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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl 2-[cyclopropyl-[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C18H23N3O4S
ethyl 2-[cyclopropyl-[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— (4R)-3-[1-(2-chlorophenyl)triazole-4-carbonyl]-N-(3-methylphenyl)-1,3-thiazolidine-4-carboxamide —— C20H18ClN5O2S
(4R)-3-[1-(2-chlorophenyl)triazole-4-carbonyl]-N-(3-methylphenyl)-1,3-thiazolidine-4-carboxamide
—— 2-(5-methylfuran-2-yl)-N-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]-1,3-thiazole-4-carboxamide —— C19H25N3O3S
2-(5-methylfuran-2-yl)-N-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]-1,3-thiazole-4-carboxamide
—— 1-(4-fluorophenyl)-N-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]-5-propan-2-ylpyrazole-4-carboxamide —— C23H31FN4O2
1-(4-fluorophenyl)-N-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]-5-propan-2-ylpyrazole-4-carboxamide
—— 1-(4-fluorophenyl)-N-[1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]-5-propan-2-ylpyrazole-4-carboxamide —— C23H31FN4O2
1-(4-fluorophenyl)-N-[1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]-5-propan-2-ylpyrazole-4-carboxamide
—— (4S)-3-[1-(4-fluorophenyl)pyrazole-3-carbonyl]-N-(3-methylphenyl)-1,3-thiazolidine-4-carboxamide —— C21H19FN4O2S
(4S)-3-[1-(4-fluorophenyl)pyrazole-3-carbonyl]-N-(3-methylphenyl)-1,3-thiazolidine-4-carboxamide
—— 1-(2-chlorophenyl)-N-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]triazole-4-carboxamide —— C19H24ClN5O2
1-(2-chlorophenyl)-N-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]triazole-4-carboxamide
—— 1-(2-chlorophenyl)-N-[1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]triazole-4-carboxamide —— C19H24ClN5O2
1-(2-chlorophenyl)-N-[1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]triazole-4-carboxamide
—— [(3S)-3-(diethylamino)pyrrolidin-1-yl]-[2-(1H-imidazol-2-yl)phenyl]methanone —— C18H24N4O
[(3S)-3-(diethylamino)pyrrolidin-1-yl]-[2-(1H-imidazol-2-yl)phenyl]methanone
—— (4S)-3-[1-(2-chlorophenyl)-5-methyl-1,2,4-triazole-3-carbonyl]-N-(3-methylphenyl)-1,3-thiazolidine-4-carboxamide —— C21H20ClN5O2S
(4S)-3-[1-(2-chlorophenyl)-5-methyl-1,2,4-triazole-3-carbonyl]-N-(3-methylphenyl)-1,3-thiazolidine-4-carboxamide
—— 2-(2,4-dimethylphenyl)-4-methyl-N-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]-1,3-thiazole-5-carboxamide —— C23H31N3O2S
2-(2,4-dimethylphenyl)-4-methyl-N-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]-1,3-thiazole-5-carboxamide
—— 1-(4-nitrophenyl)-N-[1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]pyrazole-3-carboxamide —— C20H25N5O4
1-(4-nitrophenyl)-N-[1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]pyrazole-3-carboxamide
—— [3-(4-methoxyphenyl)-5H-imidazo[1,5-c]quinazolin-6-yl]-morpholin-4-ylmethanone;hydrochloride —— C22H23ClN4O3
[3-(4-methoxyphenyl)-5H-imidazo[1,5-c]quinazolin-6-yl]-morpholin-4-ylmethanone;hydrochloride
—— 6-Chloro-2-(3-ethoxyphenyl)-3-(4-methylsulfonylphenyl)pyrazolo[1,5-a]pyridine —— C22H19ClN2O3S
6-Chloro-2-(3-ethoxyphenyl)-3-(4-methylsulfonylphenyl)pyrazolo[1,5-a]pyridine
—— 5-[(1R)-1-(3-bromopyridin-2-yl)sulfanylethyl]-3-phenyl-1,2,4-oxadiazole —— C15H12BrN3OS
5-[(1R)-1-(3-bromopyridin-2-yl)sulfanylethyl]-3-phenyl-1,2,4-oxadiazole
—— (4R)-N-(3-methylphenyl)-3-(5-methyl-1-phenylpyrazole-4-carbonyl)-1,3-thiazolidine-4-carboxamide —— C22H22N4O2S
