2-yl)anilino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-(2-{[6-(cis-3-Aminocyclobutyl)-2-pyrrolidin-1-ylpyrimidin-4-yl]amino}ethyl)-2-methylpyrimidin-4-ol —— C19H27N7O
6-(2-{[6-(cis-3-Aminocyclobutyl)-2-pyrrolidin-1-ylpyrimidin-4-yl]amino}ethyl)-2-methylpyrimidin-4-ol
—— (6Z)-6-[[3-chloro-4-[2-(3,5-dimethylphenoxy)ethoxy]-5-methoxyphenyl]methylidene]-5-imino-2-methyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C24H23ClN4O4S
(6Z)-6-[[3-chloro-4-[2-(3,5-dimethylphenoxy)ethoxy]-5-methoxyphenyl]methylidene]-5-imino-2-methyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(cis-3-aminocyclobutyl)-N-[(5-ethylpyridin-2-yl)methyl]-N-methylpyrimidin-4-amine —— C17H23N5
6-(cis-3-aminocyclobutyl)-N-[(5-ethylpyridin-2-yl)methyl]-N-methylpyrimidin-4-amine
—— 6-amino-N-[trans-3-(pyridin-2-yloxy)tetrahydro-2H-pyran-4-yl]nicotinamide —— C16H18N4O3
6-amino-N-[trans-3-(pyridin-2-yloxy)tetrahydro-2H-pyran-4-yl]nicotinamide
—— (6E)-4-chloro-3,5-dimethyl-2-nitro-6-[[(2-phenyl-1,3-benzoxazol-5-yl)amino]methylidene]cyclohexa-2,4-dien-1-one —— C22H16ClN3O4
(6E)-4-chloro-3,5-dimethyl-2-nitro-6-[[(2-phenyl-1,3-benzoxazol-5-yl)amino]methylidene]cyclohexa-2,4-dien-1-one
—— 6-[2-[2-(dimethylamino)-1-hydroxyethyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]-N-ethylnicotinamide —— C18H26N6O2
6-[2-[2-(dimethylamino)-1-hydroxyethyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]-N-ethylnicotinamide
—— 6-(3-aminocyclobutyl)-2-cyclopropyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidin-4-amine —— C16H22N6
6-(3-aminocyclobutyl)-2-cyclopropyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrimidin-4-amine
—— 6-({cis-3-[2-(dimethylamino)-6-oxo-1,6-dihydropyrimidin-4-yl]cyclobutyl}amino)-N,N-dimethylpyridine-2-carboxamide —— C18H24N6O2
6-({cis-3-[2-(dimethylamino)-6-oxo-1,6-dihydropyrimidin-4-yl]cyclobutyl}amino)-N,N-dimethylpyridine-2-carboxamide
—— 6-(cis-3-aminocyclobutyl)-N-[2-(5-methoxy-1H-benzimidazol-2-yl)ethyl]-N,2-dimethylpyrimidin-4-amine —— C20H26N6O
6-(cis-3-aminocyclobutyl)-N-[2-(5-methoxy-1H-benzimidazol-2-yl)ethyl]-N,2-dimethylpyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidine-2,4-diamine —— C13H20N8
6-(3-aminocyclobutyl)-N~4~-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~4~-(isoxazol-3-ylmethyl)pyrimidine-2,4-diamine —— C12H16N6O
6-(3-aminocyclobutyl)-N~4~-(isoxazol-3-ylmethyl)pyrimidine-2,4-diamine
—— 6-{1-[6-(3-Aminocyclobutyl)-2-(methoxymethyl)pyrimidin-4-YL]piperidin-4-YL}-2-methylpyrimidin-4-OL —— C20H28N6O2
6-{1-[6-(3-Aminocyclobutyl)-2-(methoxymethyl)pyrimidin-4-YL]piperidin-4-YL}-2-methylpyrimidin-4-OL
—— 6-(2-methylpropyl)-2-oxo-N-[(3R,4R)-4-piperidin-1-yloxolan-3-yl]-1H-pyrimidine-4-carboxamide —— C18H28N4O3
6-(2-methylpropyl)-2-oxo-N-[(3R,4R)-4-piperidin-1-yloxolan-3-yl]-1H-pyrimidine-4-carboxamide
—— 6-({4-[(4-methoxyphenoxy)methyl]piperidin-1-yl}carbonyl)pyridin-2(1H)-one —— C19H22N2O4
6-({4-[(4-methoxyphenoxy)methyl]piperidin-1-yl}carbonyl)pyridin-2(1H)-one
—— 6-ethyl-1,5-dimethyl-N-[(3R,4S)-4-(3-methylbut-2-enoxy)oxan-3-yl]-2-oxopyridine-3-carboxamide —— C20H30N2O4
