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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-2-pyrazol-1-ylbenzamide —— C18H16FN3O2
N-[(2S)-2-(4-fluorophenyl)-2-hydroxyethyl]-2-pyrazol-1-ylbenzamide
—— 1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-(2-methoxyphenyl)piperidine-4-carboxamide —— C24H27FN4O3
1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-N-(2-methoxyphenyl)piperidine-4-carboxamide
—— (1S)-N-[(5-bromofuran-2-yl)methyl]-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-methylethanamine —— C17H17BrFN3O2
(1S)-N-[(5-bromofuran-2-yl)methyl]-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-methylethanamine
—— N-[(3S)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidin-3-yl]methanesulfonamide —— C16H20F2N4O4S
N-[(3S)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidin-3-yl]methanesulfonamide
—— N-[(3R)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidin-3-yl]methanesulfonamide —— C16H20F2N4O4S
N-[(3R)-1-[[3-[2-(difluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidin-3-yl]methanesulfonamide
—— 2-[1-(3-chloro-4-methylphenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide —— C22H23ClFN3O2
2-[1-(3-chloro-4-methylphenyl)-3,5-dimethylpyrazol-4-yl]-N-[(2R)-2-(4-fluorophenyl)-2-hydroxyethyl]acetamide
—— N-[(2S)-1-piperidin-1-ylpropan-2-yl]-2-pyrazol-1-ylbenzamide —— C18H24N4O
N-[(2S)-1-piperidin-1-ylpropan-2-yl]-2-pyrazol-1-ylbenzamide
—— 2-[(3S)-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]-1,3-benzoxazole —— C23H23FN4O2
2-[(3S)-1-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]-1,3-benzoxazole
—— 3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-(4-pyridin-3-ylsulfonylpiperazin-1-yl)ethyl]-1,2,4-oxadiazole —— C20H22FN5O3S
3-(4-fluoro-3-methylphenyl)-5-[(1S)-1-(4-pyridin-3-ylsulfonylpiperazin-1-yl)ethyl]-1,2,4-oxadiazole
—— 2-[(3S)-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]-1,3-benzoxazole —— C23H23FN4O2
2-[(3S)-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]-1,3-benzoxazole
—— (1S)-N-[[3-(difluoromethoxy)-4-methoxyphenyl]methyl]-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-methylethanamine —— C21H22F3N3O3
(1S)-N-[[3-(difluoromethoxy)-4-methoxyphenyl]methyl]-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-methylethanamine
—— 4-[2-[[4-[(E)-N-[[2-(4-chlorophenyl)-1,3-oxazol-4-yl]methoxy]-C-methylcarbonimidoyl]-2,5-dimethylphenoxy]methyl]phenyl]-5-methoxy-2-methyl-1,2,4-triazol-3-one —— C31H30ClN5O5
4-[2-[[4-[(E)-N-[[2-(4-chlorophenyl)-1,3-oxazol-4-yl]methoxy]-C-methylcarbonimidoyl]-2,5-dimethylphenoxy]methyl]phenyl]-5-methoxy-2-methyl-1,2,4-triazol-3-one
—— N-[(3S)-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]methanesulfonamide —— C17H23FN4O3S
N-[(3S)-1-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperidin-3-yl]methanesulfonamide
—— 1-[5-(1-Methylcyclohexyl)-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]urea —— C34H41N5O3
1-[5-(1-Methylcyclohexyl)-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-(2-morpholin-4-ylethoxy)naphthalen-1-yl]urea
—— 4-(5-(4-methoxyphenyl)pyrazol-3-yloxy)-6-methoxy-7-(1-(2-methylsulphonylethyl)piperidin-4-ylmethoxy)quinazoline —— C28H33N5O6S
4-(5-(4-methoxyphenyl)pyrazol-3-yloxy)-6-methoxy-7-(1-(2-methylsulphonylethyl)piperidin-4-ylmethoxy)quinazoline
—— 5-(cyclopropylmethyl)-1-(3-fluorophenyl)-3-[(3S)-oxolan-3-yl]-1,2,4-triazole —— C16H18FN3O
5-(cyclopropylmethyl)-1-(3-fluorophenyl)-3-[(3S)-oxolan-3-yl]-1,2,4-triazole
—— N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]-2-(1H-imidazol-2-yl)-N-methylbenzamide —— C21H23N3O3