(4R)-N-(3-methylphenyl)-3-(5-methyl-1-phenylpyrazole-4-carbonyl)-1,3-thiazolidine-4-carboxamide
—— [(2S)-2-(3-methoxyphenyl)azetidin-1-yl]-[4-(2-methyltetrazol-5-yl)phenyl]methanone —— C19H19N5O2
[(2S)-2-(3-methoxyphenyl)azetidin-1-yl]-[4-(2-methyltetrazol-5-yl)phenyl]methanone
—— ethyl 2-[cyclopropyl-[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C18H23N3O4S
ethyl 2-[cyclopropyl-[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— 7-(1,1-Dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2,3,6-trifluorophenyl)-1,2,4-triazolo[4,3-b]pyridazine —— C20H20F3N7O
7-(1,1-Dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2,3,6-trifluorophenyl)-1,2,4-triazolo[4,3-b]pyridazine
—— ethyl 2-[cyclopropyl-[(2S)-2-(3,4-difluorophenoxy)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C19H20F2N2O4S
ethyl 2-[cyclopropyl-[(2S)-2-(3,4-difluorophenoxy)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[cyclopropyl-[(2S)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate —— C18H24N4O3S
ethyl 2-[cyclopropyl-[(2S)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-4-methyl-1,3-thiazole-5-carboxylate
—— 4-[4-(4-fluorophenyl)-2-[2-(1-phenylethylamino)propyl]-1H-imidazol-5-yl]pyrimidin-2-amine —— C24H25FN6
4-[4-(4-fluorophenyl)-2-[2-(1-phenylethylamino)propyl]-1H-imidazol-5-yl]pyrimidin-2-amine
—— 4-methoxy-3,5-dimethyl-2-[[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylmethyl]pyridine —— C23H27N3O2S
4-methoxy-3,5-dimethyl-2-[[1-[[(2S)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylmethyl]pyridine
—— 2-(5-methylfuran-2-yl)-N-[1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]-1,3-thiazole-4-carboxamide —— C19H25N3O3S
2-(5-methylfuran-2-yl)-N-[1-[[(3S)-oxolan-3-yl]methyl]piperidin-4-yl]-1,3-thiazole-4-carboxamide
—— 1-(4-nitrophenyl)-N-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]pyrazole-3-carboxamide —— C20H25N5O4
1-(4-nitrophenyl)-N-[1-[[(3R)-oxolan-3-yl]methyl]piperidin-4-yl]pyrazole-3-carboxamide
—— (3R)-1-[2-[(5-phenyl-1H-pyrazole-4-carbonyl)amino]ethyl]piperidine-3-carboxamide —— C18H23N5O2
(3R)-1-[2-[(5-phenyl-1H-pyrazole-4-carbonyl)amino]ethyl]piperidine-3-carboxamide
—— 1-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethyl 4-[(Z)-(3,5-dioxo-1,2-oxazolidin-4-ylidene)methyl]benzoate —— C23H18N2O6
1-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethyl 4-[(Z)-(3,5-dioxo-1,2-oxazolidin-4-ylidene)methyl]benzoate
—— 4-[[3-[2-(2-Phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methylsulfonyl]-1,2-dihydropyrazol-3-one —— C21H19N3O5S
4-[[3-[2-(2-Phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methylsulfonyl]-1,2-dihydropyrazol-3-one
—— 4-[4-(cyanomethyl)-3-(4-thiophen-2-ylphenyl)-1H-pyrazol-5-yl]benzenesulfonamide —— C21H16N4O2S2
4-[4-(cyanomethyl)-3-(4-thiophen-2-ylphenyl)-1H-pyrazol-5-yl]benzenesulfonamide
—— [(3R)-3-(diethylamino)pyrrolidin-1-yl]-[2-(1H-imidazol-2-yl)phenyl]methanone —— C18H24N4O
[(3R)-3-(diethylamino)pyrrolidin-1-yl]-[2-(1H-imidazol-2-yl)phenyl]methanone
—— (4R)-N-(3-methylphenyl)-3-[2-(4-pyrazol-1-ylphenyl)acetyl]-1,3-thiazolidine-4-carboxamide —— C22H22N4O2S
(4R)-N-(3-methylphenyl)-3-[2-(4-pyrazol-1-ylphenyl)acetyl]-1,3-thiazolidine-4-carboxamide
—— 4-methoxy-3,5-dimethyl-2-[[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylmethyl]pyridine —— C23H27N3O2S
4-methoxy-3,5-dimethyl-2-[[1-[[(2R)-oxolan-2-yl]methyl]-5-phenylimidazol-2-yl]sulfanylmethyl]pyridine
—— (4R)-3-[1-(2-chlorophenyl)-5-methyl-1,2,4-triazole-3-carbonyl]-N-(3-methylphenyl)-1,3-thiazolidine-4-carboxamide —— C21H20ClN5O2S