6-ethyl-1,5-dimethyl-N-[(3R,4S)-4-(3-methylbut-2-enoxy)oxan-3-yl]-2-oxopyridine-3-carboxamide
—— (6E)-4-bromo-6-[[2-(2,4,6-trichlorophenyl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C13H8BrCl3N2O
(6E)-4-bromo-6-[[2-(2,4,6-trichlorophenyl)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— 6-isopropyl-1-methyl-2-oxo-N-[rac-(1R,5R,6S,7R)-7-pyrrolidin-1-yl-2-oxabicyclo[3.2.0]hept-6-yl]-1,2-dihydropyridine-3-carboxamide —— C20H29N3O3
6-isopropyl-1-methyl-2-oxo-N-[rac-(1R,5R,6S,7R)-7-pyrrolidin-1-yl-2-oxabicyclo[3.2.0]hept-6-yl]-1,2-dihydropyridine-3-carboxamide
—— 6-(3-aminocyclobutyl)-N-(1H-benzimidazol-5-ylmethyl)pyrimidin-4-amine —— C16H18N6
6-(3-aminocyclobutyl)-N-(1H-benzimidazol-5-ylmethyl)pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-(2-chlorobenzyl)-N~4~-methylpyrimidine-2,4-diamine —— C16H20ClN5
6-(3-aminocyclobutyl)-N~4~-(2-chlorobenzyl)-N~4~-methylpyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~4~-(2,4-dichloro-6-methylbenzyl)pyrimidine-2,4-diamine —— C16H19Cl2N5
6-(3-aminocyclobutyl)-N~4~-(2,4-dichloro-6-methylbenzyl)pyrimidine-2,4-diamine
—— 6-amino-N-[(5-ethylpyridin-2-yl)methyl]nicotinamide —— C14H16N4O
6-amino-N-[(5-ethylpyridin-2-yl)methyl]nicotinamide
—— 6-fluoro-7-morpholin-4-yl-N-[rac-(1S,5R,6R)-2-oxabicyclo[3.2.0]hept-6-yl]-4-oxo-1,4-dihydroquinoline-3-carboxamide —— C20H22FN3O4
6-fluoro-7-morpholin-4-yl-N-[rac-(1S,5R,6R)-2-oxabicyclo[3.2.0]hept-6-yl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
—— 6-methyl-N-[(2-morpholin-4-yl-1,3-thiazol-4-yl)methyl]pyridine-2-carboxamide —— C15H18N4O2S
6-methyl-N-[(2-morpholin-4-yl-1,3-thiazol-4-yl)methyl]pyridine-2-carboxamide
—— 6-methoxy-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]chromane-3-carboxamide —— C21H25N3O3
6-methoxy-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]chromane-3-carboxamide
—— 6-(2-methylbutan-2-yl)-2-[[(E)-3-phenylprop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C23H28N2O2S
6-(2-methylbutan-2-yl)-2-[[(E)-3-phenylprop-2-enoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-methoxy-N-[cis-3-(6-pyrrolidin-1-ylpyrimidin-4-yl)cyclobutyl]nicotinamide —— C19H23N5O2
6-methoxy-N-[cis-3-(6-pyrrolidin-1-ylpyrimidin-4-yl)cyclobutyl]nicotinamide
—— (6Z)-6-[(3-bromoanilino)methylidene]cyclohexa-2,4-dien-1-one —— C13H10BrNO
(6Z)-6-[(3-bromoanilino)methylidene]cyclohexa-2,4-dien-1-one
—— 6-(3-aminocyclobutyl)-N-[(3-pyrazin-2-yl-1H-1,2,4-triazol-5-yl)methyl]pyrimidin-4-amine —— C15H17N9
6-(3-aminocyclobutyl)-N-[(3-pyrazin-2-yl-1H-1,2,4-triazol-5-yl)methyl]pyrimidin-4-amine
—— 6-methoxy-N-[(1S,5R,6S)-2-oxabicyclo[3.2.0]heptan-6-yl]naphthalene-2-sulfonamide —— C17H19NO4S
6-methoxy-N-[(1S,5R,6S)-2-oxabicyclo[3.2.0]heptan-6-yl]naphthalene-2-sulfonamide
—— (6E)-6-[[(2E)-2-(4-methyl-3-phenyl-1,3-thiazol-2-ylidene)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C17H15N3OS
(6E)-6-[[(2E)-2-(4-methyl-3-phenyl-1,3-thiazol-2-ylidene)hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— 6-methyl-N-[(3R,4S)-4-(3-methylbut-2-enoxy)oxan-3-yl]-4-oxo-1H-pyridine-3-carboxamide —— C17H24N2O4