N-[(1S)-1-(2,4-dimethoxyphenyl)ethyl]-2-(1H-imidazol-2-yl)-N-methylbenzamide
—— [(6R)-6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-(1-methylimidazo[1,2-b]pyrazol-7-yl)methanone —— C14H21N5O3
[(6R)-6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-(1-methylimidazo[1,2-b]pyrazol-7-yl)methanone
—— 5-(cyclopropylmethyl)-1-(3-fluorophenyl)-3-[(3R)-oxolan-3-yl]-1,2,4-triazole —— C16H18FN3O
5-(cyclopropylmethyl)-1-(3-fluorophenyl)-3-[(3R)-oxolan-3-yl]-1,2,4-triazole
—— N'-[3-(2,6-dichloro-4-methoxyphenyl)-5-ethyl-2-methylpyrazolo[1,5-a]pyrimidin-7-yl]-N-(1-pyrimidin-2-ylpiperidin-4-yl)ethane-1,2-diamine —— C27H32Cl2N8O
N'-[3-(2,6-dichloro-4-methoxyphenyl)-5-ethyl-2-methylpyrazolo[1,5-a]pyrimidin-7-yl]-N-(1-pyrimidin-2-ylpiperidin-4-yl)ethane-1,2-diamine
—— 2-[5-(methoxymethyl)-3-[(3R)-oxolan-3-yl]-1,2,4-triazol-1-yl]benzoic acid —— C15H17N3O4
2-[5-(methoxymethyl)-3-[(3R)-oxolan-3-yl]-1,2,4-triazol-1-yl]benzoic acid
—— [(6S)-6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-(1-methylimidazo[1,2-b]pyrazol-7-yl)methanone —— C14H21N5O3
[(6S)-6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]-(1-methylimidazo[1,2-b]pyrazol-7-yl)methanone
—— 1-[(5-chloro-2-methoxyphenyl)methyl]-4-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]piperazine —— C21H25ClN6O
1-[(5-chloro-2-methoxyphenyl)methyl]-4-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]piperazine
—— (5S,7R)-N-[(3S)-1,1-dioxo-2,3-dihydrothiophen-3-yl]-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide —— C17H22N4O3S
(5S,7R)-N-[(3S)-1,1-dioxo-2,3-dihydrothiophen-3-yl]-3-(1,2,4-triazol-1-yl)adamantane-1-carboxamide
—— 1-methyl-3-phenyl-4-[[(3R)-3-pyrrolidin-1-ylpyrrolidin-1-yl]methyl]pyrazole —— C19H26N4
1-methyl-3-phenyl-4-[[(3R)-3-pyrrolidin-1-ylpyrrolidin-1-yl]methyl]pyrazole
—— (5R)-3-methyl-7-[(2-propan-2-yl-1,3-oxazol-4-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H21N3O3
(5R)-3-methyl-7-[(2-propan-2-yl-1,3-oxazol-4-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— 3-[(2R)-1-[[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl]piperidin-2-yl]-5-methyl-1,2-oxazole —— C19H21FN4O
3-[(2R)-1-[[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl]piperidin-2-yl]-5-methyl-1,2-oxazole
—— 3-[(2S)-1-[[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl]piperidin-2-yl]-5-methyl-1,2-oxazole —— C19H21FN4O
3-[(2S)-1-[[5-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl]piperidin-2-yl]-5-methyl-1,2-oxazole
—— N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]-2-(1H-imidazol-2-yl)-N-methylbenzamide —— C21H23N3O3
N-[(1R)-1-(2,4-dimethoxyphenyl)ethyl]-2-(1H-imidazol-2-yl)-N-methylbenzamide
—— 1-methyl-3-phenyl-4-[[(3S)-3-pyrrolidin-1-ylpyrrolidin-1-yl]methyl]pyrazole —— C19H26N4
1-methyl-3-phenyl-4-[[(3S)-3-pyrrolidin-1-ylpyrrolidin-1-yl]methyl]pyrazole
—— N-[3-[[2-(4,5-diphenyl-1,3-oxazol-2-yl)cyclohex-2-en-1-yl]methyl]phenyl]-1-phenylmethanesulfonamide —— C35H32N2O3S
N-[3-[[2-(4,5-diphenyl-1,3-oxazol-2-yl)cyclohex-2-en-1-yl]methyl]phenyl]-1-phenylmethanesulfonamide
—— 5-[[4-[[(3R)-oxolan-3-yl]methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole —— C18H24N4O2
5-[[4-[[(3R)-oxolan-3-yl]methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— 1-[(5-chloro-2-methoxyphenyl)methyl]-4-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]piperazine —— C21H25ClN6O
1-[(5-chloro-2-methoxyphenyl)methyl]-4-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]piperazine
—— 2-[5-(methoxymethyl)-3-[(3S)-oxolan-3-yl]-1,2,4-triazol-1-yl]benzoic acid —— C15H17N3O4
2-[5-(methoxymethyl)-3-[(3S)-oxolan-3-yl]-1,2,4-triazol-1-yl]benzoic acid