(4R)-3-[1-(2-chlorophenyl)-5-methyl-1,2,4-triazole-3-carbonyl]-N-(3-methylphenyl)-1,3-thiazolidine-4-carboxamide
—— 5-[3-[6-(5-methyl-2-phenyl-4-oxazolylmethoxy)-2-benzofuranyl]propyl]-1H-tetrazole —— C23H21N5O3
5-[3-[6-(5-methyl-2-phenyl-4-oxazolylmethoxy)-2-benzofuranyl]propyl]-1H-tetrazole
—— 4-(3,4-dimethoxyphenyl)-3-tridecyl-1H-1,2,4-triazole-5-thione —— C23H37N3O2S
4-(3,4-dimethoxyphenyl)-3-tridecyl-1H-1,2,4-triazole-5-thione
—— [(2S)-2-(furan-2-yl)azepan-1-yl]-[3-(4-methylphenyl)-1H-pyrazol-5-yl]methanone —— C21H23N3O2
[(2S)-2-(furan-2-yl)azepan-1-yl]-[3-(4-methylphenyl)-1H-pyrazol-5-yl]methanone
—— 4-[4-[2-(2-Phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]sulfonyl-1,2-dihydropyrazol-3-one —— C20H17N3O5S
4-[4-[2-(2-Phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]sulfonyl-1,2-dihydropyrazol-3-one
—— N-ethyl-N-[(2R)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(2H-tetrazol-5-yl)benzamide —— C18H19N5O3
N-ethyl-N-[(2R)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(2H-tetrazol-5-yl)benzamide
—— (3R)-1-[2-[3-(2-methylpyrazol-3-yl)phenyl]pyrimidin-4-yl]piperidin-3-ol —— C19H21N5O
(3R)-1-[2-[3-(2-methylpyrazol-3-yl)phenyl]pyrimidin-4-yl]piperidin-3-ol
—— N-ethyl-N-[(2S)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(2H-tetrazol-5-yl)benzamide —— C18H19N5O3
N-ethyl-N-[(2S)-2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2-(2H-tetrazol-5-yl)benzamide
—— (3S)-1-[2-[3-(2-methylpyrazol-3-yl)phenyl]pyrimidin-4-yl]piperidin-3-ol —— C19H21N5O
(3S)-1-[2-[3-(2-methylpyrazol-3-yl)phenyl]pyrimidin-4-yl]piperidin-3-ol
—— butyl-2-[4-(4-{[(1Z)-amino(thien-2-yl)methylene]amino}phenyl)-1H-imidazol-2-yl]ethylcarbamate —— C21H25N5O2S
butyl-2-[4-(4-{[(1Z)-amino(thien-2-yl)methylene]amino}phenyl)-1H-imidazol-2-yl]ethylcarbamate
—— (3S)-1-[2-[(5-phenyl-1H-pyrazole-4-carbonyl)amino]ethyl]piperidine-3-carboxamide —— C18H23N5O2
(3S)-1-[2-[(5-phenyl-1H-pyrazole-4-carbonyl)amino]ethyl]piperidine-3-carboxamide
—— N-[(2R)-2-(azepan-1-yl)-2-phenylethyl]-2-(2,4-dimethyl-1,3-thiazol-5-yl)acetamide —— C21H29N3OS
N-[(2R)-2-(azepan-1-yl)-2-phenylethyl]-2-(2,4-dimethyl-1,3-thiazol-5-yl)acetamide
—— (3R)-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidine-3-carbonitrile —— C16H17N3S
(3R)-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidine-3-carbonitrile
—— N-[[(2R)-8-propan-2-yl-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl]-2-(1H-1,2,4-triazol-5-yl)benzamide —— C21H29N5O2
N-[[(2R)-8-propan-2-yl-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl]-2-(1H-1,2,4-triazol-5-yl)benzamide
—— (3S)-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidine-3-carbonitrile —— C16H17N3S
(3S)-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidine-3-carbonitrile
—— 1-(3,5-dimethyl-1-propylpyrazol-4-yl)-3-[[(3R)-1,1-dioxothiolan-3-yl]methyl]urea —— C14H24N4O3S
1-(3,5-dimethyl-1-propylpyrazol-4-yl)-3-[[(3R)-1,1-dioxothiolan-3-yl]methyl]urea
—— N-[[1-(2-chlorophenyl)-7-methoxy-4,5-dihydrobenzo[g]indazol-3-yl]methyl]piperidin-1-amine —— C24H27ClN4O
N-[[1-(2-chlorophenyl)-7-methoxy-4,5-dihydrobenzo[g]indazol-3-yl]methyl]piperidin-1-amine
—— 9-Heptan-4-yl-6-methyl-3-(2,4,6-trifluorophenyl)-1,3,5,9-tetrazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one —— C22H25F3N4O
9-Heptan-4-yl-6-methyl-3-(2,4,6-trifluorophenyl)-1,3,5,9-tetrazatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one