循环系统是由生物体内的细胞外液(包括血浆、淋巴和组织液)及其流动管道组成的系统。自动物形成心脏后,该系统分为两大部分:心脏和血管,称为心血管系统。循环系统作为生物体内的运输系统,负责将消化道吸收的营养物质以及由鳃或肺摄取的氧气输送到各组织器官,并通过同样的途径将这些组织器官产生的代谢产物带回血液中,再经肺、肾排出体外。此外,它还承担着输送热量到全身以维持体温和运送激素至靶器官以调节其功能的任务。
循环系统的药物主要包括抗心绞痛药、抗心律失常药、抗高血压药、用于治疗休克的血管活性药、调节血脂药及预防动脉粥样硬化的药物、周围血管扩张药、钙拮抗剂、抗心力衰竭药以及治疗慢性心功能不全的药物。
| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| 美托洛尔 | S-(-)-metoprolol | 81024-42-2 | C15H25NO3 |
| 美托洛尔 | (RS)-metoprolol | 51384-51-1 | C15H25NO3 |
| 美卡拉明 | mecamylamine | 60-40-2 | C11H21N |
| 美伐他汀 | mevastatin | 73573-88-3 | C23H34O5 |
| 罗尼帕米 | Ronipamil | 85247-77-4 | C32H48N2 |
| 罗伐他汀 | rosuvastatin | 287714-41-4 | C22H28FN3O6S |
| 缬沙坦USP杂质A | valsartan | 137862-87-4 | C24H29N5O3 |
| 缬沙坦 | N-pentanoyl-N-[[2'-(1H-tetrazol-5-yl)-[1,1'-biphenyl]-4-yl]-methyl]-(L)-valine | 137862-53-4 | C24H29N5O3 |
| 维那卡兰 | (3R)-1-[(1R,2R)-2-[2-(3,4-dimethoxyphenyl)ethoxy]cyclohexyl]pyrrolidin-3-ol | 794466-70-9 | C20H31NO4 |
| 维达列汀 | vildagliptin | 274901-16-5 | C17H25N3O2 |
| 维拉帕米 | Verapamil | 52-53-9 | C27H38N2O4 |
| 维司力农 | vesnarinone | 81840-15-5 | C22H25N3O4 |
| 索拉非尼 | sorafenib | 284461-73-0 | C21H16ClF3N4O3 |
| 索他洛尔 | sotalol | 3930-20-9 | C12H20N2O3S |
| 米贝地尔(二盐酸盐) | mibefradil | 116644-53-2 | C29H38FN3O3 |
| 米诺地尔 | minoxidil | 38304-91-5 | C9H15N5O |
| 米屈肼 | meldonium | 76144-81-5 | C6H14N2O2 |
| 米多君 | midodrine | 42794-76-3 | C12H18N2O4 |
| 米力农 | 1,6-dihydro-2-methyl-6-oxo-(3,4'-bipyridine)-5-carbonitrile | 78415-72-2 | C12H9N3O |
| 福辛普利钠 | 88889-14-9 | C30H46NNaO7P | |
| 福辛普利 | fosinopril | 98048-97-6 | C30H46NO7P |
| 磷酸肌酸 | Phosphocreatine | 67-07-2 | C4H10N3O5P |
| 磷酸川芎嗪 | Ligustrazine phosphate | 105256-26-6 | C8H15N2O4P |
| 磷酸丙吡胺 | disopyramide phosphate | 22059-60-5 | C21H29N3O*H3O4P |
| 碘化N,N,N-三甲基-2-{[2-(戊基桥氧基)丙酰]氧代}乙铵 | Piperazine, 1-[(1-pyrrolidinylcarbonyl)methyl]-4-(3,4,5-trimethoxycinnamoyl)-, maleate | 26328-04-1 | C4H4O4*C22H31N3O5 |
| 硫酸奎尼丁二水合物 | (S)-[(2R,4S,5R)-5-ethenyl-1-azabicyclo[2.2.2]octan-2-yl]-(6-methoxyquinolin-4-yl)methanol;sulfuric acid;dihydrate | 6591-63-5 | C20H30N2O8S |
| 硫酸司巴丁 | sparteine sulfate | 299-39-8 | C15H26N2*H2O4S |
| 硫酸双肼屈嗪 | dihydrazino-1,4-phthalazine sulfate | 7327-87-9 | C8H10N6*H2O4S |
| 硝酸异山梨酯 | isosorbide dinitrate | 87-33-2 | C6H8N2O8 |
| 硝苯地平 | nifedipine | 193689-82-6 | C17H18N2O6 |
| 硝普钠 | disodium;iron(4+);nitroxyl anion;pentacyanide;dihydrate | 13755-38-9 | C5H4FeN6Na2O3 |
| 盐酸阿夫唑嗪 | alfuzosin hydrochloride | 81403-68-1 | C19H27N5O4*ClH |
| 盐酸酚苄明 | phenoxybenzamine hydrochloride | 63-92-3 | C18H22ClNO*ClH |
| 盐酸酚妥拉明 | phentolamine hydrochloride | 73-05-2 | C17H19N3O*ClH |
| 盐酸贝那普利 | (3S)-1-(carboxymethyl)-<<(1S)-1-(ethoxycarbonyl)-3-phenylpropyl>amino>-2,3,4,5-tetrahydro-1H-<1>benzazepin-2-one hydrochloride | 86541-77-7 | C24H28N2O5*ClH |
| 盐酸贝那普利 | benazepril hydrochloride | 86541-74-4 | C24H28N2O5*ClH |
| 盐酸贝凡洛尔 | bevantolol hydrochloride | 42864-78-8 | C20H27NO4*ClH |
| 盐酸萘哌地尔 | Naftopidil dihydrochloride | 57149-08-3 | C24H30Cl2N2O3 |
| 盐酸莫索尼定 | 4-chloro-6-methoxy-2-methyl-5-(2-imidazolin-2-yl)aminopyrimidine hydrochloride | 75438-58-3 | C9H12ClN5O*(x)ClH |
| 盐酸茚洛秦 | 2-(7-indenyloxymethyl)-morpholine hydrochloride | 65043-22-3 | C14H17NO2*ClH |
| 盐酸艾司洛尔 | esmolol hydrochloride | 81161-17-3 | C16H25NO4*ClH |
| 盐酸胺碘酮 | amiodarone hydrochloride | 19774-82-4 | C25H29I2NO3*ClH |
| 盐酸胍法辛 | guanfacine hydrochloride | 29110-48-3 | C9H9Cl2N3O*ClH |
| 盐酸肾上腺素 | epinephrine hydrochloride | 55-31-2 | C9H13NO3*ClH |
| 盐酸肼屈嗪 | hydralazine hydrochloride | 304-20-1 | C8H8N4*ClH |
| 盐酸考来维仑 | 2-(chloromethyl)oxirane;hydron;prop-2-en-1-amine;N-prop-2-enyldecan-1-amine;trimethyl-[6-(prop-2-enylamino)hexyl]azanium;dichloride | 182815-44-7 | C31H67Cl3N4O |
| 盐酸考尼伐坦 | conivaptan hydrochloride | 168626-94-6 | C32H26N4O2*ClH |
| 盐酸美西律 | (rac)-mexiletine hydrochloride | 5370-01-4 | C11H17NO*ClH |
| 盐酸罂粟碱 | papaverine hydrochloride | 61-25-6 | C20H22NO4*Cl |
| 盐酸维拉帕米 | verapamil hydrochloride | 152-11-4 | C27H38N2O4*ClH |