6-methyl-N-[(3R,4S)-4-(3-methylbut-2-enoxy)oxan-3-yl]-4-oxo-1H-pyridine-3-carboxamide
—— 6-(3-aminocyclobutyl)-N~4~-(3-isopropoxybenzyl)pyrimidine-2,4-diamine —— C18H25N5O
6-(3-aminocyclobutyl)-N~4~-(3-isopropoxybenzyl)pyrimidine-2,4-diamine
—— 6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)thio]ethyl}pyrimidin-4-amine —— C15H23N7OS
6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)thio]ethyl}pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N-(4-methoxybenzyl)-N-methylpyrimidin-4-amine —— C17H22N4O
6-(cis-3-aminocyclobutyl)-N-(4-methoxybenzyl)-N-methylpyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine —— C15H22N6O
6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[3-(methylthio)benzyl]pyrimidine-2,4-diamine —— C17H23N5S
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[3-(methylthio)benzyl]pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~2~,N~2~-dimethyl-N~4~-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrimidine-2,4-diamine —— C15H24N8
6-(3-aminocyclobutyl)-N~2~,N~2~-dimethyl-N~4~-[3-(1H-1,2,3-triazol-1-yl)propyl]pyrimidine-2,4-diamine
—— (6E)-2,4-dibromo-6-[[2-[4-(4-nitroanilino)-6-pyrrolidin-1-yl-1,3,5-triazin-2-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C20H18Br2N8O3
(6E)-2,4-dibromo-6-[[2-[4-(4-nitroanilino)-6-pyrrolidin-1-yl-1,3,5-triazin-2-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— 6-{[2-(hydroxymethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]sulfonyl}-1,3-benzoxazol-2(3H)-one —— C14H14N4O5S
6-{[2-(hydroxymethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]sulfonyl}-1,3-benzoxazol-2(3H)-one
—— 6-ethyl-4-({2-[3-(hydroxymethyl)phenyl]-1,4,6,7-tetrahydro-5H-imidazo[4,5-c]pyridin-5-yl}carbonyl)pyridin-2(1H)-one —— C21H22N4O3
6-ethyl-4-({2-[3-(hydroxymethyl)phenyl]-1,4,6,7-tetrahydro-5H-imidazo[4,5-c]pyridin-5-yl}carbonyl)pyridin-2(1H)-one
—— 6-[[(Z)-(4-bromothiophen-2-yl)methylideneamino]-ethylamino]-3-methyl-1H-pyrimidine-2,4-dione —— C12H13BrN4O2S
6-[[(Z)-(4-bromothiophen-2-yl)methylideneamino]-ethylamino]-3-methyl-1H-pyrimidine-2,4-dione
—— 6-{(E)-2-[4-(dimethylamino)phenyl]vinyl}-1,3-dimethyl-5-nitropyrimidine-2,4(1H,3H)-dione —— C16H18N4O4
6-{(E)-2-[4-(dimethylamino)phenyl]vinyl}-1,3-dimethyl-5-nitropyrimidine-2,4(1H,3H)-dione
—— 6-(cis-3-aminocyclobutyl)-N-[(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)methyl]-2-methylpyrimidin-4-amine —— C15H24N4O2S
6-(cis-3-aminocyclobutyl)-N-[(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)methyl]-2-methylpyrimidin-4-amine
—— 6-methoxy-N-[cis-3-(6-oxo-1,6-dihydropyrimidin-4-yl)cyclobutyl]indane-5-carboxamide —— C19H21N3O3
6-methoxy-N-[cis-3-(6-oxo-1,6-dihydropyrimidin-4-yl)cyclobutyl]indane-5-carboxamide
—— 6-(3-Aminocyclobutyl)-N-(1-cyclopentylcyclopropyl)pyrimidin-4-amine —— C16H24N4
6-(3-Aminocyclobutyl)-N-(1-cyclopentylcyclopropyl)pyrimidin-4-amine
—— 6-(cis-3-aminocyclobutyl)-N~4~-(3-azepan-1-ylpropyl)-N~4~-methylpyrimidine-2,4-diamine —— C18H32N6
6-(cis-3-aminocyclobutyl)-N~4~-(3-azepan-1-ylpropyl)-N~4~-methylpyrimidine-2,4-diamine