—— N-benzyl-N-[(3S)-1,1-dioxothiolan-3-yl]-2-propyl-1,3-thiazole-4-carboxamide —— C18H22N2O3S2
N-benzyl-N-[(3S)-1,1-dioxothiolan-3-yl]-2-propyl-1,3-thiazole-4-carboxamide
—— 5-[[4-[[(3S)-oxolan-3-yl]methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole —— C18H24N4O2
5-[[4-[[(3S)-oxolan-3-yl]methyl]piperazin-1-yl]methyl]-3-phenyl-1,2,4-oxadiazole
—— 1-[(4-Methoxyphenoxy)carbonyl-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]cyclopropane-1-carboxylic acid —— C31H30N2O7
1-[(4-Methoxyphenoxy)carbonyl-[[3-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]methyl]amino]cyclopropane-1-carboxylic acid
—— N'-[9-(2,6-dichloro-4-methoxyphenyl)-2,8-dimethylpurin-6-yl]-N-(1-pyrimidin-2-ylpiperidin-4-yl)ethane-1,2-diamine —— C25H29Cl2N9O
N'-[9-(2,6-dichloro-4-methoxyphenyl)-2,8-dimethylpurin-6-yl]-N-(1-pyrimidin-2-ylpiperidin-4-yl)ethane-1,2-diamine
—— [4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-(4-fluorophenyl)methanone —— C23H24F2N4O2
[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-(4-fluorophenyl)methanone
—— 1-cycloheptyl-4-[4-(4-fluorophenyl)-5-[2-[[(1S)-1-phenylethyl]amino]pyrimidin-4-yl]-1H-imidazol-2-yl]piperidin-4-ol —— C33H39FN6O
1-cycloheptyl-4-[4-(4-fluorophenyl)-5-[2-[[(1S)-1-phenylethyl]amino]pyrimidin-4-yl]-1H-imidazol-2-yl]piperidin-4-ol
—— [4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-(4-fluorophenyl)methanone —— C23H24F2N4O2
[4-[(1R)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-(4-fluorophenyl)methanone
—— (4-fluorophenyl)-[4-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]-1,4-diazepan-1-yl]methanone —— C21H23FN6O
(4-fluorophenyl)-[4-[(1S)-1-(1-phenyltetrazol-5-yl)ethyl]-1,4-diazepan-1-yl]methanone
—— N-benzyl-N-[(3R)-1,1-dioxothiolan-3-yl]-2-propyl-1,3-thiazole-4-carboxamide —— C18H22N2O3S2
N-benzyl-N-[(3R)-1,1-dioxothiolan-3-yl]-2-propyl-1,3-thiazole-4-carboxamide
—— (5S)-3-methyl-7-[(2-propan-2-yl-1,3-oxazol-4-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one —— C14H21N3O3
(5S)-3-methyl-7-[(2-propan-2-yl-1,3-oxazol-4-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
—— (4-fluorophenyl)-[4-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]-1,4-diazepan-1-yl]methanone —— C21H23FN6O
(4-fluorophenyl)-[4-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]-1,4-diazepan-1-yl]methanone
—— tert-butyl 4-[4-(4-fluorophenyl)-5-[2-[[(1S)-1-phenylethyl]amino]pyrimidin-4-yl]-1,3-oxazol-2-yl]piperidine-1-carboxylate —— C31H34FN5O3
tert-butyl 4-[4-(4-fluorophenyl)-5-[2-[[(1S)-1-phenylethyl]amino]pyrimidin-4-yl]-1,3-oxazol-2-yl]piperidine-1-carboxylate
—— [4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-(3-methylphenyl)methanone —— C24H27FN4O2
[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]-1,4-diazepan-1-yl]-(3-methylphenyl)methanone
—— (E)-3-[2-butyl-3-[2-(carboxymethoxy)-4-methoxyphenyl]imidazol-4-yl]-2-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]prop-2-enoic acid —— C28H30N2O9
(E)-3-[2-butyl-3-[2-(carboxymethoxy)-4-methoxyphenyl]imidazol-4-yl]-2-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]prop-2-enoic acid
—— (5E)-5-[[3-(furan-2-yl)-1-phenylpyrazol-4-yl]methylidene]-2-[(E)-2-phenylethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C26H17N5O2S
(5E)-5-[[3-(furan-2-yl)-1-phenylpyrazol-4-yl]methylidene]-2-[(E)-2-phenylethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— [4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(4-methoxyphenyl)methanone —— C23H25FN4O3
[4-[(1S)-1-[3-(4-fluoro-3-methylphenyl)-1,2,4-oxadiazol-5-yl]ethyl]piperazin-1-yl]-(4-methoxyphenyl)methanone